|
|
LAVR-289, a broad-spectrum antiviral, protects immunosuppressed Syrian hamsters against lethal adenovirus challenge
Ann Tollefson
,
Anna Cline-Smith
,
Vincent Roy
,
Luigi A. Agrofoglio
,
Getahun Abate
et al.
Article dans une revue
hal-05588571v1
|
|
|
LAVR-289, an Acyclo-Nucleoside Phosphonate, Has Broad-Spectrum Activity against Herpesviruses
Sandrine Kappler-Gratias
,
Charlotte Quentin-Froignant
,
Elie Marcheteau
,
José Fernandez
,
David Boutolleau
et al.
Article dans une revue
hal-05549140v1
|
|
|
LAVR-289, an Orally Bioavailable Inhibitor of Adenovirus Replication In Vitro and In Vivo
Charlotte Quentin-Froignant
,
Ann Tollefson
,
Anna Cline-Smith
,
Sandrine Kappler-Gratias
,
Nicolas Landrein
et al.
Article dans une revue
hal-05588724v1
|
|
|
Antiviral Activity of the Acyclic Nucleoside Phosphonate Prodrug LAVR-289 against Poxviruses and African Swine Fever Virus
Elie Marcheteau
,
Estelle Mosca
,
Gaelle Frenois-Veyrat
,
Sandrine Kappler-Gratias
,
Laetitia Boutin
et al.
Article dans une revue
hal-05588572v1
|
|
|
Synthesis of LAVR-289, a new [(Z)-3-(acetoxymethyl)-4-(2,4-diaminopyrimidin-6-yl)oxy-but-2-enyl]phosphonic acid prodrug with pronounced antiviral activity against DNA viruses
Maximes Bessières
,
Vincent Roy
,
Tuniyazi Abuduani
,
Patrick Favetta
,
Robert Snoeck
et al.
Article dans une revue
hal-05588577v1
|
|
|
Molecularly Imprinted Polymeric Nanoparticles as Drug Delivery System for Tenofovir, an Acyclic Nucleoside Phosphonate Antiviral
Thomas Mathieu
,
Patrick Favetta
,
Luigi Agrofoglio
Article dans une revue
hal-04790768v1
|
|
|
Synthesis and Antiviral Evaluation of 5-(4-Aryl-1,3-butadiyn-1-yl)-uridines and Their Phosphoramidate Pronucleotides
Evan Saillard
,
Otmane Bourzikat
,
Koffi Assa
,
Vincent Roy
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588574v1
|
|
|
Lyotropic liquid crystal emulsions of LAVR-289: Influence of internal mesophase structure on cytotoxicity and in-vitro antiviral activity
Mathias Brouillard
,
Thomas Mathieu
,
Samuel Guillot
,
Fabienne Méducin
,
Vincent Roy
et al.
Article dans une revue
hal-05588575v1
|
|
|
Cobalt-assisted route to rare carbocyclic C -ribonucleosides
Andrea C. Ojeda-Porras
,
Vincent Roy
,
Otmane Bourzikat
,
Patrick Favetta
,
L. Agrofoglio
Article dans une revue
hal-04790673v1
|
|
|
Antibiotics and Antibiotic Resistance—Mur Ligases as an Antibacterial Target
Vincent Hervin
,
Vincent Roy
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588578v1
|
|
|
Nucleosides and emerging viruses: A new story
Vincent Roy
,
Luigi Agrofoglio
Article dans une revue
hal-03859490v1
|
|
|
Synthesis of Novel 3’,3’‐cyclic Dinucleotide Analogues Targeting STING Protein
Jérémy Magand
,
Vincent Roy
,
Hervé Meudal
,
Stéphanie Rose
,
Valérie Quesniaux
et al.
Article dans une revue
hal-05588712v1
|
|
|
Synthesis of novel 3’,3’‐cyclic dinucleotide analogues targeting STING protein
Jérémy Magand
,
Vincent Roy
,
Hervé Meudal
,
Stéphanie Rose
,
Valérie Quesniaux
et al.
Article dans une revue
hal-03859427v1
|
|
|
Synthesis and structure–activity relationship studies of pyrido [1,2-e]purine-2,4(1H,3H)-dione derivatives targeting Flavin-Dependent $Thymidylate\ Synthase$ in $Mycobacterium\ tuberculosis$
Nicolas G. Biteau
,
Vincent Roy
,
Cyril Nicolas
,
Hubert F Becker
,
Jean-Christophe Lambry
et al.
Article dans une revue
hal-03798565v1
|
|
|
A Tunable Approach to C-Linked Analogs of Glycosamines
Tuniyazi Abuduaini
,
Sizhe Li
,
Vincent Roy
,
Luigi A Agrofoglio
,
Olivier R Martin
et al.
Article dans une revue
hal-03798583v1
|
|
|
Chemical Approaches to Carbocyclic Nucleosides
Andrea C. Ojeda-Porras
,
Vincent Roy
,
Luigi A. Agrofoglio
Article dans une revue
hal-03890854v1
|
|
|
Molecularly Imprinted Hydrogels Selective to Ribavirin as New Drug Delivery Systems to Improve Efficiency of Antiviral Nucleoside Analogue: A Proof‐of‐Concept Study with Influenza A Virus
Mohamed Ayari
,
Patrick Favetta
,
Dawid Warszycki
,
Virginie Vasseur
,
Virginie Herve
et al.
Article dans une revue
hal-03557328v1
|
|
|
Design, synthesis and biological evaluation of 2-substituted-6-[(4-substituted-1-piperidyl)methyl]-1H-benzimidazoles as inhibitors of ebola virus infection
Maxime Bessières
,
Elżbieta Plebanek
,
Payel Chatterjee
,
Punya Shrivastava-Ranjan
,
Mike Flint
et al.
Article dans une revue
hal-03717303v1
|
|
|
Synthesis and Antiviral Evaluation of (1,4-Disubstituted-1,2,3-Triazol)-(E)-2-Methyl-but-2-Enyl Nucleoside Phosphonate Prodrugs
Tuniyazi Abuduaini
,
Vincent Roy
,
Julien Marlet
,
Catherine Gaudy-Graffin
,
Denys Brand
et al.
Article dans une revue
inserm-03412066v1
|
|
|
Vers un nouvel antiviral puissant contre les virus à ADN
Vincent Roy
,
Patrick Favetta
,
Luigi A. Agrofoglio
Microscoop. Hors-série, 2021, HS21, pp.8-9
Article dans une revue
hal-03658279v1
|
|
|
Circadian and chemotherapy-related changes in urinary modified nucleosides excretion in patients with metastatic colorectal cancer
S. Dulong
,
Q. Huang
,
P. Innominato
,
A. Karaboue
,
M. Bouchahda
et al.
Article dans une revue
hal-05588725v1
|
|
|
Synthesis of acyclic nucleoside phosphonates targeting Flavin-Dependent Thymidylate Synthase in Mycobacterium tuberculosis
Nicolas G Biteau
,
Vincent Roy
,
J.-C. Lambry
,
Hubert F Becker
,
Hannu Myllykallio
et al.
Article dans une revue
hal-03322503v1
|
|
|
Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–6
Jean Jacques Vanden Eynde
,
Arduino Aleksander Mangoni
,
Jarkko Rautio
,
Jérôme Leprince
,
Yasu-Taka Azuma
et al.
Article dans une revue
hal-03321491v1
|
|
|
Thiopurine Derivative-Induced Fpg/Nei DNA Glycosylase Inhibition: Structural, Dynamic and Functional Insights
Charlotte Rieux
,
Stéphane Goffinont
,
Franck Coste
,
Zahira Tber
,
Julien Cros
et al.
Article dans une revue
hal-05588581v1
|
|
|
Thiopurine Derivative-Induced Fpg/Nei DNA Glycosylase Inhibition: Structural, Dynamic and Functional Insights
Charlotte Rieux
,
Stéphane Goffinont
,
Franck Coste
,
Zahira Tber
,
Julien Cros
et al.
Article dans une revue
hal-03082414v1
|
|
|
Design and Synthesis of Various 5′-Deoxy-5′-(4-Substituted-1,2,3-Triazol-1-yl)-Uridine Analogues as Inhibitors of Mycobacterium tuberculosis Mur Ligases
Vincent Hervin
,
Ritu Arora
,
Jyoti Rani
,
Srinivasan Ramchandran
,
Urmi Bajpai
et al.
Article dans une revue
hal-05588580v1
|
|
|
Monitoring of phosphorylation using immobilized kinases by on-line enzyme bioreactors hyphenated with High-Resolution Mass Spectrometry
Justine Ferey
,
David da Silva
,
Cyril Colas
,
Pierre Lafite
,
Dimitrios Topalis
et al.
Article dans une revue
hal-03466045v1
|
|
|
Synthesis of imprinted hydrogel microbeads by inverse Pickering emulsion to controlled release of adenosine 5′‑monophosphate
Mohamed Ayari
,
Porkodi Kadhirvel
,
Patrick Favetta
,
Bernard Plano
,
Corinne Dejous
et al.
Article dans une revue
hal-02299722v1
|
|
|
Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–4
Arduino A Mangoni
,
Catherine Guillou
,
Jean Jacques Vanden Eynde
,
Christopher Hulme
,
Josef Jampilek
et al.
Article dans une revue
hal-02346060v1
|
|
|
Microwave-assisted Suzuki-Miyaura and Sonogashira coupling of 4-Chloro-2-(trifluoromethyl)pyrido[1,2-e]purine derivatives
Zahira Tber
,
Nicolas G. Biteau
,
Luigi Agrofoglio
,
Julien Cros
,
Stéphane Goffinont
et al.
Article dans une revue
hal-02347523v1
|
|
|
Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–5
Arduino Mangoni
,
Jean Eynde
,
Josef Jampilek
,
Dimitra Hadjipavlou-Litina
,
Hong Liu
et al.
Article dans une revue
hal-03170800v1
|
|
|
Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–6
Jean Jacques Vanden Eynde
,
Arduino Mangoni
,
Jarkko Rautio
,
Jérôme Leprince
,
Yasu-Taka Azuma
et al.
Article dans une revue
hal-05588582v1
|
|
|
Monitoring of successive phosphorylations of thymidine using free and immobilized human nucleoside/nucleotide kinases by Flow Injection Analysis with High-Resolution Mass Spectrometry
Justine Ferey
,
David da Silva
,
Cyril Colas
,
Reine Nehmé
,
Pierre Lafite
et al.
Article dans une revue
hal-02090335v1
|
|
|
Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–4
Arduino Mangoni
,
Catherine Guillou
,
Jean Vanden Eynde
,
Christopher Hulme
,
Josef Jampilek
et al.
Article dans une revue
hal-05588611v1
|
|
|
Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-3
Arduino Mangoni
,
Tiziano Tuccinardi
,
Simona Collina
,
Jean Vanden Eynde
,
Diego Muñoz-Torrero
et al.
Article dans une revue
hal-05588612v1
|
|
|
Highly convergent synthesis and antiviral activity of (E)-but-2-enyl nucleoside phosphonoamidates
Maxime Bessières
,
Vincent Hervin
,
Vincent Roy
,
Agnes Chartier
,
Robert Snoeck
et al.
Article dans une revue
hal-03090373v1
|
|
|
Synthesis and characterization of various 5′-dye-labeled ribonucleosides
Coralie de Schutter
,
Vincent Roy
,
Patrick Favetta
,
Corentin Pavageau
,
Stéphane Maisonneuve
et al.
Article dans une revue
hal-03863168v1
|
|
|
Synthesis and characterization of various 5′-dye-labeled ribonucleosides
Coralie de Schutter
,
Vincent Roy
,
Patrick Favetta
,
Corentin Pavageau
,
Stéphane Maisonneuve
et al.
Article dans une revue
hal-05588609v1
|
|
|
Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-3
Arduino A Mangoni
,
Tiziano Tuccinardi
,
Simona Collina
,
Jean Jacques Vanden Eynde
,
Diego Muñoz-Torrero
et al.
Article dans une revue
hal-02346050v1
|
|
|
Highly convergent synthesis and antiviral activity of (E)-but-2-enyl nucleoside phosphonoamidates
Maxime Bessières
,
Vincent Hervin
,
Vincent Roy
,
Agnès Chartier
,
Robert Snoeck
et al.
Article dans une revue
hal-05588607v1
|
|
|
Selective inhibition of human cathepsin S by 2,4,6-trisubstituted 1,3,5-triazine analogs
Zahira Tber
,
Mylène Wartenberg
,
Jean-Eddy Jacques
,
Vincent Roy
,
Fabien Lecaille
et al.
Article dans une revue
hal-04678746v1
|
|
|
Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–2
Diego Muñoz-Torrero
,
Arduino Mangoni
,
Hong Liu
,
Christopher Hulme
,
Jarkko Rautio
et al.
Article dans une revue
hal-05588606v1
|
|
|
Synthesis of 5,5-difluoro-5-phosphono-pent-2-en-1-yl nucleosides as potential antiviral agents
Florian Chevrier
,
Zein Chamas
,
Thierry Lequeux
,
Emmanuel Pfund
,
G. Andrei
et al.
Article dans une revue
hal-01829613v1
|
|
|
Tailor‐Made Molecularly Imprinted Polymer for Selective Recognition of the Urinary Tumor Marker Pseudouridine
Aleksandra Krstulja
,
Stefania Lettieri
,
Andrew Hall
,
Vincent Roy
,
Patrick Favetta
et al.
Article dans une revue
hal-05588614v1
|
|
|
Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-2 Molecules
Diego Muñoz-Torrero
,
Arduino A Mangoni
,
Hong Liu
,
Christopher Hulme
,
Jarkko Rautio
et al.
Article dans une revue
hal-02345682v1
|
|
|
Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–2
Diego Muñoz-Torrero
,
Arduino Mangoni
,
Hong Liu
,
Christopher Hulme
,
Jarkko Rautio
et al.
Article dans une revue
hal-05588586v1
|
|
|
Synthesis of 5,5-difluoro-5-phosphono-pent-2-en-1-yl nucleosides as potential antiviral agents
F. Chevrier
,
Z. Chamas
,
T. Lequeux
,
E. Pfund
,
G. Andrei
et al.
Article dans une revue
hal-05588613v1
|
|
|
Love Acoustic Wave-Based Devices and Molecularly-Imprinted Polymers as Versatile Sensors for Electronic Nose or Tongue for Cancer Monitoring
Corinne Dejous
,
Hamida Hallil
,
Vincent Raimbault
,
Jean-Luc Lachaud
,
Bernard Plano
et al.
Article dans une revue
hal-05588615v1
|
|
|
Sonication‐Assisted Synthesis of (E) ‐2‐Methyl‐but‐2‐enyl Nucleoside Phosphonate Prodrugs
Maxime Bessières
,
Ozkan Sari
,
Vincent Roy
,
Dawid Warszycki
,
Andrzej Bojarski
et al.
Article dans une revue
hal-05588616v1
|
|
|
Love Acoustic Wave-Based Devices and Molecularly-Imprinted Polymers as Versatile Sensors for Electronic Nose or Tongue for Cancer Monitoring
Corinne Dejous
,
Hamida Hallil
,
Vincent Raimbault
,
Jean-Luc Lachaud
,
Bernard Plano
et al.
Article dans une revue
hal-01356195v1
|
|
|
Straightforward synthesis of 2,4,6-trisubstituted 1,3,5-triazine compounds targeting cysteine cathepsins K and S
Elżbieta Plebanek
,
Florian Chevrier
,
Vincent Roy
,
Thibault Garenne
,
Fabien Lecaille
et al.
Article dans une revue
hal-05588617v1
|
|
|
Synthesis of dihydropyrimidine α,γ-diketobutanoic acid derivatives targeting HIV integrase
Ozkan Sari
,
Vincent Roy
,
Mathieu Métifiot
,
Christophe Marchand
,
Yves Pommier
et al.
Article dans une revue
hal-02904762v1
|
|
|
Synthesis of a molecularly imprinted polymer to isolate glucosamine from plant extracts by an ionic–non‐covalent dual approach
N. Henry
,
P. Favetta
,
R. Delépée
,
J.‐m. Seigneuret
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588620v1
|
|
|
Synthesis of a molecularly imprinted polymer to isolate glucosamine from plant extracts by an ionic-non-covalent dual approach
N. Henry
,
P. Favetta
,
R. Delépée
,
J.-M. Seigneuret
,
L. Agrofoglio
Article dans une revue
istex
hal-03593458v1
|
|
|
Recent Progress for the Synthesis of Selected Carbocyclic Nucleosides
Maxime Bessières
,
Florian Chevrier
,
Vincent Roy
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588619v1
|
|
|
Active site labeling of cysteine cathepsins by a straightforward diazomethylketone probe derived from the N-terminus of human cystatin C
Thibaut Garenne
,
Ahlame Saidi
,
Brendan Gilmore
,
Elżbieta Niemiec
,
Vincent Roy
et al.
Article dans une revue
istex
hal-05588618v1
|
|
|
Synthesis of Fluorine-Containing 3,3-Disubstituted Oxetanes and Alkylidene Oxetanes
Romain Laporte
,
Anais Prunier
,
Emmanuel Pfund
,
Vincent Roy
,
Luigi Agrofoglio
et al.
Article dans une revue
istex
hal-02348052v1
|
|
|
Love Wave Sensor Based on Thin Film Molecularly Imprinted Polymer: Study of VOCs Adsorption
Hamida Hallil
,
Nima Omar-Aouled
,
Bernard Plano
,
Raphaël Delépée
,
Luigi A. Agrofoglio
et al.
Journal of Integrated Circuits and Systems, 2014, 9 (2), pp.118-122
Article dans une revue
hal-01241891v1
|
|
|
Detection of urinary modified nucleosides by a bulk acoustic wave MIP sensor - Results and future work
Luigi A. Agrofoglio
,
Aleksandra Krstulja
,
Coralie de Schutter
,
Patrick Favetta
,
Raphaël Delépée
et al.
Article dans une revue
istex
hal-00988691v1
|
|
|
Evaluation of molecularly imprinted polymers using 2′,3′,5′-tri-O-acyluridines as templates for pyrimidine nucleoside recognition
Aleksandra Krstulja
,
Stefania Lettieri
,
Andrew Hall
,
Raphael Delépée
,
Patrick Favetta
et al.
Article dans une revue
hal-03593455v1
|
|
|
A convenient, highly selective and eco-friendly N-Boc protection of pyrimidines under microwave irradiation
Maxime Bessières
,
Vincent Roy
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588726v1
|
|
|
Study of gaseous compounds adsorption with a Love wave sensor based on molecularly imprinted polymer thin film
Nima Omar-Aouled
,
Naïma Lebal
,
Hamida Hallil
,
Raphael Delepee
,
Luigi A. Agrofoglio
et al.
Sensors & Transducers., 2013, 149 (2), pp.37-42
Article dans une revue
hal-00817577v1
|
|
|
Synthesis and broad spectrum antiviral evaluation of bis(POM) prodrugs of novel acyclic nucleosides
Manabu Hamada
,
Vincent Roy
,
Tamara Mcbrayer
,
Tony Whitaker
,
Cesar Urbina-Blanco
et al.
Article dans une revue
hal-05588728v1
|
|
|
Combination of computational methods, adsorption isotherms and selectivity tests for the conception of a mixed non-covalent–semi-covalent molecularly imprinted polymer of vanillin
Kinga Puzio
,
Raphaël Delépée
,
Richard Vidal
,
Luigi Agrofoglio
Article dans une revue
istex
hal-03593453v1
|
|
|
Phase I Dose‐Escalation Pharmacokinetics of AZT‐P‐ddI (IVX‐E‐59) in Patients with Human Immunodeficiency Virus
Xiao‐jian Zhou
,
Kathleen Squires
,
Xin‐ru Pan-Zhou
,
Steve Bernhard
,
Luigi A. Agrofoglio
et al.
Article dans une revue
istex
hal-05588851v1
|
|
|
Nucleosides analogs recognition by Molecularly Imprinted Polymer- coated Love wave sensor
Naïma Lebal
,
Hamida Hallil
,
Corinne Dejous
,
B. Plano
,
Aleksandra Krstulja
et al.
Article dans une revue
hal-00847369v1
|
|
|
The Preparation of Trisubstituted Alkenyl Nucleoside Phosphonates under Ultrasound-Assisted Olefin Cross-Metathesis
Ozkan Sari
,
Manabu Hamada
,
Vincent Roy
,
Steven Nolan
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588727v1
|
|
|
Synthesis of water-compatible imprinted polymers of in situ produced fructosazine and 2,5-deoxyfructosazine
Nathaly Henry
,
Raphaël Delépée
,
Jean-Marc Seigneuret
,
Luigi Agrofoglio
Article dans une revue
istex
hal-03593450v1
|
|
|
Synthesis and antiviral evaluation of bis(POM) prodrugs of (E)-[4′-phosphono-but-2′-en-1′-yl]purine nucleosides
Ugo Pradère
,
Vincent Roy
,
Aurélien Montagu
,
Ozkan Sari
,
Manabu Hamada
et al.
Article dans une revue
istex
hal-05588730v1
|
|
|
Efficient Synthesis of Unprotected C-5-Aryl/Heteroaryl-2'-deoxyuridine via a Suzuki-Miyaura Reaction in Aqueous Media
Nathalie Fresneau
,
Marie-Aude Hiebel
,
Luigi A. Agrofoglio
,
Sabine Berteina-Raboin
Article dans une revue
hal-05588729v1
|
|
|
Synthesis and antiviral evaluation of C5-substituted-(1,3-diyne)-2′-deoxyuridines
Ozkan Sari
,
Vincent Roy
,
Jan Balzarini
,
Robert Snoeck
,
Graciela Andrei
et al.
Article dans une revue
istex
hal-05588731v1
|
|
|
One-pot Sonogashira-cyclization protocol to obtain substituted furopyrimidine nucleosides in aqueous conditions
Nathalie Fresneau
,
Marie-Aude Hiebel
,
Luigi A. Agrofoglio
,
Sabine Berteina-Raboin
Article dans une revue
istex
hal-05588732v1
|
|
|
Synthesis and Anti-HIV Evaluation of 3′-Triazolo Nucleosides
Vincent Roy
,
Aleksandr Obikhod
,
Hong-Wang Zhang
,
Steven Coats
,
Brian Herman
et al.
Article dans une revue
hal-05588733v1
|
|
|
Expeditious convergent procedure for the preparation of bis(POC) prodrugs of new (E)-4-phosphono-but-2-en-1-yl nucleosides
Aurélien Montagu
,
Ugo Pradére
,
Vincent Roy
,
Steven Nolan
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588746v1
|
|
|
In Situ One-Step Method for Synthesis of “Click”-Functionalized Monolithic Stationary Phase for Capillary Electrochromatography
Aleksander Salwiński
,
Vincent Roy
,
Luigi Agrofoglio
,
Raphaël Delépée
Article dans une revue
istex
hal-03593449v1
|
|
|
Synthesis of new C5-(1-substituted-1,2,3-triazol-4 or 5-yl)-2′-deoxyuridines and their antiviral evaluation
Aurélien Montagu
,
Vincent Roy
,
Jan Balzarini
,
Robert Snoeck
,
Graciela Andrei
et al.
Article dans une revue
istex
hal-05588749v1
|
|
|
The Shortest Strategy for Generating Phosphonate Prodrugs by Olefin Cross‐Metathesis – Application to Acyclonucleoside Phosphonates
Ugo Pradère
,
Hervé Clavier
,
Vincent Roy
,
Steven Nolan
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588734v1
|
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3′-(1,2,3-Triazol-1-yl)-3′-deoxythymidine analogs as substrates for human and Ureaplasma parvum thymidine kinase for structure–activity investigations
Jay Lin
,
Vincent Roy
,
Liya Wang
,
Li You
,
Luigi A. Agrofoglio
et al.
Article dans une revue
hal-05588752v1
|
|
|
Potential and Perspectives of Cyclonucleosides
A. Mieczkowski
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588756v1
|
|
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Novel Antiviral C5-Substituted Pyrimidine Acyclic Nucleoside Phosphonates Selected as Human Thymidylate Kinase Substrates
Dimitri Topalis
,
Ugo Pradère
,
Vincent Roy
,
Christophe Caillat
,
Ahmed Azzouzi
et al.
Article dans une revue
hal-05588748v1
|
|
|
Preparation of Carbocyclic C ‐Nucleosides from α‐Chlorooxime Precursor
Ugo Pradere
,
Hiroki Kumamoto
,
Vincent Roy
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588755v1
|
|
|
Human and viral nucleoside/nucleotide kinases involved in antiviral drug activation: Structural and catalytic properties
Dominique Deville-Bonne
,
Chahrazade El Amri
,
Philippe Meyer
,
Yuxing Chen
,
Luigi A. Agrofoglio
et al.
Article dans une revue
istex
hal-05588750v1
|
|
|
Microwave-Assisted Syntheses of Nucleosides and Their Precursors
Vincent Roy
,
Ugo Pradère
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588754v1
|
|
|
Preparation of Cyclonucleosides
Adam Mieczkowski
,
Vincent Roy
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588753v1
|
|
|
Click Azide‐Alkyne Cycloaddition for the Synthesis of D ‐(–)‐1,4‐Disubstituted Triazolo‐Carbanucleosides
Julie Broggi
,
Hiroki Kumamoto
,
Sabine Berteina-Raboin
,
Steven Nolan
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588766v1
|
|
|
Phosphorylation of dGMP analogs by vaccinia virus TMP kinase and human GMP kinase.
Constance Auvynet
,
Dimitri Topalis
,
Christophe Caillat
,
Hélène Munier-Lehmann
,
Edward Seclaman
et al.
Article dans une revue
pasteur-00417244v1
|
|
|
Synthesis of (±)-1,2,3-triazolo-3′-deoxy-4′-hydroxymethyl carbanucleosides via ‘click’ cycloaddition
Julie Broggi
,
Nicolas Joubert
,
Silvia Díez-González
,
Sabine Berteina-Raboin
,
Thomas Zevaco
et al.
Article dans une revue
istex
hal-05588764v1
|
|
|
Preparation of C-5-substituted 6,5′-O-anhydrouridine by Sn–Pd transmetallation-coupling process and their use
Adam Mieczkowski
,
Jerome Blu
,
Vincent Roy
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588759v1
|
|
|
Molecular imprinting of AMP by an ionic-noncovalent dual approach
Florent Breton
,
Raphaël Delépée
,
Luigi Agrofoglio
Article dans une revue
istex
hal-03593445v1
|
|
|
A short and stereoselective synthesis of carbocyclic alpha ‐l‐dideoxyhomonucleosides
F. Girard
,
M.‐g. Lee
,
Luigi A. Agrofoglio
,
A. Fridland
Article dans une revue
hal-05588827v1
|
|
|
Preparation of C5-substituted O6,5′-cyclouridine
Adam Mieczkowski
,
Pauline Peltier
,
Thomas Zevaco
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588761v1
|
|
|
Preparation of ribavirin analogues by copper- and ruthenium-catalyzed azide-alkyne 1,3-dipolar cycloaddition
Ugo Pradere
,
Vincent Roy
,
Tamara Mcbrayer
,
Raymond Schinazi
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588767v1
|
|
|
Evaluation of C-5 Substituted Uracil Acyclic Phosphonates as Substrates or Inhibitors for DTMP and UMP–CMP Kinases and Potential Antipox Derivatives
Dimitri Topalis
,
Julie Broggi
,
Julie A.C. Alexandre
,
Ugo Pradère
,
Vincent Roy
et al.
Article dans une revue
istex
hal-05588776v1
|
|
|
Preparation of acyclo nucleoside phosphonate analogues based on cross-metathesis
Hiroki Kumamoto
,
Dimitri Topalis
,
Julie Broggi
,
Ugo Pradère
,
Vincent Roy
et al.
Article dans une revue
istex
hal-05588774v1
|
|
|
Molecularly imprinted polymer of 5-methyluridine for solid-phase extraction of pyrimidine nucleoside cancer markers in urine
Damien Jégourel
,
Raphaël Delépée
,
Florent Breton
,
Antoine Rolland
,
Richard Vidal
et al.
Article dans une revue
istex
hal-03593440v1
|
|
|
Crystal structure of poxvirus thymidylate kinase: an unexpected dimerization has implications for antiviral therapy.
Christophe Caillat
,
Dimitri Topalis
,
Luigi A. Agrofoglio
,
Sylvie Pochet
,
Jan Balzarini
et al.
Proceedings of the National Academy of Sciences of the United States of America, 2008, 105 (44), pp.16900-5. ⟨10.1073/pnas.0804525105⟩
Article dans une revue
pasteur-00347333v1
|
|
|
Study of Copper(I) Catalysts for the Synthesis of Carbanucleosides via Azide-Alkyne 1,3-Dipolar Cycloaddition
Julie Broggi
,
Silvia Díez-González
,
Jeffrey Petersen
,
Sabine Berteina-Raboin
,
Steven Nolan
et al.
Article dans une revue
hal-05588781v1
|
|
|
Synthesis and anti-HIV activity of 5-haloethynyl and 5-(1,2-dihalo)vinyl analogues of AZT and FLT
Nicolas Joubert
,
Franck Amblard
,
Kimberly Rapp
,
Raymond Schinazi
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588773v1
|
|
|
Microwave-Assisted Silylation-Amination of Uracil Acyclonucleosides to 4-Alkylamino-2(1 H )-Pyrimidinone Analogues
Vincent Roy
,
Adam Mieczkowski
,
Dimitri Topalis
,
Sabine Berteina-Raboin
,
Dominique Deville-Bonne
et al.
Article dans une revue
hal-05588770v1
|
|
|
Selective adenosine-5′-monophosphate uptake by water-compatible molecularly imprinted polymer
Florent Breton
,
Raphaël Delépée
,
Damien Jégourel
,
Dominique Deville-Bonne
,
Luigi Agrofoglio
Article dans une revue
istex
hal-03593439v1
|
|
|
Mass Spectrometry Based Methods for Analysis of Nucleosides as Antiviral Drugs and Potential Tumor Biomarkers
Luigi Agrofoglio
,
Vincent Bezy
,
Patrick Chaimbault
,
Raphaël Delépée
,
Boutaina Rhourri
et al.
Article dans une revue
hal-03593436v1
|
|
|
Specificity enhancement with LC‐positive ESI‐MS/MS for the measurement of nucleotides: application to the quantitative determination of carbovir triphosphate, lamivudine triphosphate and tenofovir diphosphate in human peripheral blood mononuclear cells
Alain Pruvost
,
Frédéric Théodoro
,
Luigi A. Agrofoglio
,
Eugenia Negredo
,
Henri Bénech
Article dans une revue
istex
hal-05588778v1
|
|
|
EFFICIENT SYNTHESIS OF D -[1′- 13 C]-RIBONUCLEOSIDES FOR INCORPORATION INTO OLIGO-RNA
Y. Saito
,
A. Nyilas
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588810v1
|
|
|
Study of different copper(I) catalysts for the "click chemistry" approach to carbanucleosides
J. Broggi
,
N. Joubert
,
Vincent Aucagne
,
T. Zevaco
,
S. Berteina-Raboin
et al.
Nucleosides, Nucleotides and Nucleic Acids, 2007, 26, pp.779-783
Article dans une revue
hal-00275217v1
|
|
|
ANALYSIS OF ANTI-HIV NUCLEOSIDE INHIBITORS BY CAPILLARY ELECTROPHORESIS-ELECTROSPRAY IONIZATION MASS SPECTROMETRY
Luigi A. Agrofoglio
,
X. Cahours
,
T. Tran
,
H. Dessans
,
C. Kieda
et al.
Article dans une revue
hal-05588817v1
|
|
|
Nucleotide binding to human UMP-CMP kinase using fluorescent derivatives - a screening based on affinity for the UMP-CMP binding site.
Dimitri Topalis
,
Hiroki Kumamoto
,
Maria-Fernanda Amaya Velasco
,
Laurence Dugué
,
Ahmed Haouz
et al.
Article dans une revue
pasteur-00166127v1
|
|
|
Cross-Metathesis Mediated Synthesis of New Acyclic Nucleoside Phosphonates
Vincent Roy
,
Hiroki Kumamoto
,
Sabine Berteina-Raboin
,
Steven Nolan
,
Dimitri Topalis
et al.
Article dans une revue
hal-05588782v1
|
|
|
Alkyne-Azide Click Chemistry Mediated Carbanucleosides Synthesis
Julie Broggi
,
Nicolas Joubert
,
Vincent Aucagne
,
Sabine Berteina-Raboin
,
S. Diez-Gonzalez
et al.
Article dans une revue
hal-04678703v1
|
|
|
Supported Synthesis and Functionnalization of 2″-Deoxyuridine by Suzuki-Miyaura Cross-Coupling
Saïd El Kazzouli
,
Sabine Berteina-Raboin
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588783v1
|
|
|
SYNTHESIS OF CARBOCYCLIC PHOSPHONONUCLEOSIDES
B. Legeret
,
Z. Sarakauskaite
,
F. Pradaux
,
Y. Saito
,
S. Tumkevicius
et al.
Article dans une revue
hal-05588814v1
|
|
|
SYNTHESIS OF CARBOCYCLIC PHOSPHONONUCLEOSIDES
B. Légeret
,
Z. Sarakauskaite
,
F. Pradaux
,
Y. Saito
,
S. Tumkevicius
et al.
Article dans une revue
hal-02061990v1
|
|
|
Looking for new pyrimidine acyclic nucleotide analogues designed for phosphorylation by human ump-cmp kinase.
Dimitri Topalis
,
Hiroki Kumamoto
,
Julie a C Alexandre
,
Laurence Dugué
,
Sylvie Pochet
et al.
Article dans une revue
pasteur-00202298v1
|
|
|
Alkyne-Azide Click Chemistry Mediated Carbanucleosides Synthesis
Julie Broggi
,
Nicolas Joubert
,
Vincent Aucagne
,
Sabine Berteina-Raboin
,
S. Diez-Gonzalez
et al.
Article dans une revue
hal-02086003v1
|
|
|
An Overview of Diazine Nucleoside Analogues
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588787v1
|
|
|
Analysis and validation of the phosphorylated metabolites of two anti‐human immunodeficiency virus nucleotides (stavudine and didanosine) by pressure‐assisted CE‐ESI‐MS/MS in cell extracts: Sensitivity enhancement by the use of perfluorinated acids and alcohols as coaxial sheath‐liquid make‐up constituents
Vincent Bezy
,
Patrick Chaimbault
,
Philippe Morin
,
Steve Unger
,
Marie‐charlotte Bernard
et al.
Article dans une revue
istex
hal-05588786v1
|
|
|
Efficient synthesis of various acycloalkenyl derivatives of pyrimidine using cross-metathesis and Pd(0) methodologies
Franck Amblard
,
Steven Nolan
,
Raymond Schinazi
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588793v1
|
|
|
Efficient Pd(0)-catalyzed synthesis of 1,2,3-triazolo-3′-deoxycarbanucleosides and their analogues
Nicolas Joubert
,
Raymond Schinazi
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588788v1
|
|
|
Metathesis strategy in nucleoside chemistry
Franck Amblard
,
Steven Nolan
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588791v1
|
|
|
Synthesis of 5-haloethynyl- and 5-(1,2-dihalo)vinyluracil nucleosides: Antiviral activity and cellular toxicity
Vanessa Escuret
,
Vincent Aucagne
,
Nicolas Joubert
,
David Durantel
,
Kimberly Rapp
et al.
Article dans une revue
istex
hal-02086013v1
|
|
|
Synthesis and antiviral activity of novel acyclic nucleosides in the 5-alkynyl- and 6-alkylfuro[2,3-d]pyrimidine series
Franck Amblard
,
Vincent Aucagne
,
Pierre Guenot
,
Raymond Schinazi
,
Luigi Agrofoglio
Article dans une revue
istex
hal-02086014v1
|
|
|
Olefin Metathesis Route to Antiviral Nucleosides
Luigi A. Agrofoglio
,
Steven Nolan
Article dans une revue
istex
hal-05588790v1
|
|
|
Highly Efficient AgNO3-Catalyzed Preparation of Substituted Furanopyrimidine Nucleosides [cf. (III)].
Vincent Aucagne
,
Franck Amblard
,
Luigi Agrofoglio
Article dans une revue
istex
hal-02086027v1
|
|
|
Simultaneous analysis of several antiretroviral nucleosides in rat-plasma by high-performance liquid chromatography with UV using acetic acid/hydroxylamine bufferTest of this new volatile medium-pH for HPLC–ESI-MS/MS
V Bezy
,
P Morin
,
P Couerbe
,
G Leleu
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588792v1
|
|
|
Highly Efficient AgNO 3 -Catalyzed Preparation of Substituted Furanopyrimidine Nucleosides
Vincent Aucagne
,
Franck Amblard
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588795v1
|
|
|
Palladium-Catalyzed Synthesis of Uridines on Polystyrene-Based Solid Supports
Vincent Aucagne
,
Sabine Berteina-Raboin
,
Pierre Guenot
,
Luigi Agrofoglio
Article dans une revue
hal-02086022v1
|
|
|
Synthesis of l-cyclopentenyl nucleosides using ring-closing metathesis and palladium-mediated allylic alkylation methodologies
Luigi A. Agrofoglio
,
Franck Amblard
,
Steven Nolan
,
Steve Charamon
,
Isabelle Gillaizeau
et al.
Article dans une revue
hal-05588796v1
|
|
|
Straightforward Synthesis of Labeled and Unlabeled Pyrimidine d4Ns via 2′,3′-Diyne seco Analogues through Olefin Metathesis Reactions
Isabelle Gillaizeau
,
Irene m. Lagoja
,
Steve p. Nolan
,
Vincent Aucagne
,
Jef Rozenski
et al.
Article dans une revue
istex
hal-02086029v1
|
|
|
Liquid chromatographic separation of phosphoramidate diastereomers on a polysaccharide-type chiral stationary phase
Nathalie Mesplet
,
Yoshio Saito
,
Philippe Morin
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588801v1
|
|
|
A new route to acyclic nucleosides via palladium-mediated allylic alkylation and cross-metathesis
Franck Amblard
,
Steven Nolan
,
Isabelle Gillaizeau
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588799v1
|
|
|
HPLC and mass spectrometry analysis of the enzymatic hydrolysis of anti-HIV pronucleotide diastereomers
Nathalie Mesplet
,
Yoshio Saito
,
Philippe Morin
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588800v1
|
|
|
Palladium-Assisted Routes to Nucleosides
Luigi A. Agrofoglio
,
Isabelle Gillaizeau
,
Yoshio Saito
Article dans une revue
hal-05588797v1
|
|
|
Synthesis of a Novel Heterocyclic System: 2H-2,3,5,6,9-Pentaazabenz[cd]azulene
Sigitas Tumkevicius
,
Luigi Agrofoglio
,
Andrius Kaminskas
,
Gintaras Urbelis
,
Thomas Zevaco
et al.
Article dans une revue
hal-05588806v1
|
|
|
Chemical synthesis of 13C labeled anti-HIV nucleosides as mass-internal standards
Yoshio Saito
,
Thomas Zevaco
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588803v1
|
|
|
Analysis of intracellular didanosine triphosphate at sub-ppb level using LC-MS/MS
Xavier Cahours
,
Thanh Thu Tran
,
Nathalie Mesplet
,
Claudine Kieda
,
Philippe Morin
et al.
Article dans une revue
istex
hal-05588816v1
|
|
|
Synthesis of isotopically labeled d-[1′-13C]ribonucleoside phosphoramidites
Yoshio Saito
,
Agnès Nyilas
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588807v1
|
|
|
Enantioselective synthesis of carba- l -furanose precursors of carbanucleosides, using ring-closing metathesis
Isabelle Gillaizeau
,
Steve Charamon
,
Luigi A. Agrofoglio
Article dans une revue
hal-05588815v1
|
|
|
Simultaneous quantitation of nucleoside HIV-1 reverse transcriptase inhibitors by short-end injection capillary electrochromatography on a β-cyclodextrin-bonded silica stationary phase
Nathalie Mesplet
,
Philippe Morin
,
Carole François
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588811v1
|
|
|
Determination at ppb level of an anti-human immunodeficiency virus nucleoside drug by capillary electrophoresis–electrospray ionization tandem mass spectrometry
Xavier Cahours
,
Hélène Dessans
,
Philippe Morin
,
Michel Dreux
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588820v1
|
|
|
Determination at ppb level of an anti-human immunodeficiency virus nucleoside drug by capillary electrophoresis–electrospray ionization tandem mass spectrometry
Xavier Cahours
,
Hélène Dessans
,
Philippe Morin
,
Michel Dreux
,
Luigi Agrofoglio
Article dans une revue
istex
hal-03298652v1
|
|
|
Synthesis of 5′-Thioalkyl, Sulfoxide and Sulfone Pyrimidine Nucleosides
Luigi A. Agrofoglio
,
F. Girard
,
F. Fleury
,
S. Léonce
Article dans une revue
hal-05588823v1
|
|
|
Chiral Synthesis of Carbocyclic Analogues of l -ribofuranosides
Peiyuan Wang
,
Luigi A. Agrofoglio
,
M. Gary Newton
,
Chung Chu
Article dans une revue
hal-05588822v1
|
|
|
Enantiomeric synthesis of nucleosides
Luigi A. Agrofoglio
,
Christine Demaison
,
Loïc Toupet
Article dans une revue
istex
hal-05588826v1
|
|
|
Stereoselective Synthesis of Carbocyclic α-L-Homonucleosides
Luigi A. Agrofoglio
,
F. Girard
,
C. Demaison
,
M-G. Lee
,
P. Roingeard
et al.
Article dans une revue
hal-05588825v1
|
|
|
Stereoselective synthesis of α-l-bicarbocyclic nucleosides as potential antiviral drugs
Christine Demaison
,
Christophe Hourioux
,
Philippe Roingeard
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588831v1
|
|
|
Asymmetric synthesis of L-cyclopentyl carbocyclic nucleosides
Peiyuan Wang
,
Luigi A. Agrofoglio
,
M. Gary Newton
,
Chung Chu
Article dans une revue
istex
hal-05588852v1
|
|
|
Synthesis of Some 5′-Thiopentofuranosylpyrimidines as Potential Anti-tumor Agents.
Frédéric Girard
,
Stephane Leonce
,
Luigi A. Agrofoglio
Article dans une revue
istex
hal-05588853v1
|
|
|
A multigram, stereoselective synthesis of d-[13C5]ribose from d-[13C6]glucose and its conversion into [13C5]nucleosides
Luigi A. Agrofoglio
,
Jean-Claude Jacquinet
,
Gérard Lancelot
Article dans une revue
istex
hal-05588855v1
|
|
|
Inhibition of human immunodeficiency virus type 1 reverse transcriptase by the 5'-triphosphate beta enantiomers of cytidine analogs
A Faraj
,
Luigi A. Agrofoglio
,
J Wakefield
,
S Mcpherson
,
C Morrow
et al.
Article dans une revue
hal-05588858v1
|
|
|
Synthesis of carbocyclic nucleosides
Luigi A. Agrofoglio
,
Edouard Suhas
,
Audrey Farese
,
Roger Condom
,
S. Richard Challand
et al.
Article dans une revue
istex
hal-05588857v1
|
|
|
Synthesis of Three New Carbocyclic Analogues of 3′-Deoxy Purine Ribonucleosides
Luigi A. Agrofoglio
,
Roger Condom
,
Roger Guedj
,
S. Richard Challand
,
John Selway
Article dans une revue
hal-05588860v1
|
|
|
Synthesis of a new exocyclic amino carbocyclic nucleoside with potential antiviral activity.
Luigi A. Agrofoglio
,
Roger Condom
,
Roger Guedj
,
Richard Challand
,
John Selway
Article dans une revue
istex
hal-05588861v1
|
|
|
Steric control of the epoxidation of 1-hydroxymethyl-3-cyclopentene using aryl or silyl hydroxyl protecting groups.
Luigi A. Agrofoglio
,
Roger Condom
,
Roger Guedj
Article dans une revue
istex
hal-05588862v1
|