Emmanuelle DREGE

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Publications

User‐friendly and Green Procedure for a Photoinduced Wohl‐Ziegler Reaction

Florent Edde , Emmanuelle Drège , Laurent Evanno

European Journal of Organic Chemistry, 2025, 28 (18), ⟨10.1002/ejoc.202500183⟩

Article dans une revue hal-05114321v1
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Correction of a Traffic-Defective Missense ABCB11 Variant Responsible for Progressive Familial Intrahepatic Cholestasis Type 2

Martine Lapalus , Elodie Mareux , Rachida Amzal , Emmanuelle Drège , Yosra Riahi et al.

International Journal of Molecular Sciences, 2025, 26 (11), pp.5232. ⟨10.3390/ijms26115232⟩

Article dans une revue hal-05293002v1

Enantioselective Total Synthesis of the Neurotoxin Caramboxin

Benoit Derrien , Karine Leblanc , Laurent Evanno , Emmanuelle Drège

Journal of Organic Chemistry, 2024, 89 (9), pp.6489-6493. ⟨10.1021/acs.joc.4c00541⟩

Article dans une revue hal-05114333v1

Metal-free synthesis of γ-ketosulfones through Brønsted acid-promoted conjugate addition of sulfinamides

Nicolas Gigant , Sami Kayal , Emmanuelle Drège , Delphine Joseph

RSC Advances, 2024, 14 (7), pp.4623-4631. ⟨10.1039/D3RA08675E⟩

Article dans une revue hal-05339308v1

The dual reactivity of Weinreb amides applied to the late-stage divergent functionalisation of meso pyrrolidines

Hamza Boufroura , Laurent Sevaille , Nicolas Gigant , Emmanuelle Drège , Delphine Joseph

New Journal of Chemistry, 2018, 42 (15), pp.12403-12411. ⟨10.1039/C8NJ01975D⟩

Article dans une revue hal-05339317v1
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Identification of a pre-active conformation of a pentameric channel receptor

Anaïs Menny , Solène N Lefebvre , Philipp Am Schmidpeter , Emmanuelle Drège , Zaineb Fourati et al.

eLife, 2017, 6, pp.e23955. ⟨10.7554/eLife.23955⟩

Article dans une revue hal-01519856v1
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Barbiturates Bind in the GLIC Ion Channel Pore and Cause Inhibition by Stabilizing a Closed State

Zaineb Fourati , Reinis Reinholds Ruza , Duncan Laverty , Emmanuelle Drège , Sandrine Delarue et al.

Journal of Biological Chemistry, 2017, 292 (5), pp.1550-1558. ⟨10.1074/jbc.M116.766964⟩

Article dans une revue pasteur-02174609v1

Microwave-assisted telescoped cross metathesis-ring closing aza-Michael reaction sequence: step-economical access to nicotine–lobeline hybrid analogues

Emmanuelle Drège , J. Oko , P.-E. Venot , N. Gigant , D. Joseph

RSC Advances, 2015, 5 (117), pp.96720-96724. ⟨10.1039/C5RA20930G⟩

Article dans une revue hal-05340115v1

Access to Highly Functionalized Sulfonated Cyclopentanes by Acid‐Promoted Rauhut–Currier Reaction with Sulfinamides

Nicolas Gigant , Emmanuelle Drège , Pascal Retailleau , Delphine Joseph

Chemistry - A European Journal, 2015, 21 (44), pp.15544-15547. ⟨10.1002/chem.201502816⟩

Article dans une revue istex hal-05340110v1

Two-Component Domino Reactions Initiated from Ketenes: Serendipitous Synthesis of Quinolizidinones Analogous to Chelated Lobeline’s Conformation

Emmanuelle Drège , Pierre-Etienne Venot , Franck Le Bideau , Pascal Retailleau , Delphine Joseph

Journal of Organic Chemistry, 2015, 80 (20), pp.10119-10126. ⟨10.1021/acs.joc.5b01727⟩

Article dans une revue hal-05340113v1

Thermodynamic epimeric equilibration and crystallisation-induced dynamic resolution of lobelanine, norlobelanine and related analogues

Z. Amara , G. Bernadat , P.-E. Venot , P. Retailleau , C. Troufflard et al.

Organic & Biomolecular Chemistry, 2014, 12 (48), pp.9797-9810. ⟨10.1039/C4OB01787K⟩

Article dans une revue hal-05340102v1

Switchable Stereocontrolled Divergent Synthesis Induced by aza‐Michael Addition of Deactivated Primary Amines under Acid Catalysis

Z. Amara , Emmanuelle Drège , C. Troufflard , P. Retailleau , M.‐e. Tran Huu-Dau et al.

Chemistry - A European Journal, 2014, 20 (48), pp.15840-15848. ⟨10.1002/chem.201404589⟩

Article dans une revue istex hal-05340107v1

Step-Economical Access to Valuable Weinreb Amide 2,5-Disubstituted Pyrrolidines by a Sequential One-Pot Two-Directional Cross-Metathesis/Cyclizing Aza-Michael Process

Hamza Boufroura , Marc Mauduit , Emmanuelle Drège , Delphine Joseph

Journal of Organic Chemistry, 2013, 78 (6), pp.2346-2354. ⟨10.1021/jo302435a⟩

Article dans une revue hal-05340097v1

Step-economical access to valuable Weinreb amide 2,5-disubstituted pyrrolidines by a sequential one-pot two-directional cross-metathesis/cyclizing aza-Michael process.

Hamza Boufroura , Marc Mauduit , Emmanuelle Drège , Delphine Joseph

Journal of Organic Chemistry, 2013, 78 (6), pp.2346-54. ⟨10.1021/jo302435a⟩

Article dans une revue hal-00881452v1

Solvent-free double aza-Michael under ultrasound irradiation: diastereoselective sequential one-pot synthesis of pyrrolidine Lobelia alkaloids analogues

Zacharias Amara , Emmanuelle Drège , Claire Troufflard , Pascal Retailleau , Delphine Joseph

Organic & Biomolecular Chemistry, 2012, 10 (35), pp.7148. ⟨10.1039/C2OB25963J⟩

Article dans une revue hal-05340094v1

Amine-mediated tandem conjugative isomerization-bridging Michael addition: concise synthesis of 1-azabicyclo[3.3.1]nonanes

Anh Ngoc Ngo , Khadija El Kassimi , Zacharias Amara , Emmanuelle Drège , Delphine Joseph

Tetrahedron Letters, 2012, 53 (26), pp.3296-3300. ⟨10.1016/j.tetlet.2012.04.069⟩

Article dans une revue istex hal-05340090v1

Solvent-free double aza-Michael under ultrasound irradiation: diastereoselective sequential one-pot synthesis of pyrrolidine Lobelia alkaloids analogues.

Zacharias Amara , Emmanuelle Drège , Claire Troufflard , Pascal Retailleau , Delphine Joseph

Organic & Biomolecular Chemistry, 2012, 10 (35), pp.7148-57. ⟨10.1039/c2ob25963j⟩

Article dans une revue hal-00798104v1

Asymmetric aza-Michael addition under ultra-high pressure: short bias to polyhydroxylated piperidines

Sidnei Moura , Christine Thomassigny , Caroline Ligeour , Christine Greck , Delphine Joseph et al.

Green Chemistry, 2011, 13 (7), pp.1812. ⟨10.1039/C1GC15097A⟩

Article dans une revue hal-05340084v1

A Facile and Stereocontrolled Synthesis of γ-Substituted γ-Fluoroglutamates by Conjugate Addition: Conflicting Effect between Fluorinated Enaminoester and Hinderered Michael Acceptor

Emmanuelle Drège , Anaïs Guillaume , Nadjia Boukhedimi , Jérôme Marrot , Claire Troufflard et al.

Journal of Organic Chemistry, 2010, 75 (22), pp.7596-7604. ⟨10.1021/jo101417c⟩

Article dans une revue hal-05340080v1

A Facile and Stereocontrolled Synthesis of γ-Substituted γ-Fluoroglutamates by Conjugate Addition: Conflicting Effect between Fluorinated Enaminoester and Hinderered Michael Acceptor.

Emmanuelle Drège , Anaïs Guillaume , Nadjia Boukhedimi , Jérôme Marrot , Claire Troufflard et al.

Journal of Organic Chemistry, 2010, 75 (22), pp.7596-7604. ⟨10.1021/jo101417c⟩

Article dans une revue hal-00551656v1

Synthetic Studies on Cyathin Terpenoids: Enantioselective Synthesis of the Tricyclic Core of Cyathin through Intramolecular Heck Cyclisation

Emmanuelle Drège , Cyrille Tominiaux , Georges Morgant , Didier Desmaële

European Journal of Organic Chemistry, 2006, 2006 (21), pp.4825-4840. ⟨10.1002/ejoc.200600429⟩

Article dans une revue hal-05340063v1

Asymmetric synthesis of the tricyclic core of cyathin diterpenoids via intramolecular Heck reaction

Emmanuelle Drège , Georges Morgant , Didier Desmaële

Tetrahedron Letters, 2005, 46 (42), pp.7263-7266. ⟨10.1016/j.tetlet.2005.07.157⟩

Article dans une revue (article de synthèse) istex hal-05339904v1