Thanh Nhat Pham

12
Documents

Publications

Publications

Design, synthesis, and structure–activity relationship studies of 6 H -benzo[ b ]indeno[1,2- d ]thiophen-6-one derivatives as DYRK1A/CLK1/CLK4/haspin inhibitors

Abdelfattah Faouzi , Alexandre Arnaud , François Hallé , Jean Roussel , Mandy Aymard et al.
RSC Medicinal Chemistry, 2025, 16 (1), pp.179-199. ⟨10.1039/D4MD00537F⟩
Article dans une revue hal-05316119 v1

Valorization of Biomass Polyphenols as Potential Tyrosinase Inhibitors

Thanh Nhat Pham , Elisabeth Anne Cazier , E. Gormally , Philip Lawrence
Drug Discovery Today, 2024, 29 (1), pp.103843. ⟨10.1016/j.drudis.2023.103843⟩
Article dans une revue hal-04598135 v1
Image document

Exploring industrial lignocellulosic waste: Sources, types, and potential as high-value molecules

Elisabeth A. Cazier , Thanh-Nhat Pham , Louis Cossus , Maher Abla , Tina Ilc et al.
Waste Management, 2024, 188, pp.11 - 38. ⟨10.1016/j.wasman.2024.07.029⟩
Article dans une revue hal-04666947 v1

Cinnamides Target Leishmania amazonensis Arginase Selectively

Edson Roberto da Silva , Júlio Abel Alfredo dos Santos Simone Come , Simone Brogi , Vincenzo Calderone , Giulia Chemi et al.
Molecules, 2020, 25 (22), pp.5271. ⟨10.3390/molecules25225271⟩
Article dans une revue hal-03409117 v1

Cinnamides Target Leishmania amazonensis Arginase Selectively

Edson Roberto da Silva , Júlio Abel Alfredo dos Santos Simone Come , Simone Brogi , Vincenzo Calderone , Giulia Chemi et al.
Molecules, 2020, 25 (22), pp.5271. ⟨10.3390/molecules25225271⟩
Article dans une revue hal-03407783 v1

Research of novel anticancer agents targeting arginase inhibition

Thanh-Nhat Pham , Bertrand Liagre , Corine Girard-Thernier , Céline Demougeot
Drug Discovery Today, 2018, 23 (4), pp.871-878. ⟨10.1016/j.drudis.2018.01.046⟩
Article dans une revue hal-03409047 v1

Investigation of Mammal Arginase Inhibitory Properties of Natural Ubiquitous Polyphenols by Using an Optimized Colorimetric Microplate Assay

Simon Bordage , Thanh-Nhat Pham , Andy Zedet , Anne-Sophie Gugglielmetti , Maude Tournier-Nappey et al.
Planta Medica, 2017, 83 (07), pp.647-653. ⟨10.1055/s-0042-118711⟩
Article dans une revue hal-03408743 v1

Cinnamide Derivatives as Mammalian Arginase Inhibitors: Synthesis, Biological Evaluation and Molecular Docking

Thanh-Nhat Pham , Simon Bordage , M. Pudlo , Céline Demougeot , Khac-Minh Thai et al.
International Journal of Molecular Sciences, 2016, 17 (10), pp.1656. ⟨10.3390/ijms17101656⟩
Article dans une revue hal-03409018 v1

Cinnamide Derivatives as Mammalian Arginase Inhibitors: Synthesis, Biological Evaluation and Molecular Docking

Thanh-Nhat Pham , Simon Bordage , M. Pudlo , Céline Demougeot , Khac-Minh Thai et al.
International Journal of Molecular Sciences, 2016, 17 (10), pp.1656. ⟨10.3390/ijms17101656⟩
Article dans une revue hal-03409019 v1

Cinnamide Derivatives as Mammalian Arginase Inhibitors: Synthesis, Biological Evaluation and Molecular Docking

Thanh-Nhat Pham , Simon Bordage , M. Pudlo , Céline Demougeot , Khac-Minh Thai et al.
International Journal of Molecular Sciences, 2016, 17 (10), pp.1656. ⟨10.3390/ijms17101656⟩
Article dans une revue hal-03409024 v1

Cinnamide Derivatives as Mammalian Arginase Inhibitors: Synthesis, Biological Evaluation and Molecular Docking

Thanh-Nhat Pham , Simon Bordage , M. Pudlo , Céline Demougeot , Khac-Minh Thai et al.
International Journal of Molecular Sciences, 2016, 17 (10), pp.1656. ⟨10.3390/ijms17101656⟩
Article dans une revue hal-03407831 v1