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GPER involvement in inflammatory pain
Baptiste Jouffre
,
Alexandre Acramel
,
Yves Jacquot
,
Laurence Daulhac
,
Christophe Mallet
Journal articles
hal-04337675v1
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Role of T CD4+ cells, macrophages, C-low threshold mechanoreceptors and spinal Cav3.2 channels in inflammation and related pain-like symptoms in murine inflammatory models
Elodie Picard
,
Nicolas Kerckhove
,
Amaury François
,
Ludivine Boudieu
,
Elisabeth Billard
Journal articles
hal-03790651v1
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An Updated Review on the Metabolite (AM404)-Mediated Central Mechanism of Action of Paracetamol (Acetaminophen): Experimental Evidence and Potential Clinical Impact
Christophe Mallet
,
Jules Desmeules
,
Rassa Pegahi
,
Alain Eschalier
Journal articles
hal-04337681v1
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Identification of a human estrogen receptor α tetrapeptidic fragment with dual antiproliferative and anti-nociceptive action
Baptiste Jouffre
,
Alexandre Acramel
,
Mathilde Belnou
,
Maria Francesca Santolla
,
Marianna Talia
Journal articles
hal-04087799v1
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Design, synthesis and biological evaluation of conformationnally-restricted analogues of E7010 as inhibitors of tubulin assembly (ITA) and vascular disrupting agents (VDA)
Vassili Prudhomme
,
Mélissa Cucca
,
Lionel Nauton
,
Elsa Andrieu
,
Mathilde Fereyrolles
Journal articles
hal-03959739v1
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Centrally expressed Cav3.2 T-type calcium channel is critical for the initiation and maintenance of neuropathic pain
Sophie L Fayad
,
Guillaume Ourties
,
Benjamin Le Gac
,
Baptiste Jouffre
,
Sylvain Lamoine
Journal articles
hal-03942925v1
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L’évaluation de la douleur chez l’animal de laboratoire
Christine Courteix
,
Alain Eschalier
,
Christophe Mallet
Journal articles
hal-03418812v1
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Paracetamol analogues conjugated by FAAH induce TRPV1-mediated antinociception without causing acute liver toxicity
Johan Å.Nilsson
,
Christophe Mallet
,
Kiseko Shionoya
,
Anders Blomgren
,
Anders Sundin
Journal articles
hal-04256629v1
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The Antitumor Peptide ERα17p Exerts Anti-Hyperalgesic and Anti-Inflammatory Actions Through GPER in Mice
Christophe Mallet
,
Ludivine Boudieu
,
Sylvain Lamoine
,
Catherine Coudert
,
Yves Jacquot
Journal articles
hal-04256623v1
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Paracetamol is a centrally acting analgesic using mechanisms located in the periaqueductal grey
David André Barrière
,
Fawzi Boumezbeur
,
Romain Dalman
,
Roberto Cadeddu
,
Damien Richard Richard
Journal articles
hal-02380187v1
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Inhibition of Cav3.2 calcium channels: A new target for colonic hypersensitivity associated with low‐grade inflammation
Elodie Picard
,
Frédéric Antonio Carvalho
,
Francina Agosti
,
Emmanuel Bourinet
,
Denis Ardid
Journal articles
hal-04317223v1
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Ethosuximide improves chronic pain-induced anxiety- and depression-like behaviors
Nicolas Kerckhove
,
Ludivine Boudieu
,
Guillaume Ourties
,
Justine Bourdier
,
Laurence Daulhac
Journal articles
hal-03488870v1
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A tetrapeptide class of biased analgesics from an Australian fungus targets the µ-opioid receptor
Zoltan Dekan
,
Setareh Sianati
,
Arsalan Yousuf
,
Katy Sutcliffe
,
Alexander Gillis
Proceedings of the National Academy of Sciences of the United States of America, 2019, 116 (44), pp.22353-22358. ⟨10.1073/pnas.1908662116⟩
Journal articles
hal-04257287v1
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The Peptide ERα17p Is a GPER Inverse Agonist that Exerts Antiproliferative Effects in Breast Cancer Cells
Rosamaria Lappano
,
Christophe Mallet
,
Bruno Rizzuti
,
Fedora Grande
,
Giulia Raffaella Galli
Cells, 2019, Molecular and Cellular Mechanisms of Cancers: Breast Cancer, 8 (6), pp.590. ⟨10.3390/cells8060590⟩
Journal articles
hal-02273130v1
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Optimization of the synthesis of a key intermediate for the preparation of glucocorticoids
Romain Jouve
,
Vincent Thery
,
Sylvie Ducki
,
Julie Helfenbein
,
Christophe Thiery
Journal articles
hal-01875170v1
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Assessment of the effectiveness and safety of Ethosuximide in the Treatment of non-Diabetic Peripheral Neuropathic Pain: EDONOT—protocol of a randomised, parallel, controlled, double-blinded and multicentre clinical trial
Nicolas Kerckhove
,
Christophe Mallet
,
Bruno Pereira
,
Chouki Chenaf
,
Christian Duale
Journal articles
hal-04337204v1
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FAAH inhibitors in the limelight, but regrettably
Christophe Mallet
,
Claude Dubray
,
Christian Dualé
International Journal of Clinical Pharmacology and Therapeutics, 2016, 54 (07), pp.498 - 501. ⟨10.5414/cp202687⟩
Journal articles
hal-04337687v1
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Colonic overexpression of the T‐type calcium channel Cav 3.2 in a mouse model of visceral hypersensitivity and in irritable bowel syndrome patients
J. Scanzi
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A. Accarie
,
E. Muller
,
Bruno Pereira
,
Y. Aissouni
Journal articles
hal-04317301v1
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Supra-spinal FAAH is required for the analgesic action of paracetamol in an inflammatory context
Romain Dalmann
,
Laurence Daulhac
,
Myriam Antri
,
Alain Eschalier
,
Christophe Mallet
Journal articles
hal-04326283v1
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Prise en charge médicamenteuse de la douleur
Christophe Mallet
,
Chouki Chenaf
Cerveau & psycho. L'essentiel, 2014, 17
Journal articles
hal-04273988v1
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Cav3.2 calcium channels: the key protagonist of the supraspinal effect of paracetamol
Nicolas Kerckhove
,
Christophe Mallet
,
Amaury François
,
Mathieu Boudes
,
Jean Chemin
Journal articles
hal-02356344v1
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Fatty Acid Amide Hydrolase-Dependent Generation of Antinociceptive Drug Metabolites Acting on TRPV1 in the Brain
David A Barrière
,
Christophe Mallet
,
Anders Blomgren
,
Charlotte Simonsen
,
Laurence Daulhac
Journal articles
hal-04337223v1
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Monoacylglycerols Activate TRPV1 – A Link between Phospholipase C and TRPV1
Peter M Zygmunt
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Anna Ermund
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Pouya Movahed
,
David A Andersson
,
Charlotte Simonsen
Journal articles
hal-04337227v1
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Mise au point sur les mécanismes de l'action antalgique du paracétamol
Christophe Mallet
,
Alain Eschalier
Urgence Pratique, 2012, 115, pp.29-31
Journal articles
hal-04273935v1
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Le paracétamol : un ancêtre plein d’avenir
Christophe Mallet
,
David Barrière
,
Alain Eschalier
Journal articles
hal-04337690v1
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Drug-induced GABA transporter currents enhance GABA release to induce opioid withdrawal behaviors
Elena Bagley
,
Jennifer Hacker
,
Vladimir Chefer
,
Christophe Mallet
,
Gavan Mcnally
Journal articles
hal-04337230v1
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TRPV1 in Brain Is Involved in Acetaminophen-Induced Antinociception
Christophe Mallet
,
David Barrière
,
Anna Ermund
,
Bo Jönsson
,
Alain Eschalier
Journal articles
hal-04326308v1
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Le paracétamol, de nouvelles cibles pour un vieux médicament
David André Barrière
,
Christophe Mallet
,
Alain Eschalier
La Lettre de l’Institut UPSA de la Douleur, 2010, 33
Journal articles
hal-04273458v1
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Endocannabinoids Can Open the Pain Gate
Macdonald Christie
,
Christophe Mallet
Journal articles
hal-04337579v1
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Endocannabinoid and serotonergic systems are needed for acetaminophen-induced analgesia
Christophe Mallet
,
Laurence Daulhac
,
Jérôme Bonnefont
,
Catherine Ledent
,
Monique Etienne
Journal articles
hal-04326295v1
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Acetaminophen recruits spinal p42/p44 mAPKs and GH/IGF-1 receptors to produce analgesia via the serotonergic system
Jérôme Bonnefont
,
Laurence Daulhac
,
Monique Etienne
,
Eric Chapuy
,
Christophe Mallet
Journal articles
hal-02659399v1
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Diabetes-Induced Mechanical Hyperalgesia Involves Spinal Mitogen-Activated Protein Kinase Activation in Neurons and Microglia via N -Methyl-D-aspartate-Dependent Mechanisms
Laurence Daulhac
,
Christophe Mallet
,
Christine Courteix
,
Monique Etienne
,
Eliane Duroux
Journal articles
hal-04326273v1
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