François-Xavier Toublet

8
Documents

Publications

Publications

A Review of Natural and Synthetic Chalcones as Anticancer Agents Targeting Topoisomerase Enzymes

François-Xavier Toublet , Aurélie Laurent , Christelle Pouget

Molecules, 2025, 30 (12), pp.2498. ⟨10.3390/molecules30122498⟩

Article dans une revue hal-05106640v1

Synthesis of a New Bichalcone via Suzuki–Miyaura Coupling Reaction

François-Xavier Toublet , Yves Champavier , Aurélie Lévêque , Catherine Fagnère , Christelle Pouget

Molbank, 2025, 2025 (2), pp.M2012. ⟨10.3390/M2012⟩

Article dans une revue hal-05084728v1
Deposit thumbnail

Synthesis and Antiproliferative Effect of 3,4,5-Trimethoxylated Chalcones on Colorectal and Prostatic Cancer Cells

Cécile Letulle , François-Xavier Toublet , Aline Pinon , Soufyane Hba , Aurélie Laurent et al.

Pharmaceuticals, 2024, 17 (9), pp.1207. ⟨10.3390/ph17091207⟩

Article dans une revue hal-04699095v1
Deposit thumbnail

Pleiotropic prodrugs: Design of a dual butyrylcholinesterase inhibitor and 5-HT6 receptor antagonist with therapeutic interest in Alzheimer’s disease

François-Xavier Toublet , Julien Lalut , Bérénice Hatat , Cédric Lecoutey , Audrey Davis et al.

European Journal of Medicinal Chemistry, 2021, 210, pp.113059. ⟨10.1016/j.ejmech.2020.113059⟩

Article dans une revue hal-03082877v1
Deposit thumbnail

Inhibiting Acetylcholinesterase to Activate Pleiotropic Prodrugs with Therapeutic Interest in Alzheimer’s Disease

François-Xavier Toublet , Cédric Lecoutey , Julien Lalut , Bérénice Hatat , Audrey Davis et al.

Molecules, 2019, 24 (15), pp.2786. ⟨10.3390/molecules24152786⟩

Article dans une revue hal-02399906v1