Christophe Mallet

Publications

Article dans une revue (33)

Commentary: harnessing the first peptidic modulator of the estrogen receptor GPER Rosamaria Lappano,Marcello Maggiolini,Christophe Mallet,Yves Jacquot Frontiers in Pharmacology, 2024, 15, pp.1413058. ⟨10.3389/fphar.2024.1413058⟩ Article dans une revue hal-04871148v1
GPER involvement in inflammatory pain Baptiste Jouffre,Alexandre Acramel,Yves Jacquot,Laurence Daulhac,Christophe Mallet Steroids, 2023, 200, pp.109311. ⟨10.1016/j.steroids.2023.109311⟩ Article dans une revue hal-04337675v1
Identification of a human estrogen receptor α tetrapeptidic fragment with dual antiproliferative and anti-nociceptive action Baptiste Jouffre,Alexandre Acramel,Mathilde Belnou,Maria Francesca Santolla,Marianna Taliaet al. Scientific Reports, 2023, 13 (1), pp.1326. ⟨10.1038/s41598-023-28062-9⟩ Article dans une revue hal-04087799v1
Role of T CD4+ cells, macrophages, C-low threshold mechanoreceptors and spinal Cav3.2 channels in inflammation and related pain-like symptoms in murine inflammatory models Elodie Picard,Nicolas Kerckhove,Amaury François,Ludivine Boudieu,Elisabeth Billardet al. British Journal of Pharmacology, 2023, 180 (4), pp.385-400. ⟨10.1111/bph.15956⟩ Article dans une revue hal-03790651v1
An Updated Review on the Metabolite (AM404)-Mediated Central Mechanism of Action of Paracetamol (Acetaminophen): Experimental Evidence and Potential Clinical Impact Christophe Mallet,Jules Desmeules,Rassa Pegahi,Alain Eschalier Journal of Pain Research, 2023, 16, pp.1081 - 1094. ⟨10.2147/jpr.s393809⟩ Article dans une revue hal-04337681v1
Centrally expressed Cav3.2 T-type calcium channel is critical for the initiation and maintenance of neuropathic pain Sophie L Fayad,Guillaume Ourties,Benjamin Le Gac,Baptiste Jouffre,Sylvain Lamoineet al. eLife, 2022, 11, pp.e79018. ⟨10.7554/elife.79018⟩ Article dans une revue hal-03942925v1
Design, synthesis and biological evaluation of conformationnally-restricted analogues of E7010 as inhibitors of tubulin assembly (ITA) and vascular disrupting agents (VDA) Vassili Prudhomme,Mélissa Cucca,Lionel Nauton,Elsa Andrieu,Mathilde Fereyrolleset al. European Journal of Medicinal Chemistry, 2022, 244, pp.114809. ⟨10.1016/j.ejmech.2022.114809⟩ Article dans une revue hal-03959739v1
The Antitumor Peptide ERα17p Exerts Anti-Hyperalgesic and Anti-Inflammatory Actions Through GPER in Mice Christophe Mallet,Ludivine Boudieu,Sylvain Lamoine,Catherine Coudert,Yves Jacquotet al. Frontiers in Endocrinology, 2021, 12, ⟨10.3389/fendo.2021.578250⟩ Article dans une revue hal-04256623v1
L’évaluation de la douleur chez l’animal de laboratoire Christine Courteix,Alain Eschalier,Christophe Mallet Douleur et Analgésie, 2021, 34 (2), pp.114-122. ⟨10.3166/dea-2021-0145⟩ Article dans une revue hal-03418812v1
Paracetamol analogues conjugated by FAAH induce TRPV1-mediated antinociception without causing acute liver toxicity Johan Å.Nilsson,Christophe Mallet,Kiseko Shionoya,Anders Blomgren,Anders Sundinet al. European Journal of Medicinal Chemistry, 2021, 213, pp.113042. ⟨10.1016/j.ejmech.2020.113042⟩ Article dans une revue hal-04256629v1
Paracetamol is a centrally acting analgesic using mechanisms located in the periaqueductal grey David André Barrière,Fawzi Boumezbeur,Romain Dalman,Roberto Cadeddu,Damien Richard Richardet al. British Journal of Pharmacology, 2020, 177 (8), pp.1773-1792. ⟨10.1111/bph.14934⟩ Article dans une revue hal-02380187v1
The Peptide ERα17p Is a GPER Inverse Agonist that Exerts Antiproliferative Effects in Breast Cancer Cells Rosamaria Lappano,Christophe Mallet,Bruno Rizzuti,Fedora Grande,Giulia Raffaella Galliet al. Cells, 2019, Molecular and Cellular Mechanisms of Cancers: Breast Cancer, 8 (6), pp.590. ⟨10.3390/cells8060590⟩ Article dans une revue hal-02273130v1
A tetrapeptide class of biased analgesics from an Australian fungus targets the µ-opioid receptor Zoltan Dekan,Setareh Sianati,Arsalan Yousuf,Katy Sutcliffe,Alexander Gilliset al. Proceedings of the National Academy of Sciences of the United States of America, 2019, 116 (44), pp.22353-22358. ⟨10.1073/pnas.1908662116⟩ Article dans une revue hal-04257287v1
Inhibition of Cav3.2 calcium channels: A new target for colonic hypersensitivity associated with low‐grade inflammation Elodie Picard,Frédéric Antonio Carvalho,Francina Agosti,Emmanuel Bourinet,Denis Ardidet al. British Journal of Pharmacology, 2019, 176 (7), pp.950-963. ⟨10.1111/bph.14608⟩ Article dans une revue hal-04317223v1
Ethosuximide improves chronic pain-induced anxiety- and depression-like behaviors Nicolas Kerckhove,Ludivine Boudieu,Guillaume Ourties,Justine Bourdier,Laurence Daulhacet al. European Neuropsychopharmacology, 2019, 29, pp.1419 - 1432. ⟨10.1016/j.euroneuro.2019.10.012⟩ Article dans une revue hal-03488870v1
Optimization of the synthesis of a key intermediate for the preparation of glucocorticoids Romain Jouve,Vincent Thery,Sylvie Ducki,Julie Helfenbein,Christophe Thieryet al. Steroids, 2018, 137, pp.14 - 21. ⟨10.1016/j.steroids.2018.06.007⟩ Article dans une revue hal-01875170v1
Colonic overexpression of the T‐type calcium channel Cav 3.2 in a mouse model of visceral hypersensitivity and in irritable bowel syndrome patients J. Scanzi,A. Accarie,E. Muller,Bruno Pereira,Y. Aissouniet al. Neurogastroenterology & Motility, 2016, 28 (11), pp.1632-1640. ⟨10.1111/nmo.12860⟩ Article dans une revue hal-04317301v1
FAAH inhibitors in the limelight, but regrettably Christophe Mallet,Claude Dubray,Christian Dualé International Journal of Clinical Pharmacology and Therapeutics, 2016, 54 (07), pp.498 - 501. ⟨10.5414/cp202687⟩ Article dans une revue hal-04337687v1
Assessment of the effectiveness and safety of Ethosuximide in the Treatment of non-Diabetic Peripheral Neuropathic Pain: EDONOT—protocol of a randomised, parallel, controlled, double-blinded and multicentre clinical trial Nicolas Kerckhove,Christophe Mallet,Bruno Pereira,Chouki Chenaf,Christian Dualeet al. BMJ Open, 2016, 6 (12), pp.e013530. ⟨10.1136/bmjopen-2016-013530⟩ Article dans une revue hal-04337204v1
Supra-spinal FAAH is required for the analgesic action of paracetamol in an inflammatory context Romain Dalmann,Laurence Daulhac,Myriam Antri,Alain Eschalier,Christophe Mallet Neuropharmacology, 2015, 91, pp.63-70. ⟨10.1016/j.neuropharm.2014.11.006⟩ Article dans une revue hal-04326283v1
Prise en charge médicamenteuse de la douleur Christophe Mallet,Chouki Chenaf Cerveau & psycho. L'essentiel, 2014, 17 Article dans une revue hal-04273988v1
Cav3.2 calcium channels: the key protagonist of the supraspinal effect of paracetamol Nicolas Kerckhove,Christophe Mallet,Amaury François,Mathieu Boudes,Jean Cheminet al. Pain, 2014, 155 (4), pp.764-772. ⟨10.1016/j.pain.2014.01.015⟩ Article dans une revue hal-02356344v1
Fatty Acid Amide Hydrolase-Dependent Generation of Antinociceptive Drug Metabolites Acting on TRPV1 in the Brain David A Barrière,Christophe Mallet,Anders Blomgren,Charlotte Simonsen,Laurence Daulhacet al. PLoS ONE, 2013, 8 (8), pp.e70690. ⟨10.1371/journal.pone.0070690⟩ Article dans une revue hal-04337223v1
Monoacylglycerols Activate TRPV1 – A Link between Phospholipase C and TRPV1 Peter M Zygmunt,Anna Ermund,Pouya Movahed,David A Andersson,Charlotte Simonsenet al. PLoS ONE, 2013, 8 (12), pp.e81618. ⟨10.1371/journal.pone.0081618⟩ Article dans une revue hal-04337227v1
Le paracétamol : un ancêtre plein d’avenir Christophe Mallet,David Barrière,Alain Eschalier Therapies, 2012, 67 (4), pp.277-281. ⟨10.2515/therapie/2012039⟩ Article dans une revue istex hal-04337690v1
Mise au point sur les mécanismes de l'action antalgique du paracétamol Christophe Mallet,Alain Eschalier Urgence Pratique, 2012, 115, pp.29-31 Article dans une revue hal-04273935v1
Drug-induced GABA transporter currents enhance GABA release to induce opioid withdrawal behaviors Elena Bagley,Jennifer Hacker,Vladimir Chefer,Christophe Mallet,Gavan Mcnallyet al. Nature Neuroscience, 2011, 14 (12), pp.1548-1554. ⟨10.1038/nn.2940⟩ Article dans une revue hal-04337230v1
TRPV1 in Brain Is Involved in Acetaminophen-Induced Antinociception Christophe Mallet,David Barrière,Anna Ermund,Bo Jönsson,Alain Eschalieret al. PLoS ONE, 2010, 5 (9), pp.e12748. ⟨10.1371/journal.pone.0012748⟩ Article dans une revue hal-04326308v1
Le paracétamol, de nouvelles cibles pour un vieux médicament David André Barrière,Christophe Mallet,Alain Eschalier La Lettre de l’Institut UPSA de la Douleur, 2010, 33 Article dans une revue hal-04273458v1
Endocannabinoids Can Open the Pain Gate Macdonald Christie,Christophe Mallet Science Signaling, 2009, 2 (88), ⟨10.1126/scisignal.288pe57⟩ Article dans une revue hal-04337579v1
Endocannabinoid and serotonergic systems are needed for acetaminophen-induced analgesia Christophe Mallet,Laurence Daulhac,Jérôme Bonnefont,Catherine Ledent,Monique Etienneet al. Pain, 2008, 139 (1), pp.190-200. ⟨10.1016/j.pain.2008.03.030⟩ Article dans une revue istex hal-04326295v1
Acetaminophen recruits spinal p42/p44 mAPKs and GH/IGF-1 receptors to produce analgesia via the serotonergic system Jérôme Bonnefont,Laurence Daulhac,Monique Etienne,Eric Chapuy,Christophe Malletet al. Molecular Pharmacology, 2007, 71 (2), pp.407-415. ⟨10.1124/mol.106.025775⟩ Article dans une revue hal-02659399v1
Diabetes-Induced Mechanical Hyperalgesia Involves Spinal Mitogen-Activated Protein Kinase Activation in Neurons and Microglia via N -Methyl-D-aspartate-Dependent Mechanisms Laurence Daulhac,Christophe Mallet,Christine Courteix,Monique Etienne,Eliane Durouxet al. Molecular Pharmacology, 2006, 70 (4), pp.1246-1254. ⟨10.1124/mol.106.025478⟩ Article dans une revue hal-04326273v1

Communication dans un congrès (1)

Paracetamol is a centrally acting analgesic using mechanisms located in the periaqueductal grey Christophe Mallet,David André Barrière,Fouad Boumezbeur,Romain Dalmann,Roberto Cadedduet al. Annual Meeting of French Society of Pharmacology and Therapeutics, Jun 2021, Online, France Communication dans un congrès hal-03745618v1

Poster de conférence (2)

Involvment of Cav3.2 calcium channels in osteoarthritis pain Guillaume Ourties,Laurence Daulhac,Alain Eschalier,Emmanuel Bourinet,Christophe Mallet European Pain Federation, Krakow Pain School, Jun 2019, Krakow (Cracovie), Poland Poster de conférence hal-04872989v1
Involvment of Cav3.2 calcium channels in oesteoarthritis pain Guillaume Ourties,Laurence Daulhac,Alain Eschalier,Christophe Mallet EFIC pain school, Jun 2019, cracovie, Poland Poster de conférence hal-02363984v1

Chapitre d'ouvrage (2)

Traitements de la douleur, Approche pharmacologique Nicolas Authier,Bénédicte Eschalier,Chouki Chenaf,Marie Zenut,Christophe Malletet al. Traité de Médecine (5ème édition), TDM, pp.S10-P01-C11, 2018, 9782901094012 Chapitre d'ouvrage hal-04273871v1
Pharmacology and Mechanism of Action of Acetaminophen Christophe Mallet,Alain Eschalier Pharmacology of Pain, IASP press, 2015, 0931092787 Chapitre d'ouvrage hal-04337640v1

Pré-publication, Document de travail (1)

Centrally expressed Cav3.2 T-type calcium channel is critical for the initiation and maintenance of neuropathic pain Sophie L Fayad,Guillaume Ourties,Benjamin Le Gac,Baptiste Jouffre,Sylvain Lamoineet al. 2022 Pré-publication, Document de travail hal-03746638v1