Pascal VERDIE

Identifiants chercheurs

IdHAL :

pascal-verdie

ORCID :

0000-0002-5807-0293

IdRef :

087809729

Publications

Article dans une revue (49)

Development of Low-Nanomolar Covalent Epoxide Inhibitors of Tubulin Detyrosinating Enzymes VASH1&2 Anthony Feral,Guillaume Marcellin,Yoann Lannay,Camille Hennebert,Yazid Soufet al. Journal of Medicinal Chemistry, 2025, 68 (17), pp.18335-18355. ⟨10.1021/acs.jmedchem.5c00980⟩ Article dans une revue hal-05328434v1
Study of the impact of histidine configuration and position on analytical separation of tripeptides Ella Tyson,Elodie Carretero,Pascal Verdié,Christine Enjalbal,Yoann Ladner Journal of Chromatography A, 2025, 1759, pp.466202. ⟨10.1016/j.chroma.2025.466202⟩ Article dans une revue hal-05184470v1
Targeting a lineage-specific PI3Kɣ–Akt signaling module in acute myeloid leukemia using a heterobifunctional degrader molecule Lois Kelly,Justine Rutter,Kevin Lin,Frank Ling,Matthieu Duchmannet al. Nature Cancer, In press, Online ahead of print. ⟨10.1038/s43018-024-00782-5⟩ Article dans une revue hal-04598240v1
The C-terminal pentapeptide acein analogue (JMV3315) stimulates dopamine release in the brain Charlène Lucas-Valmalle,Gilles Subra,Pascal Verdié,Marie-Lou Kemel,Valérie Daugéet al. Australian Journal of Chemistry, 2023, 76 (8), pp.448-454. ⟨10.1071/CH22232⟩ Article dans une revue hal-04604961v1
Amelogenin-Derived Peptide (ADP-5) Hydrogel for Periodontal Regeneration: An In Vitro Study on Periodontal Cells Cytocompatibility, Remineralization and Inflammatory Profile Nina Attik,Xavier Garric,Audrey Bethry,Gilles Subra,Charlène Chevalieret al. Journal of Functional Biomaterials, 2023, 14 (2), pp.53. ⟨10.3390/jfb14020053⟩ Article dans une revue hal-04628797v1
Fast and Cost‐Efficient 17 O‐Isotopic Labeling of Carboxylic Groups in Biomolecules: From Free Amino Acids to Peptide Chains Jessica Špačková,Ieva Goldberga,Rishit Yadav,Guillaume Cazals,Aurélien Lebrunet al. Chemistry - A European Journal, 2023, 29 (10), pp.e202203014. ⟨10.1002/chem.202203014⟩ Article dans une revue hal-04002744v1
Structural insights into recognition of chemokine receptors by Staphylococcus aureus leukotoxins Paul Lambey,Omolade Otun,Xiaojing Cong,François Hoh,Luc Brunelet al. eLife, 2022, 11, pp.e72555. ⟨10.7554/eLife.72555⟩ Article dans une revue hal-03754372v1
Peptide-guided self-assembly of polyethylene glycol-b-poly(ε-caprolactone-g-peptide) block copolymers Ayman El Jundi,Matthias Mayor,Enrique Folgado,Chaimaa Gomri,Belkacem Tarek Benkhaledet al. European Polymer Journal, 2022, 176, pp.111386. ⟨10.1016/j.eurpolymj.2022.111386⟩ Article dans une revue hal-04065895v1
Active Targeted Nanoemulsions for Repurposing of Tegaserod in Alzheimer’s Disease Treatment Line Séguy,Léna Guyon,Manon Maurel,Pascal Verdié,Audrey Daviset al. Pharmaceutics, 2021, 13 (10), pp.1626. ⟨10.3390/pharmaceutics13101626⟩ Article dans une revue hal-04570312v1
Potent Lys Patch-containing Stapled Peptides Targeting PCSK9 Kevin Bourbiaux,Baptiste Legrand,Pascal Verdié,Sergio Mallart,Géraldine Manetteet al. Journal of Medicinal Chemistry, 2021, 64 (15), pp.10834-10848. ⟨10.1021/acs.jmedchem.0c02051⟩ Article dans une revue hal-03371411v1
JMV5656, a short synthetic derivative of TLQP-21, alleviates acid-induced lung injury and fibrosis in mice Vanessa Zambelli,Laura Rizzi,Paolo Delvecchio,Elena Bresciani,Laura Molteniet al. Pulmonary Pharmacology and Therapeutics, 2020, 62, pp.101916. ⟨10.1016/j.pupt.2020.101916⟩ Article dans une revue hal-04549706v1
Star-poly(lactide)-peptide hybrid networks as bioactive materials L.V. Arsenie,Coline Pinese,Audrey Bethry,L. Valot,P. Verdieet al. European Polymer Journal, 2020, 139, pp.109990 -. ⟨10.1016/j.eurpolymj.2020.109990⟩ Article dans une revue hal-03491991v1
A Short SOX9 Peptide Mimics SOX9 Tumor Suppressor Activity and Is Sufficient to Inhibit Colon Cancer Cell Growth Philippe Blache,Lucile Canterel-Thouennon,Muriel Busson,Pascal Verdié,Gilles Subraet al. Molecular Cancer Therapeutics, 2019, 18 (8), pp.1386-1395. ⟨10.1158/1535-7163.MCT-18-1149⟩ Article dans une revue hal-04830489v1
Site-specific grafting on titanium surfaces with hybrid temporin antibacterial peptides Nicolas Masurier,Jean-Baptiste Tissot,Douae Boukhriss,Said Jebors,Coline Pineseet al. Journal of materials chemistry‎ B, 2018, 6 (12), pp.1782 - 1790. ⟨10.1039/c8tb00051d⟩ Article dans une revue hal-01742222v1
STIM Proteins and Orai Ca2+ Channels Are Involved in the Intracellular Pathways Activated by TLQP-21 in RAW264.7 Macrophages Laura Molteni,Laura Rizzi,Elena Bresciani,Ramona Meanti,Jean-Alain Fehrentzet al. Frontiers in Pharmacology, 2018, 9, ⟨10.3389/fphar.2018.01386⟩ Article dans une revue hal-02871099v1
Study of the Tissue Distribution of TLQP-21 in Mice Using [18F]JMV5763, a Radiolabeled Analog Prepared via [18F]Aluminum Fluoride Chelation Chemistry Elia Turolla,Silvia Valtorta,Elena Bresciani,Jean-Alain Fehrentz,Liliana Giulianoet al. Frontiers in Pharmacology, 2018, 9, ⟨10.3389/fphar.2018.01274⟩ Article dans une revue hal-02871096v1
JMV5656, A Novel Derivative of TLQP-21, Triggers the Activation of a Calcium-Dependent Potassium Outward Current in Microglial Cells Ilaria Rivolta,Anna Binda,Laura Molteni,Laura Rizzi,Elena Brescianiet al. Frontiers in Cellular Neuroscience, 2017, 11, pp.41. ⟨10.3389/fncel.2017.00041⟩ Article dans une revue hal-02871317v1
Systemic Delivery of Tumor-Targeted Bax-Derived Membrane-Active Peptides for the Treatment of Melanoma Tumors in a Humanized SCID Mouse Model Anastassia Karageorgis,Michaël Claron,Romain Jugé,Caroline Aspord,Fabien Thoreauet al. Molecular Therapy, 2017, 25 (2), pp.534-546. ⟨10.1016/j.ymthe.2016.11.002⟩ Article dans une revue hal-02000186v1
Bioactive peptides grafted silicone dressings: A simple and specific method Coline Pinese,Said Jebors,Pierre-Emmanuel Stoebner,Vincent Humblot,Pascal Verdiéet al. Materials Today Chemistry, 2017, 4, pp.73-83. ⟨10.1016/j.mtchem.2017.02.007⟩ Article dans une revue hal-01496701v1
Peptide synthesis: ball-milling, in solution, or on solid support, what is the best strategy? Ophélie Maurin,Pascal Verdié,Gilles Subra,Frédéric Lamaty,Jean Martinezet al. Beilstein Journal of Organic Chemistry, 2017, 13, pp.2087-2093. ⟨10.3762/bjoc.13.206⟩ Article dans une revue hal-02336152v1
Sol-gel synthesis of collagen-inspired peptide hydrogel Cécile Echalier,Said Jebors,Guillaume Laconde,Luc Brunel,Pascal Verdiéet al. Materials Today, 2017, 20 (2), pp.59-66. ⟨10.1016/j.mattod.2017.02.001⟩ Article dans une revue hal-01516237v1
[Erratum for] &quot;Palatability Can Drive Feeding Independent of AgRP Neurons Raphael Georges Denis,Aurélie Joly-Amado,Emily Webber,Fanny Langlet,Marie Schaefferet al. Cell Metabolism, 2017, 25 (4), pp.975. ⟨10.1016/j.cmet.2017.03.001⟩ Article dans une revue hal-02067393v1
Pharmacological and Biochemical Characterization of TLQP-21 Activation of a Binding Site on CHO Cells Laura Molteni,Laura Rizzi,Elena Bresciani,Roberta Possenti,Pamela Petrocchi Passeriet al. Frontiers in Pharmacology, 2017, 8, pp.167. ⟨10.3389/fphar.2017.00167⟩ Article dans une revue hal-02871330v1
A switchable stapled peptide Aleksandra Kalistratova,Baptiste Legrand,Pascal Verdié,Emilia Naydenova,Muriel Amblardet al. Journal of Peptide Science, 2016, 22 (3), pp.143-148. ⟨10.1002/psc.2851⟩ Article dans une revue istex hal-03564342v1
Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling Céline M'Kadmi,Jean-Philippe Leyris,Lauriane Onfroy,Céline Galés,Aude Saulièreet al. Journal of Biological Chemistry, 2015, 290 (45), pp.27021-27039. ⟨10.1074/jbc.M115.659250⟩ Article dans une revue hal-03564155v1
Solid-Supported Synthesis and 5-HT 7 /5-HT 1A Receptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1 H )-one Katarzyna Grychowska,Nicolas Masurier,Pascal Verdié,Grzegorz Satała,Andrzej Bojarskiet al. Chemical Biology and Drug Design, 2015, 86 (4), pp.697-703. ⟨10.1111/cbdd.12539⟩ Article dans une revue istex hal-03564059v1
Palatability Can Drive Feeding Independent of AgRP Neurons Raphael Georges Denis,Aurélie Joly-Amado,Emily Webber,Fanny Langlet,Marie Schaefferet al. Cell Metabolism, 2015, 22 (4), pp.646-657. ⟨10.1016/j.cmet.2015.07.011⟩ Article dans une revue hal-02067347v1
Solid-supported synthesis, molecular modeling, and biological activity of long-chain arylpiperazine derivatives with cyclic amino acid amide fragments as 5-HT7 and 5-HT1A receptor ligands Vittorio Canale,Paweł Guzik,Rafał Kurczab,Pascal Verdie,Grzegorz Satałaet al. European Journal of Medicinal Chemistry, 2014, 78, pp.10-22. ⟨10.1016/j.ejmech.2014.03.005⟩ Article dans une revue hal-03563396v1
N- and O-acetylation of threonine residues in the context of proteomics. Jean-Baptiste Boyer,Alain Dedieu,J. Armengaud,Pascal Verdié,Gilles Subraet al. Journal of Proteomics, 2014, 108, pp.369-372. ⟨10.1016/j.jprot.2014.06.005⟩ Article dans une revue istex hal-01025681v1
Supported oligomethionine sulfoxide and Ellman's reagent for cysteine bridges formation Luisa Ronga,Pascal Verdié,Pierre Sanchez,Christine Enjalbal,Amélie Maurraset al. Amino Acids, 2013, 44 (2), pp.733-742. ⟨10.1007/s00726-012-1397-5⟩ Article dans une revue istex hal-01563741v1
Biophysical characterization of a binding site for TLQP-21, a naturally occurring peptide which induces resistance to obesity V. Cassina,A. Torsello,A. Tempestini,D. Salerno,D. Brogioliet al. Biochimica et Biophysica Acta:Biomembranes, 2013, 1828 (2), pp.455-460. ⟨10.1016/j.bbamem.2012.10.023⟩ Article dans une revue hal-02871939v1
The pipecolic linker—an acid-labile handle for derivatization of secondary amines on a solid-support. Part 3 Paweł Zajdel,Nicolas Masurier,Vittorio Canale,Pascal Verdie,Muriel Amblardet al. Tetrahedron Letters, 2013, 54 (8), pp.998-1002. ⟨10.1016/j.tetlet.2012.12.036⟩ Article dans une revue istex hal-03563368v1
Heating and microwave assisted SPPS of C-terminal acid peptides on trityl resin: The truth behind the yield Cécile Echalier,Soultan Al-Halifa,Aude Kreiter,Christine Enjalbal,Pierre Sanchezet al. Amino Acids, 2013, 45 (6), pp.1395-1403. ⟨10.1007/s00726-013-1604-z⟩ Article dans une revue istex hal-01563742v1
Rapid sensing of circulating ghrelin by hypothalamic appetite-modifying neurons. Marie Schaeffer,Fanny Langlet,Chrystel Lafont,François Molino,David J Hodsonet al. Proceedings of the National Academy of Sciences of the United States of America, 2013, 110 (4), pp.1512-7. ⟨10.1073/pnas.1212137110⟩ Article dans une revue hal-00796900v1
How ligands and signalling proteins affect G-protein-coupled receptors' conformational landscape Sophie Mary,Jean-Alain Fehrentz,Marjorie Damian,Pascal Verdie,Jean Martinezet al. Biochemical Society Transactions, 2013, 41 (1), pp.144-147. ⟨10.1042/BST20120267⟩ Article dans une revue hal-02871941v1
Microwave-Mediated Reduction of Disulfide Bridges with Supported (Tris(2-carboxyethyl)phosphine) as Resin-Bound Reducing Agent Guillaume Miralles,Pascal Verdié,Karine Puget,Amélie Maurras,Jean Martinezet al. ACS Combinatorial Science, 2013, 15 (4), pp.169-173. ⟨10.1021/co300104k⟩ Article dans une revue hal-03563025v1
Ghrelin Receptor Ligands: Design and Synthesis of Pseudopeptides and Peptidomimetics. Aline Moulin,Luc Brunel,Pascal Verdié,Laurent Gavara,Jean Martinezet al. Current Chemical Biology, 2013, 3 (7), pp.000-000. ⟨10.2174/2212796807999131128125920⟩ Article dans une revue istex hal-01089074v1
Heterodimerization with Its Splice Variant Blocks the Ghrelin Receptor 1a in a Non-signaling Conformation Sophie Mary,Jean-Alain Fehrentz,Marjorie Damian,Gérald Gaibelet,Hélène Orcelet al. Journal of Biological Chemistry, 2013, 288 (34), pp.24656-24665. ⟨10.1074/jbc.M113.453423⟩ Article dans une revue hal-02871944v1
High Constitutive Activity Is an Intrinsic Feature of Ghrelin Receptor Protein. A study with a functional monomeric GHS-R1a receptor reconstitued in lipid discs Marjorie Damian,Jacky Marie,Jean-Philippe Leyris,Jean-Alain Fehrentz,Pascal Verdieet al. Journal of Biological Chemistry, 2012, 287 (6), pp.3630-3641. ⟨10.1074/jbc.M111.288324⟩ Article dans une revue hal-00713589v1
Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a Jean-Philippe Leyris,Thomas Roux,Eric Trinquet,Pascal Verdié,Jean-Alain Fehrentzet al. Analytical Biochemistry, 2011, 408, pp.253-262. ⟨10.1016/j.ab.2010.09.030⟩ Article dans une revue istex hal-00534262v1
cis-Apa: A Practical Linker for the Microwave-Assisted Preparation of Cyclic Pseudopeptides via RCM Cyclative Cleavage Alice Baron,Pascal Verdié,Jean Martinez,Frédéric Lamaty Journal of Organic Chemistry, 2011, 76 (3), pp.766-772. ⟨10.1021/jo101629v⟩ Article dans une revue hal-00564151v1
Oxyfold: A simple and efficient solid-supported reagent for disulfide bond formation P. Verdié,Luisa Ronga,M. Cristau,M. Amblard,S. Cantelet al. Chemistry - An Asian Journal, 2011, 6 (9), pp.2382-2389. ⟨10.1002/asia.201100202⟩ Article dans une revue istex hal-01563744v1
From Polyesters to Polyamides Via ON Acyl Migration: An Original Multi-Transfer Reaction Julien Tailhades,Sébastien Blanquer,Benjamin Nottelet,Jean Coudane,Gilles Subraet al. Macromolecular Rapid Communications, 2011, 32 (12), pp.876 - 880. ⟨10.1002/marc.201100235⟩ Article dans une revue istex hal-01833151v1
Sequencing Lys-N Proteolytic Peptides by ESI and MALDI Tandem Mass Spectrometry Mathieu Dupré,Sonia Cantel,Pascal Verdié,Jean Martinez,Christine Enjalbal Journal of The American Society for Mass Spectrometry, 2011, 22, pp.265-279. ⟨10.1007/s13361-010-0022-7⟩ Article dans une revue hal-00580756v1
Sulfonamides with the N-alkyl-N'-dialkylguaninidine moiety as 5-HT7 receptor ligands Pawel Zajdel,Gilles Subra,Pascal Verdié,Ewa Gabzdyl,Andrzej J. Bojarskiet al. Bioorganic and Medicinal Chemistry Letters, 2009, 19, pp.4827-4831. ⟨10.1016/j.bmcl.2009.06.038⟩ Article dans une revue hal-00411218v1
The influence of an ethylene spacer of the 5-HT1A and 5-HT2A receptor affinity of arylpiperazine derivatives of amides with N-acylated amino acids and 3-differently substituted pyrrolidine-2,5-diones Pawel Zajdel,Gilles Subra,Pascal Verdie,Andrzej J. Bojarski,Beata Duszynskaet al. European Journal of Medicinal Chemistry, 2009, 44, pp.800-808. ⟨10.1016/j.ejmech.2008.05.021⟩ Article dans une revue hal-00411106v1
Solid-Phase Synthesis of 4-methylcarboxy-1,4-benzodiazepine-2,5-diones Pascal Verdié,Gilles Subra,Marie-Christine Averlant-Petit,Muriel Amblard,Jean Martinez Journal of Combinatorial Chemistry, 2008, 10 (6), pp.869-874. ⟨10.1021/cc800085d⟩ Article dans une revue hal-00411034v1
Solid-phase synthesis of 5-arylhistidines via a microwave-assisted Suzuki-Miyaura cross-coupling Vanessa Cerezo,Muriel Amblard,Jean Martinez,Pascal Verdié,Marta Planaset al. Tetrahedron, 2008, 64, pp.10538-10545. ⟨10.1016/j.tet.2008.08.077⟩ Article dans une revue istex hal-00411015v1
Valuable Versatile Reactivity of Thiaisatoic Anhydrides: Expedient Solid-Phases Synthesis of Thieno[1,4]Diazepine-2,5-diones Yann Brouillette,Pascal Verdié,Jean Martinez SYNLETT, 2008, 15, pp.2360-2364. ⟨10.1055/s-2008-1078210⟩ Article dans une revue hal-00341629v1

Communication dans un congrès (2)

Marrying sol-gel and peptide chemistry to design bioactive materials Gilles Subra,Cécile Echalier,Ahmad Mehdi,Margaux Clavié,Mathilde Guerinet al. Turku Biomaterials Days 2024, Oct 2024, Turku, Finland Communication dans un congrès hal-04891598v1
Designing biomimetic materials from silylated amino acids, peptides and proteins. Gilles Subra,Cécile Echalier,Margaux Clavié,Pascal Verdié,Muriel Amblardet al. European Peptide Synthesis Conference 2023, Feb 2023, Leeds, United Kingdom Communication dans un congrès hal-04891483v1

Brevet (1)

COMPOUNDS FOR TREATING SEGMENTAL PROGEROID SYNDROMES Pierre Cau,Eric Dessaud,Muriel Amblard,Pascal Verdié,Gilles Subraet al. France, Patent n° : US2024010610. 2024 Brevet hal-04806443v1

Pré-publication, Document de travail (1)

Fast and cost-efficient approaches for 17O-isotopic labeling of carboxylic groups in biomolecules: from free amino acids to peptide chains Jessica Špačková,Ieva Goldberga,Rishit Yadav,Guillaume Cazals,Aurélien Lebrunet al. 2022 Pré-publication, Document de travail (preprint/prepublication) hal-03846579v1