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Fluorescent Antimicrobial Peptides Based on Nile Red: Effect of Conjugation Site and Chemistry on Wash-Free Staining of Bacteria
Lucille Weiss
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Acute, chronic and conditioned effects of intranasal oxytocin in the mu-opioid receptor knockout mouse model of autism: Social context matters
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The IMS Library: from IN‐Stock to Virtual
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Biased activation of the vasopressin V2 receptor probed by NMR, paramagnetic ligands, and molecular dynamics simulations
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Alared: Solvatochromic and Fluorogenic Red Amino Acid for Ratiometric Live‐cell Imaging of Bioactive Peptides
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Article dans une revue
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Fluorinated apelin-13 mediates neuroprotective effects in multiple sclerosis models
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Rational Design of Cyanine-Based Fluorogenic Dimers to Reduce Nonspecific Interactions with Albumin and Lipid Bilayers: Application to Highly Sensitive Imaging of GPCRs in Living Cells
Yann Berthomé
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Article dans une revue
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Hetero-Diels–Alder and CuAAC Click Reactions for Fluorine-18 Labeling of Peptides: Automation and Comparative Study of the Two Methods
Timothé Maujean
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Catalyst-free thia-Diels-Alder click reaction for the labeling of peptides for imaging applications
Timothé Maujean
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Rapid and Highly Selective Fluorescent Labeling of Peptides via a Thia-Diels–Alder Cycloaddition: Application to Apelin
Timothé Maujean
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Christel Valencia
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Article dans une revue
hal-04075152
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Hetero-Diels–Alder click reaction of dithioesters for a catalyst-free indirect 18 F-radiolabelling of peptides
Timothé Maujean
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Stephanie Riché
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Frédéric Boisson
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Article dans une revue
hal-03780966
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Functional Rescue of a Nephrogenic Diabetes Insipidus Causing Mutation in the V2 Vasopressin Receptor by Specific Antagonist and Agonist Pharmacochaperones
Laura Szalai
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András Sziráki
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László Sándor Erdélyi
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Kinga Bernadett Kovács
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hal-03827827
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Activating the apelin receptor with LIT01-196, a metabolically stable apelin analog, reverses AVP-induced antidiuresis and hyponatremia
Adrien Flahault
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Mathilde Keck
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Rodrigo Alvear-Perez
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LIT01-196, a Metabolically Stable Apelin-17 Analog, Normalizes Blood Pressure in Hypertensive DOCA-Salt Rats via a NO Synthase-dependent Mechanism
Adrien Flahault
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Mathilde Keck
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Pierre-Emmanuel Girault-Sotias
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Lucie Esteoulle
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A Selective Neutraligand for CXCL12/SDF-1α With Beneficial Regulatory Functions in MRL/Lpr Lupus Prone Mice
Nicolas Schall
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Nile Red-Based GPCR Ligands as Ultrasensitive Probes of the Local Lipid Microenvironment of the Receptor
Fabien Hanser
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Christel Valencia
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Pascal Villa
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The EHA Research Roadmap: Normal Hematopoiesis
Thierry Jaffredo
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Article dans une revue
hal-03463225
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Three Cheers for Nitrogen: Aza-DKPs, the Aza Analogues of 2,5-Diketopiperazines
Timothé Maujean
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Nicolas Girard
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A. Ganesan
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Mihaela Gulea
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Dominique Bonnet
Article dans une revue
hal-03441420
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Pharmacological tools to mobilize mesenchymal stromal cells into the blood promote bone formation after surgery
Tariq G Fellous
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Article dans une revue
hal-03012479
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Self‐organization Properties of a GPCR‐Binding Peptide with a Fluorinated Tail Studied by Fluorine NMR Spectroscopy
Capucine Jourdain de Muison
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Sridevi M. Ramanoudjame
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Lucie Esteoulle
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Claude Ling
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Germain Brou
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Article dans une revue
hal-03090942
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Endocyclic Enamides Derived from Aza‐Diketopiperazines as Olefin Partners in Povarov Reaction: An Access to Tetracyclic N‐Heterocycles
Timothé Maujean
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Isabelle Chataigner
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Nicolas Girard
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Mihaela Gulea
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Dominique Bonnet
Article dans une revue
hal-03441064
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A near-infrared fluorogenic dimer enables background-free imaging of endogenous GPCRs in living mice
Lucie Esteoulle
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Francois Daubeuf
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Stéphanie Riché
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Article dans une revue
hal-02922372
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Neutralization of CXCL12 attenuates established pulmonary hypertension in rats Short Title: CXCL12 neutraligands in severe PH in the rat
Jennifer Bordenave
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Ly Tu
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Article dans une revue
hal-02195697
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LIT-001, the First Nonpeptide Oxytocin Receptor Agonist that Improves Social Interaction in a Mouse Model of Autism
Marie-Céline Frantz
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Lucie P. Pellissier
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Elsa Pflimlin
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Stéphanie Loison
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Jorge Gandía
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Article dans une revue
hal-02366272
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Versatile synthetic approach for selective diversification of bicyclic aza-diketopiperazines
Florent Péron
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Philippe Breton
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Article dans une revue
hal-02366261
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Discovery of a Locally and Orally Active CXCL12 Neutraligand (LIT-927) with Anti-inflammatory Effect in a Murine Model of Allergic Airway Hypereosinophilia
Pierre Regenass
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Dayana Abboud
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François Daubeuf
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Christine Lehalle
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Patrick Gizzi
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Article dans une revue
hal-03563473
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Decreased Migration of Dendritic Cells into the Jugular-Nodose Ganglia by the CXCL12 Neutraligand Chalcone 4 in Ovalbumin-Sensitized Asthmatic Mice
Sebastian Heck
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Francois Daubeuf
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Duc dung Le
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Martina Sester
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Dominique Bonnet
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Article dans une revue
hal-02366307
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A Time-Resolved FRET Cell-Based Binding Assay for the Apelin Receptor
Christel Valencia
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Céline Dujet
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Jean-François Margathe
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Article dans une revue
hal-02153692
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From the Promiscuous Asenapine to Potent Fluorescent Ligands Acting at a Series of Aminergic G-Protein-Coupled Receptors
Candide Hounsou
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Corinne Baehr
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Vincent Gasparik
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Doria Alili
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Article dans une revue
hal-02366277
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Comparative Study of the Synthesis and Structural and Physicochemical Properties of Diketopiperazines vs Aza-diketopiperazines
Pierre Regenass
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Stéphanie Riché
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Patrick Gizzi
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Marcel Hibert
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Article dans une revue
hal-02366265
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Two distinct CXCR4 antagonists mobilize progenitor cells in mice by different mechanisms
Andia Redpath
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Moïra François
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Suet-Ping Wong
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Dominique Bonnet
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Sara Rankin
Article dans une revue
hal-02366286
v1
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Comparative Study of the Synthesis and Structural and Physicochemical Properties of Diketopiperazines vs Aza-diketopiperazines
Pierre Regenass
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Damien Bosc
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Stéphanie Riché
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Patrick Gizzi
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Marcel Hibert
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Article dans une revue
hal-03563479
v1
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Convenient Access to Fluorescent Probes by Chemoselective Acylation of Hydrazinopeptides: Application to the Synthesis of the First Far-Red Ligand for Apelin Receptor Imaging
Jean-François Margathe
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Xavier Iturrioz
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Pierre Regenass
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Iuliia Karpenko
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Nicolas Humbert
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Article dans une revue
istex
hal-02153700
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A step-economical multicomponent synthesis of 3D-shaped aza-diketopiperazines and their drug-like chemical space analysis
Pierre-Michel Regenass
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Stéphanie Riché
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Florent Péron
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Didier Rognan
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Marcel Hibert
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Article dans une revue
hal-04684621
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Push-pull dioxaborine as fluorescent molecular rotor: far-red fluorogenic probe for ligand-receptor interactions
Iuliia Karpenko
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Yosuke Niko
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Viktor P. Yakubovskyi
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Andriy O. Gerasov
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Dominique Bonnet
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Article dans une revue
hal-03536470
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New fluorescein precursors for live bacteria detection
Célia Guilini
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Corinne Baehr
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Etienne Schaeffer
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Patrick Gizzi
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Frédéric Rufi
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Article dans une revue
hal-02196002
v1
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Time-resolved FRET binding assay to investigate hetero-oligomer binding properties: proof of concept with dopamine D1/D3 heterodimer
Candide Hounsou
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Jean-François Margathe
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Nadia Oueslati
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Abderazak Belhocine
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Elodie Dupuis
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Article dans une revue
hal-01950133
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A strategy to discover decoy chemokine ligands with an anti-inflammatory activity
Dayana Abboud
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Francois Daubeuf
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Quoc Tuan Do
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Valérie Utard
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Pascal Villa
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Article dans une revue
hal-02193983
v1
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Identification of CCL17 neutraligands targeting atopic diseases
Dayana Abboud
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Francois Daubeuf
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V Utard
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Dominique Bonnet
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Marcel Hibert
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Article dans une revue
hal-05051746
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Structure–Activity Relationship Studies toward the Discovery of Selective Apelin Receptor Agonists
Jean-François Margathe
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Xavier Iturrioz
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Rodrigo Alvear-Perez
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Claire Marsol
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Stéphanie Riché
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Article dans une revue
hal-02153719
v1
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Diastereoselective Synthesis of Novel Aza-diketopiperazines via a Domino Cyclohydrocarbonylation/Addition Process
Pierre-Michel Regenass
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Jean Francois Margathe
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Andre Mann
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Jean Suffert
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Marcel Hibert
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Article dans une revue
hal-04679522
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Un neutraligand de la chimiokine CXCL12 inhibe la fibroprolifération dans un modèle de bronchiolite oblitérante après transplantation hétérotopique de trachée chez la souris
Simona Nemska
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Clément Ammouche
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François Daubeuf
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Dominique Bonnet
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Marcel Hibert
et al.
Article dans une revue
hal-05015140
v1
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An Antedrug of the CXCL12 Neutraligand Blocks Experimental Allergic Asthma without Systemic Effect in Mice
Francois Daubeuf
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Muriel Hachet-Haas
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Patrick Gizzi
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Vincent Gasparik
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Dominique Bonnet
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Article dans une revue
hal-02194500
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Exploration of the Orthosteric/Allosteric Interface in Human M1 Muscarinic Receptors by Bitopic Fluorescent Ligands
Sandrine B Daval
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Esther Kellenberger
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Dominique Bonnet
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Valérie Utard
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Jean-Luc Galzi
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Article dans une revue
hal-02193988
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Involvement of the TGFβ pathway in the regulation of α5 β1 integrins by caveolin-1 in human glioblastoma.
Erika C Cosset
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Julien Godet
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Natacha Entz-Werlé
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Eric Guérin
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Dominique Guenot
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Article dans une revue
istex
hal-00746869
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Selective Fluorescent Nonpeptidic Antagonists For Vasopressin V 2 GPCR: Application To Ligand Screening and Oligomerization Assays
Stéphanie Loison
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Martin Cottet
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Hélène Orcel
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Hélène Adihou
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Rita Rahmeh
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Article dans une revue
hal-04584099
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Fluorescent Derivatives of AC-42 To Probe Bitopic Orthosteric/Allosteric Binding Mechanisms on Muscarinic M1 Receptors
Sandrine B Daval
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Céline Valant
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Dominique Bonnet
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Esther Kellenberger
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Marcel Hibert
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Article dans une revue
hal-02193850
v1
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Les neutraligands à l'assaut des chimiokines
Muriel Hachet-Haas
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Dominique Bonnet
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Francois Daubeuf
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Marcel Hibert
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Jacques Haiech
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Biofutur, 2011, 319, pp.52-55
Article dans une revue
hal-02196019
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Prodrugs of a CXC Chemokine-12 (CXCL12) Neutraligand Prevent Inflammatory Reactions in an Asthma Model in Vivo
Vincent Gasparik
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François Daubeuf
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Muriel Hachet-Haas
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François Rohmer
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Patrick Gizzi
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Article dans une revue
hal-04748151
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Identification and pharmacological properties of E339–3D6, the first nonpeptidic apelin receptor agonist
Xavier Itturioz
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Rodrigo Alvear-Perez
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Nadia de Mota
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Christel Franchet
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Fabrice Guillier
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Article dans une revue
hal-02196074
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Homodimerization of the death-associated protein kinase catalytic domain: development of a new small molecule fluorescent reporter
Michael Zimmermann
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Cédric Atmanene
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Qingyan Xu
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Laetitia Fouillen
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Alain van Dorsselaer
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Article dans une revue
hal-04593556
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Neutralizing endogenous chemokines with small molecules : principles and potential therapeutic applications
Jean-Luc Galzi
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Muriel Hachet-Haas
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Dominique Bonnet
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Francois Daubeuf
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Sandra Lecat
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Article dans une revue
hal-02196582
v1
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Biased agonist pharmacochaperones of the AVP V2 receptor may treat congenital nephrogenic diabetes insipidus.
Frédéric Jean-Alphonse
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Sanja Perkovska
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Marie-Céline Frantz
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Thierry Durroux
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Catherine Méjean
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Article dans une revue
inserm-00421838
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Small Neutralizing Molecules to Inhibit Actions of the Chemokine CXCL12.
Muriel Hachet-Haas
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Karl Balabanian
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François Rohmer
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Françoise Pons
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Christel Franchet
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Article dans une revue
pasteur-00315588
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A Rapid and Versatile Method to Label Receptor Ligands Using “Click” Chemistry: Validation with the Muscarinic M1 Antagonist Pirenzepine
Dominique Bonnet
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Brigitte Ilien
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Jean-Luc Galzi
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Stéphanie Riché
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Cyril Antheaune
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Article dans une revue
istex
hal-02938550
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Effect of Glycoamphiphiles on the Solubilization and Dendritic Cell Uptake of a Lipopeptide: A Preliminary Study
Dominique Bonnet
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Gerhild Angyalosi
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Alexandra Demory
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Valérie Santraine
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Arnaud Boulet
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Article dans une revue
hal-02196957
v1
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Efficient preparation of carbohydrate- and related polyol-amphiphiles by hydrazone ligation
Cyrille Grandjean
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Valérie Santraine
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Nathalie Fardel
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Ange Polidori
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Bernard Pucci
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Article dans une revue
istex
hal-02197015
v1
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Solid-Phase Functionalization of Peptides by an α-Hydrazinoacetyl Group
Dominique Bonnet
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Cyrille Grandjean
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Pierre Rousselot-Pailley
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Pascal Joly
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Line Bonnet
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Article dans une revue
istex
hal-02196953
v1
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The tetrapeptide acserasplyspro (seraspenide), a hematopoietic inhibitor, may reduce the in vitro toxicity of 3'-deoxythymidine to human hematopoietic progenitors
Catherine Grillon
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Dominique Bonnet
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Jean‐Yves Mary
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Maryse Lenfant
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Albert Najman
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Article dans une revue
hal-02114633
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La reconstitution d'une forêt de protection : vers une nouvelle image des forêts des Alpes sèches
Dominique Bonnet
Article dans une revue
hal-03423749
v1
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