Kevin Cariou

Publications

Article dans une revue (38)

Design, Synthesis, and Evaluation of Organic and Organometallic Pyrazoline Derivatives as Selective Dual COX-2/5-LOX Inhibitors and Potential Anticancer Agents Elizabeth Navarrete,Tomás Cáceres M,Pilar Morales,Michelle Muñoz-Osses,Olivier Blacqueet al. Journal of Medicinal Chemistry, 2026, ⟨10.1021/acs.jmedchem.5c02815⟩ Article dans une revue hal-05450044v1
Synthesis, Characterization, and Biological Evaluation of Red Light‐Activatable BODIPY‐Caged Ceritinib Compounds Kirill M Kuznetsov,Kallol Purkait,Pierre Mesdom,Philippe Arnoux,Céline Frochotet al. Helvetica Chimica Acta, In press, ⟨10.1002/hlca.202500023⟩ Article dans une revue hal-05037869v1
A Cathepsin B‐Triggered CO‐Releasing Molecule with a Non‐Toxic Metal Core for Targeted Tumor Delivery Inga Černauskienė,Eduardo Izquierdo‐garcía,Sarah Keller,Harley Betts,Kevin Cariouet al. Angewandte Chemie International Edition, 2025, ⟨10.1002/anie.202513808⟩ Article dans une revue hal-05354488v1
Metal‐Catalyzed Cross‐Coupling for the Synthesis of β‐Lactam Drugs and Related Chemical Probes Jules Bresson,Katie Burke,Mélanie Ethève‐quelquejeu,Laura Iannazzo,Kevin Cariou ChemMedChem, 2025, 20 (9), pp.e202400960. ⟨10.1002/cmdc.202400960⟩ Article dans une revue hal-05287299v1
EGCG-like non-competitive inhibitor of DYRK1A rescues cognitive defect in a down syndrome model Jean Delabar,Marco Antônio G.B. Gomes,Marta Fructuoso,Nadège Sarrazin,Nicolas Georgeet al. European Journal of Medicinal Chemistry, 2024, 265, pp.116098. ⟨10.1016/j.ejmech.2023.116098⟩ Article dans une revue hal-05387931v1
A Near-Infrared-Absorbing Osmium(II) Complex as a Photosensitizer for Photodynamic Therapy inducing Immunogenic Cell Death Yiyi Zhang,Pierre Mesdom,Eduardo Izquierdo-García,João António,Bruno Saubameaet al. ChemRxiv, 2024, ⟨10.26434/chemrxiv-2024-6dnl2⟩ Article dans une revue hal-05389603v1
N-Metallocenyl Ynamides: Preparation, Reactivity and Synthesis of ansa[3]-Ferrocenylamides Capucine Mahe,Olivier Blacque,Gilles Gasser,Vincent Gandon,Kevin Cariou Organic Letters, 2023, ⟨10.1021/acs.orglett.2c04169⟩ Article dans une revue hal-03966748v1
Base‐Mediated Generation of Ketenimines from Ynamides: Addition of Hydrazones to Give Acetimidohydrazides** Capucine Mahe,Agathe C A d'Hollander,Kevin Cariou European Journal of Organic Chemistry, 2022, 2022 (18), pp.e202200028. ⟨10.1002/ejoc.202200028⟩ Article dans une revue hal-03721985v1
Phototherapeutic anticancer strategies with first-row transition metal complexes: a critical review Lisa Gourdon,Kevin Cariou,Gilles Gasser Chemical Society Reviews, 2022, ⟨10.1039/D1CS00609F⟩ Article dans une revue hal-03542713v1
Base-Mediated Generation of Ketenimines from Ynamides: [3+2] Annulation with Azaallyl Anions Agathe C A d'Hollander,Eugénie Romero,Kamsana Vijayakumar,Camille Le Houérou,Pascal Retailleauet al. Advanced Synthesis and Catalysis, 2021, 363 (11), pp.2903-2908. ⟨10.1002/adsc.202100047⟩ Article dans une revue hal-03227971v1
Photoinduced Aerobic Iodoarene-Catalyzed Spirocyclization of N-Oxy-Amides to N-Fused Spirolactams Loïc Habert,Kevin Cariou Angewandte Chemie International Edition, 2021, 60 (1), pp.171-175. ⟨10.1002/anie.202009175⟩ Article dans une revue hal-03367856v1
Ynamides in Free Radical Reactions Capucine Mahe,Kevin Cariou Advanced Synthesis and Catalysis, In press, ⟨10.1002/adsc.202000849⟩ Article dans une revue hal-02962628v1
Synthetic approaches towards avibactam and other diazabicyclooctane β-lactamase inhibitors Laure Peilleron,Kevin Cariou Organic & Biomolecular Chemistry, 2020, ⟨10.1039/C9OB02605C⟩ Article dans une revue hal-02466833v1
Synthesis, Characterization and Antiparasitic Activity of Organometallic Derivatives of the Anthelmintic Drug Albendazole Yan Lin,Yih Ching Ong,Sarah Keller,Rafika Bouchene,Eric Manouryet al. Dalton Transactions, 2020, 49 (20), pp.6616-6626. ⟨10.1039/d0dt01107j⟩ Article dans une revue hal-02555378v1
Synthesis of cyclic N-hydroxylated ureas and oxazolidinone oximes enabled by chemoselective iodine(III)-mediated radical or cationic cyclizations of unsaturated N-alkoxyureas Laure Peilleron,Pascal Retailleau,Kevin Cariou Advanced Synthesis and Catalysis, 2019, 361 (22), pp.5160-5169. ⟨10.1002/adsc.201901135⟩ Article dans une revue hal-02403999v1
Halonium-Induced Polyene Cyclizations Agathe D’hollander,Laure Peilleron,Tatyana Grayfer,Kevin Cariou Synthesis: Journal of Synthetic Organic Chemistry, 2019, 51 (08), pp.1753-1769. ⟨10.1055/s-0037-1612254⟩ Article dans une revue hal-02307164v1
A tutorial for the assessment of the stability of organometallic complexes in biological media Sarah Keller,Yih Ching Ong,Yan Lin,Kevin Cariou,Gilles Gasser Journal of Organometallic Chemistry, 2019, pp.121059. ⟨10.1016/j.jorganchem.2019.121059⟩ Article dans une revue hal-02393969v1
DYRK1A inhibition and cognitive rescue in a Down syndrome mouse model are induced by new fluoro-DANDY derivatives Fernanda Neumann,Stéphanie Gourdain,Christelle Albac,Alain D Dekker,Linh Chi Buiet al. Scientific Reports, 2018, 8, pp.2859. ⟨10.1038/s41598-018-20984-z⟩ Article dans une revue hal-02292094v1
Iodine(III)-mediated halogenations of acyclic monoterpenoids Laure Peilleron,Tatyana Grayfer,Joëlle Dubois,Robert H Dodd,Kevin Cariouet al. Beilstein Journal of Organic Chemistry, 2018, 14, pp.1103-1111. ⟨10.3762/bjoc.14.96⟩ Article dans une revue hal-02307167v1
Ketenimines Generated from Ynamides: Versatile Building Blocks for Nitrogen-Containing Scaffolds Robert H Dodd,Kevin Cariou Chemistry - A European Journal, 2018, 24 (10), pp.2297-2304. ⟨10.1002/chem.201704689⟩ Article dans une revue hal-02307203v1
Synthesis of Orthogonally N-Protected, C-4 Functionalized Cyclic Guanidines from L-Serine Diego Silva,Edmilson Maria,Rosa Suárez Ordóñez,Josiane Thierry,Kevin Cariouet al. SYNLETT, 2017, 28 (07), pp.815-818. ⟨10.1055/s-0036-1589935⟩ Article dans une revue hal-02307213v1
Base-Mediated Generation of Ketenimines from Ynamides: Direct Access to Azetidinimines by an Imino Staudinger Synthesis Eugénie Romero,Corinne Minard,Mohamed Benchekroun,Sandrine Ventre,Pascal ́ Retailleauet al. Chemistry - A European Journal, 2017, 23 (53), pp.12991-12994. ⟨10.1002/chem.201702545⟩ Article dans une revue hal-02307210v1
Chemodivergent, Tunable, and Selective Iodine(III)-Mediated Bromo-Functionalizations of Polyprenoids Tatyana Grayfer,Pascal ́ Retailleau,Robert H Dodd,Joëlle Dubois,Kevin Cariou Organic Letters, 2017, 19 (18), pp.4766-4769. ⟨10.1021/acs.orglett.7b02125⟩ Article dans une revue hal-02307207v1
Mallotojaponins B and C: Total Synthesis, Antiparasitic Evaluation and Preliminary SAR Studies Tatyana Grayfer,Philippe Grellier,Elisabeth Mouray,Robert H Dodd,Joëlle Duboiset al. Organic Letters, 2016, 18 (4), pp.708-711. ⟨10.1021/acs.orglett.5b03676⟩ Article dans une revue hal-02420932v1
Assessing Ligand and Counterion Effects in the Noble Metal Catalyzed Cycloisomerization Reactions of 1,6-Allenynes: a Combined Experimental and Theoretical Approach Florian Jaroschik,Antoine Simonneau,Gilles Lemiere,Kevin Cariou,Nicolas Agenetet al. ACS Catalysis, 2016, 6 (8), pp.5146-5160. ⟨10.1021/acscatal.5b02696⟩ Article dans une revue hal-01397955v1
PIFA-mediated ethoxyiodination of enamides with potassium iodide R. Beltran,S. Nocquet-Thibault,Fabian Blanchard,R. Dodd,K. Cariou Organic & Biomolecular Chemistry, 2016, 14 (36), pp.8448-8451. ⟨10.1039/C6OB01673A⟩ Article dans une revue hal-02307217v1
Halocyclization of Unsaturated Guanidines Mediated by Koser's Reagent and Lithium Halides. Marion Daniel,Florent Blanchard,Sophie Nocquet-Thibault,Kevin Cariou,Robert H Dodd Journal of Organic Chemistry, 2015, 80 (21), pp.10624-33. ⟨10.1021/acs.joc.5b01750⟩ Article dans une revue hal-03023458v1
Iodine(III)-mediated diazidation and azido-oxyamination of enamides S. Nocquet-Thibault,Anita Marie Rayar,Pascal ́ Retailleau,Kevin Cariou,Robert Dodd Chemistry - A European Journal, 2015, 21 (40), pp.14205-14210. ⟨10.1002/chem.201501782⟩ Article dans une revue istex hal-03026966v1
Selective Suzuki-Miyaura monocouplings with symmetrical dibromoarenes and aryl ditriflates for the one-pot synthesis of unsymmetrical triaryls C. Minard,C. Palacio,K. Cariou,Robert H Dodd European Journal of Organic Chemistry, 2014, 2014 (14), pp.2942-2955. ⟨10.1002/ejoc.201400090⟩ Article dans une revue istex hal-00994366v1
Iodine(III)-mediated ethoxychlorination of enamides with iron(III) chloride Sophie Nocquet-Thibault,Corinne Minard,Pascal Retailleau,Kevin Cariou,Robert H. Dodd Tetrahedron, 2014, 70 (38), pp.6769-6775. ⟨10.1016/j.tet.2014.07.066⟩ Article dans une revue hal-01067773v1
Transition-metal-free tunable chemoselective N functionalization of indoles with ynamides. Alexandre Hentz,Pascal Retailleau,Vincent Gandon,Kevin Cariou,Robert H Dodd Angewandte Chemie International Edition, 2014, 53 (32), pp.8333-8337. ⟨10.1002/anie.201402767⟩ Article dans une revue istex hal-01065687v1
Iodine(III)-Mediated Umpolung of Bromide Salts for the Ethoxybromination of Enamides. Sophie Nocquet-Thibault,Pascal Retailleau,Kevin Cariou,Robert H Dodd Organic Letters, 2013, 15 (8), pp.1842-5. ⟨10.1021/ol400453b⟩ Article dans une revue hal-00827755v1
Development of DANDYs, New 3,5-Diaryl-7-azaindoles Demonstrating Potent DYRK1A Kinase Inhibitory Activity. Stéphanie Gourdain,Julien Dairou,Clément Denhez,Linh Chi Bui,Fernando Rodrigues-Limaet al. Journal of Medicinal Chemistry, 2013, 56 (23), pp.9569-9585. ⟨10.1021/jm401049v⟩ Article dans une revue hal-00933939v1
New elements in the gold(I)-catalyzed cycloisomerization of enynyl ester derivatives embedding a cyclohexane template Youssef Harrak,Malika Makhlouf,Stéphane Azzaro,Emily Mainetti,Juan Manuel Lopez Romeroet al. Journal of Organometallic Chemistry, 2011, 696 (1), pp.388-399. ⟨10.1016/j.jorganchem.2010.10.016⟩ Article dans une revue istex hal-05415359v1
Copper(I) catalyzed regioselective asymmetric alkoxyamination of aryl enamide derivatives. Masafumi Nakanishi,Corinne Minard,Pascal Retailleau,Kevin Cariou,Robert H Dodd Organic Letters, 2011, 13 (21), pp.5792-5. ⟨10.1021/ol202367d⟩ Article dans une revue hal-00647697v1
Generation and Trapping of Cyclopentenylidene Gold Species: Four Pathways to Polycyclic Compounds Gilles Lemière,Vincent Gandon,Kevin Cariou,Alexandra Hours,Takahide Fukuyamaet al. Journal of the American Chemical Society, 2009, 131 (8), pp.2993-3006. ⟨10.1021/ja808872u⟩ Article dans une revue hal-05415340v1
Tandem Gold(I)-Catalyzed Cyclization/Electrophilic Cyclopropanation of Vinyl Allenes Gilles Lemière,Vincent Gandon,Kevin Cariou,Takahide Fukuyama,Anne-Lise Dhimaneet al. Organic Letters, 2007, 9 (11), pp.2207-2209. ⟨10.1021/ol070788r⟩ Article dans une revue hal-05415300v1
New unsaturated amino acids containing an allylsilane moiety on the lateral chain Gianna Reginato,Alessandro Mordini,Patrick Meffre,Alice Tenti,Michela Valacchiet al. Tetrahedron: Asymmetry, 2006, 17 (6), pp.922-926. ⟨10.1016/j.tetasy.2006.02.017⟩ Article dans une revue hal-02002619v1

Pré-publication, Document de travail (2)

Base-Mediated Generation of Ketenimines from Ynamides: [3+2] Annulation with Azaallyl Anions Agathe D’hollander,Eugénie Romero,Kamsana Vijayakumar,Camille Le Houérou,Pascal Retailleauet al. 2020 Pré-publication, Document de travail hal-02998846v1
Azetidinimines as a novel series of non-covalent broad-spectrum inhibitors of β-lactamases with submicromolar activities against carbapenemases of classes A, B and D Eugénie Romero,Saoussen Oueslati,Mohamed Benchekroun,Agathe D’hollander,Sandrine Ventreet al. 2020 Pré-publication, Document de travail hal-02998861v1