Gilles Hanquet

40
Documents

Publications

Publications

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Phenylseleno trifluoromethoxylation of alkenes

Clément Delobel , Armen Panossian , Gilles Hanquet , Frédéric R Leroux , Fabien Toulgoat et al.
Beilstein Journal of Organic Chemistry, 2024, 20, pp.2434-2441. ⟨10.3762/bjoc.20.207⟩
Article dans une revue hal-04711420 v1
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Unlocking the Power of Acyl Fluorides: A Comprehensive Guide to Synthesis and Properties

Clémence Bonnefoy , Adrien Gallego , Clément Delobel , Betty Raynal , Maxime Decourt et al.
European Journal of Organic Chemistry, 2024, 27 (18), pp.e202400142. ⟨10.1002/ejoc.202400142⟩
Article dans une revue hal-04591439 v1
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Selectivity of N(2)-substituted oxotriazinoindole aldose reductase inhibitors is determined by the interaction pattern with Pro301-Arg312 loop of aldehyde reductase

Lucia Kováčiková , Sunil Gaikwad , Kristína Almášiová , Ambroz Almássy , Gabriela Addová et al.
Medicinal Chemistry Research, 2024, 33 (3), pp.492-503. ⟨10.1007/s00044-024-03194-3⟩
Article dans une revue hal-04508563 v1
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Trifluoromethoxylation of Arynes using 2,4‐Dinitro‐1‐(trifluoromethoxybenzene) as Trifluoromethoxide Anion Source

Lilian Wisson , Gilles Hanquet , Fabien Toulgoat , Thierry Billard , Armen Panossian et al.
European Journal of Organic Chemistry, In press, 27 (28), pp.e202400388. ⟨10.1002/ejoc.202400388⟩
Article dans une revue hal-04591124 v1
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The Diels-Alder reaction of 1,4-quinones in hexafluoroisopropanol

Loïc Jeanmart , Kalina Mambourg , Gilles hanquet , Steve Lanners
ARKIVOC - Online Journal of Organic Chemistry, 2024, 2024 (1), ⟨10.24820/ark.5550190.p012.140⟩
Article dans une revue hal-04467685 v1
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Comprehensive Study and Development of a Metal-Free and Mild Nucleophilic Trifluoromethoxylation

Clémence Bonnefoy , Armen Panossian , Gilles Hanquet , Frédéric Leroux , Fabien Toulgoat et al.
Chemistry - A European Journal, 2023, 29 (46), ⟨10.1002/chem.202301513⟩
Article dans une revue hal-04165325 v1
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Direct Deprotonative Functionalization of α,α‐Difluoromethyl Ketones using a Catalytic Organosuperbase

Amélia Messara , Armen Panossian , Koichi Mikami , Gilles Hanquet , Frederic Leroux
Angewandte Chemie International Edition, In press, ⟨10.1002/anie.202215899⟩
Article dans une revue hal-03933942 v1
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Difluoromethoxylated Ketones as Building Blocks for the Synthesis of Challenging OCF2H‐Bearing N‐Heterocycles.

Anaïs Loison , Gilles Hanquet , Fabien Toulgoat , Thierry Billard , Armen Panossian et al.
European Journal of Organic Chemistry, 2023, 26 (42), pp.e202300695. ⟨10.1002/ejoc.202300695⟩
Article dans une revue hal-04163739 v2
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Study of Carbamoyl Fluoride: Synthesis, Properties and Applications

Clémence Bonnefoy , Emmanuel Chefdeville , Christian Tourvieille , Armen Panossian , Gilles Hanquet et al.
Chemistry - A European Journal, 2022, 28 (43), ⟨10.1002/chem.202201589⟩
Article dans une revue hal-03744602 v1
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Ketenimines as Intermediates To Access Difluoromethoxylated Scaffolds

Anaïs Loison , Gilles Hanquet , Fabien Toulgoat , Thierry Billard , Armen Panossian et al.
Organic Letters, 2022, ⟨10.1021/acs.orglett.2c03283⟩
Article dans une revue hal-03843401 v1
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Access to 12-Membered Cyclic ortho , meta -Diarylheptanoids: Total Synthesis of Actinidione via Isomyricanone

Paul Massé , Sabine Choppin , Lucia Chiummiento , Françoise Colobert , Gilles Hanquet
Journal of Organic Chemistry, 2021, 86 (3), pp.3033-3040. ⟨10.1021/acs.joc.0c02489⟩
Article dans une revue hal-03228806 v1
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Direct trifluoromethoxylation without OCF3 ‐carrier via in‐situ generation of fluorophosgene

Jérémy Saiter , Thomas Guérin , Morgan Donnard , Armen Panossian , Gilles Hanquet et al.
European Journal of Organic Chemistry, 2021, 2021 (22), ⟨10.1002/ejoc.202100429⟩
Article dans une revue hal-03228836 v1
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Recent synthetic methods towards the –OCHF2 moiety

Anaïs Loison , Fabien Toulgoat , Thierry Billard , Gilles Hanquet , Armen Panossian et al.
Tetrahedron, 2021, 99, pp.132458. ⟨10.1016/j.tet.2021.132458⟩
Article dans une revue hal-03517915 v1
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Study of a Stable “Trifluoromethoxide Anion Solution” Arising from 2,4‐Dinitro‐Trifluoromethoxybenzene

Clémence Bonnefoy , Emmanuel Chefdeville , Armen Panossian , Gilles Hanquet , Frédéric R. Leroux et al.
Chemistry - A European Journal, 2021, 27 (64), pp.15986-15991. ⟨10.1002/chem.202102809⟩
Article dans une revue hal-03582991 v1
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Practical Synthesis and Application of Halogen-Doped Pyrrole Building Blocks

Andrej Emanuel Cotman , Thomas Guérin , Ivana Kovačević , Davide Benedetto Tiz , Martina Durcik et al.
ACS Omega, 2021, 6 (14), pp.9723-9730. ⟨10.1021/acsomega.1c00331⟩
Article dans une revue hal-03228819 v1
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Aryl Fluoroalkyl Sulfoxides: Optical Stability and p K a Measurement

Amélia Messara , Nicolas Vanthuyne , Patrick Diter , Mourad Elhabiri , Armen Panossian et al.
European Journal of Organic Chemistry, 2021, 2021 (36), ⟨10.1002/ejoc.202100816⟩
Article dans une revue hal-03319682 v1

Novel substituted N-benzyl(oxotriazinoindole) inhibitors of aldose reductase exploiting ALR2 unoccupied interactive pocket

Matúš Hlaváč , Lucia Kováčiková , Marta Šoltésová Prnová , Gabriela Addová , Gilles Hanquet et al.
Bioorganic and Medicinal Chemistry, 2021, 29, pp.115885. ⟨10.1016/j.bmc.2020.115885⟩
Article dans une revue hal-03052028 v1
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Novel substituted N-benzyl(oxotriazinoindole) inhibitors of aldose reductase exploiting ALR2 unoccupied interactive pocket

Matúš Hlaváč , Lucia Kováčiková , Marta Šoltésová Prnová , Gabriela Addová , Gilles Hanquet et al.
Bioorganic and Medicinal Chemistry, 2020
Article dans une revue hal-03070904 v1
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Development of Novel Oxotriazinoindole Inhibitors of Aldose Reductase: Isosteric Sulfur/Oxygen Replacement in the Thioxotriazinoindole Cemtirestat Markedly Improved Inhibition Selectivity

Matúš Hlaváč , Lucia Kováčiková , Marta Šoltésová Prnová , Peter Sramel , Gabriela Addová et al.
Journal of Medicinal Chemistry, 2020, 63 (1), pp.369-381. ⟨10.1021/acs.jmedchem.9b01747⟩
Article dans une revue hal-03079080 v1
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Synthesis and Use of Trifluoromethylthiolated Ketenimines

Frédéric R. Leroux , Thomas Guérin , Nadiia Pikun , Ryutaro Morioka , Armen Panossian et al.
Chemistry - A European Journal, 2020, ⟨10.1002/chem.202002723⟩
Article dans une revue hal-02990038 v1
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New synthesized polyoxygenated diarylheptanoids suppress lipopolysaccharide-induced neuroinflammation

Anna Santarsiero , Antonella Bochicchio , Maria Funicello , Paolo Lupattelli , Sabine Choppin et al.
Biochemical and Biophysical Research Communications, 2020, 529 (4), pp.1117-1123. ⟨10.1016/j.bbrc.2020.06.122⟩
Article dans une revue hal-03077267 v1
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Unintended Formation of a 26-Membered Cycle in the Course of a Novel Approach to Myricanol, a Strained [7,0]-metacyclophane

Paul Massé , Sabine Choppin , Lucia Chiummiento , Gilles Hanquet , Francoise Colobert
SYNLETT, 2019, 31 (06), pp.559-564. ⟨10.1055/s-0039-1691523⟩
Article dans une revue hal-03075499 v1
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Efficient asymmetric synthesis of aryl difluoromethyl sulfoxides and their use to access enantiopure α-difluoromethyl alcohols

Chloé Batisse , Maria Cespedes Davila , Marco Castello , Amélia Messara , Bertrand Vivet et al.
Tetrahedron, 2019, 75 (23), pp.3063-3079. ⟨10.1016/j.tet.2019.04.037⟩
Article dans une revue hal-02400108 v1
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Design, Synthesis and Biological Evaluation of Antimicrobial Diarylimine and -amine Compounds Targeting the Interaction between the Bacterial NusB and NusE Proteins

Yangyi Qiu , Shu Ting Chan , Lin Lin , Tsun Lam Shek , Tsz Fung Tsang et al.
European Journal of Medicinal Chemistry, 2019, 178, pp.214-231. ⟨10.1016/j.ejmech.2019.05.090⟩
Article dans une revue hal-03079069 v1

First Total Synthesis of Pamamycin-621D

H Norouzi-Arasi , X Salom-Roig , S Lanners , Gilles Hanquet
Current Organic Synthesis, 2018, 15, pp.105-109. ⟨10.2174/1570179414666170525103947⟩
Article dans une revue hal-02167613 v1
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Access towards enantiopure α,α-difluoromethyl alcohols by means of sulfoxides as traceless chiral auxiliaries

Chloé Batisse , Armen Panossian , Gilles Hanquet , Frédéric Leroux
Chemical Communications, 2018, 54 (74), pp.10423-10426. ⟨10.1039/C8CC05571H⟩
Article dans une revue hal-02150060 v1

Convergent total synthesis of (±) myricanol, a cyclic natural diarylheptanoid

Antonella Bochicchio , Lucie Schiavo , L Chiummiento , P Lupattelli , M Funicello et al.
Organic & Biomolecular Chemistry, 2018, 16, pp.8859-8869. ⟨10.1039/C8OB02052C⟩
Article dans une revue hal-02158253 v1

Access to Wieland–Miescher Diketone-Derived Building Blocks by Stereoselective Construction of the C-9 Quaternary Carbon Center Using the Mukaiyama Aldol Reaction

Lucie Schiavo , L Lebedel , P Massé , Sabine Choppin , Gilles Hanquet
Journal of Organic Chemistry, 2018, 83 (12), pp.6247-6258. ⟨10.1021/acs.joc.7b02862⟩
Article dans une revue hal-02150059 v1

Quinoides and VEGFR2 TKIs influence the fate of hepatocellular carcinoma and its cancer stem cells

D Kahraman , Gilles Hanquet , L Jeanmart , S Lanners , Peter Sramel et al.
MedChemComm, 2017, 8, pp.81-87. ⟨10.1039/C6MD00392C⟩
Article dans une revue hal-02177405 v1

Novel CLK1 inhibitors based on N-aryloxazol-2-amine skeleton - A possible way to dual VEGFR2 TK/CLK ligands

M Murár , J Dobiaš , P Šramel , G Addová , Gilles Hanquet et al.
European Journal of Medicinal Chemistry, 2017, 126, pp.754-761. ⟨10.1016/j.ejmech.2016.11.003⟩
Article dans une revue hal-02170487 v1

FeCl3.6H2O/acetaldehyde, a versatile system for the deprotection of ketals and acetals via a transacetalization process

Lucie Schiavo , L Jeanmart , S Lanners , Sabine Choppin , Gilles Hanquet
New Journal of Chemistry, 2017, 41, pp.1421-1424. ⟨10.1039/C6NJ03439J⟩
Article dans une revue hal-02167611 v1
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Synthesis, biological evaluation and molecular modeling studies on novel quinonoid inhibitors of CDC25 phosphatases

E Evain-Bana , Lucie Schiavo , C Bour , Don Antoine Lanfranchi , S Berardozzi et al.
Journal of Enzyme Inhibition and Medicinal Chemistry, 2017, 32, pp.113-118. ⟨10.1080/14756366.2016.1238364⟩
Article dans une revue hal-02161666 v1

New Insights into the Synthesis and Biological Activity of the Pamamycin Macrodiolides

Gilles Hanquet , Xavier Salom-Roig , Steve Lanners
CHIMIA, 2016, 70 (1), pp.20-28. ⟨10.2533/chimia.2016.20⟩
Article dans une revue hal-03054586 v1

Selective Claisen rearrangement and iodination for the synthesis of polyoxygenated allyl phenol derivatives

Antonella Bochicchio , Rossella Cefola , Sabine Choppin , Françoise Colobert , Maria Antonietta Di Noia et al.
Tetrahedron Letters, 2016, 57 (36), pp.4053-4055. ⟨10.1016/j.tetlet.2016.07.079⟩
Article dans une revue hal-03054575 v1
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New Insights into the Synthesis and Biological Activity of the Pamamycin Macrodiolides

Gilles Hanquet , Xavier Salom-Roig , Steve Lanners
CHIMIA, 2016, 70 (1), pp.20-28. ⟨10.2533/chimia.2016.20⟩
Article dans une revue hal-03468389 v1

Carbamoyl fluorides: from synthesis to radiochemistry

Clémence Bonnefoy , Emmanuel Chefdeville , Armen Panossian , Gilles Hanquet , Frédéric R. Leroux et al.
57th International Conference on Medicinal Chemistry, Jul 2023, Lille, France
Poster de conférence hal-04720307 v1

Carbamoyl Fluorides: From Synthesis to Radiochemistry

Clémence Bonnefoy , Emmanuel Chefdeville , Armen Panossian , Gilles Hanquet , Frédéric R. Leroux et al.
28th French-Japanese Symposium on Medicinal & Fine Chemistry, Oct 2023, Nice, France
Poster de conférence hal-04720313 v1

Carbamoyl fluoride as a potential new tag for fluorine-18 labeling

Clémence Bonnefoy , Christian Tourvieille , Armen Panossian , Gilles Hanquet , Frédéric R. Leroux et al.
24th International Symposium on Radiopharmaceutical Sciences, May 2022, Nantes, France
Poster de conférence hal-04720303 v1

2,4-Dinitro-trifluoromethoxybenzene: a promising reagent in fluorine chemistry

Clémence Bonnefoy , Emmanuel Chefdeville , Christian Tourvielle , Armen Panossian , Gilles Hanquet et al.
55th Bürgenstock Conference, May 2022, Brunnen, Switzerland
Poster de conférence hal-04720299 v1

Modern Fluorine‐Containing Agrochemicals

Sergii Pazenok , David Bernier , Morgan Donnard , Gilles Hanquet , Armen Panossian et al.
Z. Rappoport. PATAI'S Chemistry of Functional Groups, 1, Wiley; Wiley, 2022, 9780470682531. ⟨10.1002/9780470682531.pat1013⟩
Chapitre d'ouvrage hal-03920395 v1