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Facile access to novel furoyl-based amide retroisoster inhibitors of LuxR-regulated quorum sensing: conformation analysis and docking studies
Laurent Soulère
,
Yves Queneau
Article dans une revue
hal-04709389
v1
|
|
Membrane plasticity induced by <i>myo</i>-inositol derived archaeal lipids: chemical synthesis and biophysical characterization
Johal Ruiz
,
Josephine G Loricco
,
Laurent Soulère
,
Marta Salvador-Castell
,
Axelle Grélard
et al.
Article dans une revue
hal-04391247
v1
|
|
Machine learning approaches for the identification of ligands of the autophagy marker LC3
Laurent Soulère
,
Yves Queneau
Article dans une revue
hal-04292493
v1
|
|
Towards More Practical Methods for the Chemical Synthesis of Thioamides Using Sulfuration Agents: A Decade Update
Qiang Zhang
,
Laurent Soulère
,
Yves Queneau
Article dans une revue
(article de synthèse)
hal-04079206
v1
|
|
In Silico Identification of Potential Inhibitors of the SARS-CoV-2 Main Protease among a PubChem Database of Avian Infectious Bronchitis Virus 3CLPro Inhibitors
Laurent Soulère
,
Thibaut Barbier
,
Yves Queneau
Article dans une revue
hal-04122457
v1
|
|
Importance of the 2,6-Difluorobenzamide Motif for FtsZ Allosteric Inhibition: Insights from Conformational Analysis, Molecular Docking and Structural Modifications
Thibaut Barbier
,
Oana Dumitrescu
,
Gérard Lina
,
Yves Queneau
,
Laurent Soulère
Article dans une revue
hal-04028136
v1
|
|
Synthesis and Biological Evaluation of Benzo[b]thiophene Acylhydrazones as Antimicrobial Agents against Multidrug-Resistant Staphylococcus aureus
Thibaut Barbier
,
Alexia Barbry
,
Jérémy Magand
,
Cédric Badiou
,
Floriane Davy
et al.
Article dans une revue
hal-03719638
v1
|
|
Structural Variations in the Central Heterocyclic Scaffold of Tripartite 2,6-Difluorobenzamides: Influence on Their Antibacterial Activity against MDR Staphylococcus aureus
Thibaut Barbier
,
Cédric Badiou
,
Floriane Davy
,
Yves Queneau
,
Oana Dumitrescu
et al.
Article dans une revue
hal-03923036
v1
|
|
Synthesis of phospholipids under plausible prebiotic conditions and analogies with phospholipid biochemistry or origin of life studies
Michele Fiore
,
Carolina Chieffo
,
Augustin Lopez
,
Dimitri Fayolle
,
Johal Ruiz
et al.
Article dans une revue
hal-03591985
v1
|
|
What is a supercoiling-sensitive gene? Insights from topoisomerase I inhibition in the Gram-negative bacterium Dickeya dadantii
Maïwenn Pineau
,
Shiny Martis Badiadka
,
Raphaël Forquet
,
Jessica Baude
,
Camille Villard
et al.
Article dans une revue
hal-03774489
v1
|
|
Heterocyclic Chemistry Applied to the Design of N-Acyl Homoserine Lactone Analogues as Bacterial Quorum Sensing Signals Mimics
Qiang Zhang
,
Sizhe Li
,
Maha Hachicha
,
Mohamed Boukraa
,
Laurent Soulère
et al.
Article dans une revue
hal-03378442
v1
|
|
PGRP-LB: An Inside View into the Mechanism of the Amidase Reaction
Julien Orlans
,
Carole Vincent-Monegat
,
Isabelle Rahioui
,
Catherine Sivignon
,
Agata Butryn
et al.
Article dans une revue
hal-03237949
v1
|
|
Synthesis of new 1,4‐ and 1,5‐disubstituted N ‐ethyl acetate and N ‐α‐butyro‐γ‐lactone alkylimidazole derivatives as N ‐acylhomoserine lactone analogs
Qiang Zhang
,
Si-Zhe Li
,
Yves Queneau
,
Laurent Soulère
Article dans une revue
hal-03378482
v1
|
|
Straightforward Synthesis of Chiral Terpenoid Building Blocks by Ru-Catalyzed Enantioselective Hydrogenation
Johal Ruiz
,
Phil M. Oger
,
Laurent Soulère
,
Florence Popowycz
Article dans une revue
hal-03275385
v1
|
|
Docking-based virtual screening studies aiming at the covalent inhibition of SARS-CoV-2 MPro by targeting the cysteine 145
Laurent Soulère
,
Thibaut Barbier
,
Yves Queneau
Article dans une revue
hal-03243702
v1
|
|
Computer-Assisted Conformational Analysis of Small Molecules Using VEGA ZZ, a Freely Available Software Program, as an Introduction to Molecular Modeling
Laurent Soulère
Article dans une revue
hal-04167147
v1
|
|
(2R)- and (2S)- 2-hydroxy Hexanoyl and Octanoyl-l-Homoserine Lactones: new highly potent Quorum Sensing modulators with opposite activities
Qiang Zhang
,
Erwann Jeanneau
,
Yves Queneau
,
Laurent Soulère
Article dans une revue
hal-02952061
v1
|
|
CKD Increases Carbonylation of HDL and Is Associated with Impaired Antiaggregant Properties
Nans Florens
,
Catherine Calzada
,
Sandrine Lemoine
,
Marie Michèle Boulet
,
Nicolas Guillot
et al.
Article dans une revue
hal-03046430
v1
|
|
Biological Evaluation and Docking Studies of New Carbamate, Thiocarbamate, and Hydrazide Analogues of Acyl Homoserine Lactones as Vibrio fischeri-Quorum Sensing Modulators
Zhang Qiang
,
Yves Queneau
,
Laurent Soulère
Article dans une revue
hal-02883805
v1
|
|
Esters of Glucose-2-Phosphate: Occurrence and Chemistry
Zhang Qiang
,
Si-Zhe Li
,
Mohammed Ahmar
,
Laurent Soulère
,
Yves Queneau
Article dans une revue
hal-02883902
v1
|
|
Synthesis of a non-natural glucose-2-phosphate ester able to dupe the acc system of Agrobacterium fabrum
Si-Zhe Li
,
Armelle Vigouroux
,
Mohammed Ahmar
,
Abbas El Sahili
,
Laurent Soulere
et al.
Article dans une revue
hal-02173130
v1
|
|
Conformational and docking studies of acyl homoserine lactones as a robust method to investigate bioactive conformations
Laurent Soulère
,
Yves Queneau
Article dans une revue
hal-02110869
v1
|
|
Lifestyle of the biotroph Agrobacterium tumefaciens in the ecological niche constructed on its host plant
Almudena Gonzalez-Mula
,
Julien Lang
,
Catherine Grandclément
,
Delphine Naquin
,
Mohammed Ahmar
et al.
Article dans une revue
hal-02110550
v1
|
|
Identification of novel antilipogenic agents targeting fatty acid biosynthesis through structure-based virtual screening
Laurent Soulère
,
Pascaline M. Alix
,
Marine L. Croze
,
Christophe Soulage
Article dans une revue
hal-01847387
v1
|
|
Influence of the d/l configuration of N-acyl-homoserine lactones (AHLs) and analogues on their Lux-R dependent quorum sensing activity
Si-Zhe Li
,
Rui Xu
,
Mohammed Ahmar
,
Catherine Goux-Henry
,
Yves Queneau
et al.
Article dans une revue
hal-02110506
v1
|
|
Skeletal muscle insulin resistance is induced by 4-hydroxy-2-hexenal, a by-product of n-3 fatty acid peroxidation
Christophe Soulage
,
Laura Sardón Puig
,
Laurent Soulère
,
Bader Zarrouki
,
Michel Guichardant
et al.
Article dans une revue
hal-02110460
v1
|
|
α-Eleostearic acid-containing triglycerides for a continuous assay to determine lipase sn -1 and sn -3 regio-preference
Meddy El Alaoui
,
Laurent Soulère
,
Alexandre Noiriel
,
Yves Queneau
,
Abdelkarim Abousalham
Article dans une revue
hal-04167239
v1
|
|
Exploring docking methods for virtual screening: application to the identification of neuraminidase and Ftsz potential inhibitors
Laurent Soulère
,
Christophe Soulage
Article dans une revue
hal-01600438
v1
|
|
2-Substituted Aniline as a Simple Scaffold for LuxR-Regulated QS Modulation
S. Li
,
Julien Wawrzyniak
,
Y. Queneau
,
L. Soulère
Article dans une revue
hal-02001353
v1
|
|
Liquid crystalline glycosteroids and acyl steroid glycosides (ASG)
Zonglong Yang
,
Rui Xu
,
Fahima Ali-Rachedi
,
Stéphane Chambert
,
Nuno Xavier
et al.
Article dans une revue
hal-02193065
v1
|
|
Quorum Sensing Inhibitor Activities of Celecoxib Derivatives in Pseudomonas aeruginosa
Seyhan Ulusoy
,
Sevil Senkardes
,
Inci Coskun
,
Gulgun Bosgelmez-T|naz
,
Laurent Soulère
et al.
Article dans une revue
hal-02193031
v1
|
|
Insights into the Quorum Sensing Regulon of the Acidophilic Acidithiobacillus ferrooxidans Revealed by Transcriptomic in the Presence of an Acyl Homoserine Lactone Superagonist Analog
Sigde Mamani
,
Danielle Moinier
,
Yann Denis
,
L. Soulère
,
Y. Queneau
et al.
Article dans une revue
hal-01440758
v1
|
|
A continuous spectrophotometric assay that distinguishes between phospholipase A1 and A2 activities
Meddy El Alaoui
,
L. Soulere
,
A. Noiriel
,
F. Popowycz
,
A. Khatib
et al.
Article dans une revue
hal-01477286
v1
|
|
A convenient method for phosphorylation using trially phosphate
S.L. Li
,
M. Ahmar
,
Y. Queneau
,
L. Soulère
Article dans une revue
hal-01478940
v1
|
|
A Pyranose-2-Phosphate Motif Is Responsible for Both Antibiotic Import and Quorum-Sensing Regulation in Agrobacterium tumefaciens
Abbas El Sahili
,
Si-Zhe Li
,
Julien Lang
,
Cornelia Virus
,
Sara Planamente
et al.
Article dans une revue
hal-01430779
v1
|
|
Glycoxidized HDL, HDL enriched with oxidized phospholipids and HDL from diabetic patients inhibit platelet function
Quang Huy Lê
,
Meddy El Alaoui
,
Evelyne Véricel
,
Bérénice Ségrestin
,
Laurent Soulère
et al.
Article dans une revue
inserm-01134619
v1
|
|
Development of a high-throughput assay for measuring phospholipase A activity using synthetic 1,2-a-eleostearoyl-sn-glycero-3-phosphocholine coated on microtiter plates.
Meddy El Alauoui
,
Alexandre Noiriel
,
Laurent Soulère
,
Lucie Grand
,
Yves Queneau
et al.
Article dans une revue
hal-01141494
v1
|
|
AHL signaling molecules with a large acyl chain enhance biofilm formation on sulfur and metal sulfides by the bioleaching bacterium Acidithiobacillus ferrooxidans.
Alex González
,
Sören Bellenberg
,
Sigde Mamani
,
Lina Ruiz
,
Alex Echeverría
et al.
Article dans une revue
istex
hal-00919253
v1
|
|
A new route towards fimbrolide analogues : importance of the exomethylene motif in LuxR dependent quorum sensing inhibition
Mohamad Sabbah
,
Maud Bernollin
,
Alain Doutheau
,
Laurent Soulère
,
Yves Queneau
Article dans une revue
hal-01146328
v1
|
|
N,N'-alkylated Imidazolium-derivatives act as quorum-sensing inhibitors targeting the Pectobacterium atrosepticum-induced symptoms on potato tubers.
Yannick Raoul Des Essarts
,
Mohamad Sabbah
,
Arnaud Comte
,
Laurent Soulère
,
Yves Queneau
et al.
Article dans une revue
hal-00919246
v1
|
|
At a supra-physiological concentration, human sexual hormones act as quorum-sensing inhibitors.
Amélie Beury-Cirou
,
Mélanie Tannières
,
Corinne Minard
,
Laurent Soulère
,
Tsiry Rasamiravaka
et al.
Article dans une revue
hal-00949341
v1
|
|
Synthesis and biological evaluation of new N-acyl-homoserine-lactone analogues, based on triazole and tetrazole scaffolds, acting as LuxR-dependent quorum sensing modulators.
Mohamad Sabbah
,
Fanny Fontaine
,
Lucie Grand
,
Mohamed Boukraa
,
Mohamed L Efrit
et al.
Article dans une revue
istex
hal-00919262
v1
|
|
The lipid peroxidation by-product 4-hydroxy-2-Nonenal (4-HNE) induces insulin resistance in skeletal
J. Pillon N.
,
L. Croze M.
,
E. Vella R.
,
L. Soulère
,
M. Lagarde
et al.
Article dans une revue
hal-01555917
v1
|
|
Mechanisms and synthetic modulators of AHL-dependent gene regulation.
Ann M Stevens
,
Y. Queneau
,
L. Soulère
,
Susanne von Bodman
,
A. Doutheau
Article dans une revue
hal-00695865
v1
|
|
LuxR dependent quorum sensing inhibition by N,N'-disubstituted imidazolium salts.
Mohamad Sabbah
,
Laurent Soulère
,
Sylvie Reverchon
,
Y. Queneau
,
Alain Doutheau
Article dans une revue
istex
hal-00695863
v1
|
|
AHL-dependent quorum sensing inhibition: synthesis and biological evaluation of α-(N-alkyl-carboxamide)-γ-butyrolactones and α-(N-alkyl-sulfonamide)-γ-butyrolactones.
Mohamed Boukraa
,
Mohamad Sabbah
,
Laurent Soulère
,
Mohamed L El Efrit
,
Yves Queneau
et al.
Article dans une revue
istex
hal-00695861
v1
|
|
Structural and Functional Changes in Human Insulin Induced by the Lipid Peroxidation Byproducts 4-Hydroxy-2-nonenal and 4-Hydroxy-2-hexenal
Nicolas Pillon
,
Roxane E. Vella
,
Laurent Soulère
,
Michel Becchi
,
Michel Lagarde
et al.
Article dans une revue
hal-02650408
v1
|
|
Marine natural meroterpenes: synthesis and antiproliferative activity
Annabel Simon-Levert
,
Christophe Menniti
,
Laurent Soulère
,
Anne-Marie Genevière
,
Chantal Barthomeuf
et al.
Article dans une revue
hal-02190465
v1
|
|
Quantitative structure-activity relationship for 4-hydroxy-2-alkenal induced cytotoxicity in L6 muscle cells
Nicolas J Pillon
,
Laurent Soulère
,
Roxane E Vella
,
Marine Croze
,
Bertrand R Caré
et al.
Article dans une revue
istex
hal-00759515
v1
|
|
LuxR-dependent quorum sensing: computer aided discovery of new inhibitors structurally unrelated to N-acylhomoserine lactones.
Laurent Soulère
,
Mohamad Sabbah
,
Fanny Fontaine
,
Yves Queneau
,
Alain Doutheau
Article dans une revue
istex
hal-00695871
v1
|
|
Toward Docking-Based Virtual Screening for Discovering Antitubulin Agents by Targeting Taxane and Colchicine Binding Sites
Laurent Soulère
Article dans une revue
istex
hal-04167250
v1
|
|
Rational design, solid phase synthesis and evaluation of cationic ferrocenoyl peptide bioconjugates as potential antioxidant enzyme mimics
Laurent Soulère
,
Julien Bernard
Article dans une revue
istex
hal-00374569
v1
|
|
N-Acyl-3-amino-5H-furanone derivatives as new inhibitors of LuxR-dependent quorum sensing: Synthesis, biological evaluation and binding mode study
J. Estephane
,
J. Dauvergne
,
L. Soulere
,
Sylvie Reverchon
,
Y. Queneau
et al.
Bioorganic and Medicinal Chemistry Letters, 2008, 18 (15), pp.4321-4
Article dans une revue
hal-01997033
v1
|
|
Synthetic homoserine lactone-derived sulfonylureas as inhibitors of Vibrio fischeri quorum sensing regulator
M. Frezza
,
L. Soulere
,
Sylvie Reverchon
,
N. Guiliani
,
C. Jerez
et al.
Article dans une revue
istex
hal-01997035
v1
|
|
AHL communication is a widespread phenomenon in biomining bacteria and seems to be involved in mineral-adhesion efficiency
Lina María Ruiz
,
Susana Valenzuela
,
Matias Castro
,
Alex Gonzalez
,
Marine Frezza
et al.
Article dans une revue
istex
hal-04167264
v1
|
|
Molecular insights into quorum sensing in Acidithiobacillus ferrooxidans bacteria via molecular modelling of the transcriptional regulator AfeR and of the binding mode of long-chain acyl homoserine lactones
Laurent Soulère
,
Nicolas Guiliani
,
Yves Queneau
,
Carlos Jerez
,
Alain Doutheau
Article dans une revue
istex
hal-04167257
v1
|
|
Bis-(O)-acetylated derivative of 4,5-dihydroxy-2,3-pentanedione (DPD): a convenient stable precursor of quorum sensing autoinducer AI-2
M. Frezza
,
L. Soulere
,
D. Balestrino
,
Y. Queneau
,
C. Forestier
et al.
Biorg.Med.Chem.Lett., 2007, 17, pp.1428-1431
Article dans une revue
hal-00139413
v1
|
|
Ac2-DPD, the bis-(O)-acetylated derivative of 4,5-dihydroxy-2,3-pentanedione (DPD) is a convenient stable precursor of bacterial quorum sensing autoinducer AI-2.
Marine Frezza
,
Laurent Soulère
,
Damien Balestrino
,
Michel Gohar
,
Christian Deshayes
et al.
Article dans une revue
istex
hal-00164190
v1
|
|
Exploring the active site of acyl homoserine lactones-dependent transcriptional regulators with bacterial quorum sensing modulators using molecular mechanics and docking studies
Laurent Soulère
,
Marine Frezza
,
Yves Queneau
,
Alain Doutheau
Article dans une revue
istex
hal-04167213
v1
|
|
An expeditious synthesis of 4-hydroxy-2(E)-nonenal (4-HNE), its dimethyl acetal and of related compounds
Laurent Soulère
,
Yves Queneau
,
Alain Doutheau
Article dans une revue
istex
hal-04167188
v1
|
|
Synthesis and biological evaluation of the trifluoromethyl analog of (4S)-4,5-dihydroxy-2,3-pentanedione (DPD)
M. Frezza
,
D. Balestrino
,
L. Soulère
,
S. Reverchon-Pescheux
,
Y. Queneau
et al.
European Journal of Organic Chemistry, 2006, pp.4731-4736
Article dans une revue
hal-00144011
v1
|
|
Conjugated linoleic acid, unlike other unsaturated fatty acids, strongly induces glutathione synthesis without any lipoperoxidation
J.-P. Steghens
,
K. Arab
,
A. Rossary
,
L. Soulère
British Journal of Nutrition, 2006, 96 (96), pp.811-819
Article dans une revue
hal-00144012
v1
|
|
Synthesis and biological evaluation of homoserine lactone derived ureas as antagonists of bacterial quorum sensing
M. Frezza
,
S. Castang
,
J. Estephane
,
L. Soulere
,
C. Deshayes
et al.
Bioorganic and Medicinal Chemistry, 2006, 14 (14), pp.4781-91
Article dans une revue
hal-01997034
v1
|
|
A Baylis–Hillman/ozonolysis route towards (±) 4,5-dihydroxy-2,3-pentanedione (DPD) and analogues
Marine Frezza
,
Laurent Soulère
,
Yves Queneau
,
Alain Doutheau
Article dans une revue
istex
hal-04167707
v1
|