Anthony Martin

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Publications

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Targeting pregnane X receptor with a potent agonist-based PROTAC to delay colon cancer relapse

Lucile Bansard , Guillaume Laconde , Vanessa Delfosse , Tiphaine Huet , Margaux Ayeul et al.

Oncogenesis, 2025, 14 (1), pp.34. ⟨10.1038/s41389-025-00573-2⟩

Article dans une revue hal-05238194v1
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Targeting a lineage-specific PI3Kɣ–Akt signaling module in acute myeloid leukemia using a heterobifunctional degrader molecule

Lois Kelly , Justine Rutter , Kevin Lin , Frank Ling , Matthieu Duchmann et al.

Nature Cancer, In press, Online ahead of print. ⟨10.1038/s43018-024-00782-5⟩

Article dans une revue hal-04598240v1
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Covalent-reversible peptide-based protease inhibitors. Design, synthesis, and clinical success stories

Anthony Feral , Anthony R. Martin , Alexandre Desfoux , Muriel Amblard , Lubomir Vezenkov

Amino Acids, In press, ⟨10.1007/s00726-023-03286-1⟩

Article dans une revue (article de synthèse) hal-04167336v1
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Synthesis, photophysics, and theoretical calculations of styryl-based fluorophores harboring substituted benzothiazole acceptors

Mauro Safir Filho , Emmanuel Santos Moraes , Lilian Camargo da Luz , Fabiano da Silveira Santos , Anthony Martin et al.

Journal of Photochemistry and Photobiology A: Chemistry, 2023, ⟨10.1016/j.jphotochem.2022.114287⟩

Article dans une revue hal-03781753v1
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The Unexpected Helical Supramolecular Assembly of a Simple Achiral Acetamide Tecton Generates Selective Water Channels

Dan Dumitrescu , Jordi Rull-Barull , Anthony R. Martin , Nathalie Masquelez , Maurizio Polentarutti et al.

Chemistry - A European Journal, 2022, 28 (33), pp.e202200383. ⟨10.1002/chem.202200383⟩

Article dans une revue hal-03643372v2
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Ultrasound-assisted one-pot three-component synthesis of new isoxazolines bearing sulfonamides and their evaluation against hematological malignancies

Aicha Talha , Cécile Favreau , Maxence Bourgoin , Guillaume Robert , Patrick Auberger et al.

Ultrasonics Sonochemistry, 2021, 78, pp.105748. ⟨10.1016/j.ultsonch.2021.105748⟩

Article dans une revue hal-03342490v1

Dual Covalent Inhibition of PKM and IMPDH Targets Metabolism in Cutaneous Metastatic Melanoma

Marwa Zerhouni , Anthony Martin , Nathan Furstoss , Vincent Gutierrez , Emilie Jaune et al.

Cancer Research, 2021, 81 (14), pp.3806-3821. ⟨10.1158/0008-5472.CAN-20-2114⟩

Article dans une revue hal-03869881v1
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Straightforward synthetic route to gold(I)-thiolato glycoconjugate complexes bearing NHC ligands (NHC = N-heterocyclic carbene) and their promising anticancer activity

Mauro Safir Filho , Thomas Scattolin , Pascal Dao , Nikolaos V Tzouras , Rachid Benhida et al.

New Journal of Chemistry, 2021, 45 (22), pp.9995-10001. ⟨10.1039/D1NJ02117F⟩

Article dans une revue hal-03225368v1
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Nitroreductase sensitive styryl-benzothiazole profluorescent probes for the visualization of mitochondria under normoxic conditions

Mauro Safir Filho , Pascal Dao , Anthony Martin , Rachid Benhida

Journal of Photochemistry and Photobiology A: Chemistry, In press, 396, pp.112528. ⟨10.1016/j.jphotochem.2020.112528⟩

Article dans une revue hal-02567124v1
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GAPDH Overexpression in the T Cell Lineage Promotes Angioimmunoblastic T Cell Lymphoma through an NF-κB-Dependent Mechanism

Laura Mondragón , Rana Mhaidly , Gian Marco de Donatis , Marie Tosolini , Pascal Dao et al.

Cancer Cell, 2019, 36 (3), pp.268-287.e10. ⟨10.1016/j.ccell.2019.07.008⟩

Article dans une revue hal-02323021v1
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Visualization of intracellular lipid droplets using lipophilic benzothiazole-based push-pull fluorophores at ultralow concentration

Mauro Safir Filho , Pascal Dao , Anthony Martin , Rachid Benhida

Dyes and Pigments, 2019, 167, pp.68-76. ⟨10.1016/j.dyepig.2019.04.003⟩

Article dans une revue hal-02147579v1

A straightforward and versatile FeCl 3 catalyzed Friedel–Crafts C -glycosylation process. Application to the synthesis of new functionalized C -nucleosides

Hamza Tachallait , Mauro Safir Filho , Hamid Marzag , Khalid Bougrin , Luc Demange et al.

New Journal of Chemistry, 2019, 43 (14), pp.5551-5558. ⟨10.1039/c8nj06300a⟩

Article dans une revue hal-02322851v1
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Development of highly sensitive fluorescent probes for the detection of β-galactosidase activity – application to the real-time monitoring of senescence in live cells

Mauro Safir Filho , Pascal Dao , Maeva Gesson , Anthony Martin , Rachid Benhida

Analyst, 2018, 143 (11), pp.2680-2688. ⟨10.1039/C8AN00516H⟩

Article dans une revue hal-02147544v1

In Vitro and in Vivo Evaluation of Fully Substituted (5-(3-Ethoxy-3-oxopropynyl)-4-(ethoxycarbonyl)-1,2,3-triazolyl-glycosides as Original Nucleoside Analogues to Circumvent Resistance in Myeloid Malignancies

Hella Amdouni , Guillaume Robert , Mohsine Driowya , Nathan Furstoss , Camille Métier et al.

Journal of Medicinal Chemistry, 2017, ⟨10.1021/acs.jmedchem.6b01803⟩

Article dans une revue hal-01589437v1

Assessment of new triplet forming artificial nucleobases as RNA ligands directed towards HCV IRES IIId loop

Mauro Safir Filho , Anthony R. Martin , Rachid Benhida

Bioorganic and Medicinal Chemistry Letters, 2017, ⟨10.1016/j.bmcl.2017.02.061⟩

Article dans une revue hal-01589492v1

Design, synthesis and photophysical studies of styryl-based push–pull fluorophores with remarkable solvatofluorochromism

Mauro Safir Filho , Sébastien Fiorucci , Anthony Martin , Rachid Benhida

New Journal of Chemistry, 2017, 41 (22), pp.13760-13772. ⟨10.1039/C7NJ03142D⟩

Article dans une revue hal-02545203v1

ATM, ATR, CHK1, CHK2 and WEE1 inhibitors in cancer and cancer stem cells

Cyril Ronco , Anthony R. Martin , Luc Demange , Rachid Benhida

MedChemComm, 2016, ⟨10.1039/C6MD00439C⟩

Article dans une revue hal-01589489v1

Metastatic Melanoma : Insights Into the Evolution of the Treatments and Future Challenges

Antoine Millet , Anthony R. Martin , Cyril Ronco , Stéphane Rocchi , Rachid Benhida

Medicinal Research Reviews, 2016, ⟨10.1002/med.21404⟩

Article dans une revue hal-01589727v1

Hypoxia inducible factor down-regulation, cancer and cancer stem cells (CSCs): ongoing success stories

Anthony R. Martin , Cyril Ronco , Luc Demange , Rachid Benhida

MedChemComm, 2016, ⟨10.1039/C6MD00432F⟩

Article dans une revue hal-01589485v1

Scope and limitations of the dual-gold-catalysed hydrophenoxylation of alkynes

Adrián Gómez-Suárez , Yoshihiro Oonishi , Anthony Martin , Steven Nolan

Beilstein Journal of Organic Chemistry, 2016, 12, pp.172-178. ⟨10.3762/bjoc.12.19⟩

Article dans une revue hal-04599347v1

On the Mechanism of the Digold(I)–Hydroxide‐Catalysed Hydrophenoxylation of Alkynes

Adrián Gómez-Suárez , Yoshihiro Oonishi , Anthony Martin , Sai Vummaleti , David Nelson et al.

Chemistry - A European Journal, 2015, 22 (3), pp.1125-1132. ⟨10.1002/chem.201503097⟩

Article dans une revue hal-04599370v1

DNA-templated borononucleic acid self assembly: a study of minimal complexity

Renaud Barbeyron , Anthony R. Martin , Jean Jacques Vasseur , Michael Smietana

RSC Advances, 2015, 5 (128), pp.105587-105591. ⟨10.1039/C5RA20767C⟩

Article dans une revue hal-03553272v1

Efficient and selective azidation of per-O-acetylated sugars using ultrasound activation: application to the one-pot synthesis of 1,2,3-triazole glycosides

Hamid Marzag , Soukaina Alaoui , Hella Amdouni , Anthony Martin , Khalid Bougrin et al.

New Journal of Chemistry, 2015, 39 (7), pp.5437-5444. ⟨10.1039/C5NJ00624D⟩

Article dans une revue hal-04599376v1

Resistance to sunitinib in renal clear cell carcinoma results from sequestration in lysosomes and inhibition of the autophagic flux

Sandy Giuliano , Yann Cormerais , Maeva Dufies , Renaud Grépin , Pascal Colosetti et al.

Autophagy, 2015, 11 (10), pp.1891-1904. ⟨10.1080/15548627.2015.1085742⟩

Article dans une revue hal-02108861v1

Direct Synthesis of Partially Modified 2′-O-Pivaloyloxymethyl RNAs by a Base-Labile Protecting Group Strategy and their Potential for Prodrug-Based Gene-Silencing Applications.

Annabelle Biscans , Maxence Bos , Anthony R. Martin , Nicholas Ader , Georg Sczakiel et al.

ChemBioChem, 2014, 15 (18), pp.2674-2679. ⟨10.1002/cbic.201402382⟩

Article dans une revue istex hal-01101605v1

[Au]/[Pd] Multicatalytic Processes: Direct One‐Pot Access to Benzo[ c ]chromenes and Benzo[ b ]furans

Yoshihiro Oonishi , Adrián Gómez-Suárez , Anthony Martin , Yusuke Makida , Alexandra Slawin et al.

Chemistry - A European Journal, 2014, 20 (42), pp.13507-13510. ⟨10.1002/chem.201404630⟩

Article dans une revue istex hal-04599364v1

Polyaldol Synthesis by Direct Organocatalyzed Crossed Polymerization of Bis(ketones) and Bis(aldehydes)

Na Liu , Anthony Martin , Frédéric Robert , Jean-Marc Vincent , Yannick Landais et al.

Macromolecules, 2014, 47 (2), pp.525-533. ⟨10.1021/ma402108y⟩

Article dans une revue hal-01366330v1

Organocatalyzed Step-Growth Polymerization through Desymmetrization of Cyclic Anhydrides: Synthesis of Chiral Polyesters

Anthony Martin , Frédéric Robert , Daniel Taton , Henri Cramail , Jean-Marc Vincent et al.

Chemistry - A European Journal, 2014, 20 (37), pp.11946-11953. ⟨10.1002/chem.201402373⟩

Article dans une revue istex hal-01366215v1

Efficient C–N and C–S Bond Formation Using the Highly Active [Ni(allyl)Cl(IPr* OMe )] Precatalyst

Anthony Martin , David Nelson , Sébastien Meiries , Alexandra Slawin , Steven Nolan

European Journal of Organic Chemistry, 2014, 2014 (15), pp.3127-3131. ⟨10.1002/ejoc.201402022⟩

Article dans une revue istex hal-04599359v1

Solvent-free aryl amination catalysed by [Pd(NHC)] complexes

Anthony Chartoire , Arnaud Boreux , Anthony Martin , Steven Nolan

RSC Advances, 2013, 3 (12), pp.3840. ⟨10.1039/c3ra40386f⟩

Article dans une revue hal-04599348v1

Boron and nucleic acid chemistries: merging the best of both worlds

Anthony R. Martin , Jean-Jacques Vasseur , Michael Smietana

Chemical Society Reviews, 2013, 42, pp.5684-5713. ⟨10.1039/c3cs60038f⟩

Article dans une revue hal-00833343v1

Enhanced Activity of [Ni(NHC)CpCl] Complexes in Arylamination Catalysis

Anthony Martin , Yusuke Makida , Sébastien Meiries , Alexandra Slawin , Steven Nolan

Organometallics, 2013, 32 (21), pp.6265-6270. ⟨10.1021/om4004863⟩

Article dans une revue hal-04599355v1

Hydrophenoxylation of Alkynes by Cooperative Gold Catalysis

Yoshihiro Oonishi , Adrián Gómez-Suárez , Anthony Martin , Steven Nolan

Angewandte Chemie International Edition, 2013, 52 (37), pp.9767-9771. ⟨10.1002/anie.201304182⟩

Article dans une revue istex hal-04599358v1

Straightforward synthesis of [Au(NHC)X] (NHC = N-heterocyclic carbene, X = Cl, Br, I) complexes

Alba Collado , Adrián Gómez-Suárez , Anthony Martin , Alexandra Slawin , Steven Nolan

Chemical Communications, 2013, 49 (49), pp.5541. ⟨10.1039/c3cc43076f⟩

Article dans une revue hal-04599349v1

Dynamic boronic acid-mediated autoligation of DNA strands

Michael Smietana , Anthony R. Martin , Jean-Jacques Vasseur

Pure and Applied Chemistry, 2012, 84 (7), pp.1659-1667. ⟨10.1351/PAC-CON-11-09-28⟩

Article dans une revue hal-00733354v1

Borononucleotides as Substrates/Binders for Human NMP Kinases: Enzymatic and Spectroscopic Evaluation

Chahrazade El Amri , Anthony R. Martin , Jean-Jacques Vasseur , Michael Smietana

ChemBioChem, 2012, 13, pp.1605-1612. ⟨10.1002/cbic.201200199⟩

Article dans une revue istex hal-00728768v1

Extending the utility of [Pd(NHC)(cinnamyl)Cl] precatalysts: Direct arylation of heterocycles

Anthony Martin , Anthony Chartoire , Alexandra Slawin , Steven Nolan

Beilstein Journal of Organic Chemistry, 2012, 8, pp.1637-1643. ⟨10.3762/bjoc.8.187⟩

Article dans une revue hal-04599339v1

Regioselective Synthesis of 3-Carbo-5-phosphonylpyrazoles through a One-Pot Claisen-Schmidt/1,3-Dipolar Cycloaddition/Oxidation Sequence

Anthony R. Martin , Kishor Mohanan , Loic Toupet , Jean-Jacques Vasseur , Michael Smietana

European Journal of Organic Chemistry, 2011, 2011 (17), pp.3184-3190. ⟨10.1002/ejoc.2011100167⟩

Article dans une revue hal-00616408v1

Dynamic and Programmable DNA-Templated Boronic Ester Formation

Anthony R. Martin , Ivan Barvik , Delphine Luvino , Michael Smietana , Jean-Jacques Vasseur

Angewandte Chemie International Edition, 2011, pp.4193-4196. ⟨10.1002/anie.201007170⟩

Article dans une revue istex hal-00623392v1

Three-Component Reaction Using the Bestmann-Ohira Reagent: A Regioselective Synthesis of Phosphonyl Pyrazole Rings

Kishor Mohanan , Anthony R Martin , Loic Toupet , Michael Smietana , Jean-Jacques Vasseur

Angewandte Chemie International Edition, 2010, 49 (18), pp.3196-3199. ⟨10.1002/anie.200906781⟩

Article dans une revue istex hal-00616443v1

Assessment of new 2'-O-acetalester protecting groups for regular RNA synthesis and original 2'-modified proRNA.

Anthony R. Martin , Thomas Lavergne , Jean-Jacques Vasseur , Françoise Debart

Bioorganic and Medicinal Chemistry Letters, 2009, 19, pp.4046-4049. ⟨10.1016/j.bmcl.2009.06.015⟩

Article dans une revue istex hal-00412360v1

Expanding the borononucleotide family: synthesis of borono-analogues of dCMP, dGMP and dAMP.

Anthony R. Martin , Kishor Mohanan , Delphine Luvino , Nicolas Floquet , Carine Baraguey et al.

Organic & Biomolecular Chemistry, 2009, 7 (21), pp.4369-4377. ⟨10.1039/b912616c⟩

Article dans une revue istex hal-01109915v1

A potent agonist-based PROTAC targeting Pregnane X Receptor that delays colon cancer relapse

Anthony R. Martin , Jean-Marc Pascussi

2nd workshop Chimie et Cancer, Cancéropôle Grand Sud-Ouest, Apr 2024, Toulouse, France

Communication dans un congrès hal-04847858v1

De la conception de potentialisateurs d’immunothérapies au développement d’outils fluorogéniques

Anthony R. Martin

Journée Jeunes Chercheur.e.s SCF-Occitanie Méditerranée, SCF-Occitanie Méditerranée - Pôle Chimie, Jul 2023, Montpellier, France

Communication dans un congrès hal-04847879v1