Elisabeth Davioud-Charvet

Identifiants chercheurs

IdHAL :

e-davioud-charvet

ORCID :

0000-0001-7026-4034

IdRef :

100470602

ResearcherID :

http://www.researcherid.com/rid/I-3805-2013

Présentation

Publications

Article dans une revue (54)

Synthesis of 1,2,3‐Triazole‐Methyl‐Menadione Derivatives: Evaluation of Electrochemical and Antiparasitic Properties against two Blood‐Dwelling Parasites Baptiste Dupouy,Tanja Karpstein,Cécile Häberli,Monica Cal,Matthias Rottmannet al. ChemMedChem, 2025, ⟨10.1002/cmdc.202400731⟩ Article dans une revue hal-04892049v1
The heme A synthase Cox15, as a target of redox-active 3-benzylmenadiones with antiparasitic activity Marcelo L Merli,Claudia Serot,Cindy Vallières,Julia A Cricco,Bogdan I Iorgaet al. Antimicrobial Agents and Chemotherapy, 2025, ⟨10.1128/aac.01161-25⟩ Article dans une revue hal-05426246v1
Design, Synthesis and Antiplasmodial Activities of a Library of Fluorine-Based 3-Benzylmenadiones Matthieu Roignant,Jimmy Richard,Maxime Donzel,Matthias Rottmann,Pascal Mäseret al. Molecules, 2025, 30 (11), pp.2446. ⟨10.3390/molecules30112446⟩ Article dans une revue hal-05137600v1
Proteomic Profiling of Antimalarial Plasmodione Using 3‐Benz(o)ylmenadione Affinity‐Based Probes Ilaria Iacobucci,Vittoria Monaco,Agnès Hovasse,Baptiste Dupouy,Rodrigue Keumoeet al. ChemBioChem, 2024, 25 (15), pp.e202400187. ⟨10.1002/cbic.202400187⟩ Article dans une revue hal-04728204v1
Regioselective Synthesis of Potential Non-Quinonoid Prodrugs of Plasmodione: Antiparasitic Properties Against Two Hemoglobin-Feeding Parasites and Drug Metabolism Studies Elena Cesar-Rodo,Baptiste Dupouy,Cécile Häberli,Jean-Marc Strub,David L Williamset al. Molecules, 2024, 29 (22), pp.5268. ⟨10.3390/molecules29225268⟩ Article dans une revue hal-04891107v1
3-Benzylmenadiones and their Heteroaromatic Analogues Target the Apicoplast of Apicomplexa Parasites: Synthesis and Bioimaging Studies Baptiste Dupouy,Maxime Donzel,Matthieu Roignant,Sarah Charital,Rodrigue Keumoeet al. ACS Infectious Diseases, 2024, 10 (10), pp.3553-3576. ⟨10.1021/acsinfecdis.4c00304⟩ Article dans une revue hal-04728547v1
Synthesis and anti-Chagas activity profile of a redox-active lead 3benzylmenadione revealed by high-content imaging Nathan Trometer,Jérémy Pecourneau,Liwen Feng,José A. Navarro-Huerta,Danielle Lazarin-Bidóiaet al. ACS Infectious Diseases, 2024, 10 (5), pp.1808-1838. ⟨10.1021/acsinfecdis.4c00137⟩ Article dans une revue hal-04583960v1
Click Coupling of Flavylium Dyes with Plasmodione Analogues: Towards New Redox‐Sensitive Pro‐Fluorophores Baptiste Dupouy,Leandro Cotos,Annika Binder,Lucie Slavikova,Matthias Rottmannet al. Chemistry - A European Journal, 2024, 31 (6), pp.e202403691. ⟨10.1002/chem.202403691⟩ Article dans une revue hal-04975248v1
Chemoselective Synthesis and Anti-Kinetoplastidal Properties of 2,6-Diaryl-4H-tetrahydro-thiopyran-4-one S-Oxides: Their Interplay in a Cascade of Redox Reactions from Diarylideneacetones Thibault Gendron,Don Antoine Lanfranchi,Nicole I Wenzel,Hripsimée Kessedjian,Beate Jannacket al. Molecules, 2024, 29 (7), pp.1620. ⟨10.3390/molecules29071620⟩ Article dans une revue hal-04583951v1
Synthesis and Photochemical Properties of Fluorescent Metabolites Generated from Fluorinated Benzoylmenadiones in Living Cells Nathan Trometer,Bogdan Cichocki,Quentin Chevalier,Jérémy Pécourneau,Jean-Marc Strubet al. Journal of Organic Chemistry, 2023, ⟨10.1021/acs.joc.3c00620⟩ Article dans une revue hal-04157610v1
Efficient Multigram-Scale Synthesis of 7-Substituted 3-Methyltetral-1-ones and 6-Fluoromenadione Nathan Trometer,Matthieu Roignant,Elisabeth Davioud-Charvet Organic Process Research and Development, 2022, acs.oprd.1c00421. ⟨10.1021/acs.oprd.1c00421⟩ Article dans une revue hal-03584209v1
Evaluation of ferrocenyl-containing gamma-hydroxy-gamma-lactam-derived tetramates as potential antiplasmodials Maurice Médebielle,Mourad Elhabiri,Elisabeth Davioud-Charvet,J.-P. Bouillon,Stéphane Picotet al. European Journal of Medicinal Chemistry, 2022 Article dans une revue hal-03826853v1
Evaluation of ferrocenyl-containing γ-hydroxy-γ-lactam-derived tetramates as potential antiplasmodials Nicolas Chopin,Julien Bosson,Shinya Iikawa,Stéphane Picot,Anne-Lise Bienvenuet al. European Journal of Medicinal Chemistry, 2022, 243, pp.114735. ⟨10.1016/j.ejmech.2022.114735⟩ Article dans une revue hal-03798632v1
The parasitophorous vacuole nutrient channel is critical for drug access in malaria parasites and modulates the artemisinin resistance fitness cost Paolo Mesén-Ramírez,Bärbel Bergmann,Mourad Elhabiri,Lei Zhu,Heidrun von Thienet al. Cell Host & Microbe, 2021, 29 (12), pp.1774-1787.e9. ⟨10.1016/j.chom.2021.11.002⟩ Article dans une revue hal-03544974v1
Bioinspired Photoredox Benzylation of Quinones Maxime Donzel,Mourad Elhabiri,Elisabeth Davioud-Charvet Journal of Organic Chemistry, 2021, 86 (15), pp.10055-10066. ⟨10.1021/acs.joc.1c00814⟩ Article dans une revue hal-03369963v1
Recent Advances in Direct C‐H Radical Alkylation of 1,4‐Quinones Maxime Donzel,Deniz Karabiyikli,Leandro Cotos Munoz,Mourad Elhabiri,Elisabeth Davioud-Charvet European Journal of Organic Chemistry, 2021, 2021 (25), pp.3622-3633. ⟨10.1002/ejoc.202100452⟩ Article dans une revue hal-03249134v1
Magnesium Complexes of Ladanein: A Beneficial Strategy for Stabilizing Polyphenolic Antivirals Xavier Martin Benlloch,Don Antoine Lanfranchi,Sibylle Haid,Thomas Pietschmann,Elisabeth Davioud‐charvetet al. European Journal of Inorganic Chemistry, 2021, 2021 (27), pp.2764-2772. ⟨10.1002/ejic.202100341⟩ Article dans une revue hal-03357249v1
A role for the succinate dehydrogenase in the mode of action of the redox-active antimalarial drug, plasmodione Pierre Mounkoro,Thomas Michel,Marie-Pierre Golinelli-Cohen,Stephanie Blandin,Elisabeth Davioud-Charvetet al. Free Radical Biology and Medicine, 2021, ⟨10.1016/j.freeradbiomed.2020.11.010⟩ Article dans une revue hal-03026255v1
A Class of Valuable (Pro-)Activity-Based Protein Profiling Probes: Application to the Redox-Active Antiplasmodial Agent, Plasmodione Bogdan Cichocki,Vrushali Khobragade,Maxime Donzel,Leandro Cotos Munoz,Stephanie Blandinet al. JACS Au, 2021, 1 (5), pp.669-689. ⟨10.1021/jacsau.1c00025⟩ Article dans une revue hal-03243960v1
Plasmodium falciparum Ferredoxin-NADP + Reductase-Catalyzed Redox Cycling of Plasmodione Generates Both Predicted Key Drug Metabolites: Implication for Antimalarial Drug Development Bogdan Cichocki,Maxime Donzel,Kim C. Heimsch,Mindaugas Lesanavičius,Liwen Fenget al. ACS Infectious Diseases, In press, ⟨10.1021/acsinfecdis.1c00054⟩ Article dans une revue hal-03243991v1
Repurposing Auranofin and Evaluation of a New Gold(I) Compound for the Search of Treatment of Human and Cattle Parasitic Diseases: From Protozoa to Helminth Infections Liwen Feng,Sébastien Pomel,Perle Latre de Late,Alexandre Taravaud,Philippe M Loiseauet al. Molecules, 2020, 25 (21), pp.5075. ⟨10.3390/molecules25215075⟩ Article dans une revue hal-03038691v1
Selenium Status in Elderly People: Longevity and Age-Related Diseases Harry Robberecht,Tess de Bruyne,Elisabeth Davioud-Charvet,John Mackrill,Nina Hermans Current Pharmaceutical Design, 2019, 25 (15), pp.1694-1706. ⟨10.2174/1381612825666190701144709⟩ Article dans une revue istex hal-02325568v1
Author Correction: Arylmethylamino steroids as antiparasitic agents Reimar Krieg,Esther Jortzik,Alice-Anne Goetz,Stéphanie Blandin,Sergio Wittlinet al. Nature Communications, 2019, 10 (1), ⟨10.1038/s41467-019-11018-x⟩ Article dans une revue hal-02325972v1
Investigating the mode of action of the redox-active antimalarial drug plasmodione using the yeast model Pierre Mounkoro,Thomas Michel,Stéphanie Blandin,Marie-Pierre Golinelli-Cohen,Elisabeth Davioud-Charvetet al. Free Radical Biology and Medicine, 2019, 141, pp.269-278. ⟨10.1016/j.freeradbiomed.2019.06.026⟩ Article dans une revue hal-02170571v1
Physicochemical Properties Govern the Activity of Potent Antiviral Flavones Xavier Martin-Benlloch,Sibylle Haid,Alexandra Novodomska,Frank Rominger,Thomas Pietschmannet al. ACS Omega, 2019, 4 (3), pp.4871-4887. ⟨10.1021/acsomega.8b03332⟩ Article dans une revue hal-02325555v1
Antiplasmodial Activity of Nitroaromatic Compounds: Correlation with Their Reduction Potential and Inhibitory Action on Plasmodium falciparum Glutathione Reductase Audronė Marozienė,Mindaugas Lesanavičius,Elisabeth Davioud-Charvet,Alessandro Aliverti,Philippe Grellieret al. Molecules, 2019, 24 (24), pp.4509. ⟨10.3390/molecules24244509⟩ Article dans une revue hal-03038823v1
A Mild and Versatile Friedel‐Crafts Methodology for the Diversity‐Oriented Synthesis of Redox‐Active 3‐Benzoylmenadiones with Tuneable Redox Potentials Leandro Cotos,Maxime Donzel,Mourad Elhabiri,Elisabeth Davioud-Charvet Chemistry - A European Journal, 2019, 26 (15), pp.3314-3325. ⟨10.1002/chem.201904220⟩ Article dans une revue hal-02408960v1
Synthesis of plasmodione metabolites and 13C-enriched plasmodione as chemical tools for drug metabolism investigation Liwen Feng,Don Antoine Lanfranchi,Leandro Cotos Munoz,Elena Cesar Rodo,Katharina Ehrhardtet al. Organic & Biomolecular Chemistry, 2018, 15, pp.2647-2665. ⟨10.1039/C8OB00227D⟩ Article dans une revue hal-02161631v1
AntiMalarial Mode of Action (AMMA) Database: Data Selection, Verification and Chemical Space Analysis Pavel Sidorov,Elisabeth Davioud-Charvet,Gilles Marcou,Dragos Horvath,Alexandre Varnek Molecular Informatics, 2018, 37 (9-10), pp.1800021. ⟨10.1002/minf.201800021⟩ Article dans une revue hal-02325960v1
Iron(iii) coordination properties of ladanein, a flavone lead with a broad-spectrum antiviral activity Xavier Martin Benlloch,D Jacquemin,Elisabeth Davioud-Charvet,Mourad Elhabiri,A Novodomska New Journal of Chemistry, 2018, 42 (10), pp.8074-8087. ⟨10.1039/C7NJ04867J⟩ Article dans une revue hal-02161640v1
Pharmacomodulation of the antimalarial plasmodione: synthesis of biaryl- and N-arylalkylamine analogues, antimalarial activities and physicochemical properties Karène Urgin,Mouhamad Jida,Katharina Ehrhardt,T Müller,M Lanzeret al. Molecules, 2017, 22, pp.1-32. ⟨10.3390/molecules22010161⟩ Article dans une revue hal-02177398v1
Arylmethylamino steroids as novel antiparasitic agents R Krieg,E Jortzik,Alice-Anne Goetz,Stephanie Blandin,S Wittlinet al. Nature Communications, 2017, 8, ⟨10.1038/ncomms14478⟩ Article dans une revue hal-02158243v1
A high susceptibility to redox imbalance of the transmissible stages of Plasmodium falciparum revealed with a luciferase-based mature gametocyte assay Giulia Siciliano,T.R. Santha Kumar,Roberta Bona,Grazia Camarda,Maria Maddalena Calabrettaet al. Molecular Microbiology, 2017, 104, pp.306-318. ⟨10.1111/mmi.13626⟩ Article dans une revue hal-02161655v1
A Redox-Active Fluorescent pH Indicator for Detecting Plasmodium falciparum Strains with Reduced Responsiveness to Quinoline Antimalarial Drugs Mouhamad Jida,Cecilia Sanchez,Karène Urgin,Katharina Ehrhardt,S Mounienet al. ACS Infectious Diseases, 2017, 3, pp.119-131. ⟨10.1021/acsinfecdis.5b00141⟩ Article dans une revue hal-02177403v1
QSAR modeling1. and chemical space analysis of antimalarial compounds Pavel Sidorov,B Viira,Elisabeth Davioud-Charvet,U Maran,Gilles Marcouet al. JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 2017, 31, pp.441-451. ⟨10.1007/s10822-017-0019-4⟩ Article dans une revue hal-02177404v1
In Silico Mining for Antimalarial Structure-Activity Knowledge and Discovery of Novel Antimalarial Curcuminoids Birgit Viira,Thibault Gendron,Don Antoine Lanfranchi,Sandrine Cojean,Dragos Horvathet al. Molecules, 2016, 21 (7), pp.853. ⟨10.3390/molecules21070853⟩ Article dans une revue hal-03150675v1
A Platform of Regioselective Methodologies to Access to Polysubstituted 2-Methyl-1,4-Naphthoquinones Derivatives: Scope and Limitations Elena Cesar Rodo,Liwen Feng,Mouhamad Jida,Katharina Ehrhardt,Max Bielitzaet al. European Journal of Organic Chemistry, 2016, 2016 (11), pp.1982-1993. ⟨10.1002/ejoc.201600144⟩ Article dans une revue istex hal-03537379v1
Redox Polypharmacology as an Emerging Strategy to Combat Malarial Parasites Pavel Sidorov,Israel Desta,Matthieu Chessé,Dragos Horvath,Gilles Marcouet al. ChemMedChem, 2016, 11 (12), pp.1339-1351. ⟨10.1002/cmdc.201600009⟩ Article dans une revue istex hal-03151671v1
The Redox Cycler Plasmodione Is a Fast-Acting Antimalarial Lead Compound with Pronounced Activity against Sexual and Early Asexual Blood-Stage Parasites Katharina Ehrhardt,Christiane Deregnaucourt,Alice-Anne Goetz,Tzvetomira Tzanova,Valentina Galloet al. Antimicrobial Agents and Chemotherapy, 2016, 60 (9), pp.5146-5158. ⟨10.1128/AAC.02975-15⟩ Article dans une revue hal-01455775v1
Antimalarial NADPH-Consuming Redox-Cyclers As Superior Glucose-6-Phosphate Dehydrogenase Deficiency Copycats Max Bielitza,Didier Belorgey,Katharina Ehrhardt,Laure Johann,Don Antoine Lanfranchiet al. Antioxidants and Redox Signaling, 2015, 22 (15), pp.1337-1351. ⟨10.1089/ars.2014.6047⟩ Article dans une revue hal-05016881v1
Double-drug development against antioxidant enzymes from Plasmodium falciparum Christophe Biot,Jean Dessolin,Philippe Grellier,Elisabeth Davioud-Charvet Redox Report, 2013, 8 (5), pp.280-283. ⟨10.1179/135100003225002916⟩ Article dans une revue mnhn-02867482v1
Exploring the trifluoromenadione core as a template to design antimalarial redox-active agents interacting with glutathione reductase D.A. Lanfranchi,D. Belorgey,T. Müller,H. Vezin,M. Lanzeret al. Organic & Biomolecular Chemistry, 2012, 10, pp.4795 - 4806. ⟨10.1039/C2OB25229E⟩ Article dans une revue hal-00702812v1
A Plant-Derived Flavonoid Inhibits Entry of All HCV Genotypes Into Human Hepatocytes Sibylle Haid,Alexandra Novodomská,Juliane Gentzsch,Christina Grethe,Silvia Geuenichet al. Gastroenterology, 2012, 143 (1), pp.213-222.e5. ⟨10.1053/j.gastro.2012.03.036⟩ Article dans une revue hal-05017702v1
A Glutathione Reductase-Catalyzed Cascade of Redox Reactions to Bioactivate Potent Antimalarial 1,4-Naphthoquinones - A New Strategy to Combat Malarial Parasites Tobias Müller,Laure Johann,Beate Jannack,Margit Brückner,Don Antoine Lanfranchiet al. Journal of the American Chemical Society, 2011, 133 (30), pp.11557-11571. ⟨10.1021/ja201729z⟩ Article dans une revue hal-03406270v1
Antimalarial activities of ferroquine conjugates with either glutathione reductase inhibitors or glutathione depletors via a hydrolyzable amide linker Natascha Chavain,Elisabeth Davioud-Charvet,Xavier Trivelli,Linda Mbeki,M. Rottmannet al. Bioorganic and Medicinal Chemistry, 2009, 17 (23), pp.8048-8059. ⟨10.1016/j.bmc.2009.10.008⟩ Article dans une revue istex hal-00642006v1
The aza-analogues of 1,4-naphthoquinones are potent substrates and inhibitors of plasmodial thioredoxin and glutathione reductases and of human erythrocyte glutathione reductase Christophe Morin,Tatiana Besset,Jean-Claude Moutet,Martine Fayolle,Margit Brückneret al. Organic & Biomolecular Chemistry, 2008, 6 (15), pp.2731. ⟨10.1039/B802649C⟩ Article dans une revue istex hal-02541797v1
A Fluoro Analogue of the Menadione Derivative 6-[2‘-(3‘-Methyl)-1‘,4‘-naphthoquinolyl]hexanoic Acid Is a Suicide Substrate of Glutathione Reductase. Crystal Structure of the Alkylated Human Enzyme† Holger Bauer,Karin Fritz-Wolf,Andreas Winzer,Sebastian Kühner,Susan Littleet al. Journal of the American Chemical Society, 2006, The Journal of physical chemistry, 128 (33), pp.10784-10794. ⟨10.1021/ja061155v⟩ Article dans une revue istex hal-03378811v1
Undressing of Phosphine Gold(I) Complexes as Irreversible Inhibitors of Human Disulfide Reductases Sabine Urig,Karin Fritz-Wolf,Régis Réau,Christel Herold-Mende,Katalin Tóthet al. Angewandte Chemie International Edition, 2006, 45 (12), pp.1881-1886. ⟨10.1002/anie.200502756⟩ Article dans une revue istex hal-01090379v1
Trypanosoma cruzi prolyl oligopeptidase Tc80 is involved in nonphagocytic mammalian cell invasion by trypomastigotes. P. Grellier,S. Vendeville,R. Joyeau,I. M. D. Bastos,H. Drobecqet al. Journal of Biological Chemistry, 2001, 276, pp.47078-47086 Article dans une revue hal-00086392v1
Glutathione-dependent activities of $Trypanosoma\ cruzi$ p52 makes it a new member of the thiol:disulphide oxidoreductase family Mireille Moutiez,Eric Quéméneur,Christian Sergheraert,Valérie Lucas,André Tartaret al. Biochemical Journal, 1997, 322 (1), pp.43-48. ⟨10.1042/bj3220043⟩ Article dans une revue hal-03637701v1
High sensitivity to auxin is a common feature of hairy root W.H. Shen,E. Davioud,C. David,H. Barbier-Brygoo Plant Physiology, 1990, 94, pp.554-560 Article dans une revue hal-02713794v1
Production of indole alkaloids by in vitro root cultures from Catharanthus trichophyllus E. Davioud,C. Kan,J. Hamon,J. Tempe,H.P. Husson Phytochemistry, 1989, 28 (10), pp.2675-2680 Article dans une revue hal-02722026v1
Cucumopine. A new T-DNA- encoded opine in hairy root and crown-gall E. Davioud,A. Petit,M.E. Tate,M.H. Ryder,J. Tempe Phytochemistry, 1988, 27 (8), pp.2429-2433 Article dans une revue hal-02727299v1
Structure and synthesis of cucumopine, a new crown gall and hairy-root opine E. Davioud,J.C. Quirion,M.E. Tate,J. Tempe,H.P. Husson Heterocycles, 1988, 27 (10), n.p Article dans une revue hal-02716461v1