Raphaël Tripier

227
Documents

Publications

Publications

Exploring the Coordination Chemistry and Potential Applications of PC3PA-Based Lanthanide Complexes: Synthesis, Solution Structure, Luminescence, and Relaxation Properties

Loëza Collobert , Lucile Bridou , Zoltán Garda , Olivier Maury , Éva Tóth et al.
Inorganic Chemistry, 2025, 64 (18), pp.9330-9341. ⟨10.1021/acs.inorgchem.5c01318⟩
Article dans une revue hal-05096028 v1

« Optimizing Imaging and Dose–Reponse in Radiotherapies » XVIe édition de l’atelier organisé par le réseau « Vectorisation, Imagerie, Radiothérapies » du Cancéropôle Grand-Ouest – 4–7 octobre 2023, Erquy, France

Françoise Léost , Vincent Potiron , Nicolas Lepareur , Latifa Rbah-Vidal , Emmanuel Garcion et al.
Bulletin du Cancer, 2025, ⟨10.1016/j.bulcan.2025.02.001⟩
Article dans une revue hal-04982114 v1
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Zn$^{2+}$ triazamacrocyclic chelators with methylpyridine pendant arms for B-cell apoptosis: a structure–activity study

Axia Marlin , Fiona Le Pape , Thibault Troadec , Jocelyn Le Goff , Raphaël Tripier et al.
Dalton Transactions, 2025, 54 (9), pp.3939-3951. ⟨10.1039/D4DT02962C⟩
Article dans une revue hal-05097560 v1

The continued industrial use of ethylene oxide despite health risks: An interventional radiology perspective on a broader medical challenge of balancing sterility, safety, and sustainability

Julien Ognard , Marie Schmidt , Christophe Paya , Isabelle Le Du , Camille Bourillon et al.
Diagnostic and Interventional Imaging, In press, ⟨10.1016/j.diii.2025.05.002⟩
Article dans une revue hal-05096043 v1
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Synthesis and <sup>64</sup>Cu‐Radiolabeling Strategies of Small Organic Radioconjugates Based on the AMD070 Scaffold

Marie M Le Roy , Patricia Le Saëc , Michel Chérel , Alain Faivre‐chauvet , Thibault Troadec et al.
ChemMedChem, 2025, ⟨10.1002/cmdc.202500243⟩
Article dans une revue hal-05113923 v1

Cobalt complexes as modulators against amyloid-β aggregation

Jeasang Yoo , Jong-Min Suh , Gunhee Kim , Hélène Bernard , Raphaël Tripier et al.
Journal of Inorganic Biochemistry, 2025, 271, pp.112972. ⟨10.1016/j.jinorgbio.2025.112972⟩
Article dans une revue hal-05117654 v1
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Advanced 64 Cu/67 Cu-Based Theranostics: Application of the Copper Chelator TE1PA to a Murine Model of HER2-positive Gastric Cancer

Julie Pineau , Cédric Ollier , Céline Mothes , Sarah Belderbos , Nathalie Le Bris et al.
Inorganic Chemistry, 2025, ⟨10.1021/acs.inorgchem.5c01513⟩
Article dans une revue hal-05115478 v1

Exploring the Limits of Ligand Rigidification in Transition Metal Complexes with Mono- N -Functionalized Pyclen Derivatives

Gwladys Nizou , Zoltán Garda , Enikő Molnár , David Esteban-Gómez , Mariane Le Fur et al.
Inorganic Chemistry, 2024, 63 (8), pp.3931-3947. ⟨10.1021/acs.inorgchem.3c04451⟩
Article dans une revue hal-04541998 v1

Extending the Scope of the C -Functionalization of Cyclam via Copper(I)-Catalyzed Alkyne–Azide Cycloaddition to Bifunctional Chelators of Interest

Cédric Ollier , Alejandro Méndez-Ardoy , Fernando Ortega-Caballero , José Jiménez-Blanco , Nathalie Le Bris et al.
Journal of Organic Chemistry, 2024, ⟨10.1021/acs.joc.3c02854⟩
Article dans une revue hal-04545763 v1
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A versatile fluorinated azamacrocyclic chelator enabling $^{18}$F PET or $^{19}$F MRI : a first step towards new multimodal and smart contrast agents.

Charline Sire , Vincent Meneyrol , Nathalie Saffon-Merceron , Enzo Terreno , Francesca Garello et al.
Chemical Science, 2024, 15, pp.13550. ⟨10.1039/d4sc02871f⟩
Article dans une revue hal-04665317 v1
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Selective synthesis of an elusive C-functional bis-cyclam and study of its inhibition of the CXCR4 chemokine receptor

Marie M Le Roy , Sandra Claes , Nathalie Saffon-Merceron , Dominique Schols , Thibault Troadec et al.
Organic & Biomolecular Chemistry, 2024, 22, pp.3059-3067. ⟨10.1039/D3OB02050A⟩
Article dans une revue hal-04536449 v1
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Taylor dispersion analysis for measurement of diffusivity and size of gadolinium-based contrast agents

Chutintorn Somnin , Laurent Leclercq , Joseph Chamieh , Mael Le Menedeu , Christelle Medina et al.
European Journal of Pharmaceutical Sciences, 2024, 200, pp.106831. ⟨10.1016/j.ejps.2024.106831⟩
Article dans une revue hal-04739876 v1
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Relevance of Oxocyclam from Palladium(II) Coordination to Radiopharmaceutical Development

Maher Hojorat , Julie Pineau , Cathryn Driver , David Esteban-Gómez , Marie Cordier et al.
Inorganic Chemistry, 2024, 63 (25), pp.11884-11896. ⟨10.1021/acs.inorgchem.4c01780⟩
Article dans une revue hal-04613088 v1

Upconversion Luminescence with Bis‐pyclen Yb(III) Chelates: Crown vs. Linear Polyether Linkers in Discrete Heteropolynuclear Architectures

Nadège Hamon , Léna Godec , Samuel Sanchez , Maryline Beyler , Loïc Charbonnière et al.
Angewandte Chemie International Edition, 2024, 64 (2), ⟨10.1002/anie.202414608⟩
Article dans une revue hal-04928814 v1
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Trehalose-polyamine/DNA nanocomplexes: impact of vector architecture on cell and organ transfection selectivity

Fernando Ortega-Caballero , María L Santana-Armas , Conchita Tros de Ilarduya , Christophe Di Giorgio , Raphäel Tripier et al.
Journal of materials chemistry‎ B, 2024, 12 (14), pp.3445-3452. ⟨10.1039/d3tb02889e⟩
Article dans une revue hal-04542122 v1

A versatile fluorinated azamacrocyclic chelator enabling 18 F PET or 19 F MRI: a first step towards new multimodal and smart contrast agents

Charline Sire , Vincent Meneyrol , Nathalie Saffon-Merceron , Enzo Terreno , Francesca Garello et al.
Chemical Science, 2024, ⟨10.1039/D4SC02871F⟩
Article dans une revue hal-04666501 v1
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Preclinical Evaluation of a 64Cu-Based Theranostic Approach in a Murine Model of Multiple Myeloma

Cassandra Métivier , Patricia Le Saëc , Joëlle Gaschet , Catherine Chauvet , Séverine Marionneau-Lambot et al.
Pharmaceutics, 2023, 15 (7), pp.1817. ⟨10.3390/pharmaceutics15071817⟩
Article dans une revue hal-04161269 v1

Multistep synthesis of a novel copper complex with potential for Alzheimer’s disease diagnosis

Fatma Dellal , Diego Santo Domingo Porqueras , Stacy Narayanin-Richenapin , Marine Thimotee , Vanessa Delahaye et al.
European Journal of Biochemistry, 2023, 28 (8), pp.777-790. ⟨10.1007/s00775-023-02028-8⟩
Article dans une revue hal-04543773 v1

Quid de notre empreinte iodée?

Dorra Guermazi , Raphel Jomaah , Raphaël Tripier , Jean-Alix Barrat , Julien Ognard et al.
Journal de Neuroradiologie / Journal of Neuroradiology, 2023, 50 (2), pp.139-140. ⟨10.1016/j.neurad.2023.01.057⟩
Article dans une revue hal-04545836 v1

H 3 nota Derivatives Possessing Picolyl and Picolinate Pendants for Ga 3+ Coordination and 67 Ga 3+ Radiolabeling

Axia Marlin , Angus Koller , Enikö Madarasi , Marie Cordier , David Esteban-Gómez et al.
Inorganic Chemistry, 2023, 62 (50), pp.20634-20645. ⟨10.1021/acs.inorgchem.3c01417⟩
Article dans une revue hal-04545822 v1

Iodinated disinfection byproducts: A silent threat, why should we care?

Dorra Guermazi , Àlex Rovira , Jean-Alix Barrat , Raphaël Tripier , Douraied Ben Salem
Journal de Neuroradiologie / Journal of Neuroradiology, 2023, ⟨10.1016/j.neurad.2023.10.006⟩
Article dans une revue hal-04545821 v1

Iodine footprint: Moving towards environmental responsibility

Raphel Jomaah , Jean-Alix J-A Barrat , Raphaël Tripier , Julien Ognard , Samy Ammari et al.
Journal de Neuroradiologie / Journal of Neuroradiology, 2023, 50 (1), pp.1-2. ⟨10.1016/j.neurad.2022.11.002⟩
Article dans une revue hal-04021423 v1
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Synthesis and Photophysical Properties of Lanthanide Pyridinylphosphonic Tacn and Pyclen Derivatives: From Mononuclear Complexes to Supramolecular Heteronuclear Assemblies

Nadège Hamon , Léna Godec , Elsa Jourdain , Carlos Platas-Iglesias , Maryline Beyler et al.
Inorganic Chemistry, 2023, 62 (46), pp.18940-18954. ⟨10.1021/acs.inorgchem.3c02522⟩
Article dans une revue hal-04541125 v1

Design of Bifunctional Pyclen-Based Lanthanide Luminescent Bioprobes for Targeted Two-Photon Imaging

Nadège Hamon , Lucile Bridou , Margaux Roux , Olivier Maury , Raphaël Tripier et al.
Journal of Organic Chemistry, 2023, 88 (13), pp.8286-8299. ⟨10.1021/acs.joc.3c00287⟩
Article dans une revue hal-04254162 v1
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A Phosphine Oxide-Functionalized Cyclam as a Specific Copper(II) Chelator

Marie Le Roy , Simon Héry , Nathalie Saffon-Merceron , Carlos Platas-Iglesias , Thibault Troadec et al.
Inorganic Chemistry, 2023, 62 (21), pp.8112-8122. ⟨10.1021/acs.inorgchem.3c00329⟩
Article dans une revue hal-04308620 v1

Highly inert Cu(II) complexes of C-aryl bifunctional cyclam-picolinates with remarkable Cu-64-labelling and biodistribution

Julie Pineau , Luis M P Lima , M Le Roy , Séverine Marionneau-Lambot , Marie Cordier et al.
Chemical Communications, 2023, 59 (7), pp.888-891. ⟨10.1039/d2cc06602e⟩
Article dans une revue hal-03969219 v1

Bioconjugated chelates based on (methylpyridinyl)tacn: synthesis, 64Cu labeling and in vitro evaluation for prostate cancer targeting

Axia Marlin , Ina Hierlmeier , Amaury Guillou , Mark Bartholomä , Raphaël Tripier et al.
Metallomics, 2022, ⟨10.1093/mtomcs/mfac036⟩
Article dans une revue hal-03697656 v1

Importance of ligand design in lanthanide azamacrocyclic complexes relevant to biomedical applications

Raphaël Tripier , Gyula Tircsó , Carlos Platas-Iglesias , Charlene Harriswangler
Handbook on the Physics and Chemistry of Rare Earths, 2022, Handbook on the Physics and Chemistry of Rare Earths, 61, pp.129-220. ⟨10.1016/BS.HPCRE.2022.05.001⟩
Article dans une revue hal-04545839 v1

Radiopharmaceutical Labelling for Lung Ventilation/Perfusion PET/CT Imaging: A Review of Production and Optimization Processes for Clinical Use

Frédérique Blanc-Béguin , Simon Hennebicq , Philippe Robin , Raphaël Tripier , Pierre-Yves Salaün et al.
Pharmaceuticals, 2022, 15 (5), pp.518. ⟨10.3390/ph15050518⟩
Article dans une revue hal-04545863 v1

Development and in vitro evaluation of a copper-64 radiolabeled antibody for targeting the CXCR4 receptor in human multiple myeloma

Cassandra Métivier , Patricia Le Saec , Hela Bouhsine , Séverine Marionneau-Lambot , Emmanuel Garçion et al.
Nuclear Medicine and Biology, 2022, 108-109, pp.S203-S204. ⟨10.1016/S0969-8051(22)00419-X⟩
Article dans une revue hal-04545853 v1

Copper( ii ) and zinc( ii ) complexation with N -ethylene hydroxycyclams and consequences on the macrocyclic backbone configuration

Nancy Alhaddad , Evan Lelong , Jong-Min Suh , Marie Cordier , Mi Hee Lim et al.
Dalton Transactions, 2022, 51 (22), pp.8640-8656. ⟨10.1039/D2DT00941B⟩
Article dans une revue hal-03679754 v1
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An ultrasensitive and highly selective nanomolar electrochemical sensor based on an electrocatalytic peak shift analysis approach for copper trace detection in water

Lylian Challier , Amélie Forget , Charlène Bazin , Simon Tanniou , Justine Le Doare et al.
Electrochimica Acta, 2022, 434, pp.141298. ⟨10.1016/j.electacta.2022.141298⟩
Article dans une revue hal-03841255 v1
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Palladium(II) coordination with polyazacycloalkanes

Nathalie Le Bris , Julie Pineau , Luís M.P. Lima , Raphaël Tripier
Coordination Chemistry Reviews, 2022, 455, pp.214343. ⟨10.1016/j.ccr.2021.214343⟩
Article dans une revue hal-03583088 v1
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Relevance of Palladium to Radiopharmaceutical Development Considering Enhanced Coordination Properties of TE1PA

Julie Pineau , Luís M P Lima , Carlos Platas-Iglesias , Jan Rijn Zeevaart , Cathryn H S Driver et al.
Chemistry - A European Journal, 2022, 28 (41), pp.e202200942. ⟨10.1002/chem.202200942⟩
Article dans une revue hal-04638161 v1

On the dissociation pathways of copper complexes relevant as PET imaging agents

Rocío Uzal-Varela , Véronique Patinec , Raphaël Tripier , Laura Valencia , Marcelino Maneiro et al.
Journal of Inorganic Biochemistry, 2022, 236, pp.111951. ⟨10.1016/j.jinorgbio.2022.111951⟩
Article dans une revue hal-03765239 v1

New Triazacycloalkane Derivatives as Cytotoxic Agents for CLL Treatment: From Proof of Concept to the Targeting Biomolecule

Axia Marlin , Fiona Le Pape , Jocelyn Le Goff , Nadège Hamon , Thibault Troadec et al.
Bioconjugate Chemistry, 2022, ⟨10.1021/acs.bioconjchem.2c00227⟩
Article dans une revue hal-03697659 v1

“Imaging of diagnostic and therapeutic biomarkers in oncology” XIIIe édition du workshop organisé par le réseau « Vectorisation, Imagerie, Radiothérapies » du Cancéropôle Grand-Ouest, 25–28 septembre 2019, Le Bono, France

Françoise Léost , Michel Chérel , Igor Chourpa , Sara Lacerda , Rbah-Vadal Latifa et al.
Bulletin du Cancer, 2022, 109 (10), pp.1094-1100. ⟨10.1016/j.bulcan.2022.05.010⟩
Article dans une revue (compte-rendu de lecture) hal-04188521 v1
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Electrocatalytic reduction of CO 2 in water by a C -functionalized Ni–cyclam complex grafted onto carbon

Amélie Forget , Matthieu Regnacq , Christophe Orain , Ewen Touzé , Evan Lelong et al.
Chemical Communications, 2022, 58 (48), pp.6785-6788. ⟨10.1039/D2CC01667B⟩
Article dans une revue hal-03679753 v1

Design of polyazamacrocyclic Gd3+ theranostic agents combining magnetic resonance imaging and two-photon photodynamic therapy

Laura Abad Galán , Nadège Hamon , Christophe Nguyen , Enikő Molnár , János Kiss et al.
Inorganic Chemistry Frontiers, 2021, 8 (9), pp.2213-2224. ⟨10.1039/D0QI01519A⟩
Article dans une revue hal-03137794 v1
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Fully Automated 68Ga-Labeling and Purification of Macroaggregated Albumin Particles for Lung Perfusion PET Imaging

Frédérique Blanc-Béguin , Julien Masset , Philippe Robin , Raphaël Tripier , Simon Hennebicq et al.
Frontiers in Nuclear Medicine, 2021, 1 (6), pp.409-411. ⟨10.3389/fnume.2021.778191⟩
Article dans une revue hal-04545867 v1

A roadmap towards pollution prevention and sustainable development of Gadolinium

Julien Ognard , Jean-Alix J-A Barrat , François Cotton , Asim Mian , Stéphane Kremer et al.
Journal de Neuroradiologie / Journal of Neuroradiology, 2021, 48 (6), pp.409-411. ⟨10.1016/j.neurad.2021.08.002⟩
Article dans une revue hal-03429112 v1

Tuning the lipophilic nature of pyclen-based 90Y3+ radiopharmaceuticals for β-radiotherapy

Mariane Le Fur , Olivier Fougère , Nicolas Lepareur , Olivier Rousseaux , Raphaël Tripier et al.
Metallomics, 2021, 13 (12), ⟨10.1093/mtomcs/mfab070⟩
Article dans une revue hal-03468303 v1
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Cyclam-Based Chelators Bearing Phosphonated Pyridine Pendants for 64 Cu-PET Imaging: Synthesis, Physicochemical Studies, Radiolabeling, and Bioimaging

Richard C Knighton , Thibault Troadec , Valérie Mazan , Patricia Le Saëc , Séverine Marionneau-Lambot et al.
Inorganic Chemistry, 2021, 60 (4), pp.2634-2648. ⟨10.1021/acs.inorgchem.0c03492⟩
Article dans une revue hal-03123032 v1

Pyclen-Based Ligands Bearing Pendant Picolinate Arms for Gadolinium Complexation

Gwladys Nizou , Enikő Molnár , Nadège Hamon , Ferenc Krisztián Kálmán , Olivier Fougère et al.
Inorganic Chemistry, 2021, ⟨10.1021/acs.inorgchem.0c03277⟩
Article dans une revue hal-03122227 v1
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Complexation of Mn(II) by Rigid Pyclen Diacetates: Equilibrium, Kinetic, Relaxometric, Density Functional Theory, and Superoxide Dismutase Activity Studies

Zoltán Garda , Enikő Molnár , Nadège Hamon , José Luis Barriada , David Esteban-Gómez et al.
Inorganic Chemistry, 2021, ⟨10.1021/acs.inorgchem.0c03276⟩
Article dans une revue hal-03094039 v1

Complexation of C -Functionalized Cyclams with Copper(II) and Zinc(II): Similarities and Changes When Compared to Parent Cyclam Analogues

Evan Lelong , Jong-Min Suh , Gunhee Kim , David Esteban-Gómez , Marie Cordier et al.
Inorganic Chemistry, 2021, 60 (15), pp.10857-10872. ⟨10.1021/acs.inorgchem.1c01572⟩
Article dans une revue hal-03320076 v1
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In Vivo Albumin‐Binding of a C ‐Functionalized Cyclam Platform for 64 Cu‐PET/CT Imaging in Breast Cancer Model

Thomas Le Bihan , Cathryn Driver , Thomas Ebenhan , Nathalie Le Bris , Jan Rijn Zeevaart et al.
ChemMedChem, 2020, ⟨10.1002/cmdc.202000800⟩
Article dans une revue hal-03079054 v1

A different approach: highly encapsulating macrocycles being used as organic tectons in the building of CPs

Agustín Esteban-Muriel , Carlos Laglera-Gándara , Marta Mato-Iglesias , Raphaël Tripier , Maryline Beyler et al.
CrystEngComm, 2020, ⟨10.1039/D0CE01499K⟩
Article dans une revue hal-03053378 v1
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Efficient luminescence control in dithienylethene functionalized cyclen macrocyclic lanthanide complexes

Hassan Al Sabea , Nadège Hamon , Olivier Galangau , Lucie Norel , Olivier Maury et al.
Inorganic Chemistry Frontiers, 2020, 7 (16), pp.2979-2989. ⟨10.1039/D0QI00354A⟩
Article dans une revue hal-02903552 v1
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Synthesis, Conformational Analysis, and Complexation Study of an Iminosugar-Aza-Crown, a Sweet Chiral Cyclam Analog

Alexandra Bordes , Ana Poveda , Thibault Troadec , Antonio Franconetti , Ana Arda et al.
Organic Letters, 2020, 22 (6), pp.2344-2349. ⟨10.1021/acs.orglett.0c00503⟩
Article dans une revue hal-02504835 v1
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Cationic Biphotonic Lanthanide Luminescent Bioprobes Based on Functionalized Cross‐Bridged Cyclam Macrocycles.

Jonathan Mendy , Anh Thy Bui , Amandine Roux , Jean-Christophe Mulatier , Damien Curton et al.
ChemPhysChem, 2020, 21 (10), pp.1036-1043. ⟨10.1002/cphc.202000085⟩
Article dans une revue hal-02533027 v1

Enabling Indium Channels for Mass Cytometry by Using Reinforced Cyclam-Based Chelating Polylysine

Laura Grenier , Maryline Beyler , Taunia Closson , Nick Zabinyakov , Alexandre Bouzekri et al.
Bioconjugate Chemistry, 2020, 31 (9), pp.2103-2115. ⟨10.1021/acs.bioconjchem.0c00267⟩
Article dans une revue hal-02925847 v1

Reactivities of cyclam derivatives with metal–amyloid-β

Gunhee Kim , Evan Lelong , Juhye Kang , Jong-Min Suh , Nathalie Le Bris et al.
Inorganic Chemistry Frontiers, 2020, ⟨10.1039/D0QI00791A⟩
Article dans une revue hal-02961463 v1
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Unexpected Trends in the Stability and Dissociation Kinetics of Lanthanide(III) Complexes with Cyclen-Based Ligands across the Lanthanide Series

Zoltán Garda , Viktória Nagy , Aurora Rodríguez-Rodríguez , Rosa Pujales-Paradela , Véronique Patinec et al.
Inorganic Chemistry, 2020, 59 (12), pp.8184-8195. ⟨10.1021/acs.inorgchem.0c00520⟩
Article dans une revue hal-02564517 v1

Pyclen-Based Ln(III) Complexes as Highly Luminescent Bioprobes for In Vitro and In Vivo One- and Two-Photon Bioimaging Applications

Nadège Hamon , Amandine Roux , Maryline Beyler , Jean-Christophe Mulatier , Chantal Andraud et al.
Journal of the American Chemical Society, 2020, ⟨10.1021/jacs.0c03496⟩
Article dans une revue hal-02616978 v1
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Formation of Heteropolynuclear Lanthanide Complexes Using Macrocyclic Phosphonated Cyclam-Based Ligands

Richard Knighton , Lohona Soro , Thibault Troadec , Valérie Mazan , Aline Nonat et al.
Inorganic Chemistry, 2020, 59 (14), pp.10311-10327. ⟨10.1021/acs.inorgchem.0c01456⟩
Article dans une revue hal-02903590 v1
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Reply to the 'Comment on "Investigation of Zr(IV) and 89 Zr(IV) complexation with hydroxamates: progress towards designing a better chelator than desferrioxamine B for immuno-PET imaging"' by A. Bianchi and M. Savastano, Chem. Commun., 2020, 56, D0CC01189D

François Guérard , Yong-Sok Lee , Raphaël Tripier , Lawrence Szajek , Jeffrey Deschamps et al.
Chemical Communications, 2020, Online ahead of print. ⟨10.1039/d0cc03594g⟩
Article dans une revue inserm-02947405 v1

A Squaraine-based Dipicolylamine Derivative Acting as a Turn-on Mercury(II) Fluorescent Probe in Water

Catarina Esteves , Hélène Bernard , Judite Costa , Raphaël Tripier , Rita Delgado
New Journal of Chemistry, 2020, ⟨10.1039/D0NJ00852D⟩
Article dans une revue hal-02533107 v1

68Ga-Labelled Carbon Nanoparticles for Ventilation PET/CT Imaging: Physical Properties Study and Comparison with Technegas®

Frédérique Blanc-Béguin , Philippe Eliès , Philippe Robin , Raphaël Tripier , Nelly Kervarec et al.
Molecular Imaging and Biology, 2020, ⟨10.1007/s11307-020-01532-6⟩
Article dans une revue hal-02961527 v1

Synthesis of Orthogonal N -Protected C -Functional Side-Bridged Cyclams to Give Access to Unsymmetrical Constrained BCAs

Thomas Le Bihan , Nathalie Le Bris , Hélène Bernard , Carlos Platas-Iglesias , Raphaël Tripier
European Journal of Organic Chemistry, 2019, ⟨10.1002/ejoc.201901013⟩
Article dans une revue hal-02270928 v1

Highly stable and inert complexation of Indium(III) by reinforced cyclam dipicolinate and a bifunctional derivative for bead encoding in mass cytometry

Laura Grenier , Maryline Beyler , Carlos Platas-Iglesias , Taunia Closson , David Esteban Gómez et al.
Chemistry - A European Journal, 2019, ⟨10.1002/chem.201903969⟩
Article dans une revue hal-02281241 v1

Methylthiazolyl Tacn Ligands for Copper Complexation and Their Bifunctional Chelating Agent Derivatives for Bioconjugation and Copper-64 Radiolabeling: An Example with Bombesin

Amaury Guillou , Luis M P Lima , David Esteban-Gómez , Nicolas Le Poul , Mark Bartholomä et al.
Inorganic Chemistry, 2019, 58 (4), pp.2669-2685. ⟨10.1021/acs.inorgchem.8b03280⟩
Article dans une revue hal-01997423 v1

Endo- versus Exocyclic Coordination in Copper Complexes with Methylthiazolylcarboxylate Tacn Derivatives

Amaury Guillou , Luis M P Lima , David Esteban , Rita Delgado , Carlos Platas-Iglesias et al.
Dalton Transactions, 2019, ⟨10.1039/C9DT01366K⟩
Article dans une revue hal-02142992 v1
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TE1PA as innovating chelator for 64Cu immuno-TEP imaging: a comparative in vivo study with DOTA/NOTA by conjugation on 9E7.4 mAb in a syngeneic multiple myeloma model

Anne-Sophie Navarro , Thomas Le Bihan , Patricia Le Saec , Nathalie Le Bris , Clément Bailly et al.
Bioconjugate Chemistry, 2019, ⟨10.1021/acs.bioconjchem.9b00510⟩
Article dans une revue inserm-02266369 v1
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Picolinate-Appended Tacn Complexes for Bimodal Imaging: radiolabeling, relaxivity, photophysical and electrochemical studies

Amaury Guillou , Margaux Galland , Amandine Roux , Balázs Váradi , Réka Anna Gogolák et al.
Journal of Inorganic Biochemistry, 2019, 205, pp.110978. ⟨10.1016/j.jinorgbio.2019.110978⟩
Article dans une revue inserm-02436868 v1
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What is the Best Radionuclide for Immuno-PET of Multiple Myeloma? A Comparison Study Between 89Zr- and 64Cu-Labeled Anti-CD138 in a Preclinical Syngeneic Model

Clément Bailly , Sébastien Gouard , François Guérard , Benjamin Chalopin , Thomas Carlier et al.
International Journal of Molecular Sciences, 2019, 20 (10), pp.2564. ⟨10.3390/ijms20102564⟩
Article dans une revue hal-02141555 v1

Phosphate and polyphosphate anions recognition by a dinuclear copper(II) complex of an unsymmetrical squaramide

Catarina Esteves , Judite Costa , David Esteban , Pedro Lamosa , Hélène Bernard et al.
Dalton Transactions, 2019, ⟨10.1039/C9DT01434A⟩
Article dans une revue hal-02145467 v1
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Design and Synthesis of Hybrid PEGylated Metal Monopicolinate Cyclam Ligands for Biomedical Applications

Fatima Aouidat , Zakaria Halime , Rosalba Moretta , Ilaria Rea , Stefania Filosa et al.
ACS Omega, 2019, 4 (2), pp.2500-2509. ⟨10.1021/acsomega.8b03266⟩
Article dans une revue hal-02337561 v1

A “Multi‐Heavy‐Atom” Approach Toward Biphotonic Photosensitizers With Improved Singlet Oxygen Generation Properties

Margaux Galland , Tangui Le Bahers , Akos Banyasz , Noëlle Lascoux , Alain Duperray et al.
Chemistry - A European Journal, 2019, 25 (38), pp.9026-9034. ⟨10.1002/chem.201901047⟩
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Steric Effects on the Binding of Phosphate and Polyphosphate Anions by Zinc(II) and Copper(II) Dinuclear Complexes of m -Xylyl-bis-cyclen

Catarina Esteves , David Esteban-Gomez , Carlos Platas-Iglesias , Raphaël Tripier , Rita Delgado
Inorganic Chemistry, 2018, ⟨10.1021/acs.inorgchem.8b00539⟩
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Expanding the Family of Pyclen-Based Ligands Bearing Pendant Picolinate Arms for Lanthanide Complexation

Mariane Le Fur , Enikő Molnár , Maryline Beyler , Olivier Fougere , David Esteban-Gomez et al.
Inorganic Chemistry, 2018, ⟨10.1021/acs.inorgchem.8b00598⟩
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Kinetics are crucial when targeting copper ions to fight Alzheimer's disease: an illustration with azamacrocyclic ligands

Amandine Conte-Daban , Maryline Beyler , Raphaël Tripier , Christelle Hureau
Chemistry - A European Journal, 2018, 24 (33), pp.8447-8452. ⟨10.1002/chem.201801520⟩
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Combining a pyclen framework with conjugated antenna for the design of europium and samarium luminescent bioprobes

Nadège Hamon , Margaux Galland , Mariane Le Fur , Amandine Roux , Alain Duperray et al.
Chemical Communications, 2018, 54 (48), pp.6173-6176. ⟨10.1039/c8cc02035c⟩
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Stable and Inert Yttrium(III) Complexes with Pyclen-Based Ligands Bearing Pendant Picolinate Arms: Toward New Pharmaceuticals for β-Radiotherapy

Mariane Le Fur , Maryline Beyler , Enikő Molnár , Olivier Fougere , David Esteban-Gómez et al.
Inorganic Chemistry, 2018, 57 (4), pp.2051-2063. ⟨10.1021/acs.inorgchem.7b02953⟩
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Synthesis of C-functionalized TE1PA and comparison with its analogues. An example of bioconjugation on 9E7.4 mAb for multiple myeloma 64 Cu-PET imaging

Thomas Le Bihan , Anne-Sophie Navarro , Nathalie Le Bris , Patricia Le Saec , Sébastien Gouard et al.
Organic & Biomolecular Chemistry, 2018, Epub ahead of print. ⟨10.1039/c8ob00499d⟩
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Biodistribution, Imaging and Metabolism Studies of 64-Copper Radiolabelled Monoclonal Antibody : Comparison of DOTA and TE1PA Chelating Agents in a Murine Model of Multiple Myeloma

A. Navarro , T. Le Bihan , Patricia Remaud-Le Saëc , Sébastien Gouard , N. Le Bris et al.
European Journal of Nuclear Medicine and Molecular Imaging, 2018, 45 (1), pp.S119-S120
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Comparison of Immuno-PET of CD138 and PET imaging with 64CuCl2 and 18F-FDG in a preclinical syngeneic model of multiple myeloma

Clément Bailly , Sébastien Gouard , Marie Lacombe , Patricia Remaud-Le Saëc , Benjamin Chalopin et al.
Oncotarget, 2018, 9, pp.9061-9072. ⟨10.18632/oncotarget.23886⟩
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A Coordination Chemistry Approach to Fine-Tune the Physicochemical Parameters of Lanthanide Complexes Relevant to Medical Applications

Mariane Le Fur , Eniko Molnar , Maryline Beyler , Ferenc K Kalman , Olivier Fougère et al.
Chemistry - A European Journal, 2018, Chemistry, an European journal, 24 (13), pp.3127-3131. ⟨10.1002/chem.201705528⟩
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PET Imaging of Multiple Myeloma : Comparison of 89Zr- and 64Cu-labeled anti-CD138 Conjugates to 64CuCl2 and 18F-FDG in a Preclinical Syngeneic Model

Clément Bailly , Sébastien Gouard , Benjamin Chalopin , Thomas M Carlier , Catherine Sai-Maurel et al.
European Journal of Nuclear Medicine and Molecular Imaging, 2018, 45 (1), pp.S20-S21
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Near infrared two photon imaging using a bright cationic Yb(III) bioprobe spontaneously internalized into live cells

Anh Thy Bui , Maryline Beyler , Alexei Grichine , Alain Duperray , Jean-Christophe Mulatier et al.
Chemical Communications, 2017, 53, pp.6005-6008 ⟨10.1039/C7CC02835K⟩
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Definition of the Labile Capping Bond Effect in Lanthanide Complexes

Aurora Rodriguez-Rodriguez , Martin Regueiro-Figueroa , David Esteban-Gomez , Teresa Rodriguez-Blas , Véronique Patinec et al.
Chemistry - A European Journal, 2017, 23 (5), pp.1110 - 1117. ⟨10.1002/chem.201604390⟩
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Tuning the copper( ii ) coordination properties of cyclam by subtle chemical modifications

Nathalie Le Bris , Nathalie Camus , Selbi Nuryyeva , Matthieu Chessé , David Esteban-Gómez et al.
Dalton Transactions, 2017, 46 (34), pp.11479 - 11490. ⟨10.1039/C7DT00750G⟩
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The role of the capping bond effect on pyclen Y-nat(3+)/Y-90(3+) chelates: full control of the regiospecific N-functionalization makes the difference

Mariane Le Fur , Maryline Beyler , Eniko Molnar , Olivier Fougere , David Esteban-Gomez et al.
Chemical Communications, 2017, 53 (69), pp.9534-9537. ⟨10.1039/c7cc05088g⟩
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Investigation of the complexation of nat Zr(IV) and 89 Zr(IV) by hydroxypyridinones for the development of chelators for PET imaging applications

François Guérard , Maryline Beyler , Y.-S Lee , Raphaël Tripier , Jean-François Gestin et al.
Dalton Transactions, 2017, 46, pp.4749-4758. ⟨10.1039/c6dt04625h⟩
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Cyclam te1pa for 64 Cu PET imaging. Bioconjugation to antibody, radiolabeling and preclinical application in xenografted colorectal cancer

Mathieu Frindel , Patricia Le Saec , Maryline Beyler , Anne-Sophie Navarro , Catherine Sai-Maurel et al.
RSC Advances, 2017, 7, pp.9272-9283. ⟨10.1039/c6ra26003a⟩
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Spectroscopic Properties of a Family of Mono- to Trinuclear Lanthanide Complexes

Mohamadou Sy , David Esteban-Gómez , Carlos Platas-Iglesias , Aurora Rodríguez-Rodríguez , Raphaël Tripier et al.
European Journal of Inorganic Chemistry, 2017, 2017 (14), pp.2122 - 2129. ⟨10.1002/ejic.201601516⟩
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1,4,7-Triazacyclononane-Based Bifunctional Picolinate Ligands for Efficient Copper Complexation

Amaury Guillou , Luís M. P. Lima , Mélissa Roger , David Esteban-Gomez , Rita Delgado et al.
European Journal of Inorganic Chemistry, 2017, 2017 (18), pp.2435 - 2443. ⟨10.1002/ejic.201700176⟩
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Cationic Two-Photon Lanthanide Bioprobes Able to Accumulate in Live Cells

Anh Thy Bui , Maryline Beyler , Yuan-Yuan Liao , Alexei Grichine , Alain Duperray et al.
Inorganic Chemistry, 2016, 55 (14), pp.7020 - 7025. ⟨10.1021/acs.inorgchem.6b00891⟩
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Improving the stability and inertness of Cu( ii ) and Cu( i ) complexes with methylthiazolyl ligands by tuning the macrocyclic structure

Mariane Le Fur , Maryline Beyler , Nicolas Le Poul , Luís M. P. Lima , Yves Le Mest et al.
Dalton Transactions, 2016, 45 (17), pp.7406 - 7420. ⟨10.1039/C6DT00385K⟩
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Correction: New synthesis of phenyl-isothiocyanate C-functionalised cyclams. Bioconjugation and 64Cu phenotypic PET imaging studies of multiple myeloma with the te2a derivative

Zakaria Halime , M. Frindel , N. Camus , Pierre Yves Orain , M. Lacombe et al.
Organic & Biomolecular Chemistry, 2016, 14 (15), pp.3838. ⟨10.1039/c6ob90046a⟩
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Catching anions with coloured assemblies: binding of pH indicators by a giant-size polyammonium macrocycle for anion naked-eye recognition

Nathalie Le Bris , Francesco Bartoli , Andrea Bencini , Luca Conti , Claudia Giorgi et al.
Organic & Biomolecular Chemistry, 2016, 14 (35), pp.8309 - 8321. ⟨10.1039/c6ob01474g⟩
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Complexation of Ln 3+ Ions with Cyclam Dipicolinates: A Small Bridge that Makes Huge Differences in Structure, Equilibrium, and Kinetic Properties

Aurora Rodriguez-Rodriguez , Martin Regueiro-Figueroa , David Esteban-Gomez , Raphaël Tripier , Gyula Tircso et al.
Inorganic Chemistry, 2016, 55 (5), pp.2227 - 2239. ⟨10.1021/acs.inorgchem.5b02627⟩
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Intracellular Transport Studies of Picolinate Macrocyclic Copper and Lanthanide Complexes

Diego Santo Domingo Porqueras , Maryline Beyler , Raphaël Tripier , Milena Salerno
ChemistrySelect, 2016, 1 (15), pp.4423 - 4429. ⟨10.1002/slct.201600990⟩
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Pyclen Tri- n -butylphosphonate Ester as Potential Chelator for Targeted Radiotherapy: From Yttrium(III) Complexation to 90 Y Radiolabeling

Mariane Le Fur , Maryline Beyler , Nicolas Lepareur , Olivier Fougère , Carlos Platas-Iglesias et al.
Inorganic Chemistry, 2016, 55 (16), pp.8003 - 8012. ⟨10.1021/acs.inorgchem.6b01135⟩
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The Relationship between NMR Chemical Shifts of Thermally Polarized and Hyperpolarized 89 Y Complexes and Their Solution Structures

Yixun Xing , Ashish K. Jindal , Martin Regueiro-Figueroa , Mariane Le Fur , Nelly Kervarec et al.
Chemistry - A European Journal, 2016, 22 (46), pp.16657 - 16667. ⟨10.1002/chem.201602901⟩
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Cyclams with Ambidentate Methylthiazolyl Pendants for Stable, Inert, and Selective Cu(II) Coordination

Aurora Rodríguez-Rodríguez , Zakaria Halime , Luís M. P. Lima , Maryline Beyler , David Deniaud et al.
Inorganic Chemistry, 2016, 55 (2), pp.619-632. ⟨10.1021/acs.inorgchem.5b01779⟩
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Targeting amyloid peptide using metal complexes

Diego Santo Domingo Porqueras , Raphaël Tripier , Maryline Beyler , Milena Salerno
Alzheimer's & Dementia : the Journal of the Alzheimer's Association, 2015, 11 (7), ⟨10.1016/j.jalz.2015.06.355⟩
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New synthesis of phenyl-isothiocyanate C-functionalised cyclams. Bioconjugation and 64 Cu phenotypic PET imaging studies of multiple myeloma with the te2a derivative †

Zakaria Halime , Mathieu Frindel , Nathalie Camus , Pierre-Yves Orain , Marie Lacombe et al.
Organic & Biomolecular Chemistry, 2015, 13 (46), pp.11302-14. ⟨10.1039/c5ob01618e⟩
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Investigating the Complexation of the Pb 2+ /Bi 3+ Pair with Dipicolinate Cyclen Ligands

Luís M. P. Lima , Maryline Beyler , Rita Delgado , Carlos Platas-Iglesias , Raphaël Tripier
Inorganic Chemistry, 2015, 54 (14), pp.7045 - 7057. ⟨10.1021/acs.inorgchem.5b01079⟩
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A [two-step/one week] synthesis of C-functionalized homocyclens and cyclams. Application to the preparation of conjugable BCAs without chelating properties alteration

Nathalie Camus , Zakaria Halime , Nathalie Le Bris , Hélène Bernard , Maryline Beyler et al.
RSC Advances, 2015, 5 (104), pp.85898 - 85910. ⟨10.1039/c5ra17133d⟩
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Dalton Discussion 15 – Metal ions in medical imaging: optical, radiopharmaceutical and MRI contrast, 8 th –10 th September 2014, York

Stephen J. Archibald , Raphaël Tripier
Dalton Transactions, 2015, 44 (11), pp.4789 - 4790. ⟨10.1039/C5DT90036K⟩
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Straightforward and mild deprotection methods of N-mono- and N1,N7-functionalised bisaminal cyclens

Fatima Oukhatar , Maryline Beyler , Raphaël Tripier
Tetrahedron, 2015, 71 (23), pp.3857 - 3862. ⟨10.1016/j.tet.2015.04.021⟩
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Chelator free gallium-68 radiolabelling of silica coated iron oxide nanorods via surface interactions

Benjamin P. Burke , Neazar Baghdadi , Alicja E. Kownacka , Shubhanchi Nigam , Goncalo S. Clemente et al.
Nanoscale, 2015, 7 (36), pp.14889 - 14896. ⟨10.1039/C5NR02753E⟩
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Stable Mn 2+ , Cu 2+ and Ln 3+ complexes with cyclen-based ligands functionalized with picolinate pendant arms

Aurora Rodríguez-Rodríguez , Zoltán Garda , Erika Ruscsák , David Esteban-Gómez , Andrés de Blas et al.
Dalton Transactions, 2015, 44 (11), pp.5017 - 5031. ⟨10.1039/C4DT02985B⟩
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Gd 3+ -Based Magnetic Resonance Imaging Contrast Agent Responsive to Zn 2+

Martin Regueiro-Figueroa , Serhat Gunduz , Véronique Patinec , Nikos K. Logothetis , David Esteban-Gomez et al.
Inorganic Chemistry, 2015, 54 (21), pp.10342 - 10350. ⟨10.1021/acs.inorgchem.5b01719⟩
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Full Control of the Regiospecific N -Functionalization of C -Functionalized Cyclam Bisaminal Derivatives and Application to the Synthesis of their TETA, TE2A, and CB-TE2A Analogues

Nathalie Le Bris , Nathalie Camus , Zakaria Halime , Hélène Bernard , Carlos Platas-Iglesias et al.
Journal of Organic Chemistry, 2014, 79 (5), pp.1885 - 1899. ⟨10.1021/jo4028566⟩
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Picolinate-Containing Macrocyclic Mn 2+ Complexes as Potential MRI Contrast Agents

Enikő Molnár , Nathalie Camus , Véronique Patinec , Gabriele A. Rolla , Mauro Botta et al.
Inorganic Chemistry, 2014, 53 (10), pp.5136 - 5149. ⟨10.1021/ic500231z⟩
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Supramolecular Luminescent Lanthanide Dimers for Fluoride Sequestering and Sensing

Hong Tao Liu , Aline M. Nonat , Maryline Beyler , Martin Regueiro-Figueroa , Katia Nchimi Nono et al.
Angewandte Chemie, 2014, 53 (28), pp.7259-7263. ⟨10.1002/anie.201404847⟩
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Monopicolinate Cross-Bridged Cyclam Combining Very Fast Complexation with Very High Stability and Inertness of Its Copper(II) Complex

Luís M. P. Lima , Zakaria Halime , Ronan Marion , Nathalie Camus , Rita Delgado et al.
Inorganic Chemistry, 2014, 53 (10), pp.5269 - 5279. ⟨10.1021/ic500491c⟩
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Lanthanide Complexes with Heteroditopic Ligands as Fluorescent Zinc Sensors

Mélissa Roger , Martín Regueiro-Figueroa , Chams Ben Azzeddine , Véronique Patinec , Célia S. Bonnet et al.
European Journal of Inorganic Chemistry, 2014, 2014 (6), pp.1072-1081. ⟨10.1002/ejic.201301426⟩
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Radiolabeling of HTE1PA: A new monopicolinate cyclam derivative for Cu-64 phenotypic imaging. In vitro and in vivo stability studies in mice

Mathieu Frindel , Nathalie Camus , Aurore Rauscher , Mickaël Bourgeois , Cyrille Alliot et al.
Nuclear Medicine and Biology, 2014, 41, pp.e49 - e57. ⟨10.1016/j.nucmedbio.2013.12.009⟩
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H2Me-do2pa: an attractive chelator with fast, stable and inert nat Bi 3+ and 213 Bi 3+ complexation for potential α-radioimmunotherapy applications

Luís M. P. Lima , Maryline Beyler , Fatima Oukhatar , Patricia Le Saec , Alain Faivre-Chauvet et al.
Chemical Communications, 2014, 50 (82), pp.12371 - 12374. ⟨10.1039/C4CC05529B⟩
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Synthesis of an unsymmetrical N-functionalized triazacyclononane ligand and its Cu(II) complex

Mélissa Roger , Véronique Patinec , Raphaël Tripier , Smail Triki , Nicolas Le Poul et al.
Inorganica Chimica Acta, 2014, 417, pp.201--207. ⟨10.1016/j.ica.2013.12.036⟩
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Investigation of Zr( iv ) and 89 Zr( iv ) complexation with hydroxamates: progress towards designing a better chelator than desferrioxamine B for immuno-PET imaging

François Guérard , Yong-Sok Lee , Raphaël Tripier , Lawrence P. Szajek , Jeffrey R. Deschamps et al.
Chemical Communications, 2013, 49 (10), pp.1002 - 1004. ⟨10.1039/C2CC37549D⟩
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A new bis-tetraamine ligand with a chromophoric 4-(9-anthracenyl)-2,6-dimethylpyridinyl linker for glyphosate and ATP sensing

Jacky Pouessel , Nathalie Le Bris , Sabah Abada , Mourad Elhabiri , Loïc J. Charbonnière et al.
Dalton Transactions, 2013, 42 (14), ⟨10.1039/c3dt32325k⟩
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Monopicolinate-dipicolyl Derivative of Triazacyclononane for Stable Complexation of Cu 2+ and 64 Cu 2+

Melissa Roger , Luis M. P. Lima , Mathieu Frindel , Carlos Platas-Iglesias , Jean-François Gestin et al.
Inorganic Chemistry, 2013, 52 (9), pp.5246 - 5259. ⟨10.1021/ic400174r⟩
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Lanthanide(III) Complexes with Ligands Derived from a Cyclen Framework Containing Pyridinecarboxylate Pendants. The Effect of Steric Hindrance on the Hydration Number

Aurora Rodriguez-Rodriguez , David Esteban-Gomez , Andrés de Blas , Teresa Rodriguez-Blas , Marianna Fekete et al.
Inorganic Chemistry, 2012, 51 (4), pp.2509 - 2521. ⟨10.1021/ic202436j⟩
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exo-Diastereoisomer of 10-aryl-1,4,7-triazabicyclo[5.2.1]decane as intermediary in specific derivatisation of triazacyclononane

Mélissa Roger , Véronique Patinec , Martine Bourgeois , Raphaël Tripier , Smail Triki et al.
Tetrahedron, 2012, 68 (27-28), pp.5637 - 5643. ⟨10.1016/j.tet.2012.04.057⟩
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Polyaminoquinoline iron chelators for vectorization of antiproliferative agents: design, synthesis, and validation.

Vincent Corcé , Emmanuelle Morin , Solène Guihéneuf , Eric Renault , Stéphanie Renaud et al.
Bioconjugate Chemistry, 2012, 23 (9), pp.1952-68. ⟨10.1021/bc300324c⟩
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Monopicolinate Cyclen and Cyclam Derivatives for Stable Copper(II) Complexation

Luís M. P. Lima , David Esteban-Gómez , Rita Delgado , Carlos Platas-Iglesias , Raphaël Tripier
Inorganic Chemistry, 2012, 51 (12), pp.6916 - 6927. ⟨10.1021/ic300784v⟩
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Glyphosate and ATP binding by mononuclear Zn(ii) complexes with non-symmetric ditopic polyamine ligands

Jacky Pouessel , Nathalie Le Bris , Andrea Bencini , Claudia Giorgi , Barbara Valtancoli et al.
Dalton Transactions, 2012, 41 (35), ⟨10.1039/C2DT31110K⟩
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Solution Structure of Ln(III) Complexes with Macrocyclic Ligands Through Theoretical Evaluation of 1 H NMR Contact Shifts

Aurora Rodríguez-Rodríguez , David Esteban-Gómez , Andrés de Blas , Teresa Rodríguez-Blas , Mauro Botta et al.
Inorganic Chemistry, 2012, 51 (24), pp.13419 - 13429. ⟨10.1021/ic302322r⟩
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1,2,4-Triazine method of bipyridine ligand synthesis for the preparation of new luminescent Eu(III) complexes

Nathalie Le Bris , Anton Prokhorov , Valery N. Kozhevnikov , Dmitry S. Kopchuk , Hélène Bernard et al.
Tetrahedron, 2011, 67 (3), pp.597 - 607. ⟨10.1016/j.tet.2010.11.058⟩
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Selective Binding of Glyphosate by a Ditopic Cyclic-Open-Chain Polyazaligand in Aqueous Solution

Nathalie Le Bris , Jacky Pouessel , Andrea Bencini , Claudia Giorgi , Henri Handel et al.
European Journal of Organic Chemistry, 2011, 2011 (34), pp.6965 - 6973. ⟨10.1002/ejoc.201100972⟩
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Synthesis, complexation and NMR relaxation properties of Gd3+ complexes of Mes(DO3A)3

Pascal Miéville , Hugues Jaccard , Felipe Reviriego , Raphaël Tripier , Lothar Helm
Dalton Transactions, 2011, 40 (16), ⟨10.1039/C0DT01597K⟩
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trans-Methylpyridine cyclen versus cross-bridged trans-methylpyridine cyclen. Synthesis, acid–base and metal complexation studies (metal = Co2+, Cu2+, and Zn2+)

Nicolas Bernier , Judite Costa , Rita Delgado , Vítor Félix , Guy Royal et al.
Dalton Transactions, 2011, ⟨10.1039/C0DT01191F⟩
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Positively Charged Lanthanide Complexes with Cyclen-Based Ligands : Synthesis, Solid-State and Solution Structure, and Fluoride Interaction

Luis M.P Lima , Alexandre Lecointre , Jean-François Morfin , Andres de Blas , Dimitris Visvikis et al.
Inorganic Chemistry, 2011, 50 (24), pp.12508-12521. ⟨10.1021/ic201447c⟩
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Exploring New Molecular Architectures for Anion Recognition: Synthesis and ATP Binding Properties of New Cyclam-Based Ditopic Polyammonium Receptors.

Nathalie Le Bris , Jacky Pouessel , Carla Bazzicalupi , Andrea Bencini , Hélène Bernard et al.
Chemistry - An Asian Journal, 2011, 6 (6), pp.1582 - 1594. ⟨10.1002/asia.201100046⟩
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Cyclen-Based Lanthanide Complexes as Luminescent Anion Receptors

Luis M. P. Lima , Raphaël Tripier
Current Inorganic Chemistrye, 2011, 1 (1), pp.36 - 60. ⟨10.2174/1877944111101010036⟩
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Towards Fluoride Sensing with Positively Charged Lanthanide Complexes

Raphaël Tripier , Carlos Platas-Iglesias , Anne Boos , Jean-François Morfin , Loïc Charbonnière
European Journal of Inorganic Chemistry, 2010, 2010 (18), pp.2735 - 2745. ⟨10.1002/ejic.200901045⟩
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From Flexible to Constrained Tris(tetraamine) Ligands: Synthesis, Acid-Base Properties, and Structural Effect on the Coordination Process with Nucleotides

Anne-Sophie Delépine , Raphaël Tripier , Michel Le Baccon , Henri Handel
European Journal of Organic Chemistry, 2010, 2010 (28), pp.5380 - 5390. ⟨10.1002/ejoc.201000495⟩
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A Tris-Macrocycle with Proton Sponge Characteristics as Efficient Receptor for Inorganic Phosphate and Nucleotide Anions

Andrea Bencini , Silvia Biagini , Claudia Giorgi , Henri Handel , Michel Le Baccon et al.
European Journal of Organic Chemistry, 2009, 2009 (32), pp.5610 - 5621. ⟨10.1002/ejoc.200900770⟩
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Selective mono-N-alkylation of triethylenetetraamine. A new versatile route to polylinear aza-ligands

Nathalie Le Bris , Anne-Sophie Delépine , Raphaël Tripier , Hélène Bernard , Henri Handel
Tetrahedron Letters, 2009, 50 (21), pp.2521 - 2524. ⟨10.1016/j.tetlet.2009.03.088⟩
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Bismuth(III) complexes with tetra-pyridylmethyl-cyclen

Jean-François Morfin , Raphaël Tripier , Michel Le Baccon , Henri Handel
Inorganica Chimica Acta Reviews, 2009, 362 (6), pp.1781 - 1786. ⟨10.1016/j.ica.2008.08.013⟩
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ATP and triphosphate anions complexation by bis-linear tetraamines: Strong interactions at neutral pH

Nathalie Le Bris , Anne-Sophie Delépine , Raphaël Tripier , Hélène Bernard , Aurelien Honraedt et al.
Inorganica Chimica Acta Reviews, 2009, 362 (10), pp.3829 - 3834. ⟨10.1016/j.ica.2009.05.003⟩
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Macrocycle-Based Spin-Crossover Materials

Fatima El Hajj , Ghania Sebki , Véronique Patinec , Mathieu Marchivie , Smail Triki et al.
Inorganic Chemistry, 2009, 48 (21), pp.10416 - 10423. ⟨10.1021/ic9012476⟩
Article dans une revue hal-01580280 v1

Selective mono-N-alkylation of triethylenetetraamine. A new versatile route to polylinear aza-ligands

Nathalie Le Bris , Anne-Sophie Delépine , Raphaël Tripier , Hélène Bernard , Henri Handel
Tetrahedron Letters, 2009, 50 (21), pp.2521 - 2524. ⟨10.1016/j.tetlet.2009.03.088⟩
Article dans une revue istex hal-01629513 v1

Bismuth (III) coordination to cyclen and cyclam bearing four appended groups

Jean-François Morfin , Raphaël Tripier , Michel Le Baccon , Henri Handel
Polyhedron, 2009, 28 (17), pp.3691 - 3698. ⟨10.1016/j.poly.2009.08.003⟩
Article dans une revue istex hal-01580260 v1

Cyclen-based bismacrocycles for biological anion recognition. A potentiometric and NMR study of AMP, ADP and ATP nucleotide complexation

Anne-Sophie Delépine , Raphaël Tripier , Henri Handel
Organic & Biomolecular Chemistry, 2008, 6 (10), ⟨10.1039/b719514a⟩
Article dans une revue istex hal-01580393 v1

Polyamines : études et applications

Franck Denat , David Deniaud , Raphaël Tripier
L'Actualité Chimique, 2008, pp.10-21
Article dans une revue hal-00458572 v1

Electrochemically-driven conformational shift in mono- and di-copper constrained macrotricyclic cyclen receptors

Antonio Doménech , Enrique García-España , Nicolas Bernier , Raphaël Tripier , Henri Handel
Dalton Transactions, 2008, 24, ⟨10.1039/b718163a⟩
Article dans une revue istex hal-01580422 v1

Proton-sponge behaviour of new pendant armed cross-bridged bis-cyclens: Synthesis, NMR, X-ray, and potentiometric investigations

Raphaël Tripier , Véronique Patinec , Michel Le Baccon , Henri Handel , Nicolas Bernier
Comptes Rendus. Chimie, 2007, 10 (9), pp.832 - 838. ⟨10.1016/j.crci.2007.03.016⟩
Article dans une revue istex hal-01581385 v1

Monopropionate analogues of DOTA4– and DTPA5–: kinetics of formation and dissociation of their lanthanide(iii) complexes

Edina Balogh , Raphaël Tripier , Petra Fousková , Felipe Reviriego , Henri Handel et al.
Dalton Transactions, 2007, 32, ⟨10.1039/B706353A⟩
Article dans une revue istex hal-01581370 v1

A potentiometric and NMR investigation of triphosphate recognition by linear and bismacrocyclic octaamines possessing a 1,4-xylenyl linker

Nathalie Le Bris , Hélène Bernard , Raphaël Tripier , Henri Handel
Inorganica Chimica Acta Reviews, 2007, 360 (9), pp.3026 - 3032. ⟨10.1016/j.ica.2007.02.041⟩
Article dans une revue istex hal-01629525 v1

Complexation of the triphosphate anion: tuning the structure of cyclen based macrotricycles with 1,3-dimethylbenzene and 2,6-dimethylpyridine linkers. A potentiometric and NMR study

Stéphanie Develay , Raphaël Tripier , Nicolas Bernier , Michel Le Baccon , Véronique Patinec et al.
Dalton Transactions, 2007, 10, ⟨10.1039/B616862K⟩
Article dans une revue istex hal-01581204 v1
Image document

Lipophosphoramidates as Lipidic Part of Lipospermines for Gene Delivery

François Lamarche , Mathieu Mével , Tristan Montier , Laure Burel-Deschamps , Philippe Giamarchi et al.
Bioconjugate Chemistry, 2007, 18 (5), pp.1575-1582. ⟨10.1021/bc070070w⟩
Article dans une revue istex hal-01581383 v1

Unexpected Aggregation of Neutral, Xylene-Cored Dinuclear Gd(III) Chelates in Aqueous Solution

Jérôme Costa , Edina Balogh , Véronique Turcry , Raphaël Tripier , Michel Le Baccon et al.
Chemistry - A European Journal, 2006, 12 (26), pp.6841 - 6851. ⟨10.1002/chem.200501335⟩
Article dans une revue istex hal-01582907 v1

Reaction of polyamines with diethyloxalate: a convenient route for the synthesis of tetraazacycloalkanes

Franck Denat , Raphaël Tripier , Frédéric Boschetti , Enrique Espinosa , Roger Guilard
ARKIVOC - Online Journal of Organic Chemistry, 2006, pp.212-233. ⟨10.3998/ark.5550190.0007.415⟩
Article dans une revue hal-00458543 v1

New side-bridged bismacrocycles and cross-bridged macrotricycles. Syntheses and Cu(ii) complexation study

Nicolas Bernier , Mustapha Allali , Raphaël Tripier , Françoise Conan , Véronique Patinec et al.
New Journal of Chemistry, 2006, 30 (3), ⟨10.1039/B515150C⟩
Article dans une revue istex hal-01582163 v1

Reaction of polyamines with diethyloxalate: A convenient route for the synthesis of tetraazacycloalkanes

F. Denat , R. Tripier , F. Boschetti , E. Espinosa , R. Guilard
ARKIVOC - Online Journal of Organic Chemistry, 2006, 4, pp.212-233
Article dans une revue hal-00204589 v1

Host–guest interaction between cyclen based macrotricyclic ligands and phosphate anions. A potentiometric investigation

Stéphanie Develay , Raphaël Tripier , Michel Le Baccon , Véronique Patinec , Guy Serratrice et al.
Dalton Transactions, 2006, 28, pp.3418 - 3426. ⟨10.1039/b517695f⟩
Article dans une revue istex hal-01582849 v1

Cyclen based bis-macrocyclic ligands as phosphates receptors. A potentiometric and NMR study

S. Develay , Raphaël Tripier , M.L. Baccon , Véronique Patinec , G. Serratrice et al.
Dalton Transactions, 2005, 18, pp.3016-3024. ⟨10.1039/b507819a⟩
Article dans une revue istex hal-01763759 v1

Kinetics of formation and dissociation of lanthanide(III) complexes with the 13-membered macrocyclic ligand TRITA

E. Balogh , Raphaël Tripier , R. Ruloff , É. Tóth
Dalton Transactions, 2005, 6, pp.1058-1065. ⟨10.1039/b418991d⟩
Article dans une revue istex hal-01763750 v1

Mono- and dinuclear CuII and ZnII complexes of cyclen-based Bis(macrocycles) containing two aminoalkyl pendant arms of different lengths

C. Anda , A. Bencini , E. Berni , S. Ciattini , F. Chuburu et al.
European Journal of Inorganic Chemistry, 2005, 11, pp.2044-2053. ⟨10.1002/ejic.200400896⟩
Article dans une revue istex hal-01763741 v1

Phenylglyoxal for polyamines modification and cyclam synthesis

Raphaël Tripier , F. Chuburu , M. Le Baccon , Henri Handel
Tetrahedron, 2003, 59 (25), pp.4573-4579. ⟨10.1016/S0040-4020(03)00656-2⟩
Article dans une revue istex hal-01763908 v1

Bis-aminals of linear tetraamines: Kinetic and thermodynamic aspects of the condensation reaction

F. Chuburu , Raphaël Tripier , M. Le Baccon , Henri Handel
European Journal of Organic Chemistry, 2003, 6, pp.1050-1055
Article dans une revue hal-01763890 v1

A new versatile synthesis of macrotricyclic tetraazacycloalkane-based ligands from bis-aminal derivatives

S. Develay , Raphaël Tripier , F. Chuburu , M. Le Baccon , Henri Handel
European Journal of Organic Chemistry, 2003, 16, pp.3047-3050
Article dans une revue hal-01763899 v1

Accelerating water exchange for GdIII chelates by steric compression around the water binding site.

Robert Ruloff , Éva Tóth , Rosario Scopelliti , Raphaël Tripier , Henri Handel et al.
Chemical Communications, 2002, 22, pp.2630-1
Article dans une revue hal-02080840 v1

Harnessing the Pyclen Macrocycle for Advanced Two-Photon Bioimaging

Nadège Hamon , Dina Akl , Baptiste Chartier , Maryline Beyler , Magali Gary-Bobo et al.
Coordination Chemistry Days 2025, Jan 2025, Université Paris-Saclay, France
Communication dans un congrès hal-04928885 v1

Design of Luminescent Lanthanide-Based Bioprobes for Two-Photon NIR-to-NIR Imaging in Vivo Applications

Loeza Collobert , Maryline Beyler , Raphaël Tripier , Olivier Sénèque , Olivier Maury
GECOM-CONCOORD 2025, May 2025, Metabief, France
Communication dans un congrès hal-05114221 v1

Chélateurs azamacrocycliques de cations métalliques : exemples d’applications en biologie

Nadège Hamon , Maryline Beyler , Raphaël Tripier
IBSAM 2025, Jan 2025, Brest, France
Communication dans un congrès hal-04928895 v1

Design and evaluation of mono-N-functionalized pyclen for gallium-68 PET imaging

Maël Le Ménédeu , Nicolas Lepareur , Olivier Fougère , Olivier Rousseaux , Maryline Beyler et al.
6th SCIENTIFIC DAYS OF THE RESEARCH NETWORK ON MOLECULAR IMAGING AGENTS - GDR AIM, Oct 2024, Lyon, France
Communication dans un congrès hal-05111602 v1

A competitive chelating agent for the development of radiopharmaceuticals in personalized nuclear medicine

Julie Pineau , Nathalie Le Bris , Raphaël Tripier
GECOM-CONCOORD 2024, May 2024, Ax-les-Thermes, France
Communication dans un congrès hal-04547260 v1

Optimisation d’un Agent Chélatant Avancé pour la Production de Radiopharmaceutiques en Médecine Nucléaire Personnalisée

Julie Pineau , Nathalie Le Bris , Raphaël Tripier
Journée IBSAM, Mar 2024, Brest, France
Communication dans un congrès hal-04547231 v1

Strategies for Matching Chelators with Cationic Radiometals in Nuclear Medicine: Approaches and Justifications

Raphaël Tripier
Cycle de Conférences de la Société Chimique de France, section Centre-Auvergne, Société Chimique de France, section Centre-Auvergne, Jun 2024, Clermont-Ferrand, France
Communication dans un congrès hal-04613091 v1

Quel(s) chélate(s) aujourd’hui pour quel(s) radioélément(s), avec un focus particulier sur ceux utilisés / utilisables en médecine nucléaire

Raphaël Tripier
Club Français des Radiopharmaceutiques, Session de Printemps, Club Français des Radiopharmaceutiques, May 2024, Montpellier, France
Communication dans un congrès hal-04581205 v1

Dual 18F PET/19F MRI imaging enabled by trifluoroborate prosthetic groups on an azamacrocyclic chelator for metallic cations

Thibault Troadec , Charline Sire , Lorenzo Tei , Emmanuelle Jestin , Raphaël Tripier
Journées de Chimie de Coordination SCF - Journées Franco-Italiennes de Chimie de Coordination, DCC - Société Chimique de France, Jan 2024, Strasbourg, France
Communication dans un congrès hal-04544119 v1

New CuAAC-based method to reach bifunctional cyclam derivatives application in cancer imaging and therapy

Cédric Ollier , Nathalie Le Bris , Raphaël Tripier
SCF Western section, Jun 2024, Logonna-Daoulas, France
Communication dans un congrès hal-04547240 v1

MCTs as new potential targets in oncology: a preliminary investigation in nuclear medicine exploiting both fluorine and copper

Raphaël Tripier , Véronique Patinec
International Symposium on Thermodynamics of Metal Complexes (ISMEC 2024), Jun 2024, Nice (06000), France
Communication dans un congrès hal-04606015 v1

TE1PA: A Powerful Chelator Driving Advances in Copper-Based Radiopharmaceuticals for Enhanced Cancer Diagnosis and Therapy

Raphaël Tripier
International Conference on Coordination Chemistry, Colorado State University (United States), Jul 2024, For Collins, United States
Communication dans un congrès hal-04675574 v1

Trifluoroborated azamacrocylic chelators as valuable tracers for medical imaging

Charline Sire , Vincent Meneyrol , Lorenzo Tei , Emmanuelle Jestin , Raphaël Tripier et al.
Journée de l'Ecole Doctorale S3M, May 2024, Rennes, France
Communication dans un congrès hal-05095846 v1

Trifluoroborated azamacrocylic chelators as valuable tracers for medical imaging

Charline Sire , Vincent Meneyrol , Lorenzo Tei , Emmanuelle Jestin , Raphaël Tripier et al.
SECO 2024, May 2024, Pornichet - La Baule, France
Communication dans un congrès hal-05095842 v1

Advanced Bioimaging: Improved Lanthanide Luminescent Bioprobes Through Pyclen Regiofunctionalization

Nadège Hamon , Lucile Bridou , Margaux Roux , Baptiste Chartier , Magali Gary-Bobo et al.
Journées Scientifiques CenTRA 2024, 2024, Saint-Aubin, France
Communication dans un congrès hal-04541489 v1

Synthèse de chélateurs polyazotés porteurs de groupements fluorés pour des applications théranostiques

Charline Sire , Raphaël Tripier , Thibault Troadec
Colloque de l'IBSAM, Jun 2023, Brest, France
Communication dans un congrès hal-05095774 v1

Functionalization of TE1PA derivatives via CuAAC for cancer imaging and therapy

Cédric Ollier , Nathalie Le Bris , Raphaël Tripier
SECO, May 2023, Arëches-Beaufort, France
Communication dans un congrès hal-04547205 v1

Designing Ln3+ luminescent pyclen complexes for optical imaging: from proof of concept to biological application

Nadège Hamon , Lucile Bridou , Margaux Roux , Maryline Beyler , Magali Gary-Bobo et al.
FrenchBIC, 2023, Logonna-Daoulas, France
Communication dans un congrès hal-04541487 v1

Zr(IV) chelators for innovative diagnostic methods

Alexandra Loubières , Maryline Beyler , Raphaël Tripier
Workshop du réseau VIR "Optimizing Imaging and Dose-Response in RadiotherapieS", Oct 2023, Erquy, France
Communication dans un congrès hal-04546909 v1

Vers de nouveaux radiopharmaceutiques au cuivre pour l’imagerie TEP et la thérapie des cancers

Cédric Ollier , Nathalie Le Bris , Raphaël Tripier
Journée IBSAM, Nov 2023, Brest, France
Communication dans un congrès hal-04547221 v1

Chélatants perfectionnés pour des techniques de diagnostic innovantes

Alexandra Loubières , Maryline Beyler , Raphaël Tripier
Canceropôle Grand Ouest, Journée scientifique annuelle du réseau « Vectorisation, Imagerie, Radiothérapies », Jun 2023, Nantes, France
Communication dans un congrès hal-04546892 v1

Polyazamacrocyclic chelators bearing trifluoroborate arms for the preparation of innovative theranostic radiopharmaceuticals

Charline Sire , Vincent Meneyrol , Emmanuelle Jestin , Raphaël Tripier , Thibault Troadec
GECOM-CONCOORD 2023, May 2023, Fournols, France
Communication dans un congrès hal-05095769 v1

Cyclam as Relevant Platform to Design 99mTc, 64Cu, or 109Pd Radiopharmaceuticals in Nuclear Medicine

Maher Hojorat , Nathalie Le Bris , Raphaël Tripier
ISMEC, Jun 2023, Urbino, Italy
Communication dans un congrès hal-04547213 v1

Design of specific regio-functionnalized pyclen-based Ln(III) complexes for two-photon excitation and application to imaging or theranostic

Nadège Hamon , Laura Abad Galán , Cyrille Monnereau , Maryline Beyler , Magali Gary-Bobo et al.
16th European Biological Inorganic Chemistry Conference, 2022, Grenoble, France
Communication dans un congrès hal-04541482 v1

DUALITE DU FLUOR EN IMAGERIE : NOUVEAUX CHELATEURS FLUORES INTELLIGENTS POUR LA TEP [18F] ET L’IRM [19F]

Thibault Troadec , Emmanuelle Jestin , Lorenzo Tei , Raphaël Tripier
Journées de Recherche en Imagerie et Technologies pour la Santé (RITS) 2022, Société Française de Génie Biologique et Médical, May 2022, Brest, France
Communication dans un congrès hal-04544063 v1

Search and destroy with azamacrocycles

Raphaël Tripier
18èmes Journées de l’axe Vectorisation du Cancéropole Grand Ouest, May 2022, rennes, France
Communication dans un congrès hal-04545887 v1

Tracking CXCR4 with a small synthetic organic vector: chelator conjugation, 64Cu radiolabeling and in vivo targeted-PET imaging

Marie Le Roy , Thibault Troadec , Raphaël Tripier
New Modalities in Cancer Imaging and Therapy, Canceropole Grand Ouest, Oct 2022, Erquy, France
Communication dans un congrès hal-04544142 v1

Imagerie 64Cu-TEP ciblée de CXCR4 par des radiopharmaceutiques synthétiques combinant chélateur du cuivre et petites molecules

Marie Le Roy , Thibault Troadec , Raphaël Tripier
Colloque annuel de l’IBSAM, IBSAM - Université de Bretagne Occidentale, Jun 2022, Brest, France
Communication dans un congrès hal-04544141 v1

Designing lanthanide based tetraazamacrocyclic chelates to improve imaging and therapy.

Raphaël Tripier
10th International Conference on f-Elements (ICFE-11), Aug 2022, Strasbourg, France
Communication dans un congrès hal-04545881 v1

Macrocyclic Zn(II) chelators for biological interests

Axia Marlin , Thibault Troadec , Fiona Le Pape , Christian Berthou , Véronique Patinec et al.
Scientific Days of the French Society of Chemistry (SCF), Western Section (BPL), Sep 2021, Rennes, France
Communication dans un congrès hal-05098291 v1

IMAGE’IN” Imagerie TEP in vivo des cancers, vectorisée par un antagoniste des récepteurs CXCR4 radiomarqués au cuivre-64

Marie Le Roy , Thibault Troadec , Raphaël Tripier
17ème journée scientifique du réseau Vectorisation, Imagerie, Radiothérapies, Canceropole Grand Ouest, May 2021, Webinaire, France
Communication dans un congrès hal-04544133 v1

Développement de radiopharmaceutiques à base de cyclam pour l'imagerie TEP au cuivre-64 et la thérapie des cancers

Nathalie Le Bris , Julie Pineau , Raphaël Tripier
Journée de l'Ecole Doctorale 3M, May 2021, Webinaire, France
Communication dans un congrès hal-04547151 v1

Novel 64Cu/109Pd theranostic pair for a TE1PA-based trifunctional chelating agent

Julie Pineau , Nathalie Le Bris , Raphaël Tripier
SCF western section, Sep 2021, Rennes, France
Communication dans un congrès hal-04547167 v1

IMAGE’IN” In vivo PET imaging of cancers, targeted by an innovative 64Cu-radiolabeled CXCR4 antagonist

Marie Le Roy , Thibault Troadec , Raphaël Tripier
Journée de l’école doctorale Matière, Molécule et Matériaux, Ecole Doctorale S3M, Nov 2021, Nantes, France
Communication dans un congrès hal-04544136 v1

In vivo albumin-binding of a cyclam-based platform for imaging and therapy of cancers

Julie Pineau , Nathalie Le Bris , Raphaël Tripier
GECOM Mini, Jul 2021, Webinaire, France
Communication dans un congrès hal-04547156 v1
Image document

Towards sustainable catalysis enabled by first-row complexes displaying enzyme-inspired features

Tanguy Debaud , Thibault Troadec , Raphaël Tripier , Rafael Gramage-Doria
Jourée de l'Ecole Doctorale (S3M), Apr 2025, Rennes (Campus de Beaulieu), France
Poster de conférence hal-05099970 v1

Harnessing the Pyclen Macrocycle for Advanced Two-Photon Bioimaging

Nadège Hamon , Dina Akl , Baptiste Chartier , Maryline Beyler , Magali Gary-Bobo et al.
5th Scientific Days of the GDR AIM, Oct 2024, Lyon, France
Poster de conférence hal-04928874 v1

New pyclen-based lanthanides complexes for radiotherapy

Maël Le Ménédeu , Olivier Rousseaux , Olivier Fougère , Maryline Beyler , Raphaël Tripier
Journée de la science, Jan 2024, Brest, France
Poster de conférence hal-04550186 v1

Development of pyclen-based lanthanide complexes for deep in vivo biphotonic bioimaging

Loeza Collobert , Maryline Beyler , Raphaël Tripier
Summer School – CS2fE, Jun 2024, Aussois, France
Poster de conférence hal-04606018 v1

Pyclen-based ligands for the complexation of gallium(III)

Raphaël Tripier , Maël Le Ménédeu , Lepareur Nicolas , Olivier Fougère , Olivier Rousseaux et al.
International Symposium on Thermodynamics of Metal Complexes (ISMEC 2024), Jun 2024, Nice, France
Poster de conférence hal-04606016 v1

Fluorinated Azamacrocycles with Dual 19F MRI/18F PET Probe as Potential imaging and Theranostic Tracers : Synthesis, Coordination Chemistry, Radiolabeling and Relaxometry

Thibault Troadec , Charline Sire , Lorenzo Tei , Emmanuelle Jestin , Raphaël Tripier
Journées Scientifiques du Cancéropole Grand Ouest - Réseau Vectorisation, Imagerie, Radiothérapies, Oct 2023, Erquy, France
Poster de conférence hal-04544089 v1

Zr(IV) chelators for innovative diagnostic methods

Alexandra Loubières , Maryline Beyler , Raphaël Tripier
Congrès SCF2023, Jun 2023, Nantes, France
Poster de conférence hal-04546899 v1

Does simplifying the design of macrocyclic lanthanide chelates lead to convincing results in luminescence?

Loeza Collobert , Maryline Beyler , Raphaël Tripier , Lucile Bridou , Olivier Maury
FrenchBic annual meeting 2023, May 2023, Logonna-Daoulas, France
Poster de conférence hal-04550889 v1

64Cu/*Pd-GluCAB: an in vivo albumin-binding theranostic radiopharmaceutical for dual active and passive targeting of breast cancer

Nathalie Le Bris , Raphaël Tripier
International Symposium on Trends in Radiopharmaceuticals, Apr 2023, Vienna, Austria
Poster de conférence hal-04547303 v1

New pyclen-based lanthanides complexes for radiotherapy

Maël Le Ménédeu , Olivier Rousseaux , Olivier Fougère , Maryline Beyler , Raphaël Tripier
ICFE, Aug 2023, Strasbourg, France
Poster de conférence hal-04550168 v1

Zr(IV) chelators for innovative diagnostic methods

Alexandra Loubières , Maryline Beyler , Raphaël Tripier
S3M Doctoral School Day (JED), May 2023, Rennes, France
Poster de conférence hal-04546883 v1

Neutral Copper(II) TE1PA-based chelate for 64Cu-PET imaging: when an additional carboxyl group makes the difference

Julie Pineau , Nathalie Le Bris , Raphaël Tripier
New Modalities in Cancer Imaging and Therapy. Cancéropôle Grand-Ouest, Oct 2022, Erquy, France
Poster de conférence hal-04547281 v1

Relevance of palladium to radiopharmaceutical development considering enhanced.

Julie Pineau , Nathalie Le Bris , Raphaël Tripier
New Modalities in Cancer Imaging and Therapy. Cancéropôle Grand Ouest, Oct 2022, Erquy, France
Poster de conférence hal-04547294 v1

Innovative 64Cu-cyclam-based radiopharmaceuticals for cancer targeting PET imaging with a CXCR4 antagonist

Marie Le Roy , Thibault Troadec , Raphaël Tripier
16th European Biological Inorganic Chemistry Conference (EUROBIC 16), Jul 2022, Grenoble, France
Poster de conférence hal-04544158 v1

Chélates du 89Zr pour des méthodes de diagnostic innovantes

Alexandra Loubières , Maryline Beyler , Raphaël Tripier
Colloque IBSAM, Jun 2022, Brest, France
Poster de conférence hal-04546873 v1

“In vivo 64Cu-PET imaging of cancers, targeted by a CXCR4 receptor antagonist”

Marie Le Roy , Thibault Troadec , Raphaël Tripier
Journée de l’Ecole Doctorale Matière, Molécule et Matériaux, Webinaire, May 2021, Webinaire, France
Poster de conférence hal-04544147 v1

Innovative 64Cu-cyclam-based radiopharmaceuticals for cancer targeting PET imaging with a CXCR4 antagonist

Marie Le Roy , Thibault Troadec , Raphaël Tripier
Journées scientifiques de la SCF section Bretagne Pays de Loire, Sep 2021, Rennes, France
Poster de conférence hal-04544152 v1

New pyclen-based Ln(III) complexes for two-photon microscopy

Nadège Hamon , Mariane Le Fur , Margaux Galland , Amandine Roux , Maryline Beyler et al.
Journées de Chimie de Coordination de la Société Chimique de France, Brest, France., 2018, Brest, France
Poster de conférence hal-04541435 v1

Pyclen-based Eu(III) complex for two-photon microscopy

Nadège Hamon , Mariane Le Fur , Margaux Galland , Maryline Beyler , Olivier Maury et al.
6ème journée du GPOL, 2017, Roscoff (29680), France
Poster de conférence hal-04541432 v1

New pyclen-based Ln(III) complexes for two-photon microscopy

Nadège Hamon , Mariane Le Fur , Margaux Galland , Amandine Roux , Maryline Beyler et al.
Is multimodal imaging an invention for the future? The input of chemistry, 2017, Orléans, France
Poster de conférence hal-04541430 v1

Lanthanide and Other Transition Metal Ion Complexes and Nanoparticles in Magnetic Resonance Imaging

Carlos F.G.C. Geraldes , Raphaël Tripier , Maryline Beyler
Lanthanide and Other Transition Metal Ion Complexes and Nanoparticles in Magnetic Resonance Imaging, 1, CRC Press, 2024, 9781003374688. ⟨10.1201/9781003374688⟩
Chapitre d'ouvrage hal-05096141 v1

Polyamine Drug Discovery. Edited by Patrick Woster and Robert A. Casero, Jr.

Raphaël Tripier
Polyamine Drug Discovery. Edited by Patrick Woster and Robert A. Casero, Jr, 7 (10), , pp.1859 - 1860, 2012, 978-1-84973-190-4. ⟨10.1002/cmdc.201200294⟩
Chapitre d'ouvrage istex hal-01556787 v1

PICOLINATE CYCLAM PALLADIUM CHELATES AND USES THEREOF

Raphaël Tripier , Nathalie Le Bris , Julie Pineau
France, Patent n° : EP 4 273 142 A1. 2022
Brevet hal-04545875 v1

REINFORCED MACROCYCLIC LIGANDS, COMPLEXES THEREOF, AND USES OF SAME

Mariane Le Fur , Gwladys Nizou , Maryline Beyler , Olivier Rousseaux , Raphaël Tripier
France, Patent n° : brevet d'invention FRANCE No.17 55933 WO2019002505 Application: Jun 28, 2018, WO 2018-EP67482. 2019
Brevet hal-02088679 v1

PYCLEN-BASED MACROCYCLIC LIGANDS, CHELATES THEREOF AND USES THEREOF

Nadège Hamon , Maryline Beyler , Raphaël Tripier , Olivier Maury , Janah Shaya
France, Patent n° : WO2019185901. 2019
Brevet hal-04859774 v1

Pyclen-based macrocyclic ligands, chelates thereof and uses thereof.

Nadège Hamon , Maryline Beyler , Olivier Maury , Raphaël Tripier
France, Patent n° : EP 18 305 380.0. 2018
Brevet hal-02089669 v1

Bifunctional do2pa derivatives, chelates with metallic cations and use thereof

Fatima Oukhatar , Maryline Beyler , Raphaël Tripier
France, Patent n° : EP 14 196 637.4. 2016
Brevet hal-01532109 v1

Chelates of Lead (II) and Bismuth (III) Based on Trans-Di-N-Picolinate Tetraazacycloalkanes

Raphaël Tripier , Carlos Platas-Iglesias , Luis M P Lima , Maryline Beyler
France, Patent n° : WO2014195416 - 2014-12-11, PCT/EP2014061723 - 2014-06-05  . 2016
Brevet hal-01532038 v1

Picolinate cross-bridged cyclam, chelate with metallic cations and use thereof

Raphaël Tripier , Zakaria Halime
France, Patent n° : WO2015071334 -2015-05-21. 2015
Brevet hal-01620527 v1

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