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Elisabeth Davioud-Charvet

22
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Publications

38052
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Synthesis and Photochemical Properties of Fluorescent Metabolites Generated from Fluorinated Benzoylmenadiones in Living Cells

Nathan Trometer , Bogdan Cichocki , Quentin Chevalier , Jérémy Pécourneau , Jean-Marc Strub
Journal of Organic Chemistry, 2023, ⟨10.1021/acs.joc.3c00620⟩
Article dans une revue hal-04157610v1
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Efficient Multigram-Scale Synthesis of 7-Substituted 3-Methyltetral-1-ones and 6-Fluoromenadione

Nathan Trometer , Matthieu Roignant , Elisabeth Davioud-Charvet
Organic Process Research and Development, 2022, acs.oprd.1c00421. ⟨10.1021/acs.oprd.1c00421⟩
Article dans une revue hal-03584209v1
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Evaluation of ferrocenyl-containing γ-hydroxy-γ-lactam-derived tetramates as potential antiplasmodials

Nicolas Chopin , Julien Bosson , Shinya Iikawa , Stéphane Picot , Anne-Lise Bienvenu
European Journal of Medicinal Chemistry, 2022, 243, pp.114735. ⟨10.1016/j.ejmech.2022.114735⟩
Article dans une revue hal-03798632v1
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The parasitophorous vacuole nutrient channel is critical for drug access in malaria parasites and modulates the artemisinin resistance fitness cost

Paolo Mesén-Ramírez , Bärbel Bergmann , Mourad Elhabiri , Lei Zhu , Heidrun von Thien
Cell Host & Microbe, 2021, 29 (12), pp.1774-1787.e9. ⟨10.1016/j.chom.2021.11.002⟩
Article dans une revue hal-03544974v1
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Plasmodium falciparum Ferredoxin-NADP + Reductase-Catalyzed Redox Cycling of Plasmodione Generates Both Predicted Key Drug Metabolites: Implication for Antimalarial Drug Development

Bogdan Cichocki , Maxime Donzel , Kim C. Heimsch , Mindaugas Lesanavičius , Liwen Feng
ACS Infectious Diseases, inPress, ⟨10.1021/acsinfecdis.1c00054⟩
Article dans une revue hal-03243991v1
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A Class of Valuable (Pro-)Activity-Based Protein Profiling Probes: Application to the Redox-Active Antiplasmodial Agent, Plasmodione

Bogdan Cichocki , Vrushali Khobragade , Maxime Donzel , Leandro Cotos Munoz , Stephanie Blandin
JACS Au, 2021, 1 (5), pp.669-689. ⟨10.1021/jacsau.1c00025⟩
Article dans une revue hal-03243960v1
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Recent Advances in Direct C‐H Radical Alkylation of 1,4‐Quinones

Maxime Donzel , Deniz Karabiyikli , Leandro Cotos Munoz , Mourad Elhabiri , Elisabeth Davioud-Charvet
European Journal of Organic Chemistry, 2021, 2021 (25), pp.3622-3633. ⟨10.1002/ejoc.202100452⟩
Article dans une revue hal-03249134v1
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Magnesium Complexes of Ladanein: A Beneficial Strategy for Stabilizing Polyphenolic Antivirals

Xavier Martin‐benlloch , Don Antoine Lanfranchi , Sibylle Haid , Thomas Pietschmann , Elisabeth Davioud‐charvet
European Journal of Inorganic Chemistry, 2021, 2021 (27), pp.2764-2772. ⟨10.1002/ejic.202100341⟩
Article dans une revue hal-03357249v1
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Repurposing Auranofin and Evaluation of a New Gold(I) Compound for the Search of Treatment of Human and Cattle Parasitic Diseases: From Protozoa to Helminth Infections

Liwen Feng , Sébastien Pomel , Perle Latre de Late , Alexandre Taravaud , Philippe M Loiseau
Molecules, 2020, 25 (21), pp.5075. ⟨10.3390/molecules25215075⟩
Article dans une revue hal-03038691v1
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Antiplasmodial Activity of Nitroaromatic Compounds: Correlation with Their Reduction Potential and Inhibitory Action on Plasmodium falciparum Glutathione Reductase

Audronė Marozienė , Mindaugas Lesanavičius , Elisabeth Davioud-Charvet , Alessandro Aliverti , Philippe Grellier
Molecules, 2019, 24 (24), pp.4509. ⟨10.3390/molecules24244509⟩
Article dans une revue hal-03038823v1

Physicochemical Properties Govern the Activity of Potent Antiviral Flavones

Xavier Martin-Benlloch , Sibylle Haid , Alexandra Novodomska , Frank Rominger , Thomas Pietschmann
ACS Omega, 2019, 4 (3), pp.4871-4887. ⟨10.1021/acsomega.8b03332⟩
Article dans une revue hal-02325555v1
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Investigating the mode of action of the redox-active antimalarial drug plasmodione using the yeast model

Pierre Mounkoro , Thomas Michel , Stéphanie Blandin , Marie-Pierre Golinelli-Cohen , Elisabeth Davioud-Charvet
Free Radical Biology and Medicine, 2019, 141, pp.269-278. ⟨10.1016/j.freeradbiomed.2019.06.026⟩
Article dans une revue hal-02170571v1

AntiMalarial Mode of Action (AMMA) Database: Data Selection, Verification and Chemical Space Analysis

Pavel Sidorov , Elisabeth Davioud-Charvet , Gilles Marcou , Dragos Horvath , Alexandre Varnek
Molecular Informatics, 2018, 37 (9-10), pp.1800021. ⟨10.1002/minf.201800021⟩
Article dans une revue hal-02325960v1

A Redox-Active Fluorescent pH Indicator for Detecting Plasmodium falciparum Strains with Reduced Responsiveness to Quinoline Antimalarial Drugs

Mouhamad Jida , Cecilia Sanchez , Karène Urgin , Katharina Ehrhardt , S Mounien
ACS Infectious Diseases, 2017, 3, pp.119-131. ⟨10.1021/acsinfecdis.5b00141⟩
Article dans une revue hal-02177403v1

Arylmethylamino steroids as novel antiparasitic agents

R Krieg , E Jortzik , Alice-Anne Goetz , Stephanie Blandin , S Wittlin
Nature Communications, 2017, 8, ⟨10.1038/ncomms14478⟩
Article dans une revue hal-02158243v1

A high susceptibility to redox imbalance of the transmissible stages of Plasmodium falciparum revealed with a luciferase-based mature gametocyte assay

G Siciliano , T Kumar , R Bona , G Camarda , M Calabretta
Molecular Microbiology, 2017, 104, pp.306-318. ⟨10.1111/mmi.13626⟩
Article dans une revue hal-02161655v1

QSAR modeling1. and chemical space analysis of antimalarial compounds

Pavel Sidorov , B Viira , Elisabeth Davioud-Charvet , U Maran , Gilles Marcou
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 2017, 31, pp.441-451. ⟨10.1007/s10822-017-0019-4⟩
Article dans une revue hal-02177404v1

Pharmacomodulation of the antimalarial plasmodione: synthesis of biaryl- and N-arylalkylamine analogues, antimalarial activities and physicochemical properties

Karène Urgin , Mouhamad Jida , Katharina Ehrhardt , T Müller , M Lanzer
Molecules, 2017, 22, pp.1-32. ⟨10.3390/molecules22010161⟩
Article dans une revue hal-02177398v1

Redox Polypharmacology as an Emerging Strategy to Combat Malarial Parasites

Pavel Sidorov , Israel Desta , Matthieu Chessé , Dragos Horvath , Gilles Marcou
ChemMedChem, 2016, 11 (12), pp.1339-1351. ⟨10.1002/cmdc.201600009⟩
Article dans une revue hal-03151671v1

The Redox Cycler Plasmodione Is a Fast-Acting Antimalarial Lead Compound with Pronounced Activity against Sexual and Early Asexual Blood-Stage Parasites

Katharina Ehrhardt , Christiane Deregnaucourt , Alice-Anne Goetz , Tzvetomira Tzanova , Valentina Gallo
Antimicrobial Agents and Chemotherapy, 2016, 60 (9), pp.5146-5158. ⟨10.1128/AAC.02975-15⟩
Article dans une revue hal-01455775v1
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A Platform of Regioselective Methodologies to Access to Polysubstituted 2-Methyl-1,4-Naphthoquinones Derivatives: Scope and Limitations

Elena Cesar Rodo , Liwen Feng , Mouhamad Jida , Katharina Ehrhardt , Max Bielitza
European Journal of Organic Chemistry, 2016, 2016 (11), pp.1982-1993. ⟨10.1002/ejoc.201600144⟩
Article dans une revue hal-03537379v1
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In Silico Mining for Antimalarial Structure-Activity Knowledge and Discovery of Novel Antimalarial Curcuminoids

Birgit Viira , Thibault Gendron , Don Antoine Lanfranchi , Sandrine Cojean , Dragos Horvath
Molecules, 2016, 21 (7), pp.853. ⟨10.3390/molecules21070853⟩
Article dans une revue hal-03150675v1