Marc Le Borgne

Identifiants chercheurs

IdHAL :

marc-le-borgne

ORCID :

0000-0003-1398-075X

IdRef :

095367829

ResearcherID :

http://www.researcherid.com/rid/H-1036-2014

Présentation

Publications

Article dans une revue (121)

Synthesis of Indeno[1,2-b]indole-9,10-diones: Toward a One-Pot, Two-Step Reaction Johana Charles,Marc Le Borgne,Ema Verel,Jean Guillon,Noël Pinaudet al. Synthesis: Journal of Synthetic Organic Chemistry, 2026, ⟨10.1055/a-2764-1257⟩ Article dans une revue hal-05487827v1
Identification of an N-methylpyrazole derivative as a selective inhibitor of breast cancer resistance protein (BCRP/ABCG2) Andrezza Braiane Ferreira Siridó,Arthur Henrique Gomes de Oliveira,Julia Poletto,Thales Kronenberger,Fabiane Gomes de Moraes Regoet al. Archives of Biochemistry and Biophysics, 2026, 779, pp.110761. ⟨10.1016/j.abb.2026.110761⟩ Article dans une revue hal-05528887v1
Functionalized nitrogen- and chalcogen-containing heterocyclic compounds as aromatase inhibitors: Design, synthesis and biological evaluation Chang Ha Park,Marc Le Borgne,Marouan Rami,Martin Fossart,Patricia Melnyket al. European Journal of Medicinal Chemistry, 2026, 302, ⟨10.1016/j.ejmech.2025.118298⟩ Article dans une revue hal-05432136v1
Crystallographic Fragment Screening with CK2α’, an Isoform of Human Protein Kinase CK2 Catalytic Subunit, and Its Use to Obtain a CK2α’/Heparin Complex Structure Christian Werner,Tatjana Barthel,Hugo Harasimowicz,Christelle Marminon,Manfred S Weisset al. Kinases and Phosphatases, 2026, 4 (1), pp.1. ⟨10.3390/kinasesphosphatases4010001⟩ Article dans une revue hal-05487842v1
Design, synthesis, and structure–activity relationship studies of 6 H -benzo[ b ]indeno[1,2- d ]thiophen-6-one derivatives as DYRK1A/CLK1/CLK4/haspin inhibitors Abdelfattah Faouzi,Alexandre Arnaud,François Hallé,Jean Roussel,Mandy Aymardet al. RSC Medicinal Chemistry, 2025, 16 (1), pp.179-199. ⟨10.1039/d4md00537f⟩ Article dans une revue hal-04961871v1
Formulation and Evaluation of Alginate Microcapsules Containing an Uncompetitive Nanomolar Dimeric Indenoindole Inhibitor of the Human Breast Cancer Resistance Pump ABCG2 with Different Excipients Krisztina Bodnár,Christelle Marminon,Florent Perret,Ádám Haimhoffer,Boglárka Pappet al. Pharmaceutics, 2025, 17 (12), pp.1587. ⟨10.3390/pharmaceutics17121587⟩ Article dans une revue hal-05487860v1
From toxic materials to food-grade materials: A major challenge for battery design – A mini review Marina Le Borgne,Perrine Ximenes,Marc Le Borgne De Remediis, 2025, 2 (1), ⟨10.71116/7qz2f897⟩ Article dans une revue hal-05487879v1
Exploring the biological potential of the brominated indenoindole MC11 and its interaction with protein kinase CK2 Christelle Marminon,Christian Werner,Alexander Gast,Lars Herfindal,Johana Charleset al. Biological Chemistry, 2025, 406 (3-4), pp.125-138. ⟨10.1515/hsz-2024-0160⟩ Article dans une revue hal-05002241v2
Kinetics of benzophenone-3 release from clay minerals or organosilicates for sun protection formulation Saddam Charaabi,Samar Issa,Anne-Marie Pensé-Lhéritier,Marc Le Borgne International Journal of Pharmaceutics, 2025, 682, pp.125920. ⟨10.1016/j.ijpharm.2025.125920⟩ Article dans une revue hal-05159385v1
To be or not to be manipulated by our bacteria? Marina Le Borgne,Kézia Sossou-Echavidre,Christine Janssen,Marc Le Borgne De Remediis, 2024, 1 (1), pp.25-38. ⟨10.71116/vj4jx563⟩ Article dans une revue hal-04880866v1
New 2,4-bis[(substituted-aminomethyl)phenyl]phenylquinazoline and 2,4-bis[(substituted-aminomethyl)phenyl]phenylquinoline derivatives: synthesis and biological evaluation as novel anticancer agents by targeting G-quadruplex Jean Guillon,Marc Le Borgne,Vittoria Milano,Aurore Guédin-Beaurepaire,Stéphane Moreauet al. Pharmaceuticals, 2024, 17 (1), pp.30. ⟨10.3390/ph17010030⟩ Article dans une revue hal-04390485v1
Efficient synthesis, crystallographic study, antimicrobial activity and in silico studies of novel bioactive α-aminophosphonates based on pyridine moiety Ismahene Grib,Malika Berredjem,Seif-Eddine Djouad,Chahrazed Benzaid,Khadidja Otmane Rachediet al. Journal of Molecular Structure, 2024, 1309, pp.138138. ⟨10.1016/j.molstruc.2024.138138⟩ Article dans une revue hal-04775535v1
Antibody–drug conjugates: prospects for the next generation Meriem Grairi,Marc Le Borgne Drug Discovery Today, 2024, 29 (12), pp.104241. ⟨10.1016/j.drudis.2024.104241⟩ Article dans une revue hal-04880853v1
L’Europe révise sa période de transition pour l’usage des alliages dentaires cobalt-chrome Christine Janssen,Marc Le Borgne,Brigitte Grosgogeat Biomatériaux Cliniques Dentaires, 2024, 9 (2), pp.90-91 Article dans une revue hal-04880822v1
Formulation and Investigation of CK2 Inhibitor-Loaded Alginate Microbeads with Different Excipients Boglárka Papp,Marc Le Borgne,Florent Perret,Christelle Marminon,Liza Józsaet al. Pharmaceutics, 2023, Dosage Form Formulation Technologies for Improving Bioavailability, 15 (12), pp.2701. ⟨10.3390/pharmaceutics15122701⟩ Article dans une revue hal-04314651v1
Drug candidates targeting multidrug resistance in cancer and infections Marc Le Borgne,Pierre Falson,Ahcène Boumendjel European Journal of Medicinal Chemistry, 2023, 249, pp.115173. ⟨10.1016/j.ejmech.2023.115173⟩ Article dans une revue hal-03972628v1
Inhibitors of ABCG2-mediated multidrug resistance: Lead generation through computer-aided drug design Laura Goracci,Alessandra Nurisso,Emile Roussel,Basile Pérès,Vincent Chaptalet al. European Journal of Medicinal Chemistry, 2023, 248, pp.115070. ⟨10.1016/j.ejmech.2022.115070⟩ Article dans une revue hal-03939266v1
Tetanus Toxin Fragment C: Structure, Drug Discovery Research and Production Caroline Bayart,Angélique Mularoni,Nada Hemmani,Soumeya Kerachni,Joachim Joseet al. Pharmaceuticals, 2022, 15 (6), pp.756. ⟨10.3390/ph15060756⟩ Article dans une revue hal-03718458v1
Toxicological Risks of the Cobalt–Chromium Alloys in Dentistry: A Systematic Review Brigitte Grosgogeat,Alina Vaicelyte,Rémy Gauthier,Christine Janssen,Marc Le Borgne Materials, 2022, 15 (17), pp.5801. ⟨10.3390/ma15175801⟩ Article dans une revue hal-03815561v1
Improved biological performance of ketoprofen using novel modified halloysite clay nanotubes Dounia Sid,Milad Baitiche,Lekhmici Arrar,Ferhat Djerboua,Riadh Bourzamiet al. Applied Clay Science, 2022, 216, pp.106341. ⟨10.1016/j.clay.2021.106341⟩ Article dans une revue hal-03475833v1
4,5,7‐trisubstituted indeno[1,2‐ b ]indole inhibits CK2 activity in tumor cells equivalent to CX‐4945 and shows strong anti‐migratory effects Robin Birus,Ehab El‐awaad,Laurens Ballentin,Faten Alchab,Dagmar Aicheleet al. FEBS Open Bio, 2022, 12 (2), pp.394-411. ⟨10.1002/2211-5463.13346⟩ Article dans une revue hal-03471998v1
Adsorption studies of benzophenone-3 onto clay minerals and organosilicates: Kinetics and modelling Saddam Charaabi,Rafik Absi,Anne-Marie Pensé-Lhéritier,Marc Le Borgne,Samar Issa Applied Clay Science, 2021, 202, pp.105937. ⟨10.1016/j.clay.2020.105937⟩ Article dans une revue hal-03088439v1
Brain safety concerns of nanomedicines: The need for a specific regulatory framework Bartlomiej Szabat-Iriaka,Marc Le Borgne Drug Discovery Today, 2021, 26 (11), pp.2502-2507. ⟨10.1016/j.drudis.2021.06.011⟩ Article dans une revue hal-03311532v1
Alliages dentaires cobalt-chrome : compatibilité entre le cadre réglementaire européen et la convention nationale ? Christine Janssen,Alina Vaicelyte,Marc Le Borgne,Brigitte Grosgogeat Biomatériaux Cliniques Dentaires, 2021, 6 (1), pp.104-107 Article dans une revue hal-03475825v1
Ninhydrins inhibit carbonic anhydrases directly binding to the metal ion Abdeslem Bouzina,Malika Berredjem,Alessio Nocentini,Silvia Bua,Zouhair Bouazizet al. European Journal of Medicinal Chemistry, 2021, 209, pp.112875. ⟨10.1016/j.ejmech.2020.112875⟩ Article dans une revue hal-02963341v1
Broad-Spectrum Anticancer Activity and Pharmacokinetic Properties of a Prenyloxy-Substituted Indeno[1,2-b]indole Derivative, Discovered as CK2 Inhibitor Ehab El-Awaad,Robin Birus,Christelle Marminon,Zouhair Bouaziz,Laurens Ballentinet al. Pharmaceuticals, 2021, 14 (6), pp.542. ⟨10.3390/ph14060542⟩ Article dans une revue hal-03311530v1
Uncompetitive nanomolar dimeric indenoindole inhibitors of the human breast cancer resistance pump ABCG2 Nathalie Guragossian,Billel Belhani,Alexis Moreno,Magda Teixeira Nunes,Lucia Gonzalez-Lobatoet al. European Journal of Medicinal Chemistry, 2021, 211, pp.113017. ⟨10.1016/j.ejmech.2020.113017⟩ Article dans une revue hal-03032952v1
Solubility enhancement of mefenamic acid by inclusion complex with β-cyclodextrin: in silico modelling, formulation, characterisation, and in vitro studies Dounia Sid,Milad Baitiche,Zineb Elbahri,Ferhat Djerboua,Mokhtar Boutahalaet al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2021, 36 (1), pp.605-617. ⟨10.1080/14756366.2020.1869225⟩ Article dans une revue hal-03161350v1
Mechanistic basis of breast cancer resistance protein inhibition by new indeno[1,2-b]indoles Diogo Henrique Kita,Nathalie Guragossian,Ingrid Fatima Zattoni,Vivian Rotuno Moure,Fabiane Gomes de Moraes Regoet al. Scientific Reports, 2021, 11 (1), pp.1788. ⟨10.1038/s41598-020-79892-w⟩ Article dans une revue hal-03126318v1
Microwave-accelerated multicomponent synthesis and X-ray characterization of novel benzothiadiazinone dioxide derivatives, analogues of Monastrol Abdeslem Bouzina,Malika Berredjem,Billel Belhani,Sofiane Bouacida,Christelle Marminonet al. Research on Chemical Intermediates, 2021, ⟨10.1007/s11164-020-04378-3⟩ Article dans une revue hal-03112770v1
Improved Surface Display of Human Hyal1 and Identification of Testosterone Propionate and Chicoric Acid as New Inhibitors Isabelle Lengers,Fabian Herrmann,Marc Le Borgne,Joachim Jose Pharmaceuticals, 2020, 13 (4), pp.54. ⟨10.3390/ph13040054⟩ Article dans une revue hal-02539544v1
QSAR Model of Indeno[1,2-b]indole Derivatives and Identification of N-isopentyl-2-methyl-4,9-dioxo-4,9-Dihydronaphtho[2,3-b]furan-3-carboxamide as a Potent CK2 Inhibitor Samer Haidar,Christelle Marminon,Dagmar Aichele,Abdelhamid Nacereddine,Wael Zeinyehet al. Molecules, 2020, 25 (1), pp.97. ⟨10.3390/molecules25010097⟩ Article dans une revue hal-02424862v1
Fragment Linking Strategies for Structure-Based Drug Design Alexandre Bancet,Claire Raingeval,Thierry Lomberget,Marc Le Borgne,Jean-François Guichouet al. Journal of Medicinal Chemistry, 2020, 63 (20), pp.11420-11435. ⟨10.1021/acs.jmedchem.0c00242⟩ Article dans une revue hal-02909120v1
Synthesis of new piperazinyl-pyrrolo[1,2- a ]quinoxaline derivatives as inhibitors of Candida albicans multidrug transporters by a Buchwald–Hartwig cross-coupling reaction Jean Guillon,Shweta Nim,Stéphane Moreau,Luisa Ronga,Solène Savrimoutouet al. RSC Advances, 2020, 10 (5), pp.2915-2931. ⟨10.1039/C9RA09348F⟩ Article dans une revue hal-02449065v1
Synthesis, Optimization, Antifungal Activity, Selectivity, and CYP51 Binding of New 2-Aryl-3-azolyl-1-indolyl-propan-2-ols Nicolas Lebouvier,Fabrice Pagniez,Young Min Na,Da Shi,Patricia Pinsonet al. Pharmaceuticals, 2020, 13 (8), ⟨10.3390/ph13080186⟩ Article dans une revue hal-03389414v1
Cobalt–Chromium Dental Alloys: Metal Exposures, Toxicological Risks, CMR Classification, and EU Regulatory Framework Alina Vaicelyte,Christine Janssen,Marc Le Borgne,Brigitte Grosgogeat Crystals, 2020, 10 (12), pp.1151. ⟨10.3390/cryst10121151⟩ Article dans une revue hal-03088443v1
Synthesis, Optimization, Antifungal Activity, Selectivity, and CYP51 Binding of New 2-Aryl-3-azolyl-1-indolyl-propan-2-ols Nicolas Lebouvier,Fabrice Pagniez,Young Min Na,Da Shi,Patricia Pinsonet al. Pharmaceuticals, 2020, 13 (8), 186 (32 p.). ⟨10.3390/ph13080186⟩ Article dans une revue hal-02913479v2
Biological exploration of a novel 1,2,4-triazole-indole hybrid molecule as antifungal agent Fabrice Pagniez,Nicolas Lebouvier,Young Min Na,Isabelle Ourliac-Garnier,Carine Picotet al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2020, 35 (1), pp.398-403. ⟨10.1080/14756366.2019.1705292⟩ Article dans une revue hal-02455791v2
A comparative adsorption study of benzophenone-3 onto synthesized lipophilic organosilicate, Laponite and montmorillonite Saddam Charaabi,Lucien Tchara,Christelle Marminon,Zouhair Bouaziz,Gérard Holtzingeret al. Applied Clay Science, 2019, 170, pp.114-124. ⟨10.1016/j.clay.2019.01.005⟩ Article dans une revue hal-02004994v1
Synthesis and biological evaluation of new dipicolylamine zinc chelators as metallo-β-lactamase inhibitors Anthony Prandina,Sylvie Radix,Marc Le Borgne,Lars Petter Jordheim,Zineb Bousfihaet al. Tetrahedron, 2019, 75 (11), pp.1525-1540. ⟨10.1016/j.tet.2019.02.004⟩ Article dans une revue hal-02054167v1
Behaviour of Tetrabenazine in Acid Medium: Reassessment and Impact on Formulation Laurent Ettouati,Zoé Senta-Loys,Sandrine Bourgeois,Bernard Fenet,Marc Le Borgneet al. Pharmaceutics, 2019, 11 (1), pp.44. ⟨10.3390/pharmaceutics11010044⟩ Article dans une revue hal-01987081v1
Carbazole scaffolds in cancer therapy: a review from 2012 to 2018 Samar Issa,Anthony Prandina,Nicolas Bedel,Pal Rongved,Saïd Youset al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2019, 34 (1), pp.1321-1346. ⟨10.1080/14756366.2019.1640692⟩ Article dans une revue hal-02190476v1
Diacritic Binding of an Indenoindole Inhibitor by CK2α Paralogs Explored by a Reliable Path to Atomic Resolution CK2α′ Structures Dirk Lindenblatt,Anna Nickelsen,Violetta M Applegate,Jennifer Hochscherf,Benedict Witulskiet al. ACS Omega, 2019, 4 (3), pp.5471-5478. ⟨10.1021/acsomega.8b03415⟩ Article dans une revue hal-02077897v1
1D NMR WaterLOGSY as an efficient method for fragment-based lead discovery Claire Raingeval,Olivier Cala,Béatrice Brion,Marc Le Borgne,Roderick Eliot Hubbardet al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2019, 34 (1), pp.1218-1225. ⟨10.1080/14756366.2019.1636235⟩ Article dans une revue hal-02188259v1
Comparison of SEC and AF4 analytical tools for size estimation of typhoid Vi polysaccharides Caroline Bayart,Elisa Jean,Marie Paillagot,Alexia Renoud,Alice Raillardet al. Analytical Methods, 2019, ⟨10.1039/C9AY00145J⟩ Article dans une revue hal-02288665v1
Synthesis and biological evaluation of zinc chelating compounds as metallo-β-lactamase inhibitors Geir Kildahl-Andersen,Christian Schnaars,Anthony Prandina,Sylvie Radix,Marc Le Borgneet al. MedChemComm, 2019, 10 (4), pp.528-537. ⟨10.1039/C8MD00578H⟩ Article dans une revue hal-02077900v1
2-Aminothiazole derivatives as selective allosteric modulators of the protein kinase CK2. Part 2: Structure–based optimization and investigation of effects specific to the allosteric mode of action Benoît Bestgen,Irina Kufareva,Weiguang Seetoh,Chris Abell,Rolf W Hartmannet al. Journal of Medicinal Chemistry, 2019, 62 (4), pp.1817-1836. ⟨10.1021/acs.jmedchem.8b01765⟩ Article dans une revue hal-02004987v1
In vitro modulation of multidrug resistance by pregnane steroids and in vivo inhibition of tumour development by 7α-OBz-11α(R)-OTHP-5β-pregnanedione in K562/R7 and H295R cell xenografts Ghina Alameh,Agnès Emptoz-Bonneton,Marc Rolland de Ravel,Eva Matera,Elisabeth Mappuset al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2019, 34 (1), pp.684-691. ⟨10.1080/14756366.2019.1575825⟩ Article dans une revue hal-02077612v1
Discovery of holoenzyme-disrupting chemicals as substrate-selective CK2 inhibitors Irina Kufareva,Benoît Bestgen,Paul Brear,Renaud Prudent,Béatrice Laudetet al. Scientific Reports, 2019, 9 (1), pp.15893. ⟨10.1038/s41598-019-52141-5⟩ Article dans une revue hal-02348673v1
2-Aminothiazole derivatives as selective allosteric modulators of the protein kinase CK2. Part 1: Identification of an allosteric binding site Benoît Bestgen,Isabelle Krimm,Irina Kufareva,Ahmed Kamal,Wei Guang Seetohet al. Journal of Medicinal Chemistry, 2019, 62 (4), pp.1803-1816. ⟨10.1021/acs.jmedchem.8b01766⟩ Article dans une revue hal-02004986v1
2-Aminothiazole Derivatives as Selective Allosteric Modulators of the Protein Kinase CK2. 2. Structure-Based Optimization and Investigation of Effects Specific to the Allosteric Mode of Action Benoît Bestgen,Irina Kufareva,Weiguang Seetoh,Chris Abell,Rolf Hartmannet al. Journal of Medicinal Chemistry, 2019, 62 (4), pp.1817-1836. ⟨10.1021/acs.jmedchem.8b01765⟩ Article dans une revue hal-02465880v1
Self-Assembled Supramolecular Nanoparticles Improve the Cytotoxic Efficacy of CK2 Inhibitor THN7 Abdelhamid Nacereddine,Andre Bollacke,Eszter Roka,Christelle Marminon,Zouhair Bouazizet al. Pharmaceuticals, 2018, 11 ((1)10), ⟨10.3390/ph11010010⟩ Article dans une revue hal-01694352v1
Enhancement of iodinin solubility by encapsulation into cyclodextrin nanoparticles Anthony Prandina,Lars Herfindal,Sylvie Radix,Pal Rongved,Stein Døskelandet al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2018, 33 (1), pp.370 - 375. ⟨10.1080/14756366.2017.1421638⟩ Article dans une revue hal-01688994v1
Synthesis and preclinical evaluation of TPA-based zinc chelators as metallo-β-lactamase inhibitors Christian Schnaars,Geir Kildahl-Andersen,Anthony Prandina,Roya Popal,Sylvie Large Radixet al. ACS Infectious Diseases, 2018, ⟨10.1021/acsinfecdis.8b00137⟩ Article dans une revue hal-01844562v1
Inhibition of Shiga toxin-converting bacteriophage development by novel antioxidant compounds Sylwia Bloch,Bożena Nejman-Faleńczyk,Karolina Pierzynowska,Ewa Piotrowska,Alicja Węgrzynet al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2018, 33 (1), pp.639 - 650. ⟨10.1080/14756366.2018.1444610⟩ Article dans une revue hal-01736468v1
Synthesis, Spectroscopic Characterization, and In Vitro Antibacterial Evaluation of Novel Functionalized Sulfamidocarbonyloxyphosphonates Abdeslem Bouzina,Khaoula Bechlem,Hajira Berredjem,Billel Belhani,Imène Bechekeret al. Molecules, 2018, 23 (7), ⟨10.3390/molecules23071682⟩ Article dans une revue hal-01839215v1
Structure-based design and profiling of novel 17β-HSD14 inhibitors Florian Braun,Nicole Bertoletti,Gabriele Möller,Jerzy Adamski,Martin Frotscheret al. European Journal of Medicinal Chemistry, 2018, 155, pp.61-76. ⟨10.1016/j.ejmech.2018.05.029⟩ Article dans une revue hal-01801297v1
Synthesis, X-ray structure, in silico calculation, and carbonic anhydrase inhibitory properties of benzylimidazole metal complexes Mehdi Bouchouit,Sofiane Bouacida,Bachir Zouchoune,Hocine Merazig,Silvia Buaet al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2018, 33 (1), pp.1150 - 1159. ⟨10.1080/14756366.2018.1481404⟩ Article dans une revue hal-01839213v1
Development of Pharmacophore Model for Indeno[1,2-b]indoles as Human Protein Kinase CK2 Inhibitors and Database Mining Samer Haidar,Zouhair Bouaziz,Christelle Marminon,Tuomo Laitinen,Antti Posoet al. Pharmaceuticals, 2017, An Updated View on an Emerging Target: Selected Papers from the 8th International Conference on Protein Kinase CK2, 10 ((1)8), ⟨10.3390/ph10010008⟩ Article dans une revue hal-01683291v1
Ebisilc® Organosilicate Particles for Innovative Galenic Formulation Saddam Charaabi,Pata-Eting Kougnassoukou Tchara,Zouhair Bouaziz,Christelle Marminon,Gérard Holtzingeret al. Annals of Pharmacology and Pharmaceutics, 2017, 2(10), pp.1103 Article dans une revue hal-01806454v1
Sequential MCR/Fisher indolization strategy for the construction of polycyclic carbazole derivatives Esma Lamera,Sofiane Bouacida,Marc Le Borgne,Zouhair Bouaziz,Abdelmalek Bouraiou Tetrahedron Letters, 2017, 58 (13), pp.1305 - 1307. ⟨10.1016/j.tetlet.2017.02.047⟩ Article dans une revue istex hal-01683348v1
Unexpected Binding Mode of a Potent Indeno[1,2-b]indole-Type Inhibitor of Protein Kinase CK2 Revealed by Complex Structures with the Catalytic Subunit CK2α and Its Paralog CK2α′ Jennifer Hochscherf,Dirk Lindenblatt,Benedict Witulski,Robin Birus,Dagmar Aicheleet al. Pharmaceuticals, 2017, 10 ((4)98), ⟨10.3390/ph10040098⟩ Article dans une revue hal-01683237v1
Editorial: An Updated View on an Emerging Target: Selected Papers from the 8th International Conference on Protein Kinase CK2 Joachim Jose,Marc Le-Borgne,Lorenzo Pinna,Mathias Montenarh Pharmaceuticals, 2017, Pharmaceuticals, 10 ((2)33), pp.33 - 33. ⟨10.3390/ph10020033⟩ Article dans une revue hal-01683242v1
Sleep Disorders and Therapeutic Management: A Survey in a French Population of Prisoners Anaïs Goudard,Laure Lalande,Camille Bertin,Marie Sautereau,Marc Le Borgneet al. Journal of Correctional Health Care, 2017, 23 (2), pp.193 - 202. ⟨10.1177/1078345817700163⟩ Article dans une revue hal-01683241v1
The combined use of analytical tools for exploring tetanus toxin and tetanus toxoid structures Caroline Bayart,Sébastien Peronin,Elisa Jean,Joseph Paladino,Philippe Talagaet al. Journal of Chromatography B - Analytical Technologies in the Biomedical and Life Sciences, 2017, 1054, pp.80 - 92. ⟨10.1016/j.jchromb.2017.04.009⟩ Article dans une revue hal-01683240v1
In Search of Small Molecule Inhibitors Targeting the Flexible CK2 Subunit Interface Benoît Bestgen,Zakia Belaid-Choucair,Thierry Lomberget,Marc Le Borgne,Odile Filholet al. Pharmaceuticals, 2017, An Updated View on an Emerging Target: Selected Papers from the 8th International Conference on Protein Kinase CK2, 10 ((1)16), ⟨10.3390/ph10010016⟩ Article dans une revue hal-01683243v1
DMAP as a new efficient catalyst for the one-pot synthesis of condensed phthalazines Esma Lamera,Sofiane Bouacida,Hocine Merazig,Aïssa Chibani,Marc Le Borgneet al. Zeitschrift fur Naturforschung B, 2017, 72 ((5)b), pp.361-368. ⟨10.1515/znb-2016-0262⟩ Article dans une revue hal-01683401v1
Screening of indeno[1,2-b]indoloquinones by MALDI-MS: a new set of potential CDC25 phosphatase inhibitors brought to light Faten Alchab,Estelle Sibille,Laurent Ettouati,Emilie Bana,Zouhair Bouazizet al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2016, 31 (sup3), pp.25-32. ⟨10.1080/14756366.2016.1201480⟩ Article dans une revue hal-01655213v1
2-Indolylmethylenebenzofuranones as first effective inhibitors of ABCC2 Elisabeta Baiceanu,Kim-Anh Nguyen,Lucia Gonzalez-Lobato,Rachad Nasr,Hélène Baubichon-Cortayet al. European Journal of Medicinal Chemistry, 2016, 122, pp.408 - 418. ⟨10.1016/j.ejmech.2016.06.039⟩ Article dans une revue istex hal-01683292v1
Toward selective CK2alpha and CK2alpha’ inhibitors: Development of a novel whole-cell kinase assay by Autodisplay of catalytic CK2alpha’ Andre Bollacke,Christian Nienberg,Marc Le Borgne,Joachim Jose Journal of Pharmaceutical and Biomedical Analysis, 2016, 121, pp.253 - 260. ⟨10.1016/j.jpba.2016.01.011⟩ Article dans une revue istex hal-01683296v1
Candidate Molecule Selection Based on In Silico Predicted ADMET Properties of 12 Indenoindole Derivatives Nathalie Guragossian,Gustavo Jabor Gozzi,Bruno Fouillet,Marie-Paule Gustin,Raphaël Terreuxet al. Chemical Informatics, 2016, 2 ((2)6), ⟨10.21767/2470-6973.100020⟩ Article dans une revue hal-01683399v1
Functional display of heterotetrameric human protein kinase CK2 on Escherichia coli: a novel tool for drug discovery Andre Gratz,Andre Bollacke,Sara Stephan,Christian Nienberg,Marc Le Borgneet al. Microbial Cell Factories, 2015, 14 (74), ⟨10.1186/s12934-015-0263-z⟩ Article dans une revue hal-01683300v1
Converting potent indeno[1,2-b]indole inhibitors of protein kinase CK2 into selective inhibitors of the breast cancer resistance protein ABCG2 Gustavo Jabor Gozzi,Zouhair Bouaziz,Evelyn Winter,Nathalia Daflon-Yunes,Dagmar Aicheleet al. Journal of Medicinal Chemistry, 2015, 58 (1), pp.265-77. ⟨10.1021/jm500943z⟩ Article dans une revue hal-01174925v1
Synthesis of New Steroidal Inhibitors of P-Glycoprotein-Mediated Multidrug Resistance and Biological Evaluation on K562/R7 Erythroleukemia Cells Marc Rolland de Ravel,Ghina Alameh,Maxime Melikian,Zahia Mahiout,Agnès Emptoz-Bonnetonet al. Journal of Medicinal Chemistry, 2015, 58 (4), pp.1832 - 1845. ⟨10.1021/jm501676v⟩ Article dans une revue hal-01683301v1
Microwave-assisted oxidation of indan-1-ones into ninhydrins Christelle Marminon,Abdelhamid Nacereddine,Zouhair Bouaziz,Pascal Nebois,Joachim Joseet al. Tetrahedron Letters, 2015, 56 (14), pp.1840 - 1842. ⟨10.1016/j.tetlet.2015.02.086⟩ Article dans une revue istex hal-01683347v1
Biomimetic synthesis of Tramadol Florine Lecerf-Schmidt,Romain Haudecoeur,Basile Peres,Marc Ferreira Queiroz,Marc Marcourtet al. Chemical Communications, 2015, 51 (77), pp.14451 - 14453. ⟨10.1039/c5cc05948h⟩ Article dans une revue hal-01683298v1
Mechanisms of depolymerization and activation of a polysialic acid and its tetramer by hydrogen peroxide Christophe Neyra,Joseph Paladino,Marc Le Borgne Carbohydrate Polymers, 2015, 115, pp.494 - 501. ⟨10.1016/j.carbpol.2014.08.112⟩ Article dans une revue hal-01683316v1
Phenolic indeno[1,2-b]indoles as ABCG2-selective potent and non-toxic inhibitors stimulating basal ATPase activity. Gustavo Jabor Gozzi,Zouhair Bouaziz,Evelyn Winter,Nathalia Daflon-Yunes,Mylène Honoratet al. Drug Design, Development and Therapy, 2015, 9, pp.3481-3495. ⟨10.2147/DDDT.S84982⟩ Article dans une revue hal-01179426v1
Biologically active carbazole derivatives: focus on oxazinocarbazoles and related compounds Zouhair Bouaziz,Samar Issa,Jacques Gentili,Andre Gratz,Andre Bollackeet al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2015, 30 (2), pp.180 - 188. ⟨10.3109/14756366.2014.899594⟩ Article dans une revue hal-01683306v1
Synthesis, Biological Evaluation and Molecular Modeling of Substituted Indeno[1,2-b]indoles as Inhibitors of Human Protein Kinase CK2. Faten Alchab,Laurent Ettouati,Zouhair Bouaziz,Andre Bollacke,Jean-Guy Delcroset al. Pharmaceuticals, 2015, 8 (2), pp.279-302. ⟨10.3390/ph8020279⟩ Article dans une revue hal-01164133v1
A one-pot three-component synthesis of novel α-sulfamidophosphonates under ultrasound irradiation and catalyst-free conditions Billel Belhani,Malika Berredjem,Marc Le Borgne,Zouhair Bouaziz,Jacques Lebretonet al. RSC Advances, 2015, 5 (49), pp.39324 - 39329. ⟨10.1039/C5RA03473F⟩ Article dans une revue hal-01694993v1
Crystal structure of 13-phenyl-2,3,4,13-tetrahydro-1 H -indazolo[1,2- b ]phthalazine-1,6,11-trione Esma Lamera,Saida Benzerka,Abdelmalek Bouraiou,Sofiane Bouacida,Hocine Meraziget al. Acta crystallographica Section E : Crystallographic communications [2015-..], 2015, 71 (12), pp.o1036 - o1037. ⟨10.1107/S2056989015023452⟩ Article dans une revue hal-01683294v1
Oxidation of sialic acid using hydrogen peroxide as a new method to tune the reducing activity Christophe Neyra,Joseph Paladino,Marc Le Borgne Carbohydrate Research, 2014, 386, pp.92 - 98. ⟨10.1016/j.carres.2014.01.007⟩ Article dans une revue hal-01683314v1
Structural elucidation of two photolytic degradation products of tetrabenazine Zouaoui Bourezg,Nathalie Cartiser,Laurent Ettouati,Jean Guillon,Aline Lacoudreet al. Journal of Pharmaceutical and Biomedical Analysis, 2014, 91, pp.138 - 143. ⟨10.1016/j.jpba.2013.12.032⟩ Article dans une revue istex hal-01655151v1
Discovery of 7-Aryl-Substituted (1,5-Naphthyridin-4-yl)ureas as Aurora Kinase Inhibitors Julien Defaux,Maud Antoine,Marc Le Borgne,Tilmann Schuster,Irene Seipeltet al. ChemMedChem, 2014, 9 (1), pp.217 - 232. ⟨10.1002/cmdc.201300384⟩ Article dans une revue istex hal-01683307v1
Discovery of (7-aryl-1,5-naphthyridin-2-yl)ureas as dual inhibitors of ERK2 and Aurora B kinases with antiproliferative activity against cancer cells Julien Defaux,Maud Antoine,Cédric Logé,Marc Le Borgne,Tilmann Schusteret al. Bioorganic and Medicinal Chemistry Letters, 2014, 24 (16), pp.3748 - 3752. ⟨10.1016/j.bmcl.2014.06.078⟩ Article dans une revue hal-01683305v1
Synthesis and biological evaluation of novel substituted pyrrolo[1,2-a]quinoxaline derivatives as inhibitors of the human protein kinase CK2 Jean Guillon,Marc Le Borgne,Charlotte Rimbault,Stéphane Moreau,Solène Savrimoutouet al. European Journal of Medicinal Chemistry, 2013, 65, pp.205 - 222. ⟨10.1016/j.ejmech.2013.04.051⟩ Article dans une revue hal-01683308v1
Preparation and characterization of CK2 inhibitor-loaded cyclodextrin nanoparticles for drug delivery Florent Perret,Christelle Marminon,Wael Zeinyeh,Pascal Nebois,Andre Bollackeet al. International Journal of Pharmaceutics, 2013, 441 (1-2), pp.491 - 498. ⟨10.1016/j.ijpharm.2012.11.004⟩ Article dans une revue istex hal-01683336v1
Indenoindoles and cyclopentacarbazoles as bioactive compounds: Synthesis and biological applications Pal Rongved,Gilbert Kirsch,Zouhair Bouaziz,Joachim Jose,Marc Le Borgne European Journal of Medicinal Chemistry, 2013, 69, pp.465 - 479. ⟨10.1016/j.ejmech.2013.08.049⟩ Article dans une revue istex hal-01524692v1
Occurrence of the Synthetic Analgesic Tramadol in an African Medicinal Plant. Ahcène Boumendjel,Germain Sotoing Taïwe,Elisabeth Ngo Bum,Tanguy Chabrol,Chantal Beneyet al. Angewandte Chemie International Edition, 2013, 52 (45), pp.11780-4. ⟨10.1002/anie.201305697⟩ Article dans une revue istex inserm-00874145v1
A safe and practical method for the preparation of 7α-thioether and thioester derivatives of spironolactone Géraldine Agusti,Sandrine Bourgeois,Nathalie Cartiser,Hatem Fessi,Marc Le Borgneet al. Steroids, 2013, 78 (1), pp.102 - 107. ⟨10.1016/j.steroids.2012.09.005⟩ Article dans une revue hal-01683309v1
African tree gets to the root of pain Ahcène Boumendjel,Germain Sotoing Taïwe,Elisabeth Ngo Gum,Tanguy Chabrol,Chantal Beneyet al. Nature, 2013, 501 (7467), pp.285 - 285. ⟨10.1038/501285b⟩ Article dans une revue hal-01683403v1
1H and 13C NMR assignments of bioactive indeno[1,2-b]indole-10-one derivatives Faten Alchab,Bernard Fenet,Marc Le Borgne,Joachim Jose,Noël Pinaudet al. Magnetic Resonance in Chemistry, 2013, 51 (12), pp.837 - 841. ⟨10.1002/mrc.4016⟩ Article dans une revue istex hal-01655126v1
Novel indeno[1,2-b]indoloquinones as inhibitors of the human protein kinase CK2 with antiproliferative activity towards a broad panel of cancer cell lines Claas Hundsdörfer,Hans-Jörg Hemmerling,Janina Hamberger,Marc Le Borgne,Patrick Bednarskiet al. Biochemical and Biophysical Research Communications, 2012, 424 (1), pp.71 - 75. ⟨10.1016/j.bbrc.2012.06.068⟩ Article dans une revue istex hal-01683311v1
Indeno[1,2-b]indole derivatives as a novel class of potent human protein kinase CK2 inhibitors Claas Hundsdörfer,Hans-Jörg Hemmerling,Claudia Götz,Frank Totzke,Patrick Bednarskiet al. Bioorganic and Medicinal Chemistry, 2012, 20 (7), pp.2282 - 2289. ⟨10.1016/j.bmc.2012.02.017⟩ Article dans une revue istex hal-01683312v1
Design, Synthesis, and in vitro Antifungal Activity of 1-[(4-Substituted-benzyl)methylamino]-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ols Rémi Guillon,Fabrice Pagniez,Francis Giraud,Damien Crépin,Carine Picotet al. ChemMedChem, 2011, 6 (5), pp.816 - 825. ⟨10.1002/cmdc.201000530⟩ Article dans une revue istex hal-01689176v1
Design, synthesis and evaluation of 3-(imidazol- 1-ylmethyl)indoles as antileishmanial agents. Part II Francis Giraud,Cédric Logé,Fabrice Pagniez,Damien Crépin,Sophie Barreset al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2009, 24 (5), pp.1067 - 1075. ⟨10.1080/14756360802610795⟩ Article dans une revue hal-01689191v1
Synthesis and structure–activity relationships of 2-phenyl-1-[(pyridinyl- and piperidinylmethyl)amino]-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as antifungal agents Francis Giraud,Rémi Guillon,Cédric Logé,Fabrice Pagniez,Carine Picotet al. Bioorganic and Medicinal Chemistry Letters, 2009, 19 (2), pp.301 - 304. ⟨10.1016/j.bmcl.2008.11.101⟩ Article dans une revue istex hal-01689192v1
Design of new antifungal agents: synthesis and evaluation of 1-[(1H-indol-5-ylmethyl)amino]-2-phenyl-3-(1H-1,2,4-triazol-1-yl)propan-2-ols Rémi Guillon,Francis Giraud,Cédric Logé,Marc Le Borgne,Carine Picotet al. Bioorganic and Medicinal Chemistry Letters, 2009, 19 (20), pp.5833 - 5836. ⟨10.1016/j.bmcl.2009.08.089⟩ Article dans une revue istex hal-01689189v1
Design, synthesis, and evaluation of 1-(N-benzylamino)-2-phenyl-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as antifungal agents Francis Giraud,Cédric Logé,Fabrice Pagniez,Damien Crépin,Patrice Le Papeet al. Bioorganic and Medicinal Chemistry Letters, 2008, 18 (6), pp.1820 - 1824. ⟨10.1016/j.bmcl.2008.02.027⟩ Article dans une revue istex hal-01689196v1
Synthesis of 6- or 4-functionalized indoles via a reductive cyclization approach and evaluation as aromatase inhibitors Marie-Pierre Lézé,Anja Palusczak,Rolf W Hartmann,Marc Le Borgne Bioorganic and Medicinal Chemistry Letters, 2008, 18 (16), pp.4713 - 4715. ⟨10.1016/j.bmcl.2008.06.094⟩ Article dans une revue istex hal-01689195v1
Synthesis and biological evaluation of 3-(azolylmethyl)-1 H -indoles and 3-(α-azolylbenzyl)-1 H -indoles as selective aromatase inhibitors Marc Le Borgne,Pascal Marchand,Marie-Renée Nourrisson,Denis Loquet,Martina Palzeret al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2007, 22 (5), pp.667 - 676. ⟨10.1080/14756360701652658⟩ Article dans une revue hal-01689199v1
Synthesis and antifungal activities of new fluconazole analogues with azaheterocycle moiety Nicolas Lebouvier,Fabrice Pagniez,Muriel Duflos,Patrice Le Pape,Young Min Naet al. Bioorganic and Medicinal Chemistry Letters, 2007, 17 (13), pp.3686 - 3689. ⟨10.1016/j.bmcl.2007.04.038⟩ Article dans une revue istex hal-01689197v1
A 3D-QSAR CoMSIA study on 3-azolylmethylindoles as anti-leishmanial agents Francis Giraud,Cédric Logé,Marc Le Borgne,Fabrice Pagniez,Young Min Naet al. SAR and QSAR in Environmental Research, 2006, 17 (3), pp.299 - 309. ⟨10.1080/10659360600787494⟩ Article dans une revue hal-01689291v1
Efficient microwave-assisted synthesis of 1-(1H-indol-1-yl)-2-phenyl-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as antifungal agents Nicolas Lebouvier,Francis Giraud,Typhanie Corbin,Young Min Na,Guillaume Le Bautet al. Tetrahedron Letters, 2006, 47 (36), pp.6479 - 6483. ⟨10.1016/j.tetlet.2006.03.199⟩ Article dans une revue istex hal-01689208v1
Synthesis and biological evaluation of 5-[(aryl)(1H-imidazol-1-yl)methyl]-1H-indoles: Potent and selective aromatase inhibitors Marie-Pierre Lézé,Marc Le Borgne,Patricia Pinson,Anja Palusczak,Muriel Dufloset al. Bioorganic and Medicinal Chemistry Letters, 2006, 16 (5), pp.1134 - 1137. ⟨10.1016/j.bmcl.2005.11.099⟩ Article dans une revue istex hal-01689230v1
Antileishmanial activities and mechanisms of action of indole-based azoles Fabrice Pagniez,Hiam Abdala-Valencia,Pascal Marchand,Marc Le Borgne,Guillaume Le Bautet al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2006, 21 (3), pp.277 - 283. ⟨10.1080/14756360600700517⟩ Article dans une revue hal-01689215v1
Three-dimensional model of cytochrome P450 human aromatase Cédric Logé,Marc Le Borgne,Pascal Marchand,Jean-Michel Robert,Guillaume Le Bautet al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2005, 20 (6), pp.581 - 585. ⟨10.1080/14756360500220574⟩ Article dans une revue hal-01689233v1
2- and 3-[(Aryl)(azolyl)methyl]indoles as Potential Non-steroidal Aromatase Inhibitors Marie-Pierre Lézé,Marc Le Borgne,Pascal Marchand,Denis Loquet,Manuela Kogleret al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2004, 19 (6), pp.549 - 557. ⟨10.1080/14756360400004631⟩ Article dans une revue hal-01689238v1
Synthesis and Antileishmanial Activity of 3-Imidazolylalkylindoles. Part I Young Min Na,Nicolas Lebouvier,Marc Le Borgne,Fabrice Pagniez,Nidia Alvarezet al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2004, 19 (6), pp.451 - 457. ⟨10.1080/14756360412331280509⟩ Article dans une revue hal-01689240v1
Synthesis and antifungal activity of new 1-halogenobenzyl-3-imidazolylmethylindole derivatives Young Min Na,Marc Le Borgne,Fabrice Pagniez,Guillaume Le Baut,Patrice Le Pape European Journal of Medicinal Chemistry, 2003, 38 (1), pp.75 - 87. ⟨10.1016/S0223-5234(02)00005-3⟩ Article dans une revue istex hal-01689264v1
Retinoic Acid Metabolism Inhibition by 3-Azolylmethyl-1 H -indoles and 2, 3 or 5-(α-Azolylbenzyl)-1 H -indoles Marc Le Borgne,Pascal Marchand,Guillaume Le Baut,Masoud Ahmadi,H. John Smithet al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2003, 18 (2), pp.155 - 158. ⟨10.1080/1475636032000069819⟩ Article dans une revue hal-01689267v1
Preparation and pharmacological profile of 7-(α-Azolylbenzyl)-1H-indoles and indolines as new aromatase inhibitors Pascal Marchand,Marc Le Borgne,Martina Palzer,Guillaume Le Baut,Rolf W Hartmann Bioorganic and Medicinal Chemistry Letters, 2003, 13 (9), pp.1553 - 1555. ⟨10.1016/S0960-894X(03)00182-3⟩ Article dans une revue istex hal-01689266v1
Synthesis and Antileishmanial Activity of 3-(α-Azolylbenzyl)indoles Pascal Marchand,Marc Le Borgne,Young Min Na,Fabrice Pagniez,Hiam Abdalaet al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2002, 17 (6), pp.353 - 358. ⟨10.1080/1475636021000005613⟩ Article dans une revue hal-01689261v1
In Vitro Activity of a New Antifungal Azolyl-substituted Indole Against Aspergillus fumigatus Fabrice Pagniez,Marc Le Borgne,Pascal Marchand,Young Min Na,Guillaume Le Bautet al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2002, 17 (6), pp.425 - 429. ⟨10.1080/1475636021000005686⟩ Article dans une revue hal-01689259v1
Potential application of plant lipid transfer proteins for drug delivery Christine Pato,Marc Le Borgne,Guillaume Le Baut,Patrice Le Pape,Didier Marionet al. Biochemical Pharmacology, 2001, 62 (5), pp.555 - 560. ⟨10.1016/S0006-2952(01)00708-0⟩ Article dans une revue istex hal-01689248v1
Dérivés indoliques à activités anti-inflammatoire ou antitumorale Marc Le Borgne,Muriel Duflos,Guillaume Le Baut,Paul J Nicholls Annales Pharmaceutiques Françaises, 2000, 58 (5), pp.316 - 320 Article dans une revue hal-01689246v1
New selective nonsteroidal aromatase inhibitors: Synthesis and inhibitory activity of 2,3 or 5-(α-azolylbenzyl)-1H-indoles Marc Le Borgne,Pascal Marchand,Bénédicte Delevoye-Seiller,Jean-Michel Robert,Guillaume Le Bautet al. Bioorganic and Medicinal Chemistry Letters, 1999, 9 (3), pp.333 - 336. ⟨10.1016/S0960-894X(98)00737-9⟩ Article dans une revue istex hal-01689251v1
3-(Azolylmethyl)-1H-indoles as Selective P450 Aromatase Inhibitors Pascal Marchand,Marc Le Borgne,Muriel Duflos,Sylvie Piessard-Robert,Guillaume Le Bautet al. Pharmacy and Pharmacology Communications, 1998, 4 (4), pp.211 - 218. ⟨10.1111/j.2042-7158.1998.tb00337.x⟩ Article dans une revue istex hal-01689256v1
Comparison of the In-vitro Aromatase Inhibitory Activity of 3-(Azolylmethyl)-1H-indoles Marc Le Borgne,Pascal Marchand,Muriel Duflos,Sylvie Piessard-Robert,Guillaume Le Bautet al. Pharmacy and Pharmacology Communications, 1997, 3 (5-6), pp.279 - 281. ⟨10.1111/j.2042-7158.1997.tb00264.x⟩ Article dans une revue istex hal-01689254v1
Synthesis andIn Vitro Evaluation of 3-(1-Azolylmethyl)-1H-indoles and 3-(1-Azolyl-1-phenylmethyl)-1H-indoles as Inhibitors of P450 arom Marc Le Borgne,Pascal Marchand,Muriel Duflos,Bénédicte Delevoye-Seiller,Sylvie Piessard-Robertet al. Archiv der Pharmazie / Chemistry in Life Sciences, 1997, 330 (5), pp.141 - 145. ⟨10.1002/ardp.19973300506⟩ Article dans une revue istex hal-01689244v1

Communication dans un congrès (12)

The Journey Towards Solubility Assessment of Small Molecules Using HPLC-DAD Nada Hemmani,Anaïs Cacilie Martin,Andy Larivière,Mathis Tresallet,Kensa Tchanget al. 8th International Electronic Conference on Medicinal Chemistry, Nov 2022, Bâle, Switzerland. ⟨10.3390/ECMC2022-13143⟩ Communication dans un congrès hal-03840347v2
Triazole-indole hybrid molecules as antifungal agents: Design, synthesis and biological activity, and beyond Nicolas Lebouvier,Fabrice Pagniez,Young Min Na,Angélique Mularoni,Marie Brossieret al. 7th International Electronic Conference on Medicinal Chemistry, Nov 2021, Sciforum.net, France. pp.11577, ⟨10.3390/ECMC2021-11577⟩ Communication dans un congrès hal-03556313v1
Biological evaluation of 4,5,7-trisubstituted Indeno[1,2-b]indoles reveals a potent inhibitor of protein kinase CK2 in tumor cells with diverse anti-cancer effects and preferential cytoplasmic localization Robin Birus,Ehab El-Awaad,Laurens Ballentin,Faten Alchab,Dagmar Aicheleet al. 7th International Electronic Conference on Medicinal Chemistry, Nov 2021, Basel, Switzerland. pp.11450, ⟨10.3390/ECMC2021-11450⟩ Communication dans un congrès hal-03552581v1
Development of water-soluble ternary system for enhancing biological activities of mefenamic acid Dounia Sid,Milad Baitiche,Zineb Elbahri,Ferhat Djerboua,Mokhtar Boutahalaet al. 6th International Electronic Conference on Medicinal Chemistry, Nov 2020, Basel, Switzerland. pp.7461, ⟨10.3390/ECMC2020-07461⟩ Communication dans un congrès hal-03566171v1
Indeno[1,2-<em>b</em>]indole scaffold in drug discovery: An effective template in kinase inhibitor medicinal chemistry Robin Birus,Christelle Marminon,Dagmar Aichele,Samer Haidar,Marine Oussetet al. 6th International Electronic Conference on Medicinal Chemistry, Nov 2020, Basel, Switzerland. pp.7433, ⟨10.3390/ECMC2020-07433⟩ Communication dans un congrès hal-03566434v1
Isoform specific inhibition of human protein kinase CK2α and CK2α’ by an indenoindole derivative Anna Nickelsen,Dirk Lindenblatt,Violetta Applegate,Jennifer Hochscherf,Benedict Witulskiet al. 6th International Electronic Conference on Medicinal Chemistry, Nov 2020, Bâle, Switzerland. pp.7505, ⟨10.3390/ECMC2020-07505⟩ Communication dans un congrès hal-03566145v1
Investigation of pharmacokinetic properties of CK2 Inhibitors with an Indeno[1,2-b]indole scaffold Robin Birus,Marc Le Borgne,Joachim Jose 5th International Electronic Conference on Medicinal Chemistry, Nov 2019, Basel, Switzerland Communication dans un congrès hal-02480385v1
Design, Synthesis, X-ray Structure and Evaluation of Functionalized Hexacyclic Carbazoles as New Inhibitors of ABCG2 Transporter Isadora da Silva Zanzarini,Esma Lamera,Sofiane Bouacida,Ingrid Fatima Zattoni,Diogo Henrique Kitaet al. 5th International Electronic Conference on Medicinal Chemistry, Nov 2019, Basel, Switzerland Communication dans un congrès hal-02480387v1
25th Conference of GP2A Joachim Jose,Marc Le Borgne,Karsten Niefind 25th Conference of GP2A, Aug 2017, Liverpool, United Kingdom. pp.9-10/2.12, ⟨10.3390/ph10040097⟩ Communication dans un congrès hal-01683410v1
Indeno[1,2-b]indole Inhibitors of Human Protein Kinase CK2 and Their Impact on Different Tumor Cell Lines (A021) Dagmar Aichele,Marc Le Borgne,Joachim Jose Second International Electronic Conference on Medicinal Chemistry (ECMC-2), Nov 2016, Bâle, Switzerland. pp.15/A021, ⟨10.3390/ph10010020⟩ Communication dans un congrès hal-01683452v1
Development of Pharmacophore Model for Indeno[1,2-b]indoles as Human Protein Kinase CK2 Inhibitors and Database Mining Samer Haidar,Zouhair Bouaziz,Christelle Marminon,Tiomo Laitinen,Anti Posoet al. 3rd International Electronic Conference on Medicinal Chemistry, Nov 2017, Basel, Switzerland Communication dans un congrès hal-02480388v1
Advances in peptidomimetics as inhibitors of ABC transporters Laurent Ettouati,Marie-Emmanuelle Million,Ophélie Arnaud,Géraldine Agusti,Waël Zeinyehet al. 1st International Electronic Conference on Medicinal Chemistry, Nov 2015, sciforum.net, France. ⟨10.3390/ecmc-1-A043⟩ Communication dans un congrès hal-01710182v1

Ouvrages (1)

An Updated View on an Emerging Target: Selected Papers from the 8 th International Conference on Protein Kinase CK2 Joachim Jose,Marc Le Borgne,Lorenzo A Pinna,Mathias Montenarh MDPI AG, 2017, 978-3-03842-413-0 Ouvrages hal-01700408v1