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Christophe Mallet

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Publications

GPER involvement in inflammatory pain

Baptiste Jouffre , Alexandre Acramel , Yves Jacquot , Laurence Daulhac , Christophe Mallet
Steroids, 2023, 200, pp.109311. ⟨10.1016/j.steroids.2023.109311⟩
Journal articles hal-04337675v1

Role of T CD4+ cells, macrophages, C-low threshold mechanoreceptors and spinal Cav3.2 channels in inflammation and related pain-like symptoms in murine inflammatory models

Elodie Picard , Nicolas Kerckhove , Amaury François , Ludivine Boudieu , Elisabeth Billard
British Journal of Pharmacology, 2023, 180 (4), pp.385-400. ⟨10.1111/bph.15956⟩
Journal articles hal-03790651v1
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An Updated Review on the Metabolite (AM404)-Mediated Central Mechanism of Action of Paracetamol (Acetaminophen): Experimental Evidence and Potential Clinical Impact

Christophe Mallet , Jules Desmeules , Rassa Pegahi , Alain Eschalier
Journal of Pain Research, 2023, 16, pp.1081 - 1094. ⟨10.2147/jpr.s393809⟩
Journal articles hal-04337681v1
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Identification of a human estrogen receptor α tetrapeptidic fragment with dual antiproliferative and anti-nociceptive action

Baptiste Jouffre , Alexandre Acramel , Mathilde Belnou , Maria Francesca Santolla , Marianna Talia
Scientific Reports, 2023, 13 (1), pp.1326. ⟨10.1038/s41598-023-28062-9⟩
Journal articles hal-04087799v1

Design, synthesis and biological evaluation of conformationnally-restricted analogues of E7010 as inhibitors of tubulin assembly (ITA) and vascular disrupting agents (VDA)

Vassili Prudhomme , Mélissa Cucca , Lionel Nauton , Elsa Andrieu , Mathilde Fereyrolles
European Journal of Medicinal Chemistry, 2022, 244, pp.114809. ⟨10.1016/j.ejmech.2022.114809⟩
Journal articles hal-03959739v1
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Centrally expressed Cav3.2 T-type calcium channel is critical for the initiation and maintenance of neuropathic pain

Sophie L Fayad , Guillaume Ourties , Benjamin Le Gac , Baptiste Jouffre , Sylvain Lamoine
eLife, 2022, 11, pp.e79018. ⟨10.7554/elife.79018⟩
Journal articles hal-03942925v1
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L’évaluation de la douleur chez l’animal de laboratoire

Christine Courteix , Alain Eschalier , Christophe Mallet
Douleur et Analgésie, 2021, 34 (2), pp.114-122. ⟨10.3166/dea-2021-0145⟩
Journal articles hal-03418812v1
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Paracetamol analogues conjugated by FAAH induce TRPV1-mediated antinociception without causing acute liver toxicity

Johan Å.Nilsson , Christophe Mallet , Kiseko Shionoya , Anders Blomgren , Anders Sundin
European Journal of Medicinal Chemistry, 2021, 213, pp.113042. ⟨10.1016/j.ejmech.2020.113042⟩
Journal articles hal-04256629v1

The Antitumor Peptide ERα17p Exerts Anti-Hyperalgesic and Anti-Inflammatory Actions Through GPER in Mice

Christophe Mallet , Ludivine Boudieu , Sylvain Lamoine , Catherine Coudert , Yves Jacquot
Frontiers in Endocrinology, 2021, 12, ⟨10.3389/fendo.2021.578250⟩
Journal articles hal-04256623v1

Paracetamol is a centrally acting analgesic using mechanisms located in the periaqueductal grey

David André Barrière , Fawzi Boumezbeur , Romain Dalman , Roberto Cadeddu , Damien Richard Richard
British Journal of Pharmacology, 2020, 177 (8), pp.1773-1792. ⟨10.1111/bph.14934⟩
Journal articles hal-02380187v1
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Inhibition of Cav3.2 calcium channels: A new target for colonic hypersensitivity associated with low‐grade inflammation

Elodie Picard , Frédéric Antonio Carvalho , Francina Agosti , Emmanuel Bourinet , Denis Ardid
British Journal of Pharmacology, 2019, 176 (7), pp.950-963. ⟨10.1111/bph.14608⟩
Journal articles hal-04317223v1
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Ethosuximide improves chronic pain-induced anxiety- and depression-like behaviors

Nicolas Kerckhove , Ludivine Boudieu , Guillaume Ourties , Justine Bourdier , Laurence Daulhac
European Neuropsychopharmacology, 2019, 29, pp.1419 - 1432. ⟨10.1016/j.euroneuro.2019.10.012⟩
Journal articles hal-03488870v1
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A tetrapeptide class of biased analgesics from an Australian fungus targets the µ-opioid receptor

Zoltan Dekan , Setareh Sianati , Arsalan Yousuf , Katy Sutcliffe , Alexander Gillis
Proceedings of the National Academy of Sciences of the United States of America, 2019, 116 (44), pp.22353-22358. ⟨10.1073/pnas.1908662116⟩
Journal articles hal-04257287v1
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The Peptide ERα17p Is a GPER Inverse Agonist that Exerts Antiproliferative Effects in Breast Cancer Cells

Rosamaria Lappano , Christophe Mallet , Bruno Rizzuti , Fedora Grande , Giulia Raffaella Galli
Cells, 2019, Molecular and Cellular Mechanisms of Cancers: Breast Cancer, 8 (6), pp.590. ⟨10.3390/cells8060590⟩
Journal articles hal-02273130v1

Optimization of the synthesis of a key intermediate for the preparation of glucocorticoids

Romain Jouve , Vincent Thery , Sylvie Ducki , Julie Helfenbein , Christophe Thiery
Steroids, 2018, 137, pp.14 - 21. ⟨10.1016/j.steroids.2018.06.007⟩
Journal articles hal-01875170v1
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Assessment of the effectiveness and safety of Ethosuximide in the Treatment of non-Diabetic Peripheral Neuropathic Pain: EDONOT—protocol of a randomised, parallel, controlled, double-blinded and multicentre clinical trial

Nicolas Kerckhove , Christophe Mallet , Bruno Pereira , Chouki Chenaf , Christian Duale
BMJ Open, 2016, 6 (12), pp.e013530. ⟨10.1136/bmjopen-2016-013530⟩
Journal articles hal-04337204v1
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FAAH inhibitors in the limelight, but regrettably

Christophe Mallet , Claude Dubray , Christian Dualé
International Journal of Clinical Pharmacology and Therapeutics, 2016, 54 (07), pp.498 - 501. ⟨10.5414/cp202687⟩
Journal articles hal-04337687v1

Colonic overexpression of the T‐type calcium channel Cav 3.2 in a mouse model of visceral hypersensitivity and in irritable bowel syndrome patients

J. Scanzi , A. Accarie , E. Muller , Bruno Pereira , Y. Aissouni
Neurogastroenterology & Motility, 2016, 28 (11), pp.1632-1640. ⟨10.1111/nmo.12860⟩
Journal articles hal-04317301v1

Supra-spinal FAAH is required for the analgesic action of paracetamol in an inflammatory context

Romain Dalmann , Laurence Daulhac , Myriam Antri , Alain Eschalier , Christophe Mallet
Neuropharmacology, 2015, 91, pp.63-70. ⟨10.1016/j.neuropharm.2014.11.006⟩
Journal articles hal-04326283v1

Prise en charge médicamenteuse de la douleur

Christophe Mallet , Chouki Chenaf
Cerveau & psycho. L'essentiel, 2014, 17
Journal articles hal-04273988v1
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Cav3.2 calcium channels: the key protagonist of the supraspinal effect of paracetamol

Nicolas Kerckhove , Christophe Mallet , Amaury François , Mathieu Boudes , Jean Chemin
Pain, 2014, 155 (4), pp.764-772. ⟨10.1016/j.pain.2014.01.015⟩
Journal articles hal-02356344v1
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Fatty Acid Amide Hydrolase-Dependent Generation of Antinociceptive Drug Metabolites Acting on TRPV1 in the Brain

David A Barrière , Christophe Mallet , Anders Blomgren , Charlotte Simonsen , Laurence Daulhac
PLoS ONE, 2013, 8 (8), pp.e70690. ⟨10.1371/journal.pone.0070690⟩
Journal articles hal-04337223v1
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Monoacylglycerols Activate TRPV1 – A Link between Phospholipase C and TRPV1

Peter M Zygmunt , Anna Ermund , Pouya Movahed , David A Andersson , Charlotte Simonsen
PLoS ONE, 2013, 8 (12), pp.e81618. ⟨10.1371/journal.pone.0081618⟩
Journal articles hal-04337227v1

Mise au point sur les mécanismes de l'action antalgique du paracétamol

Christophe Mallet , Alain Eschalier
Urgence Pratique, 2012, 115, pp.29-31
Journal articles hal-04273935v1

Le paracétamol : un ancêtre plein d’avenir

Christophe Mallet , David Barrière , Alain Eschalier
Therapies, 2012, 67 (4), pp.277-281. ⟨10.2515/therapie/2012039⟩
Journal articles hal-04337690v1

Drug-induced GABA transporter currents enhance GABA release to induce opioid withdrawal behaviors

Elena Bagley , Jennifer Hacker , Vladimir Chefer , Christophe Mallet , Gavan Mcnally
Nature Neuroscience, 2011, 14 (12), pp.1548-1554. ⟨10.1038/nn.2940⟩
Journal articles hal-04337230v1

TRPV1 in Brain Is Involved in Acetaminophen-Induced Antinociception

Christophe Mallet , David Barrière , Anna Ermund , Bo Jönsson , Alain Eschalier
PLoS ONE, 2010, 5 (9), pp.e12748. ⟨10.1371/journal.pone.0012748⟩
Journal articles hal-04326308v1

Le paracétamol, de nouvelles cibles pour un vieux médicament

David André Barrière , Christophe Mallet , Alain Eschalier
La Lettre de l’Institut UPSA de la Douleur, 2010, 33
Journal articles hal-04273458v1

Endocannabinoids Can Open the Pain Gate

Macdonald Christie , Christophe Mallet
Science Signaling, 2009, 2 (88), ⟨10.1126/scisignal.288pe57⟩
Journal articles hal-04337579v1

Endocannabinoid and serotonergic systems are needed for acetaminophen-induced analgesia

Christophe Mallet , Laurence Daulhac , Jérôme Bonnefont , Catherine Ledent , Monique Etienne
Pain, 2008, 139 (1), pp.190-200. ⟨10.1016/j.pain.2008.03.030⟩
Journal articles hal-04326295v1

Acetaminophen recruits spinal p42/p44 mAPKs and GH/IGF-1 receptors to produce analgesia via the serotonergic system

Jérôme Bonnefont , Laurence Daulhac , Monique Etienne , Eric Chapuy , Christophe Mallet
Molecular Pharmacology, 2007, 71 (2), pp.407-415. ⟨10.1124/mol.106.025775⟩
Journal articles hal-02659399v1

Diabetes-Induced Mechanical Hyperalgesia Involves Spinal Mitogen-Activated Protein Kinase Activation in Neurons and Microglia via N -Methyl-D-aspartate-Dependent Mechanisms

Laurence Daulhac , Christophe Mallet , Christine Courteix , Monique Etienne , Eliane Duroux
Molecular Pharmacology, 2006, 70 (4), pp.1246-1254. ⟨10.1124/mol.106.025478⟩
Journal articles hal-04326273v1

Traitements de la douleur, Approche pharmacologique

Nicolas Authier , Bénédicte Eschalier , Chouki Chenaf , Marie Zenut , Christophe Mallet
Traité de Médecine (5ème édition), TDM, pp.S10-P01-C11, 2018, 9782901094012
Book sections hal-04273871v1

Pharmacology and Mechanism of Action of Acetaminophen

Christophe Mallet , Alain Eschalier
Pharmacology of Pain, IASP press, 2015, 0931092787
Book sections hal-04337640v1