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Synthesis and Photochemical Properties of Fluorescent Metabolites Generated from Fluorinated Benzoylmenadiones in Living Cells
Nathan Trometer
,
Bogdan Cichocki
,
Quentin Chevalier
,
Jérémy Pécourneau
,
Jean-Marc Strub
Article dans une revue
hal-04157610v1
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Efficient Multigram-Scale Synthesis of 7-Substituted 3-Methyltetral-1-ones and 6-Fluoromenadione
Nathan Trometer
,
Matthieu Roignant
,
Elisabeth Davioud-Charvet
Article dans une revue
hal-03584209v1
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Evaluation of ferrocenyl-containing γ-hydroxy-γ-lactam-derived tetramates as potential antiplasmodials
Nicolas Chopin
,
Julien Bosson
,
Shinya Iikawa
,
Stéphane Picot
,
Anne-Lise Bienvenu
Article dans une revue
hal-03798632v1
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The parasitophorous vacuole nutrient channel is critical for drug access in malaria parasites and modulates the artemisinin resistance fitness cost
Paolo Mesén-Ramírez
,
Bärbel Bergmann
,
Mourad Elhabiri
,
Lei Zhu
,
Heidrun von Thien
Article dans une revue
hal-03544974v1
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Plasmodium falciparum Ferredoxin-NADP + Reductase-Catalyzed Redox Cycling of Plasmodione Generates Both Predicted Key Drug Metabolites: Implication for Antimalarial Drug Development
Bogdan Cichocki
,
Maxime Donzel
,
Kim C. Heimsch
,
Mindaugas Lesanavičius
,
Liwen Feng
Article dans une revue
hal-03243991v1
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A Class of Valuable (Pro-)Activity-Based Protein Profiling Probes: Application to the Redox-Active Antiplasmodial Agent, Plasmodione
Bogdan Cichocki
,
Vrushali Khobragade
,
Maxime Donzel
,
Leandro Cotos Munoz
,
Stephanie Blandin
Article dans une revue
hal-03243960v1
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Recent Advances in Direct C‐H Radical Alkylation of 1,4‐Quinones
Maxime Donzel
,
Deniz Karabiyikli
,
Leandro Cotos Munoz
,
Mourad Elhabiri
,
Elisabeth Davioud-Charvet
Article dans une revue
hal-03249134v1
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Magnesium Complexes of Ladanein: A Beneficial Strategy for Stabilizing Polyphenolic Antivirals
Xavier Martin‐benlloch
,
Don Antoine Lanfranchi
,
Sibylle Haid
,
Thomas Pietschmann
,
Elisabeth Davioud‐charvet
Article dans une revue
hal-03357249v1
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Repurposing Auranofin and Evaluation of a New Gold(I) Compound for the Search of Treatment of Human and Cattle Parasitic Diseases: From Protozoa to Helminth Infections
Liwen Feng
,
Sébastien Pomel
,
Perle Latre de Late
,
Alexandre Taravaud
,
Philippe M Loiseau
Article dans une revue
hal-03038691v1
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Antiplasmodial Activity of Nitroaromatic Compounds: Correlation with Their Reduction Potential and Inhibitory Action on Plasmodium falciparum Glutathione Reductase
Audronė Marozienė
,
Mindaugas Lesanavičius
,
Elisabeth Davioud-Charvet
,
Alessandro Aliverti
,
Philippe Grellier
Article dans une revue
hal-03038823v1
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Physicochemical Properties Govern the Activity of Potent Antiviral Flavones
Xavier Martin-Benlloch
,
Sibylle Haid
,
Alexandra Novodomska
,
Frank Rominger
,
Thomas Pietschmann
Article dans une revue
hal-02325555v1
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Investigating the mode of action of the redox-active antimalarial drug plasmodione using the yeast model
Pierre Mounkoro
,
Thomas Michel
,
Stéphanie Blandin
,
Marie-Pierre Golinelli-Cohen
,
Elisabeth Davioud-Charvet
Article dans une revue
hal-02170571v1
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AntiMalarial Mode of Action (AMMA) Database: Data Selection, Verification and Chemical Space Analysis
Pavel Sidorov
,
Elisabeth Davioud-Charvet
,
Gilles Marcou
,
Dragos Horvath
,
Alexandre Varnek
Article dans une revue
hal-02325960v1
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A Redox-Active Fluorescent pH Indicator for Detecting Plasmodium falciparum Strains with Reduced Responsiveness to Quinoline Antimalarial Drugs
Mouhamad Jida
,
Cecilia Sanchez
,
Karène Urgin
,
Katharina Ehrhardt
,
S Mounien
Article dans une revue
hal-02177403v1
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Arylmethylamino steroids as novel antiparasitic agents
R Krieg
,
E Jortzik
,
Alice-Anne Goetz
,
Stephanie Blandin
,
S Wittlin
Article dans une revue
hal-02158243v1
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A high susceptibility to redox imbalance of the transmissible stages of Plasmodium falciparum revealed with a luciferase-based mature gametocyte assay
G Siciliano
,
T Kumar
,
R Bona
,
G Camarda
,
M Calabretta
Article dans une revue
hal-02161655v1
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QSAR modeling1. and chemical space analysis of antimalarial compounds
Pavel Sidorov
,
B Viira
,
Elisabeth Davioud-Charvet
,
U Maran
,
Gilles Marcou
Article dans une revue
hal-02177404v1
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Pharmacomodulation of the antimalarial plasmodione: synthesis of biaryl- and N-arylalkylamine analogues, antimalarial activities and physicochemical properties
Karène Urgin
,
Mouhamad Jida
,
Katharina Ehrhardt
,
T Müller
,
M Lanzer
Article dans une revue
hal-02177398v1
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Redox Polypharmacology as an Emerging Strategy to Combat Malarial Parasites
Pavel Sidorov
,
Israel Desta
,
Matthieu Chessé
,
Dragos Horvath
,
Gilles Marcou
Article dans une revue
hal-03151671v1
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The Redox Cycler Plasmodione Is a Fast-Acting Antimalarial Lead Compound with Pronounced Activity against Sexual and Early Asexual Blood-Stage Parasites
Katharina Ehrhardt
,
Christiane Deregnaucourt
,
Alice-Anne Goetz
,
Tzvetomira Tzanova
,
Valentina Gallo
Article dans une revue
hal-01455775v1
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A Platform of Regioselective Methodologies to Access to Polysubstituted 2-Methyl-1,4-Naphthoquinones Derivatives: Scope and Limitations
Elena Cesar Rodo
,
Liwen Feng
,
Mouhamad Jida
,
Katharina Ehrhardt
,
Max Bielitza
Article dans une revue
hal-03537379v1
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In Silico Mining for Antimalarial Structure-Activity Knowledge and Discovery of Novel Antimalarial Curcuminoids
Birgit Viira
,
Thibault Gendron
,
Don Antoine Lanfranchi
,
Sandrine Cojean
,
Dragos Horvath
Article dans une revue
hal-03150675v1
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