Bastien Michelet

41
Documents

Publications

Publications

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Activation of N-containing olefins and alkynes with superacids

Delphine Pichon-Barré , Hélène Carreyre , Frédéric Lecornué , Agnès Martin-Mingot , Bastien Michelet et al.
Comptes Rendus. Chimie, 2025, 28, pp.727-754. ⟨10.5802/crchim.416⟩
Article dans une revue (compte-rendu de lecture) hal-05321953 v1
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Regulating the Acidity of HF/Pyridine Media to Control the Chemodivergent Fluoro- and Hydro-Heteroalkylation of Olefins

Mélissa Longuet , Fabien Naullet , Alexandre Pérochon , Agnès Martin-Mingot , Frédéric Guégan et al.
Journal of the American Chemical Society, 2025, 147 (32), pp.29079-29087. ⟨10.1021/jacs.5c07526⟩
Article dans une revue hal-05221813 v1
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Benzophenone-Based Phenylogous Peptide Linkage via Friedel–Crafts Acylation

Hao Wu , Yuko Otani , Ying Zhou , Bastien Michelet , Sebastien Thibaudeau et al.
Organic Letters, In press, ⟨10.1021/acs.orglett.5c03833⟩
Article dans une revue hal-05321949 v1
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Superacid-Synthesized Fluorinated Diamines Act as Selective hCA IV Inhibitors

Emanuela Berrino , Bastien Michelet , Kassandra Vitse , Alessio Nocentini , Gianluca Bartolucci et al.
Journal of Medicinal Chemistry, 2024, ⟨10.1021/acs.jmedchem.4c01795⟩
Article dans une revue hal-04753033 v1
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Determination of the Hammett Acidity of HF/Base Reagents

Mélissa Longuet , Kassandra Vitse , Agnès Martin-Mingot , Bastien Michelet , Frédéric Guégan et al.
Journal of the American Chemical Society, 2024, ⟨10.1021/jacs.4c02344⟩
Article dans une revue (article de synthèse) hal-04552304 v1

Glycosylium Ions in Superacid Mimic the Transition State of Enzyme Reactions

Mathilde Armand , Alba Nin-Hill , Ana Ardá , Emanuela Berrino , Jérôme Désiré et al.
Journal of the American Chemical Society, 2024, 146 (47), pp.32618-32626. ⟨10.1021/jacs.4c11677⟩
Article dans une revue hal-05326476 v1
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Glycosylium Ions in Superacid Mimic the Transition State of Enzyme Reactions

Mathilde Armand , Alba Nin-Hill , Ana Ardá , Emanuela Berrino , Jérôme Désiré et al.
Journal of the American Chemical Society, 2024, 146 (47), pp.32618-32626. ⟨10.1021/jacs.4c11677⟩
Article dans une revue hal-05176253 v1
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Leveraging long-lived arenium ions in superacid for meta-selective methylation

Paul Bourbon , Kassandra Vitse , Agnès Martin-Mingot , Hugo Geindre , Frédéric Guégan et al.
Nature Communications, 2024, 15 (1), pp.7435. ⟨10.1038/s41467-024-49421-8⟩
Article dans une revue hal-04680872 v1
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Exploring Superacid‐Promoted Skeletal Reorganization of Aliphatic Nitrogen‐Containing Compounds

Maxime Artault , Thomas Cantin , Mélissa Longuet , Kassandra Vitse , Christ Daniel Matatu Mbengo et al.
Angewandte Chemie International Edition, 2023, 63 (1), pp.e202316458. ⟨10.1002/anie.202316458⟩
Article dans une revue hal-04520297 v1
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Enantioselective Organocatalysis and Superacid Activation: Challenges and Opportunities

Bastien Michelet , Agnès Martin-Mingot , Jean Rodriguez , Sébastien Thibaudeau , Damien Bonne
Chemistry - A European Journal, 2023, 29 (35), pp.e202300440. ⟨10.1002/chem.202300440⟩
Article dans une revue hal-04047011 v1
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Exploring F/CF3 substituted oxocarbenium ions for the diastereoselective assembly of highly substituted tetrahydrofurans

Anthony J Fernandes , Bastien Michelet , Armen Panossian , Agnès Martin-Mingot , Frédéric R Leroux et al.
Chemical Communications, 2023, 59 (27), pp.4083-4086. ⟨10.1039/d2cc06521e⟩
Article dans une revue hal-04046996 v1

A general synthesis of azetidines by copper-catalysed photoinduced anti-Baldwin radical cyclization of ynamides

Clément Jacob , Hajar Baguia , Amaury Dubart , Samuel Oger , Pierre Thilmany et al.
Nature Communications, 2022, 13 (1), pp.560. ⟨10.1038/s41467-022-28098-x⟩
Article dans une revue hal-03798007 v1
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Hidden Heptacyclic Chiral N-Acyl Iminium Ions: a New Entry to Enantioenriched Polycyclic Azepanes and Azocanes by Superacid-Promoted Intramolecular Pictet-Spengler Reaction

Yasmin Reviriot , Bastien Michelet , Rodolphe Beaud , Agnès Martin-Mingot , Frédéric Guégan et al.
Chemistry - A European Journal, 2022, 28 (25), pp.e202200432. ⟨10.1002/chem.202200432⟩
Article dans une revue hal-03769652 v1
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Superacid‐Mediated Late‐Stage Aromatic Polydeuteration of Pharmaceuticals

Emeline Appert , Agnès Martin-Mingot , Omar Karam , Fabien Zunino , Bastien Michelet et al.
Chemistry - A European Journal, 2022, 28 (49), pp.e202201583. ⟨10.1002/chem.202201583⟩
Article dans une revue hal-03769665 v1
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Formation of synthetically relevant CF3-substituted phenonium ions in superacid media

Anthony J Fernandes , Bastien Michelet , Armen Panossian , Agnès Martin-Mingot , Frédéric R. Leroux et al.
RSC Advances, 2021, 11 (41), pp.25695 - 25699. ⟨10.1039/d1ra04901a⟩
Article dans une revue hal-03325280 v1
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Complementary Site-Selective Sulfonylation of Aromatic Amines by Superacid Activation

Paul Bourbon , Emeline Appert , Agnès Martin-Mingot , Bastien Michelet , Sébastien Thibaudeau
Organic Letters, 2021, 23 (11), pp.4115-4120. ⟨10.1021/acs.orglett.1c00994⟩
Article dans une revue hal-03358394 v1
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CF3-substituted carbocations: underexploited intermediates with great potential in modern synthetic chemistry

Anthony J Fernandes , Armen Panossian , Bastien Michelet , Agnès Martin-Mingot , Frédéric Leroux et al.
Beilstein Journal of Organic Chemistry, 2021, 17, pp.343-378. ⟨10.3762/bjoc.17.32⟩
Article dans une revue hal-03154651 v1
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Insight into the Ferrier rearrangement by combining flash chemistry and superacids

Naresh Bhuma , Ludivine Lebedel , Hiroki Yamashita , Yutaka Shimizu , Zahra Abada et al.
Angewandte Chemie International Edition, 2021, 60 (4), pp.2036-2041. ⟨10.1002/anie.202010175⟩
Article dans une revue hal-03007376 v1
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Modulating the Efficacy of Carbonic Anhydrase Inhibitors through Fluorine Substitution

Emanuela Berrino , Bastien Michelet , Agnès Martin-Mingot , Fabrizio Carta , Claudiu T Supuran et al.
Angewandte Chemie International Edition, 2021, 60 (43), pp.23068-23082. ⟨10.1002/anie.202103211⟩
Article dans une revue hal-03358401 v1
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Enantioenriched Methylene-Bridged Benzazocanes Synthesis by Organocatalytic and Superacid Activations

Rodolphe Beaud , Bastien Michelet , Yasmin Reviriot , Agnès Martin-Mingot , Jean Rodriguez et al.
Angewandte Chemie International Edition, 2020, 59 (3), pp.1279-1285. ⟨10.1002/anie.201912043⟩
Article dans une revue hal-02436747 v1
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Access to Optically-Pure Benzosultams by Superelectrophilic Activation

Bastien Michelet , Ugo Castelli , Emeline Appert , Maude Boucher , Kassandra Vitse et al.
Organic Letters, 2020, 22 (13), pp.4944-4948. ⟨10.1021/acs.orglett.0c01301⟩
Article dans une revue hal-03016554 v1

[(DPEPhos)(bcp)Cu]PF<sub>6</sub>: A General and Broadly Applicable Copper-Based Photoredox Catalyst

Hajar Baguia , Christopher Deldaele , Bastien Michelet , Jérôme Beaudelot , Cédric Theunissen et al.
Journal of visualized experiments : JoVE, 2019, 147, ⟨10.3791/59739⟩
Article dans une revue hal-03007750 v1

Direct and Selective C-H Carbamoylation of (Hetero)aromatics with TMSOTf-Activated Carbamoyl Chloride

Ayaka Uehara , Sandra Olivero , Bastien Michelet , Agnès Martin-Mingot , Sébastien Thibaudeau et al.
European Journal of Organic Chemistry, 2019, 2019 (1), pp.46-49. ⟨10.1002/ejoc.201801338⟩
Article dans une revue hal-03007761 v1

Superelectrophilic activation in superacid HF/SbF5: Expanding molecular diversity in nitrogen-containing compounds series by fluorination

Bastien Michelet , Hélène Carreyre , Frédéric Lecornué , Agnès Mingot , Sébastien Thibaudeau
Journal of Fluorine Chemistry, 2018, 214, pp.68-79. ⟨10.1016/j.jfluchem.2018.04.017⟩
Article dans une revue hal-03007791 v1

Copper-Catalyzed Photoinduced Radical Domino Cyclization of Ynamides and Cyanamides: A Unified Entry to Rosettacin, Luotonin A, and Deoxyvasicinone

Hajar Baguia , Christopher Deldaele , Eugénie Romero , Bastien Michelet , Gwilherm Evano
Synthesis: Journal of Synthetic Organic Chemistry, 2018, 50 (15), pp.3022-3030. ⟨10.1055/s-0037-1610134⟩
Article dans une revue hal-03007805 v1

A General Copper-based Photoredox Catalyst for Organic Synthesis: Scope, Application in Natural Product Synthesis and Mechanistic Insights

Christopher Deldaele , Bastien Michelet , Hajar Baguia , Sofia Kajouj , Eugenie Romero et al.
CHIMIA, 2018, 72 (9), pp.621-629. ⟨10.2533/chimia.2018.621⟩
Article dans une revue hal-03007774 v1

A General Copper Catalyst for Photoredox Transformations of Organic Halides

Bastien Michelet , Christopher Deldaele , Sofia Kajouj , Cécile Moucheron , Gwilherm Evano
Organic Letters, 2017, 19 (13), pp.3576-3579. ⟨10.1021/acs.orglett.7b01518⟩
Article dans une revue hal-03007815 v1

The anionic chemistry of ynamides: A review

Gwilherm Evano , Bastien Michelet , Chunyang Zhang
Comptes Rendus. Chimie, 2017, 20 (6), pp.648-664. ⟨10.1016/j.crci.2016.12.002⟩
Article dans une revue hal-03007821 v1

Catalytic Activity of Gold(I) Complexes with Hemilabile P,N Ligands

Bastien Michelet , David Lebœuf , Christophe Bour , Karel Škoch , Filip Horký et al.
ChemPlusChem, 2017, 82 (3), pp.442-448. ⟨10.1002/cplu.201600562⟩
Article dans une revue hal-03007828 v1

Catalytic applications of [IPr·GaX 2 ][SbF 6 ] and related species

Bastien Michelet , Shun Tang , Guillaume Thiery , Julien Monot , Huijing Li et al.
Organic Chemistry Frontiers, 2016, 3 (12), pp.1603-1613. ⟨10.1039/C6QO00470A⟩
Article dans une revue hal-03007837 v1

A Journey in the Chemistry of Ynamides: From Synthesis to Applications

Gwilherm Evano , Nicolas Blanchard , Guillaume Compain , Alexis Coste , Charles Demmer et al.
Chemistry Letters, 2016, 45 (6), pp.574-585. ⟨10.1246/cl.160260⟩
Article dans une revue hal-03007853 v1

Harnessing the Lewis Acidity of HFIP through its Cooperation with a Calcium(II) Salt: Application to the Aza-Piancatelli Reaction

David Lebøeuf , Lucile Marin , Bastien Michelet , Alejandro Perez-Luna , Régis Guillot et al.
Chemistry - A European Journal, 2016, 22 (45), pp.16165--16171. ⟨10.1002/chem.201603592⟩
Article dans une revue istex hal-01712359 v1

Non-Innocent Behavior of Substrate Backbone Esters in Metal-Catalyzed Carbocyclizations and Friedel–Crafts Reactions of Enynes and Arenynes

Bastien Michelet , Guillaume Thiery , Christophe Bour , Vincent Gandon
Journal of Organic Chemistry, 2015, 80 (21), pp.10925-10938. ⟨10.1021/acs.joc.5b02052⟩
Article dans une revue hal-03007863 v1
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Dibromoindium( iii ) cations as a π-Lewis acid: characterization of [IPr·InBr 2 ][SbF 6 ] and its catalytic activity towards alkynes and alkenes

Bastien Michelet , Jean-Rémy Colard-Itté , Guillaume Thiery , Régis Guillot , Christophe Bour et al.
Chemical Communications, 2015, 51 (34), pp.7401-7404. ⟨10.1039/C5CC00740B⟩
Article dans une revue hal-03007870 v1

Ca II -Catalyzed Alkenylation of Alcohols with Vinylboronic Acids

David Lebœuf , Marc Presset , Bastien Michelet , Christophe Bour , Sophie Bezzenine-Lafollée et al.
Chemistry - A European Journal, 2015, 21 (31), pp.11001-11005. ⟨10.1002/chem.201501677⟩
Article dans une revue istex hal-03007865 v1

Gallium-Assisted Transfer Hydrogenation of Alkenes

Bastien Michelet , Christophe Bour , Vincent Gandon
Chemistry - A European Journal, 2014, 20 (44), pp.14488-14492. ⟨10.1002/chem.201404139⟩
Article dans une revue istex hal-03007877 v1

Cationic Gallium(III) Halide Complexes: A New Generation of π-Lewis Acids

Shun Tang , Julien Monot , Ahmad El-Hellani , Bastien Michelet , Régis Guillot et al.
Chemistry - A European Journal, 2012, 18 (33), pp.10239-10243. ⟨10.1002/chem.201201202⟩
Article dans une revue istex hal-03007906 v1

Four-Membered Rings With Two Nitrogen Atoms

Frédéric Lecornué , Bastien Michelet
David StC Black; Janine Cossy; Christian V. Stevens. Comprehensive Heterocyclic Chemistry IV, Volume 2: Four-membered Heterocycles, and all Fused Systems with a Four-membered Heterocyclic Ring, 2, Elsevier, pp.403-457, 2022, 978-0-12-818656-5. ⟨10.1016/B978-0-12-818655-8.00153-0⟩
Chapitre d'ouvrage hal-03363494 v1

Gallium Trichloride

Masahiko Yamaguchi , Shigeki Matsunaga , Masakatsu Shibasaki , Bastien Michelet , Christophe Bour et al.
Encyclopedia of Reagents for Organic Synthesis, John Wiley & Sons, Ltd, 2014, ⟨10.1002/047084289X.rn00118u.pub3⟩
Chapitre d'ouvrage hal-03007900 v1