Pierre-Olivier Delaye

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Publications

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Emerging therapeutics: The imidazo[1,2-b]pyridazine scaffold as a novel drug candidate for eumycetoma, a neglected tropical disease

Lamis Yahia Mohamed Elkheir , Pierre-Olivier Delaye , Mélanie Penichon , Kimberly Eadie , Magdi Awadalla Mohamed et al.
European Journal of Medicinal Chemistry, 2024, 277, pp.116720. ⟨10.1016/j.ejmech.2024.116720⟩
Article dans une revue hal-04995966 v1
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Mechanochemical Suzuki‐Miyaura Cross‐Coupling with Natural Deep Eutectic Solvent as Liquid‐Assisted Grinding Additive: Merging Two Fields for a Greener Strategy

Emilie Thiery , Pierre‐olivier Delaye , Jérôme Thibonnet , Leslie Boudesocque‐delaye
European Journal of Organic Chemistry, 2023, 26, ⟨10.1002/ejoc.202300727⟩
Article dans une revue hal-04969276 v1

Cassia sieberiana root bark used in traditional medicine in Togo: Anthelmintic property against Haemonchus contortus and tannins composition

Iwaba Kpabi , Thibaut Munsch , Amégninou Agban , Isabelle Théry-Koné , Joelle Dorat et al.
South African Journal of Botany, 2022, 151 (part B), pp.549-558. ⟨10.1016/j.sajb.2022.05.055⟩
Article dans une revue hal-03918718 v1
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Bioinspired imidazo[1,2-a:4,5-c’]dipyridines with dual antiproliferative and anti-migrative properties in human cancer cells: The SAR investigation

Abdulrahim Alzain , Lucie Brisson , Pierre-Olivier Delaye , Mélanie Pénichon , Stéphanie Chadet et al.
European Journal of Medicinal Chemistry, 2021, 218, pp.113258. ⟨10.1016/j.ejmech.2021.113258⟩
Article dans une revue hal-03202963 v1
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Imidazo[1,2-b]pyridazine as privileged scaffold in medicinal chemistry: An extensive review

Amanda Garrido , Gonzalo Vera , Pierre-Olivier Delaye , Cécile Enguehard-Gueiffier
European Journal of Medicinal Chemistry, 2021, 226, pp.113867. ⟨10.1016/j.ejmech.2021.113867⟩
Article dans une revue hal-04951716 v1

Direct Access to Highly Functionalised Benzimidazoles and Benzoxazoles from a Common Precursor

Amanda Garrido , Pierre-Olivier Delaye , François Quintin , Mohamed Abarbri , Pedro Lameiras et al.
Synthesis: Journal of Synthetic Organic Chemistry, 2019, 51 (21), pp.4006-4013. ⟨10.1055/s-0039-1690153⟩
Article dans une revue hal-03533721 v1
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Natural Deep Eutectic Solvents as sustainable solvent for Suzuki-Miyaura cross- coupling reactions applied to imidazo-fused heterocycles

Pierre-Olivier Delaye , Mélanie Pénichon , Leslie Boudesocque-Delaye , Cécile Enguehard-Gueiffier , Alain Gueiffier
SynOpen, 2018, 2 (04), pp.306 - 311. ⟨10.1055/s-0037-1610400⟩
Article dans une revue hal-02172280 v1
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Gold-silver catalyzed straightforward one pot synthesis of pyrano[3,4- b]pyrrol-7(1H)-ones

Pierre-Olivier Delaye , J. Petrignet , Emilie Thiery , Jérome Thibonnet
Organic & Biomolecular Chemistry, 2017, 15 (35), pp.7290-7295. ⟨10.1039/c7ob01849e⟩
Article dans une revue hal-02170750 v2
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Discovery of imidazo[1,2-a]pyridine-based anthelmintic targeting cholinergic receptors of Haemonchus Contortus

Jean-Paul Déto Ursul N'Guessan , Pierre-Olivier Delaye , Mélanie Pénichon , Claude L. Charvet , Cédric Neveu et al.
Bioorganic and Medicinal Chemistry, 2017, 25 (24), pp.6695-6706. ⟨10.1016/j.bmc.2017.11.012⟩
Article dans une revue hal-02628509 v1
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Regiocontrolled functionalization of 2,3-dihalogenoimidazo[1,2-a] pyridines by Suzuki-Miyaura and Sonogashira cross-coupling reactions

Pierre-Olivier Delaye , Mélanie Pouvreau , Hassan Allouchi , Cécile Enguehard-Gueiffier , Alain Gueiffier
Organic & Biomolecular Chemistry, 2017, 15 (19), pp.4199-4204. ⟨10.1039/c7ob00624a⟩
Article dans une revue hal-01605432 v1
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Domino 6-endo-dig Cyclization/Halogenation Reactions: Three-Component Synthesis of 1,3-Disubstituted 4-Haloimidazo[1,2-a:4,5-c′]dipyridines

Cécile Enguehard-Gueiffier , Pierre-Olivier Delaye , Mélanie Pénichon , Caroline Denevault-Sabourin , Hassan Allouchi et al.
Synthesis: Journal of Synthetic Organic Chemistry, 2015, 47 (24), pp.3983-3989. ⟨10.1055/s-0035-1560089⟩
Article dans une revue hal-02389894 v1

Cyclopropene Derivatives as Precursors to Enantioenriched Cyclopropanols and n-Butenals Possessing Quaternary Carbon Stereocenters

Marwan Simaan , Pierre-Olivier Delaye , Min Shi , Ilan Marek
Angewandte Chemie International Edition, 2015, 54 (42), pp.12345 - 12348. ⟨10.1002/anie.201412440⟩
Article dans une revue istex hal-02631404 v1

Selective Carbon-Carbon Bond Cleavage for the Stereoselective Synthesis of Acyclic Systems

Ilan Marek , Ahmad Masarwa , Pierre-Olivier Delaye , Markus Leibeling
Angewandte Chemie International Edition, 2015, 54 (2), pp.414 - 429. ⟨10.1002/anie.201405067⟩
Article dans une revue istex hal-02637631 v1

Modulable and Highly Diastereoselective Carbometalations of Cyclopropenes

Dorian Didier , Pierre-Olivier Delaye , Marwan Simaan , Biana Island , Guillaume Eppe et al.
Chemistry - A European Journal, 2014, 20 (4), pp.1038 - 1048. ⟨10.1002/chem.201303569⟩
Article dans une revue istex hal-02641468 v1

Diastereodivergent Carbometalation/Oxidation/Selective Ring Opening: Formation of All-Carbon Quaternary Stereogenic Centers in Acyclic Systems

Pierre-Olivier Delaye , Dorian Didier , Ilan Marek
Angewandte Chemie International Edition, 2013, 52 (20), pp.5333 - 5337. ⟨10.1002/anie.201300664⟩
Article dans une revue istex hal-02648492 v1

Switching Regioselectivity in the Allylation of Imines by N-Side Chain Tuning

Pierre-Olivier Delaye , Jean-Luc Vasse , Jan Szymoniak
Organic Letters, 2012, 14 (12), pp.3004 - 3007. ⟨10.1021/ol301026w⟩
Article dans une revue hal-02651225 v1

Improved Enantioselective Synthesis of ( − )-Linderol A: Hindered Rotation about Aryl−Csp 3 Bond

Pierre-Olivier Delaye , Pedro Lameiras , Nelly Kervarec , Catherine Mirand , Hatice Berber
Journal of Organic Chemistry, 2010, 75 (8), pp.2501-2509. ⟨10.1021/jo902567y⟩
Article dans une revue hal-04941424 v1