Céline Crauste

42
Documents

Publications

Publications

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Physicochemical and Computational Study of the Encapsulation of Resv-4′-LA and Resv-4′-DHA Lipophenols by Natural and HP-β-CDs

Ana Belén Hernández-Heredia , Dennis Alexander Silva-Cullishpuma , José Pedro Cerón-Carrasco , Ángel Gil-Izquierdo , Jordan Lehoux et al.

International Journal of Molecular Sciences, 2025, 26 (15), pp.7454. ⟨10.3390/ijms26157454⟩

Article dans une revue hal-05236440v1
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Mapping of Mycobacterial Enzymes Involved in Triacylglycerol Accumulation as Intrabacterial Lipid Inclusions Using Activity-Based Multitarget Inhibitor Probes

Romain Avellan , Jordan Lehoux , Thomas Francis , Tonia Dargham , Léa Celik et al.

ACS Infectious Diseases, 2025, 11 (6), pp.1589-1605. ⟨10.1021/acsinfecdis.5c00127⟩

Article dans une revue hal-05090485v1
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The polyamino‐isoprenyl enhancer NV716 enables the antibacterial activity of two families of multi‐target inhibitors against the ESKAPEE bacterium Enterobacter cloacae

Emma Forest , Jordan Lehoux , Alexandre Guy , Thierry Durand , Stéphane Audebert et al.

mLife, 2025, 4 (3), pp.259-274. ⟨10.1002/mlf2.70014⟩

Article dans une revue hal-05131779v1
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Total Synthesis and Analysis of Phenolic Phytoprostanes, Oxidized Derivatives of Lipophenols

Jordan Lehoux , Ángel Sánchez-Illana , Pablo Miralles , Valérie Bultel-Poncé , Thierry Durand et al.

Chemistry - A European Journal, 2025, pp.e02206. ⟨10.1002/chem.202502206⟩

Article dans une revue hal-05318121v1
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Mycobacterial cell division arrest and smooth‐to‐rough envelope transition using CRISPRi ‐mediated genetic repression systems

Vanessa Point , Wafaa Achache , Janïs Laudouze , Eliana Sepulveda Ramos , Mickaël Maziero et al.

FEBS Open Bio, 2025, ⟨10.1002/2211-5463.70172⟩

Article dans une revue hal-05513141v1
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Chemo-Enzymatic Synthesis of Mixed Docosahexaenoic Acid Phosphatidylcholine Conjugates

Jordan Lehoux , Felix Grosjean , Alexandre Lobo , Michel Lagarde , Nathalie Bernoud-Hubac et al.

European Journal of Organic Chemistry, 2025, ⟨10.1002/ejoc.202500083⟩

Article dans une revue hal-04994006v1
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Fluorescence‐based CRISPR interference system for controlled genetic repression and live single‐cell imaging in mycobacteria

Janïs Laudouze , Vanessa Point , Wafaa Achache , Céline Crauste , Stéphane Canaan et al.

FEBS Letters, 2024, 599 (4), pp.488-501. ⟨10.1002/1873-3468.15071⟩

Article dans une revue hal-04818719v1
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Antitubercular potential and p H ‐driven mode of action of salicylic acid derivatives

Janïs Laudouze , Thomas Francis , Emma Forest , Frédérique Mies , Jean‐michel Bolla et al.

FEBS Open Bio, 2024, 15 (3), pp.383-398. ⟨10.1002/2211-5463.13944⟩

Article dans une revue hal-04818672v1

A novel lipophenol quercetin derivative to prevent macular degeneration: Intravenous and oral formulations for preclinical pharmacological evaluation

Maxime Vincent , Jordan Lehoux , Claire Desmarty , Esperance Moine , Philippe Legrand et al.

International Journal of Pharmaceutics, 2024, 651, pp.123740. ⟨10.1016/j.ijpharm.2023.123740⟩

Article dans une revue hal-04386862v1
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Overview of alkyl quercetin lipophenol synthesis and its protective effect against carbonyl stress involved in neurodegeneration

Léa Otaegui , Jordan Lehoux , Leo Martin , Laurent Givalois , Thierry Durand et al.

Organic & Biomolecular Chemistry, In press, ⟨10.1039/d4ob00066h⟩

Article dans une revue hal-04520041v1
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Hydroxytyrosol fatty acid esters as new candidate markers for detecting olive oil inadequate storage conditions by UHPLC-QqQ-MS/MS

Sonia Medina , David Auñón , Jordan Lehoux , Thierry Durand , Céline Crauste et al.

Microchemical Journal, 2022, 181, pp.107656. ⟨10.1016/j.microc.2022.107656⟩

Article dans une revue hal-04102912v1

Synthesis of Fatty Acid Bioconjugates and Related Derivatives

Céline Crauste , Jean-Marie Galano , Alexandre Guy , Jordan Lehoux , Thierry Durand et al.

European Journal of Organic Chemistry, 2022, 2022 (21), pp.e202101502. ⟨10.1002/ejoc.202101502⟩

Article dans une revue hal-03692908v1
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Formulation and Evaluation of SNEDDS Loaded with Original Lipophenol for the Oral Route to Prevent Dry AMD and Stragardt’s Disease

Maxime Vincent , Laurianne Simon , Philippe Brabet , Philippe Legrand , Christophe Dorandeu et al.

Pharmaceutics, 2022, 14 (5), pp.1029. ⟨10.3390/pharmaceutics14051029⟩

Article dans une revue hal-03681400v1
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Unravelling the capacity of hydroxytyrosol and its lipophenolic derivates to modulate the H2O2-induced isoprostanoid profile of THP-1 monocytes by UHPLC-QqQ-MS/MS lipidomic workflow

Carolina Alemán-Jiménez , Raúl Domínguez-Perles , Federico Fanti , Juana Gallego-Gómez , Agustín Simonelli-Muñoz et al.

Microchemical Journal, 2021, 170, pp.106703. ⟨10.1016/j.microc.2021.106703⟩

Article dans une revue hal-03374014v1
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New lipophenols prevent carbonyl and oxidative stresses involved in macular degeneration

Espérance Moine , Manel Boukhallat , David Cia , Nathalie Jacquemot , Laurent Guillou et al.

Free Radical Biology and Medicine, 2021, 162, pp.367-382. ⟨10.1016/j.freeradbiomed.2020.10.316⟩

Article dans une revue hal-03067208v1
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Fatty Acid Hydroxytyrosyl Esters of Olive Oils Are Bioaccessible According to Simulated In Vitro Gastrointestinal Digestion: Unraveling the Role of Digestive Enzymes on Their Stability

Carolina Alemán-Jiménez , Raúl Domínguez-Perles , Juana I. Gallego-Gómez , Agustín Simonelli-Muñoz , Espérance Moine et al.

Journal of Agricultural and Food Chemistry, 2021, 69 (47), pp.14165-14175. ⟨10.1021/acs.jafc.1c05373⟩

Article dans une revue hal-04102919v1
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Isopropyl‐phloroglucinol‐DHA protects outer retinal cells against lethal dose of all‐ trans ‐retinal

Aurelie Cubizolle , David Cia , Espérance Moine , Nathalie Jacquemot , Laurent Guillou et al.

Journal of Cellular and Molecular Medicine, 2020, 24 (9), pp.5057-5069. ⟨10.1111/jcmm.15135⟩

Article dans une revue hal-02593070v1
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Preclinical pharmacology of a lipophenol in a mouse model of light-induced retinopathy

Nicolas Taveau , Aurélie Cubizolle , Laurent Guillou , Nicolas Pinquier , Espérance Moine et al.

Experimental & Molecular Medicine, 2020, 52 (7), pp.1090-1101. ⟨10.1038/s12276-020-0460-7⟩

Article dans une revue hal-04837096v1
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Combination of Lutein and Zeaxanthin, and DHA Regulated Polyunsaturated Fatty Acid Oxidation in H2O2-Stressed Retinal Cells

Ho Hang Leung , Jean-Marie Galano , Céline Crauste , Thierry Durand , Jetty Chung-Yung Lee

Neurochemical Research, 2020, 45 (5), pp.1007-1019. ⟨10.1007/s11064-020-02994-4⟩

Article dans une revue hal-02592871v1
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Dissecting the antibacterial activity of oxadiazolone-core derivatives against Mycobacterium abscessus

Abdeldjalil Madani , Ivy Mallick , Alexandre Guy , Céline Crauste , Thierry Durand et al.

PLoS ONE, 2020, 15 (9), pp.e0238178. ⟨10.1371/journal.pone.0238178⟩

Article dans une revue hal-02950695v1
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Targeted lipidomics profiling reveals the generation of hydroxytyrosol-fatty acids in hydroxytyrosol-fortified oily matrices: new analytical methodology and cytotoxicity evaluation

Sonia Medina , Raúl Dominguez-Perles , David Auñon , Espérance Moine , Thierry Durand et al.

Journal of Agricultural and Food Chemistry, 2020, ⟨10.1021/acs.jafc.0c01938⟩

Article dans une revue hal-04102923v1
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Bis-allylic Deuterated DHA Alleviates Oxidative Stress in Retinal Epithelial Cells

Mélissa Rosell , Martin Giera , Philippe Brabet , Mikhail S Shchepinov , Michel Guichardant et al.

Antioxidants , 2019, 8 (10), pp.447. ⟨10.3390/antiox8100447⟩

Article dans une revue hal-02308917v1
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New Lipophenol Antioxidants Reduce Oxidative Damage in Retina Pigment Epithelial Cells

Espérance Moine , Philippe Brabet , Laurent Guillou , Thierry Durand , Joseph Vercauteren et al.

Antioxidants , 2018, 7 (12), pp.197. ⟨10.3390/antiox7120197⟩

Article dans une revue hal-02308918v1
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LipG a bifunctional phospholipase/thioesterase involved in mycobacterial envelope remodeling

Pierre Santucci , Vanessa Point , Isabelle Poncin , Alexandre Guy , Céline Crauste et al.

Bioscience Reports, 2018, 38 (6), pp.BSR20181953. ⟨10.1042/BSR20181953⟩

Article dans une revue hal-01990097v1
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Oxadiazolone derivatives, new promising multi-target inhibitors against M. tuberculosis

Phuong Chi Nguyen , Vincent Delorme , Anaïs Benarouche , Alexandre Guy , Valérie Landry et al.

Bioorganic Chemistry, 2018, 81, pp.414-424. ⟨10.1016/j.bioorg.2018.08.025⟩

Article dans une revue hal-01875577v1
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Resveratrol-Linoleate protects from exacerbated endothelial permeability via a drastic inhibition of the MMP-9 activity

Aly Shamseddin , Céline Crauste , Erwann Durand , Pierre Villeneuve , Grégor Dubois et al.

Bioscience Reports, 2018, 38 (4), pp.BSR20171712. ⟨10.1042/BSR20171712⟩

Article dans une revue hal-01935636v1
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Resveratrol formulated with a natural deep eutectic solvent inhibits active matrix metalloprotease-9 in hormetic conditions.

Aly Shamseddin , Céline Crauste , Erwann Durand , Pierre Villeneuve , Gregor Dubois et al.

European Journal of Lipid Science and Technology, 2017, pp.1700171. ⟨10.1002/ejlt.201700171⟩

Article dans une revue hal-02308915v1
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Total Syntheses of Two bis-Allylic-Deuterated DHA Analogues

Mélissa Rosell , Maxime Villa , Thierry Durand , Jean-Marie Galano , Joseph Vercauteren et al.

Asian Journal of Organic Chemistry, 2017, 6 (3), pp.322 - 334. ⟨10.1002/ajoc.201600565⟩

Article dans une revue hal-01622325v1
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Phloroglucinol protects retinal pigment epithelium and photoreceptor against all-trans-retinal-induced toxicity and inhibits A2E formation

David Cia , Aurelie Cubizolle , Céline Crauste , Nathalie Jacquemot , Laurent Guillou et al.

Journal of Cellular and Molecular Medicine, 2016, 20 (9), pp.1651-1663. ⟨10.1111/jcmm.12857⟩

Article dans une revue hal-01871969v1
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Extra Virgin Olive Oil Reduced Polyunsaturated Fatty Acid and Cholesterol Oxidation in Rodent Liver: Is This Accounted for Hydroxytyrosol-Fatty Acid Conjugation?

Yiu Yiu Lee , Céline Crauste , Hualin Wang , Ho Hang Leung , Joseph Vercauteren et al.

Chemical Research in Toxicology, 2016, 29 (10), pp.1689-1698. ⟨10.1021/acs.chemrestox.6b00214⟩

Article dans une revue hal-01622331v1
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Omega-3 polyunsaturated lipophenols, how and why?

Céline Crauste , Mélissa Rosell , Thierry Durand , Joseph Vercauteren Article dans une revue hal-02309676v1
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Ligand Efficiency Driven Design of New Inhibitors of Mycobacterium tuberculosis Transcriptional Repressor EthR Using Fragment Growing, Merging, and Linking Approaches

Baptiste Villemagne , Marion Flipo , Nicolas Blondiaux , Celine Crauste , Sandra Malaquin et al.

Journal of Medicinal Chemistry, 2014, 57 (11), pp.4876-4888. ⟨10.1021/jm500422b⟩

Article dans une revue hal-02309782v1
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Unconventional surface plasmon resonance signals reveal quantitative inhibition of transcriptional repressor EthR by synthetic ligands

Céline Crauste , Nicolas Willand , Baptiste Villemagne , Marion Flipo , Eve Willery et al.

Analytical Biochemistry, 2014, 452, pp.54-66. ⟨10.1016/j.ab.2014.02.011⟩

Article dans une revue hal-02309788v1
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Synthesis and Evaluation of Polyunsaturated Fatty Acid-Phenol Conjugates as Anti-Carbonyl-Stress Lipophenols

Céline Crauste , Claire Vigor , Philippe Brabet , Madeleine Picq , Michel Lagarde et al.

European Journal of Organic Chemistry, 2014, 2014 (21), pp.4548-4561. ⟨10.1002/ejoc.201402282⟩

Article dans une revue istex hal-02309885v1
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Tuberculosis: The drug development pipeline at a glance

Baptiste Villemagne , Céline Crauste , Marion Flipo , Alain R. Baulard , Benoit Déprez et al.

European Journal of Medicinal Chemistry, 2012, 51, pp.1-16. ⟨10.1016/j.ejmech.2012.02.033⟩

Article dans une revue hal-02309791v1
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Synthesis of 2′,3′-Dideoxynucleoside Phosphoesters Using H-Phosphonate Chemistry on Soluble Polymer Support

Céline Crauste , Christian Périgaud , Suzanne Peyrottes

Journal of Organic Chemistry, 2011, 76 (3), pp.997-1000. ⟨10.1021/jo1022958⟩

Article dans une revue hal-02309881v1
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Asymmetric Synthesis of New β-Lactam Lipopeptides as Bacterial Signal Peptidase I Inhibitors

Céline Crauste , Matheus Froeyen , Jozef Anné , Piet Herdewijn

European Journal of Organic Chemistry, 2011, 2011 (19), pp.3437-3449. ⟨10.1002/ejoc.201100148⟩

Article dans une revue hal-02309796v1
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Insights into the Soluble PEG-Supported Synthesis of Cytosine-Containing Nucleoside 5′-Mono-, Di-, and Triphosphates

Céline Crauste , Christian Périgaud , Suzanne Peyrottes

Journal of Organic Chemistry, 2009, 74 (23), pp.9165-9172. ⟨10.1021/jo901931z⟩

Article dans une revue hal-02309892v1
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Development of a sensitive and selective LC/MS/MS method for the simultaneous determination of intracellular 1-beta-d-arabinofuranosylcytosine triphosphate (araCTP), cytidine triphosphate (CTP) and deoxycytidine triphosphate (dCTP) in a human follicular lymphoma cell line

Céline Crauste , Isabelle Lefebvre , Michael Hovaneissian , Jean Yves Puy , Béatrice Roy et al.

Journal of Chromatography B Biomedical Sciences and Applications, 2009, 877 (14-15), pp.1417-1425. ⟨10.1016/j.jchromb.2009.02.071⟩

Article dans une revue hal-02309584v1
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Magnesium(II)-coordinated Claisen rearrangement: a direct approach towards ulosonic acid derivatives

Claude Grison , Tomasz Krzysztof Olszewski , Céline Crauste , Alain Fruchier , Claude Didierjean et al.

Tetrahedron Letters, 2006, 47 (37), pp.6583-6586. ⟨10.1016/j.tetlet.2006.07.022⟩

Article dans une revue hal-02309971v1

Lipophenols as new therapeutics toward retinal degeneration: in vitro and in vivo pharmacological studies

Espérance Moine , Nicolas Taveau , Maxime Vincent , Laurent Guillou , Sylvie Bégu et al.

Annual Meeting of the Association for Research in Vision and Ophthalmology (ARVO 2020), Association for Research in Vision and Ophthalmology (ARVO), May 2020, En ligne (Etats-Unis), France. pp.4939

Communication dans un congrès hal-04570694v1