Pierre Milbeo

Publications

Article dans une revue (12)

Asymmetric α-Fluoroalkyl-α-Amino Acids: Recent Advances in Their Synthesis and Applications Nathan Picois,Yazid Boutahri,Pierre Milbeo,Chiara Zanato,Nathalie Lensenet al. Molecules, 2024, 29 (6), pp.1408. ⟨10.3390/molecules29061408⟩ Article dans une revue (article de synthèse) hal-04516441v1
Bimodal use of chiral α‐Trifluoromethylalanine in Aib Foldamers: study of the position impact towards the helical screw‐sense preference Nathan Picois,Lizeth Bodero,Pierre T Milbeo,Thierry Brigaud,Grégory Chaume Chemistry - A European Journal, In press, 30 (27), ⟨10.1002/chem.202400540⟩ Article dans une revue hal-04516499v1
An Organocatalytic and Stereoselective Vinylogous Domino Process Towards Thiochromans Pierre Milbeo,Arthur Lebrêne,Mariia Savchuk,Giang Vo-Thanh,Sylvain Oudeyeret al. Chemistry - A European Journal, 2023, pp.e202301311. ⟨10.1002/chem.202301311⟩ Article dans une revue hal-04102949v1
Next generation Glucose-1-phosphate thymidylyltransferase (RmlA) inhibitors: An extended SAR study to direct future design Ganyuan Xiao,Magnus Alphey,Fanny Tran,Lisa Pirrie,Pierre Milbeoet al. Bioorganic and Medicinal Chemistry, 2021, 50, pp.116477. ⟨10.1016/j.bmc.2021.116477⟩ Article dans une revue hal-05087058v1
1-Aminobicyclo[2.2.2]octane-2-carboxylic acid and derivatives as chiral constrained bridged scaffolds for foldamers and chiral catalysts Pierre Milbeo,Jean Martinez,Muriel Amblard,Monique Calmès,Baptiste Legrand Accounts of Chemical Research, 2021, 54 (3), pp.685-696. ⟨10.1021/acs.accounts.0c00680⟩ Article dans une revue hal-03371473v1
Synthesis, characterisation and cytotoxic activity evaluation of new metal-salen complexes based on the 1,2-bicyclo[2.2.2]octane bridge Pierre Milbeo,François Quintin,Laure Moulat,Claude Didierjean,Jean Martinezet al. Tetrahedron Letters, 2021, 63, pp.152706. ⟨10.1016/j.tetlet.2020.152706⟩ Article dans une revue hal-03103305v1
Radical‐Mediated Acyl Thiol‐Ene Reaction for Rapid Synthesis of Biomolecular Thioester Derivatives Joshua Mclean,Pierre Milbeo,Dylan Lynch,Lauren Mcsweeney,Eoin Scanlan European Journal of Organic Chemistry, 2021, 2021 (29), pp.4148-4160. ⟨10.1002/ejoc.202100615⟩ Article dans une revue hal-05087069v1
A bicyclic unit reversal to stabilize the 12/14-helix in mixed homochiral oligoureas Pierre Milbeo,Matthieu Simon,Claude Didierjean,Emmanuel Wenger,Emmanuel Aubertet al. Chemical Communications, 2020, 56 (57), pp.7921-7924. ⟨10.1039/d0cc02902e⟩ Article dans une revue hal-03080580v1
12/10‐Helix in Mixed β‐Peptides Alternating Bicyclic and Acyclic β‐Amino Acids: Probing the Relationship between Bicyclic Side Chain and Helix Stability Matthieu Simon,Pierre Milbeo,Hongtao Liu,Christophe Andre,Emmanuel Wengeret al. Chemistry - A European Journal, 2018, 24 (70), pp.18795-18800. ⟨10.1002/chem.201804404⟩ Article dans une revue hal-02403147v1
C 1 -Symmetric 1,2-Diaminobicyclo[2.2.2]octane Ligands in Copper-Catalyzed Asymmetric Henry Reaction: Catalyst Development and DFT Studies Pierre Milbeo,Laure Moulat,Claude Didierjean,Emmanuel Aubert,Jean Martinezet al. European Journal of Organic Chemistry, 2018, 2018 (2), pp.178-187. ⟨10.1002/ejoc.201701452⟩ Article dans une revue hal-02419329v1
Synthesis of Enantiopure 1,2-Diaminobicyclo[2.2.2]octane Derivatives, C 1 -Symmetric Chiral 1,2-Diamines with a Rigid Bicyclic Backbone Pierre Milbeo,Laure Moulat,Claude Didierjean,Emmanuel Aubert,Jean Martinezet al. Journal of Organic Chemistry, 2017, 82 (6), pp.3144 - 3151. ⟨10.1021/acs.joc.7b00122⟩ Article dans une revue hal-01552321v1
N-Pyrrolidine-based alpha/beta-peptides incorporating ABOC, a constrained bicyclic beta-amino acid, for asymmetric aldol reaction catalysis Pierre Milbeo,Kelly Maurent,Laure Moulat,Aurelien Lebrun,Claude Didierjeanet al. Tetrahedron, 2016, 72 (13), pp.1706-1715. ⟨10.1016/j.tet.2016.02.027⟩ Article dans une revue hal-01532027v1

Chapitre d'ouvrage (1)

The Thiol-ene “Click” Reaction for Synthesis of Biomolecular Thioether and Thioester Derivatives Pierre Milbéo,Chiara Zanato Topics Heterocyclic Chemistry. Modern Advances in Click Chemistry: Synthesis of Compounds, Springer Berlin Heidelberg, In press, Topics in Heterocyclic Chemistry, ⟨10.1007/7081_2025_98⟩ Chapitre d'ouvrage hal-05479896v1

Thèse (1)

Synthèse de bicycles contraints originaux pour l’élaboration de nouveaux catalyseurs chiraux et de nouveaux foldamères Pierre Milbéo Chimie organique. Université Montpellier, 2017. Français. ⟨NNT : 2017MONTT209⟩ Thèse tel-03824580v1