Pascal Dumy

170
Documents

Publications

Publications

A bioinspired approach for the modulation of electroosmotic flow and protein–surface interactions in capillary electrophoresis using silylated amino‐amides blocks and covalent grafting

Jérémie Gouyon , Margaux Clavié , Raquel Gutiérrez-Climente , Giang Ngo , Pascal Dumy et al.
Electrophoresis, 2024, 45 (5-6), pp.557-572. ⟨10.1002/elps.202300168⟩
Article dans une revue hal-04368764 v1
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Sol-gel polymerization of silylated amino acids around a protein template yields selective biomimetic imprints

Raquel Gutiérrez-Climente , Giang Ngo , Margaux Clavié , Jérémie Gouyon , Yoann Ladner et al.
Materials Today Chemistry, 2023, 27 (19), pp.101317. ⟨10.1016/j.mtchem.2022.101317⟩
Article dans une revue hal-04825773 v1

The Institute of Biomolecules Max Mousseron: A Timely Move

Michael Smietana , Pascal Dumy
European Journal of Organic Chemistry, 2022, 2022 (21), ⟨10.1002/ejoc.202101322⟩
Article dans une revue hal-04699425 v1
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Multiplexed Imaging Reveals the Spatial Relationship of the Extracellular Acidity-Targeting pHLIP with Necrosis, Hypoxia, and the Integrin-Targeting cRGD Peptide

Zhao-Hui Jin , Atsushi Tsuji , Mélissa Degardin , Pascal Dumy , Didier Boturyn et al.
Cells, 2022, 11 (21), pp.3499. ⟨10.3390/cells11213499⟩
Article dans une revue hal-03986732 v1
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Development of Amino Acids Functionalized SBA-15 for the Improvement of Protein Adsorption

Raquel Gutiérrez-Climente , Margaux Clavié , Jérémie Gouyon , Giang Ngo , Yoann Ladner et al.
Molecules, 2021, 26 (19), pp.6085. ⟨10.3390/molecules26196085⟩
Article dans une revue hal-03375545 v1
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Design of PEGylated Three Ligands Silica Nanoparticles for Multi-Receptor Targeting

Manon Maurel , Titouan Montheil , Julie Martin , Line Chaar , Veronica Guzman-Gonzalez et al.
Nanomaterials, 2021, 11 (1), pp.177. ⟨10.3390/nano11010177⟩
Article dans une revue hal-03108193 v1

Sol–gel process: the inorganic approach in protein imprinting

Raquel Gutiérrez-Climente , Margaux Clavié , Pascal Dumy , Ahmad Mehdi , Gilles Subra
Journal of materials chemistry‎ B, 2021, 9 (9), pp.2155-2178. ⟨10.1039/D0TB02941F⟩
Article dans une revue hal-03166750 v1

Benzoxaboroles: New Potent Inhibitors of the Carbonic Anhydrases of the Pathogenic Bacterium Vibrio cholerae

Alessandro Bonardi , Alessio Nocentini , Roberta Cadoni , Sonia del Prete , Pascal Dumy et al.
ACS Medicinal Chemistry Letters, 2020, 11 (11), pp.2277-2284. ⟨10.1021/acsmedchemlett.0c00403⟩
Article dans une revue hal-03527027 v1

Metal-free synthesis of imino-disaccharides and calix-iminosugars by photoinduced radical thiol–ene coupling (TEC)

Renaud Zelli , Pascal Dumy , Alberto Marra
Organic & Biomolecular Chemistry, 2020, 18 (13), pp.2392-2397. ⟨10.1039/d0ob00198h⟩
Article dans une revue hal-04554416 v1
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Radiotheranostic Agent 64Cu-cyclam-RAFT-c(-RGDfK-)4 for Management of Peritoneal Metastasis in Ovarian Cancer

Zhao-Hui Jin , Atsushi Tsuji , Mélissa Degardin , Aya Sugyo , Satoshi Obara et al.
Clinical Cancer Research, 2020, 26 (23), pp.6230-6241. ⟨10.1158/1078-0432.CCR-20-1205⟩
Article dans une revue hal-02943140 v1
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Multivalent Carbonic Anhydrases Inhibitors

Fabrizio Carta , Pascal Dumy , Claudiu Supuran , Jean‐yves Winum
International Journal of Molecular Sciences, 2019, 20 (21), pp.5352. ⟨10.3390/ijms20215352⟩
Article dans une revue hal-03527051 v1
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Self-mineralization and assembly of a bis-silylated Phe–Phe pseudodipeptide to a structured bioorganic–inorganic material

Said Jebors , Laurine Valot , Cécile Echalier , Baptiste Legrand , Remi Mikhaleff et al.
Materials Horizons, 2019, 6 (10), pp.2040-2046. ⟨10.1039/c9mh00580c⟩
Article dans une revue hal-02372976 v1
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Photomodulation of DNA-Templated Supramolecular Assemblies

Jenifer Rubio-Magnieto , Tuan-Anh Phan , Mathieu Fossépré , Valérie Matot , Jeremie Knoops et al.
Chemistry - A European Journal, 2018, 24, pp.706-714. ⟨10.1002/chem.201704538⟩
Article dans une revue hal-01666843 v1
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Uniform intratumoral distribution of radioactivity produced using two different radioagents, 64Cu-cyclam-RAFT-c(-RGDfK-)4 and 64Cu-ATSM, improves therapeutic efficacy in a small animal tumor model

Zhao-Hui Jin , Atsushi Tsuji , Melissa Degardin , Aya Sugyo , Yukie Yoshii et al.
EJNMMI Research, 2018, 8 (1), ⟨10.1186/s13550-018-0407-3⟩
Article dans une revue hal-02565825 v1
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Biomolecular dynamic covalent polymers for DNA complexation and siRNA delivery

Camille Bouillon , Yannick Bessin , Florian Poncet , Magali Gary-Bobo , Pascal Dumy et al.
Journal of materials chemistry‎ B, 2018, 6 (44), pp.7239-7246. ⟨10.1039/C8TB01278D⟩
Article dans une revue hal-01944488 v1

Self-assembly and chiroptical properties in supramolecular complexes of adenosine phosphates and guanidinium-bispyrene

Marie Trevisan , Mathieu Fossépré , Delphine Paolantoni , Jenifer Rubio-Magnieto , Pascal Dumy et al.
Chirality, 2018, 30 (6), pp.719-729. ⟨10.1002/chir.22852⟩
Article dans une revue hal-02322046 v1
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Carbonic anhydrases from Trypanosoma cruzi and Leishmania donovani chagasi are inhibited by benzoxaboroles

Alessio Nocentini , Roberta Cadoni , Pascal Dumy , Claudiu Supuran , Jean-Yves Winum
Journal of Enzyme Inhibition and Medicinal Chemistry, 2018, 33 (1), pp.286-289. ⟨10.1080/14756366.2017.1414808⟩
Article dans une revue hal-03621735 v1
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Systemic Delivery of Tumor-Targeted Bax-Derived Membrane-Active Peptides for the Treatment of Melanoma Tumors in a Humanized SCID Mouse Model

Anastassia Karageorgis , Michaël Claron , Romain Jugé , Caroline Aspord , Fabien Thoreau et al.
Molecular Therapy, 2017, 25 (2), pp.534-546. ⟨10.1016/j.ymthe.2016.11.002⟩
Article dans une revue hal-02000186 v1

67Cu-Radiolabeling of a multimeric RGD peptide for αVβ3 integrin-targeted radionuclide therapy

Zhao-Hui Jin , Takako Furukawa , Tomoyuki Ohya , Melissa Degardin , Aya Sugyo et al.
Nuclear Medicine Communications, 2017, 38 (4), pp.347 - 355. ⟨10.1097/MNM.0000000000000646⟩
Article dans une revue hal-01636938 v1
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Polyhedral Oligomeric Silsesquioxane (POSS) Bearing Glyoxylic Aldehyde as Clickable Platform Towards Multivalent Conjugates

Nasreddine Kanfar , Ahmad Mehdi , Pascal Dumy , Sebastien Ulrich, , Jean-Yves Winum
Chemistry - A European Journal, 2017, 23, pp.1-4. ⟨10.1002/chem.201703794⟩
Article dans une revue hal-01611638 v1

Effective Access to Multivalent Inhibitors of Carbonic Anhydrases Promoted by Peptide Bioconjugation

Nasreddine Kanfar , Muhammet Tanc , Pascal Dumy , Claudiu Supuran , Sébastien Ulrich et al.
Chemistry - A European Journal, 2017, 23 (28), pp.6788-6794. ⟨10.1002/chem.201700241⟩
Article dans une revue hal-03621631 v1

Benzoxaboroles as Efficient Inhibitors of the β-Carbonic Anhydrases from Pathogenic Fungi: Activity and Modeling Study

Alessio Nocentini , Roberta Cadoni , Sonia del Prete , Clemente Capasso , Pascal Dumy et al.
ACS Medicinal Chemistry Letters, 2017, 8 (11), pp.1194-1198. ⟨10.1021/acsmedchemlett.7b00369⟩
Article dans une revue hal-03549153 v1

One-Pot Self-Assembly of Peptide-Based Cage-Type Nanostructures Using Orthogonal Ligations

Eline Bartolami , Jérémie Knoops , Yannick Bessin , Mathieu Fossépré , Joseph Chamieh et al.
Chemistry - A European Journal, 2017, 23 (57), pp.14323-14331. ⟨10.1002/chem.201702974⟩
Article dans une revue hal-03542994 v1
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An oxime-based glycocluster microarray

Antoine Hoang , Eugénie Laigre , David Goyard , Eric Defrancq , Françoise Vinet et al.
Organic & Biomolecular Chemistry, 2017, 15 (24), pp.5135-5139. ⟨10.1039/c7ob00889a⟩
Article dans une revue hal-03323886 v1

Auto-assemblage dynamique de clusters cationiques pour la complexation et la vectorisation d’acides nucléiques

Sébastien Ulrich , Eline Bartolami , Pascal Dumy
L'Actualité Chimique, 2017, 417, pp.40-44
Article dans une revue hal-03622994 v1

Phthalimide-Oxy Derivatives for 3′- or 5′-Conjugation of Oligonucleotides by Oxime Ligation and Circularization of DNA by “Bis- or Tris-Click” Oxime Ligation

Albert Meyer , Jean-Jacques Vasseur , Pascal Dumy , François Morvan
European Journal of Organic Chemistry, 2017, 2017 (46), pp.6931-6941. ⟨10.1002/ejoc.201701317⟩
Article dans une revue hal-02197164 v1

Cover Feature: Polyhedral Oligomeric Silsesquioxane (POSS) Bearing Glyoxylic Aldehyde as Clickable Platform Towards Multivalent Conjugates (Chem. Eur. J. 71/2017)

Nasreddine Kanfar , Ahmad Mehdi , Pascal Dumy , Sébastien Ulrich , Jean‐Yves Winum
Chemistry - A European Journal, 2017, 23 (71), pp.17837-17837. ⟨10.1002/chem.201704700⟩
Article dans une revue hal-04728247 v1

Bioactive clusters promoting cell penetration and nucleic acid complexation for drug and gene delivery applications: from designed to self-assembled and responsive systems

Eline Bartolami , Camille Bouillon , Pascal Dumy , Sébastien Ulrich
Chemical Communications, 2016, 52 (23), pp.4257-4273. ⟨10.1039/C5CC09715K⟩
Article dans une revue hal-03621868 v1

Positron emission tomography of cerebral angiogenesis and TSPO expression in a mouse model of chronic hypoxia

Iwao Kanno , Chie Seki , Hiroyuki Takuwa , Zhao-Hui Jin , Didier Boturyn et al.
Journal of Cerebral Blood Flow and Metabolism, 2016, 38 (4), pp.687-696. ⟨10.1177/0271678X16689800⟩
Article dans une revue hal-01649350 v1

Benzoxaborole as a new chemotype for carbonic anhydrase inhibition

Vincenzo Alterio , Roberta Cadoni , Davide Esposito , Daniela Vullo , Anna Di Fiore et al.
Chemical Communications, 2016, 52 (80), pp.11983-11986. ⟨10.1039/c6cc06399c⟩
Article dans une revue hal-03549186 v1
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A metal-free synthetic approach to peptide-based iminosugar clusters as novel multivalent glycosidase inhibitors

Renaud Zelli , Eline Bartolami , Jean-François Longevial , Yannick Bessin , Pascal Dumy et al.
RSC Advances, 2016, 6 (3), pp.2210-2216. ⟨10.1039/c5ra20420h⟩
Article dans une revue hal-03547008 v1

Corrigendum to “Clustering and Internalization of Integrin αvβ3 With a Tetrameric RGD-synthetic Peptide”

Lucie Sancey , Elisabeth C Garanger , Stéphanie Deville-Foillard , Guy Schoehn , Amandine Hurbin et al.
Molecular Therapy, 2016, 17 (7), pp.1301. ⟨10.1038/mt.2009.109⟩
Article dans une revue hal-04837283 v1

αVβ3 Integrin-Targeted Radionuclide Therapy with 64Cu-cyclam-RAFT-c(-RGDfK-)4

Z.-H. Jin , T. Furukawa , M. Degardin , A. Sugyo , A. B. Tsuji et al.
Molecular Cancer Therapeutics, 2016, 15 (9), pp.2076 - 2085. ⟨10.1158/1535-7163.MCT-16-0040⟩
Article dans une revue hal-01645391 v1

Influence of Pre-organised Architecture on Cell Adhesion by Using Multivalent RGD Compounds

Adrien Grassin , Muriel Jourdan , Pascal Dumy , Didier Boturyn
ChemBioChem, 2016, 17 (6), pp.515 - 520. ⟨10.1002/cbic.201500495⟩
Article dans une revue istex hal-01644671 v1

A Click Ligation Based on SuFEx for the Metal-Free Synthesis of Sugar and Iminosugar Clusters

Renaud Zelli , Stefano Tommasone , Pascal Dumy , Alberto Marra , Alessandro Dondoni
European Journal of Organic Chemistry, 2016, 2016 (30), pp.5102-5116. ⟨10.1002/ejoc.201600732⟩
Article dans une revue istex hal-03546885 v1

Synthesis of α-PNA containing a functionalized triazine as nucleobase analogue

Eline Bartolami , Arnaud Gilles , Pascal Dumy , Sébastien Ulrich
Tetrahedron Letters, 2015, 56 (18), pp.2319-2323. ⟨10.1016/j.tetlet.2015.03.072⟩
Article dans une revue hal-03621582 v1
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A Dynamic Combinatorial Approach for Identifying Side Groups that Stabilize DNA-Templated Supramolecular Self-Assemblies

Delphine Paolantoni , Sonia Cantel , Pascal Dumy , Sebastien Ulrich,
International Journal of Molecular Sciences, 2015, 16 (2), pp.3609-3625. ⟨10.3390/ijms16023609⟩
Article dans une revue hal-03574646 v1

Hydroxylamine-O-sulfonamide is a versatile lead compound for the development of carbonic anhydrase inhibitors

Anna Di Fiore , Alessandro Vergara , Marco Caterino , Vincenzo Alterio , Simona Maria Monti et al.
Chemical Communications, 2015, 51 (57), pp.11519-11522. ⟨10.1039/C5CC03711E⟩
Article dans une revue hal-03546192 v1

Carbonic Anhydrase Glycoinhibitors belonging to the Aminoxysulfonamide Series

Joanna Ombouma , Daniella Vullo , Pascal Dumy , Claudiu Supuran , Jean-Yves Winum
ACS Medicinal Chemistry Letters, 2015, 6 (7), pp.819-821. ⟨10.1021/acsmedchemlett.5b00175⟩
Article dans une revue hal-03621576 v1

Dynamic Expression of DNA Complexation with Self-assembled Biomolecular Clusters

Eline Bartolami , Yannick Bessin , Virginie Gervais , Pascal Dumy , Sebastien Ulrich,
Angewandte Chemie International Edition, 2015, 54 (35), pp.10183-10187. ⟨10.1002/anie.201504047⟩
Article dans une revue istex hal-03546810 v1

Emerging trends in enzyme inhibition by multivalent nanoconstructs

Nasreddine Kanfar , Eline Bartolami , Renaud Zelli , Alberto Marra , Jean-Yves Winum et al.
Organic & Biomolecular Chemistry, 2015, 13 (39), pp.9894-9906. ⟨10.1039/C5OB01405K⟩
Article dans une revue hal-03621855 v1

Synthesis and biological properties of multivalent iminosugars

Renaud Zelli , Jean-François Longevial , Pascal Dumy , Alberto Marra
New Journal of Chemistry, 2015, 39 (7), pp.5050-5074. ⟨10.1039/C5NJ00462D⟩
Article dans une revue hal-03621912 v1
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Fluorescent Silica Nanoparticles with Multivalent Inhibitory Effects towards Carbonic Anhydrases

Nadia Touisni , Nasreddine Kanfar , Sebastien Ulrich, , Pascal Dumy , Claudiu T Supuran et al.
Chemistry - A European Journal, 2015, ⟨10.1002/chem.201501037⟩
Article dans une revue istex hal-01206436 v1
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Multivalent DNA recognition by self-assembled clusters: deciphering structural effects by fragments screening and evaluation as siRNA vectors

Eline Bartolami , Yannick Bessin , Nadir Bettache , Magali Gary-Bobo , Marcel Garcia et al.
Organic & Biomolecular Chemistry, 2015, 13 (36), pp.9427 - 9438. ⟨10.1039/c5ob01404b⟩
Article dans une revue hal-03116768 v1
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PET imaging and biodistribution analysis of the effects of succinylated gelatin combined with l-lysine on renal uptake and retention of 64Cu-cyclam-RAFT-c(-RGDfK-)4 in vivo

Zhao-Hui Jin , Takako Furukawa , Chizuru Sogawa , Michaël Claron , Winn Aung et al.
European Journal of Pharmaceutics and Biopharmaceutics, 2014, 86 (3), pp.478 - 486. ⟨10.1016/j.ejpb.2013.11.006⟩
Article dans une revue hal-01652343 v1

Access to bifunctionalized biomolecular platforms using oxime ligation

Karel Křen , Radek Gažák , Gour Chand Daskhan , Julian Garcia , Michele Fiore et al.
Carbohydrate Research, 2014, 393, pp.9 - 14. ⟨10.1016/j.carres.2014.04.020⟩
Article dans une revue hal-01652160 v1
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N-glycosyl-N-hydroxysulfamides as potent inhibitors of Brucella suis carbonic anhydrases

Joanna Ombouma , Daniela Vullo , Stephan Köhler , Pascal Dumy , Claudiu T. Supuran et al.
Journal of Enzyme Inhibition and Medicinal Chemistry, 2014, 30 (6), pp.1010-1012. ⟨10.3109/14756366.2014.986119⟩
Article dans une revue hal-02425102 v1

Retraction of “Synthesis of Multivalent Glycoconjugates Containing the Immunoactive LELTE Peptide: Effect of Glycosylation on Cellular Activation and Natural Killing by Human Peripheral Blood Mononuclear Cells”

Olivier Renaudet , Karel Křen , Isabelle Bossu , Pascal Dumy , Alan Kádek et al.
Journal of the American Chemical Society, 2014, 136 (3), pp.1156 - 1156. ⟨10.1021/ja4081277⟩
Article dans une revue hal-01652507 v1
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Re-Evaluation of Binding Properties of Recombinant Lymphocyte Receptors NKR-P1A and CD69 to Chemically Synthesized Glycans and Peptides

Daniel Rozbeský , Jan Krejzová , Karel Křen , Jan Prchal , Richard Hrabal et al.
International Journal of Molecular Sciences, 2014, 15 (1), pp.1271 - 1283. ⟨10.3390/ijms15011271⟩
Article dans une revue hal-01660558 v1

Thiol-ene and thiol-yne-based synthesis of glycodendrimers as nanomolar inhibitors of wheat germ agglutinin

Mattia Ghirardello , Kim Öberg , Samuele Staderini , Olivier Renaudet , Nathalie Berthet et al.
Journal of Polymer Science Part A: Polymer Chemistry, 2014, 52 (17), pp.2422 - 2433. ⟨10.1002/pola.27262⟩
Article dans une revue istex hal-01652509 v1
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Co-liposomes comprising a lipidated multivalent RGD-peptide and a cationic gemini cholesterol induce selective gene transfection in αvβ3 and αvβ5 integrin receptor-rich cancer cells

Santosh Misra , Paturu Kondaiah , Santanu Bhattacharya , Didier Boturyn , Pascal Dumy
Journal of materials chemistry‎ B, 2014, 2 (35), pp.5758 - 5767. ⟨10.1039/C4TB00701H⟩
Article dans une revue hal-01652173 v1
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Inhibition of β -carbonic anhydrases from Brucella suis with C -cinnamoyl glycosides incorporating the phenol moiety

Leonardo Riafrecha , Daniela Vullo , Safia Ouahrani-Bettache , Stephan Köhler , Pascal Dumy et al.
Journal of Enzyme Inhibition and Medicinal Chemistry, 2014, 30 (6), pp.1017-1020. ⟨10.3109/14756366.2014.986120⟩
Article dans une revue hal-02425101 v1

Oxime Ligation: A Chemoselective Click-Type Reaction for Accessing Multifunctional Biomolecular Constructs

Sébastien Ulrich , Didier Boturyn , Alberto Marra , Olivier Renaudet , Pascal Dumy
Chemistry - A European Journal, 2014, 20 (1), pp.34 - 41. ⟨10.1002/chem.201302426⟩
Article dans une revue istex hal-01652331 v1

Probing secondary interactions in biomolecular recognition by dynamic combinatorial chemistry

Sébastien Ulrich , Pascal Dumy
Chemical Communications, 2014, 50 (44), pp.5810-5825. ⟨10.1039/C4CC00263F⟩
Article dans une revue hal-03621883 v1

Probing the importance of π-stacking interactions in DNA-templated self-assembly of bisfunctionalized guanidinium compounds

Delphine Paolantoni , Jenifer Rubio-Magnieto , Sonia Cantel , Jean Martinez , Pascal Dumy et al.
Chemical Communications, 2014, 50 (91), pp.14257-14260. ⟨10.1039/c4cc05706f⟩
Article dans une revue hal-03564868 v1

Degradable Hybrid Materials Based on Cationic Acylhydrazone Dynamic Covalent Polymers Promote DNA Complexation through Multivalent Interactions

Camille Bouillon , Delphine Paolantoni , Jennifer Rote , Yannick Bessin , Larryn Peterson et al.
Chemistry - A European Journal, 2014, 20 (45), pp.14705-14714. ⟨10.1002/chem.201403695⟩
Article dans une revue istex hal-03545958 v1

Redox-Driven Host-Guest Interactions Allow the Controlled Release of Captured Cells on RGD-Functionalized Surfaces

Dhruv Thakar , Liliane Coche-Guérente , Michaël Claron , Christiane H. F. Wenk , Jérôme Dejeu et al.
ChemBioChem, 2014, 15 (3), pp.377 - 381. ⟨10.1002/cbic.201300636⟩
Article dans une revue istex hal-01652366 v1
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Thiyl Glycosylation of Propargylated Octasilsesquioxane: Synthesis and Lectin-Binding Properties of Densely Glycosylated Clusters on a Cubic Platform

Alberto Marra , Samuele Staderini , Nathalie Berthet , Pascal Dumy , Olivier Renaudet et al.
European Journal of Organic Chemistry, 2013, 2013 (6), pp.1144 - 1149. ⟨10.1002/ejoc.201201453⟩
Article dans une revue istex hal-01653059 v1

Synthesis of multi-antigenic platforms as vaccine candidates against cancers

Michele Fiore , Baptiste Thomas , Vincent Dulery , Pascal Dumy , Olivier Renaudet
New Journal of Chemistry, 2013, 37 (2), pp.286 - 289. ⟨10.1039/c2nj40972k⟩
Article dans une revue hal-01653057 v1

Engineering of biomolecules for sensing and imaging applications

Sébastien Ulrich , Pascal Dumy , D. Boturyn , O. Renaudet
JOURNAL OF DRUG DELIVERY SCIENCE AND TECHNOLOGY, 2013, 23 (1), pp.5 - 16. ⟨10.1016/S1773-2247(13)50001-3⟩
Article dans une revue hal-01653232 v1

Multivalent glyco(cyclo)peptides

M. Carmen Galan , Pascal Dumy , Olivier Renaudet
Chemical Society Reviews, 2013, 42 (11), pp.4599 - 4612. ⟨10.1039/c2cs35413f⟩
Article dans une revue hal-01652834 v1
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In vivo molecular imaging of atherosclerotic lesions in ApoE-/- mice using VCAM-1-specific, 99mTc-labeled peptidic sequences.

Julien Dimastromatteo , Alexis Broisat , Pascale Perret , Mitra Ahmadi , Didier Boturyn et al.
Journal of Nuclear Medicine, 2013, 54 (8), pp.1442-9. ⟨10.2967/jnumed.112.115675⟩
Article dans une revue inserm-00831631 v1

Micro-positron emission tomography/contrast-enhanced computed tomography imaging of orthotopic pancreatic tumor-bearing mice using the αvβ₃ integrin tracer ⁶⁴Cu-labeled cyclam-RAFT-c(-RGDfK-)₄.

Winn Aung , Zhao-Hui Jin , Takako Furukawa , Michael Claron , Didier Boturyn et al.
Molecular Imaging, 2013, 12 (6), pp.376-87. ⟨10.2310/7290.2013.00054⟩
Article dans une revue hal-03618140 v1

Expanding the scope of oxime ligation: facile synthesis of large cyclopeptide-based glycodendrimers

Baptiste Thomas , Nathalie Berthet , Julian Garcia , Pascal Dumy , Olivier Renaudet
Chemical Communications, 2013, 49 (92), ⟨10.1039/c3cc45368e⟩
Article dans une revue hal-01652802 v1

High affinity glycodendrimers for the lectin LecB from <i>Pseudomonas aeruginosa</i>

Nathalie Berthet , Baptiste Thomas , Isabelle Bossu , Emilie Dufour , Emilie Gillon et al.
Bioconjugate Chem., 2013, pp.1598-1611. ⟨10.1021/bc400239m⟩
Article dans une revue hal-00903491 v1

Integrin and matrix metalloprotease dual-targeting with an MMP substrate–RGD conjugate

Christiane Wenk , Veronique Josserand , Pascal Dumy , Jean-Luc Coll , Didier Boturyn
Organic & Biomolecular Chemistry, 2013, 11 (3), pp.448 - 452. ⟨10.1039/c2ob26926k⟩
Article dans une revue hal-01652823 v1

Near-infrared optical guided surgery of highly infiltrative fibrosarcomas in cats using an anti-αvß3 integrin molecular probe

Christiane H.F. Wenk , Frédérique Ponce , Stéphanie Guillermet , Corinne Tenaud , Didier Boturyn et al.
Cancer Letters, 2013, 334 (2), pp.188 - 195. ⟨10.1016/j.canlet.2012.10.041⟩
Article dans une revue istex hal-01652839 v1

Tetravalent glycocyclopeptide with nanomolar affinity to wheat germ agglutinin

Michele Fiore , Nathalie Berthet , Alberto Marra , Emilie Gillon , Pascal Dumy et al.
Organic & Biomolecular Chemistry, 2013, 11 (41), pp.7113-7122. ⟨10.1039/C3OB41203B⟩
Article dans une revue hal-00903486 v1

Glycoside and peptide clustering around the octasilsesquioxane scaffold via photoinduced free-radical thiol–ene coupling. The observation of a striking glycoside cluster effect

Mauro Lo Conte , Samuele Staderini , Angela Chambery , Nathalie Berthet , Pascal Dumy et al.
Organic & Biomolecular Chemistry, 2012, 10 (16), ⟨10.1039/c2ob07078b⟩
Article dans une revue hal-01654849 v1

Synthesis of heteroglycoclusters by using orthogonal chemoselective ligations

Baptiste Thomas , Michele Fiore , Isabelle Bossu , Pascal Dumy , Olivier Renaudet
Beilstein Journal of Organic Chemistry, 2012, 8, pp.421 - 427. ⟨10.3762/bjoc.8.47⟩
Article dans une revue hal-01654997 v1

Positron emission tomography imaging of tumor angiogenesis and monitoring of antiangiogenic efficacy using the novel tetrameric peptide probe 64Cu-cyclam-RAFT-c(-RGDfK-)4

Zhao-Hui Jin , Takako Furukawa , Michaël Claron , Didier Boturyn , Jean-Luc Coll et al.
Angiogenesis, 2012, 15 (4), pp.569 - 580. ⟨10.1007/s10456-012-9281-1⟩
Article dans une revue hal-01654932 v1

Double threading through DNA: NMR structural study of a bis-naphthalene macrocycle bound to a thymine–thymine mismatch

Muriel Jourdan , Anton Granzhan , Régis Guillot , Pascal Dumy , Marie-Paule Teulade-Fichou
Nucleic Acids Research, 2012, 40 (11), pp.5115 - 5128. ⟨10.1093/nar/gks067⟩
Article dans une revue hal-01654807 v1

Reduction of renal uptake of 111In-DOTA-labeled and A700-labeled RAFT-RGD during integrin αvβ3 targeting using single photon emission computed tomography and optical imaging

Arnaud Briat , Christiane H. F. Wenk , Mitra Ahmadi , Michaël Claron , Didier Boturyn et al.
Cancer Science, 2012, 103 (6), pp.1105 - 1110. ⟨10.1111/j.1349-7006.2012.02286.x⟩
Article dans une revue hal-01661937 v1

Multilayer assemblies of polyelectrolyte–gold nanoparticles for the electrocatalytic oxidation and detection of arsenic(III)

M.M. Ottakam Thotiyl , Hajra Basit , Julio A. Sánchez , Cédric Goyer , Liliane Coche-Guerente et al.
Journal of Colloid and Interface Science, 2012, 383 (1), pp.130 - 139. ⟨10.1016/j.jcis.2012.06.033⟩
Article dans une revue hal-01654891 v1

Amphipol mediated surface immobilization of FhuA: a platform for label-free detection of the bacteriophage protein pb5

Hajra Basit , K. Shivaji Sharma , Angéline van Der Heyden , Chantal Gondran , Cécile Breyton et al.
Chemical Communications, 2012, 48 (48), ⟨10.1039/C2CC31107K⟩
Article dans une revue hal-01654783 v1

Redox strategy for reversible attachment of biomolecules using bifunctional linkers

Galina Dubacheva , Mathieu Galibert , Liliane Coche-Guerente , Pascal Dumy , Didier Boturyn et al.
Chemical Communications, 2011, 47 (12), ⟨10.1039/c0cc05647b⟩
Article dans une revue hal-01655562 v1

X-Ray Structure of the Key Synthetic Intermediate of a Cancer-Related Sialyl-Tn Antigen Analogue

Olivier Renaudet , Christian Philouze , Corinne Bailly , André Durif , Pascal Dumy
Journal of Chemical Crystallography, 2011, 41 (2), pp.204 - 208. ⟨10.1007/s10870-010-9864-x⟩
Article dans une revue istex hal-01655660 v1

Controlled Density Patterning of Tolylterpyridine-Tagged Oligonucleotides

Nunzio Tuccitto , Nicoletta Giamblanco , Sumana Ghosh , Valentina Spampinato , Pierre Labbé et al.
Langmuir, 2011, 27 (14), pp.8595 - 8599. ⟨10.1021/la2003468⟩
Article dans une revue hal-01655222 v1

Improvement of porphyrins for G-quadruplex DNA targeting

Carmen Romera , Oriane Bombarde , Romaric Bonnet , Dennis Gomez , Pascal Dumy et al.
Biochimie, 2011, 93 (8), pp.1310 - 1317. ⟨10.1016/j.biochi.2011.06.008⟩
Article dans une revue istex hal-01655267 v1

Cyclic neoglycodecapeptides: how to increase their inhibitory activity and selectivity on lectin/toxin binding to a glycoprotein and cells

Sabine André , Olivier Renaudet , Isabelle Bossu , Pascal Dumy , Hans-Joachim Gabius
Journal of Peptide Science, 2011, 17 (6), pp.427 - 437. ⟨10.1002/psc.1338⟩
Article dans une revue istex hal-01655225 v1

Noninvasive visualization and quantification of tumor αVβ3 integrin expression using a novel positron emission tomography probe, 64Cu-cyclam-RAFT-c(-RGDfK-)4

Zhao-Hui Jin , Takako Furukawa , Mathieu Galibert , Didier Boturyn , Jean-Luc Coll et al.
Nuclear Medicine and Biology, 2011, 38 (4), pp.529 - 540. ⟨10.1016/j.nucmedbio.2010.11.008⟩
Article dans une revue istex hal-01655293 v1

The Use of a Peptidic Scaffold for the Formation of Stable Guanine Tetrads: Control of a H-bonded Pattern in Water

Pierre Murat , Béatrice Gennaro , Julian Garcia , Nicolas Spinelli , Pascal Dumy et al.
Chemistry - A European Journal, 2011, 17 (21), pp.5791 - 5795. ⟨10.1002/chem.201003556⟩
Article dans une revue istex hal-01655632 v1

Synthesis of Glycocyclopeptides by Click Chemistry and Inhibition Assays with Lectins

Isabelle Bossu , Nathalie Berthet , Pascal Dumy , Olivier Renaudet
Journal of Carbohydrate Chemistry, 2011, 30 (7-9), pp.458 - 468. ⟨10.1080/07328303.2011.590260⟩
Article dans une revue hal-01655621 v1

Tethered Bilayer Lipid Membranes on Mixed Self-Assembled Monolayers of a Novel Anchoring Thiol: Impact of the Anchoring Thiol Density on Bilayer Formation

Hajra Basit , Angéline van Der Heyden , Chantal Gondran , Bernard Nysten , Pascal Dumy et al.
Langmuir, 2011, 27 (23), pp.14317 - 14328. ⟨10.1021/la202847r⟩
Article dans une revue hal-01655629 v1

Versatile Introduction of Azido Moiety into Oligonucleotides through Diazo Transfer Reaction

Rémy Lartia , Pierre Murat , Pascal Dumy , Eric Defrancq
Organic Letters, 2011, 13 (20), pp.5672 - 5675. ⟨10.1021/ol202397e⟩
Article dans une revue hal-01655654 v1

Hepatocyte Targeting and Intracellular Copper Chelation by a Thiol-Containing Glycocyclopeptide

Anais M Pujol , Martine Cuillel , Olivier Renaudet , Colette Lebrun , Peggy Charbonnier et al.
Journal of the American Chemical Society, 2011, 133 (2), pp.286-296. ⟨10.1021/ja106206z⟩
Article dans une revue hal-01138626 v1

Dendri-RAFTs: a second generation of cyclopeptide-based glycoclusters

Isabelle Bossu , Miroslav Šulc , Karel Křen , Emilie Dufour , Julian Garcia et al.
Organic & Biomolecular Chemistry, 2011, 9 (6), ⟨10.1039/c0ob00772b⟩
Article dans une revue hal-01655233 v1

Access to Biomolecular Assemblies through One-Pot Triple Orthogonal Chemoselective Ligations

Mathieu Galibert , Olivier Renaudet , Pascal Dumy , Didier Boturyn
Angewandte Chemie International Edition, 2011, 50 (8), pp.1901 - 1904. ⟨10.1002/anie.201006867⟩
Article dans une revue istex hal-01655191 v1

Amyloidogenesis highlighted by designed peptides forming supramolecular self-assemblies

Myriam Ouberai , Gunnar T. Dolphin , Pascal Dumy , Julian Garcia
Chemical Science, 2011, 2 (7), ⟨10.1039/c1sc00016k⟩
Article dans une revue hal-01655194 v1

Clicked tacrine conjugates as acetylcholinesterase and β-amyloid directed compounds

Myriam Ouberai , Kristoffer Brännström , Monika Vestling , Anders Olofsson , Pascal Dumy et al.
Organic & Biomolecular Chemistry, 2011, 9 (4), pp.1140 - 1147. ⟨10.1039/c0ob00393j⟩
Article dans une revue hal-01655212 v1
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Targeted delivery of a proapoptotic peptide to tumors in vivo.

Sandrine Dufort , Lucie Sancey , Amandine Hurbin , Stéphanie Foillard , Didier Boturyn et al.
Journal of Drug Targeting, 2011, 19 (7), pp.582-8. ⟨10.3109/1061186X.2010.542245⟩
Article dans une revue inserm-00559542 v1

RGD–cyclam conjugate: Synthesis and potential application for positron emission tomography

Mathieu Galibert , Zhao-Hui Jin , Takako Furukawa , Toshimitsu Fukumura , Tsuneo Saga et al.
Bioorganic and Medicinal Chemistry Letters, 2010, 20 (18), pp.5422 - 5425. ⟨10.1016/j.bmcl.2010.07.114⟩
Article dans une revue istex hal-01658572 v1

Molecular engineering of biomolecules for nanobio-sciences

Olivier Renaudet , Julian Garcia , Didier Boturyn , Nicolas Spinelli , Eric Defrancq et al.
International Journal of Nanotechnology, 2010, 7 (4/5/6/7/8), ⟨10.1504/IJNT.2010.031742⟩
Article dans une revue hal-01658284 v1

Synthesis of Multivalent Glycoconjugates Containing the Immunoactive LELTE Peptide: Effect of Glycosylation on Cellular Activation and Natural Killing by Human Peripheral Blood Mononuclear Cells

Olivier Renaudet , Karel Křen , Isabelle Bossu , Pascal Dumy , Alan Kádek et al.
Journal of the American Chemical Society, 2010, 132 (19), pp.6800 - 6808. ⟨10.1021/ja101296t⟩
Article dans une revue hal-01658615 v1

Cell adhesion through clustered ligand on fluid supported lipid bilayers

Ludivine Sandrin , Liliane Coche-Guerente , Amandine Bernstein , Hajra Basit , Pierre Labbé et al.
Organic & Biomolecular Chemistry, 2010, 8 (7), ⟨10.1039/b924523e⟩
Article dans une revue istex hal-01657947 v1

Oligonucleotide sequential bis-conjugation via click-oxime and click-Huisgen procedures.

Albert Meyer , Nicolas Spinelli , Pascal Dumy , Jean-Jacques Vasseur , François Morvan et al.
Journal of Organic Chemistry, 2010, 75, pp.3927-3930. ⟨10.1021/jo100599m⟩
Article dans une revue hal-00519475 v1

Unlimited growth of host–guest multilayer films based on functionalized neutral polymers

Galina Dubacheva , Pascal Dumy , Rachel Auzély , Pierre Schaaf , Fouzia Boulmedais et al.
Soft Matter, 2010, 6 (16), ⟨10.1039/c0sm00324g⟩
Article dans une revue istex hal-01658644 v1
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Application of click-click chemistry to the synthesis of new multivalent RGD conjugates.

Mathieu Galibert , Lucie Sancey , Olivier Renaudet , Jean-Luc Coll , Pascal Dumy et al.
Organic & Biomolecular Chemistry, 2010, 8 (22), pp.5133-8. ⟨10.1039/c0ob00070a⟩
Article dans une revue inserm-00559554 v1

Template-Assembled Synthetic G-Quadruplex (TASQ): A Useful System for Investigating the Interactions of Ligands with Constrained Quadruplex Topologies

Pierre Murat , Romaric Bonnet , Angéline Van der heyden , Nicolas Spinelli , Pierre Labbé et al.
Chemistry - A European Journal, 2010, 16 (20), pp.6106 - 6114. ⟨10.1002/chem.200903456⟩
Article dans une revue istex hal-01658627 v1

Electrochemically controlled adsorption of Fc-functionalized polymers on beta-CD-modified self-assembled monolayers

Galina Dubacheva , Angéline van der Heyden , Pascal Dumy , Oznur Kaftan , Rachel Auzély-Velty et al.
Langmuir, 2010, 26 (17), pp.13976-13986. ⟨10.1021/la102026h⟩
Article dans une revue hal-00524345 v1

In vivo molecular imaging of myocardial angiogenesis using the αvβ3 integrin-targeted tracer 99mTc-RAFT-RGD

Julien Dimastromatteo , Laurent M. Riou , Mitra Ahmadi , Guillaume Pons , Eric Pellegrini et al.
Journal of Nuclear Cardiology, 2010, 17 (3), pp.435 - 443. ⟨10.1007/s12350-010-9191-9⟩
Article dans une revue istex hal-01658043 v1

Linear and Branched Glyco-Lipopeptide Vaccines Follow Distinct Cross-Presentation Pathways and Generate Different Magnitudes of Antitumor Immunity

Olivier Renaudet , Gargi Dasgupta , Ilham Bettahi , Alda Shi , Anthony B. Nesburn et al.
PLoS ONE, 2010, 5 (6), ⟨10.1371/journal.pone.0011216⟩
Article dans une revue hal-01658280 v1

Highly efficient cell adhesion on beads functionalized with clustered peptide ligands

Stéphanie Foillard , Pascal Dumy , Didier Boturyn
Organic & Biomolecular Chemistry, 2009, 7 (20), ⟨10.1039/b911440h⟩
Article dans une revue istex hal-01658989 v1

Biomolecular assembly by iterative oxime ligations

Olivier Renaudet , Didier Boturyn , Pascal Dumy
Bioorganic and Medicinal Chemistry Letters, 2009, 19 (14), pp.3880 - 3883. ⟨10.1016/j.bmcl.2009.03.119⟩
Article dans une revue istex hal-01658952 v1

One-Pot Approach to Well-Defined Biomolecular Assemblies by Orthogonal Chemoselective Ligations

Mathieu Galibert , Pascal Dumy , Didier Boturyn
Angewandte Chemie International Edition, 2009, 48 (14), pp.2576 - 2579. ⟨10.1002/anie.200806223⟩
Article dans une revue hal-01659013 v1

Design and synthesis of novel hybrid metal complex-DNA conjugates: key building blocks for mutimetallic linear DNA nanoarrays

S. Ghosh , I. Pignot-Paintrand , P. Dumy , E. Defrancq
Organic & Biomolecular Chemistry, 2009, pp.2729-2737
Article dans une revue hal-00413878 v1

Antitumor activity of a self-adjuvanting glyco-lipopeptide vaccine bearing B cell, CD4+ and CD8+ T cell epitopes

Ilham Bettahi , Gargi Dasgupta , Olivier Renaudet , Aziz Alami Chentoufi , Xiuli Zhang et al.
Cancer Immunology, Immunotherapy, 2009, 58 (2), pp.187 - 200. ⟨10.1007/s00262-008-0537-y⟩
Article dans une revue istex hal-01658946 v1

Design and synthesis of novel hybrid metal complex–DNA conjugates: key building blocks for multimetallic linear DNA nanoarrays

Sumana Ghosh , Isabelle Pignot-Paintrand , Pascal Dumy , Eric Defrancq
Organic & Biomolecular Chemistry, 2009, 7 (13), ⟨10.1039/b904758a⟩
Article dans une revue istex hal-01658958 v1

Efficient conjugation of oligonucleotides through aromatic oxime formation

Pierre Murat , Nicolas Spinelli , Pascal Dumy , Eric Defrancq
Bioorganic and Medicinal Chemistry Letters, 2009, 19 (23), pp.6534 - 6537. ⟨10.1016/j.bmcl.2009.10.048⟩
Article dans une revue istex hal-01658963 v1

Design and synthesis of novel hybrid metal complex-DNA conjugates: key building blocks for mutimetallic linear DNA nanoarrays

S. Ghosh , I. Pignot-Paintrand , P. Dumy , E. Defrancq
Organic & Biomolecular Chemistry, 2009, pp.2729-2737
Article dans une revue hal-00440002 v1

Oligonucleotide Duplexes with Tethered Photoreactive Ruthenium(II) Complexes: Influence of the Ligands and Their Linker on the Photoinduced Electron Transfer and Crosslinking Processes of the Two Strands

Stéphanie Deroo , Stéphane Le Gac , Sumana Ghosh , Mathilde Villien , Pascal Gerbaux et al.
European Journal of Inorganic Chemistry, 2009, 2009 (4), pp.524 - 532. ⟨10.1002/ejic.200801083⟩
Article dans une revue hal-01659008 v1

Synthesis and Biological Evaluation of Clicked Curcumin and Clicked KLVFFA Conjugates as Inhibitors of β-Amyloid Fibril Formation

Myriam Ouberai , Pascal Dumy , Sabine Chierici , Julian Garcia
Bioconjugate Chemistry, 2009, 20 (11), pp.2123 - 2132. ⟨10.1021/bc900281b⟩
Article dans une revue hal-01659035 v1

A gadolinium-binding cyclodecapeptide with a large high-field relaxivity involving second-sphere water.

Célia Bonnet , P.H. Fries , Serge Crouzy , Olivier Sénèque , Federico - Cisnetti et al.
Chemistry - A European Journal, 2009, 15 (29), pp.7083-7093. ⟨10.1002/chem.200900636⟩
Article dans une revue istex hal-00414404 v1

Chemical synthesis, DNA incorporation and biological study of a new photocleavable 2'-deoxyadenosine mimic

N. Berthet , C. Crey-Desbiolles , M. Kotera , P. Dumy
Nucleic Acids Research, 2009, 37 (16), pp.5237 - 5245. ⟨10.1093/nar/gkp562⟩
Article dans une revue hal-01658955 v1

Phenolic Oxime Oligomers Inhibit Alzheimer's Amyloid Fibril Formation and Disaggregate Fibrils In Vitro

Gunnar Dolphin , Olivier Renaudet , Myriam Ouberai , Pascal Dumy , Julian Garcia et al.
ChemBioChem, 2009, 10 (8), pp.1325 - 1329. ⟨10.1002/cbic.200900044⟩
Article dans une revue hal-01659020 v1

Artificial enzyme-based biosensors

Laurent Vial , Pascal Dumy
New Journal of Chemistry, 2009, 33 (5), pp.939. ⟨10.1039/b822966j⟩
Article dans une revue istex hal-04822668 v1
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Drug development in oncology assisted by noninvasive optical imaging.

Lucie Sancey , Sandrine Dufort , Véronique Josserand , Michelle Keramidas , Christian A. Righini et al.
International Journal of Pharmaceutics, 2009, 379 (2), pp.309-16. ⟨10.1016/j.ijpharm.2009.05.034⟩
Article dans une revue inserm-00390608 v1

Targeted delivery of activatable fluorescent pro-apoptotic peptide into live cells

Stéphanie Foillard , Lucie Sancey , Jean-Luc Coll , Didier Boturyn , Pascal Dumy
Organic & Biomolecular Chemistry, 2009, 7 (2), pp.221 - 224. ⟨10.1039/b817251j⟩
Article dans une revue istex hal-01659051 v1

Functionalization of the A ring of pyridoacridine as a route toward greater structural diversity. Synthesis of an octacyclic analogue of eilatin

Laurent Bouffier , Rodica Dinica , Julien Debray , Pascal Dumy , Martine Demeunynck
Bioorganic and Medicinal Chemistry Letters, 2009, 19 (16), pp.4836 - 4838. ⟨10.1016/j.bmcl.2009.06.039⟩
Article dans une revue istex hal-01658979 v1

Synthesis and evaluation of fused bispyrimidinoacridines as novel pentacyclic analogues of quadruplex-binder BRACO-19

Julien Debray , Walid Zeghida , Muriel Jourdan , David Monchaud , Marie-Louise Dheu-Andries et al.
Organic & Biomolecular Chemistry, 2009, 7 (24), pp.5219. ⟨10.1039/B912716J⟩
Article dans une revue istex hal-02125664 v1
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Clustering and internalization of integrin alphavbeta3 with a tetrameric RGD-synthetic peptide.

Lucie Sancey , Elisabeth Garanger , Stéphanie Foillard , Guy Schoehn , Amandine Hurbin et al.
Molecular Therapy, 2009, 17 (5), pp.837-43. ⟨10.1038/mt.2009.29⟩
Article dans une revue inserm-00369024 v1

Promotion of sugar–lectin recognition through the multiple sugar presentation offered by regioselectively addressable functionalized templates (RAFT): a QCM-D and SPR study

Marie Wilczewski , Angéline van der Heyden , Olivier Renaudet , Pascal Dumy , Liliane Coche-Guérente et al.
Organic & Biomolecular Chemistry, 2008, 6 (6), pp.1114. ⟨10.1039/b716214f⟩
Article dans une revue istex hal-04827930 v1

Towards a Self‐Adjuvanting Multivalent B and T cell Epitope Containing Synthetic Glycolipopeptide Cancer Vaccine

Olivier Renaudet , Lbachir Benmohamed , Gargi Dasgupta , Ilham Bettahi , Pascal Dumy
ChemMedChem, 2008, 3 (5), pp.737-741. ⟨10.1002/cmdc.200700315⟩
Article dans une revue istex hal-04823512 v1

Use of γ-aminopropyl-coated glass surface for the patterning of oligonucleotides through oxime bond formation

Nabil Dendane , Antoine Hoang , Éric Defrancq , Françoise Vinet , Pascal Dumy
Bioorganic and Medicinal Chemistry Letters, 2008, 18 (8), pp.2540-2543. ⟨10.1016/j.bmcl.2008.03.054⟩
Article dans une revue istex hal-04827091 v1

A Novel Conformationally Constrained Parallel G Quadruplex

Pierre Murat , Delphine Cressend , Nicolas Spinelli , Angéline van der Heyden , Pierre Labbé et al.
ChemBioChem, 2008, 9 (16), pp.2588-2591. ⟨10.1002/cbic.200800457⟩
Article dans une revue hal-04823402 v1

Concise Synthesis of 2-Amino-4(3 H )-quinazolinones from Simple (Hetero)aromatic Amines

Walid Zeghida , Julien Debray , Sabine Chierici , Pascal Dumy , Martine Demeunynck
Journal of Organic Chemistry, 2008, 73 (6), pp.2473-2475. ⟨10.1021/jo7026883⟩
Article dans une revue istex hal-04398317 v1

Synthesis and Biological Characterisation of Targeted Pro-Apoptotic Peptide.

Stéphanie Foillard , Zhao-Hui Jin , Elisabeth Garanger , Didier Boturyn , Marie-Christine Favrot et al.
ChemBioChem, 2008, epub ahead of print. ⟨10.1002/cbic.200800327⟩
Article dans une revue istex inserm-00314521 v1

A cyclodecapeptide ligand to vitamin B12

Vincent Duléry , Nicolas Uhlich , Noélie Maillard , Viviana Fluxá , Julian Garcia et al.
Organic & Biomolecular Chemistry, 2008, 6 (22), pp.4134. ⟨10.1039/b811234g⟩
Article dans une revue istex hal-04829716 v1

Oxime‐Based Synthesis of New Chromogenic and Fluorogenic Oligosaccharides

Olivier Renaudet , Pascal Dumy
European Journal of Organic Chemistry, 2008, 2008 (32), pp.5383-5386. ⟨10.1002/ejoc.200800855⟩
Article dans une revue istex hal-04823666 v1

A Multimeric Quinacrine Conjugate as a Potential Inhibitor of Alzheimer's β‐Amyloid Fibril Formation

Gunnar Dolphin , Sabine Chierici , Myriam Ouberai , Pascal Dumy , Julian Garcia
ChemBioChem, 2008, 9 (6), pp.952-963. ⟨10.1002/cbic.200700602⟩
Article dans une revue istex hal-04398267 v1

Randomized Combinatorial Library of Heteroglycoclusters (hGC)

Vincent Duléry , Olivier Renaudet , Marie Wilczewski , Angéline van der Heyden , Pierre Labbé et al.
Journal of Combinatorial Chemistry, 2008, 10 (3), pp.368-371. ⟨10.1021/cc800029v⟩
Article dans une revue hal-04827382 v1

1-Ethoxyethylidene, a New Group for the Stepwise SPPS of Aminooxyacetic Acid Containing Peptides

Stéphanie Foillard , Martin Ohsten Rasmussen , Jesus Razkin , Didier Boturyn , Pascal Dumy
Journal of Organic Chemistry, 2008, 73 (3), pp.983-991. ⟨10.1021/jo701628k⟩
Article dans une revue istex hal-04827625 v1
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Cyclic peptides bearing a side-chain tail: A tool to model the structure and reactivity of protein zinc sites.

Olivier Sénèque , Emilie Bourlès , Vincent Lebrun , Estelle Bonnet , Pascal Dumy et al.
Angewandte Chemie International Edition, 2008, 47 (36), pp.6888-6891. ⟨10.1002/anie.200800677⟩
Article dans une revue istex hal-00373744 v1

Surface patterning of (bio)molecules onto the inner wall of fused-silica capillary tubes

Nabil Dendane , Antoine Hoang , Olivier Renaudet , Françoise Vinet , Pascal Dumy et al.
Lab on a Chip, 2008, 8 (12), pp.2161. ⟨10.1039/b811786a⟩
Article dans une revue istex hal-04829839 v1

Synthesis of N-acridinyl-N′-alkylguanidines: Dramatic influence of amine to guanidine replacement on the physicochemical properties

Walid Zeghida , Julien Debray , Carine Michel , Anne Milet , Pascal Dumy et al.
Bioorganic and Medicinal Chemistry Letters, 2008, 18 (17), pp.4779 - 4782. ⟨10.1016/j.bmcl.2008.07.100⟩
Article dans une revue istex hal-01900192 v1
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Chemical and biological evaluations of an (111)in-labeled RGD-peptide targeting integrin alpha(V) beta(3) in a preclinical tumor model.

Mitra Ahmadi , Lucie Sancey , Arnaud Briat , Laurent M. Riou , Didier Boturyn et al.
Cancer Biotherapy & Radiopharmaceuticals, 2008, 23 (6), pp.691-700. ⟨10.1089/cbr.2008.0528⟩
Article dans une revue inserm-00333439 v1

Activatable probes for non-invasive small animal fluorescence imaging.

I. Texier , Jesus Razkin , V. Josserand , Didier Boturyn , Pascal Dumy et al.
Nuclear Instruments and Methods in Physics Research Section A: Accelerators, Spectrometers, Detectors and Associated Equipment, 2007, 571, pp.165-168
Article dans une revue hal-00174220 v1

Efficient Surface Patterning of Oligonucleotides Inside a Glass Capillary through Oxime Bond Formation.

Nabil Dendane , Antoine Hoang , Ludovic Guillard , Eric Defrancq , Francoise Vinet et al.
Bioconjugate Chemistry, 2007, 18, pp.671-676
Article dans une revue hal-00174221 v1

In vivo noninvasive optical imaging of receptor-mediated RGD internalization using self-quenched Cy5-labeled RAFT-c(-RGDfK-)(4).

Zhao-Hui Jin , Jesus Razkin , Veronique Josserand , Didier Boturyn , Alexeï Grichine et al.
Molecular Imaging, 2007, 6 (1), pp.43-55
Article dans une revue inserm-00313766 v1

Designed Amyloid β Peptide Fibril—A Tool for High‐Throughput Screening of Fibril Inhibitors

Gunnar Dolphin , Myriam Ouberai , Pascal Dumy , Julian Garcia
ChemMedChem, 2007, 2 (11), pp.1613-1623. ⟨10.1002/cmdc.200700103⟩
Article dans une revue istex hal-04832101 v1

In Vivo Noninvasive Optical Imaging of Receptor-Mediated RGD Internalization Using Self-Quenched Cy5-Labeled RAFT-c(-RGDfK-)(4)

Zhao-Hui Jin , Jesus Razkin , V. Josserand , Didier Boturyn , Alexei Grichine et al.
Molecular Imaging, 2007, 6, pp.43-55
Article dans une revue hal-00174224 v1

The oxime bond formation as an efficient tool for the conjugation of ruthenium complexes to oligonucleotides and peptides

Mathilde Villien , Stéphanie Deroo , Etienne Gicquel , Éric Defrancq , Cécile Moucheron et al.
Tetrahedron, 2007, 63 (46), pp.11299-11306. ⟨10.1016/j.tet.2007.08.088⟩
Article dans une revue istex hal-04830500 v1

New solid support for the synthesis of 3 '-oligonucleotide conjugates through glyoxylic oxime bond formation

Nicolas Spinelli , Om Prakash Edupuganti , Eric Defrancq , Pascal Dumy
Organic Letters, 2007, 9, pp.219-222. ⟨10.1021/ol062607b⟩
Article dans une revue hal-00169469 v1

Molecular imaging of vascular cell adhesion molecule-1 expression in experimental atherosclerotic plaques with radiolabelled B2702-p

A. Broisat , Laurent Riou , V. Ardisson , Didier Boturyn , Pascal Dumy et al.
European Journal of Nuclear Medicine and Molecular Imaging, 2007, 34 (6), pp.830-840. ⟨10.1007/s00259-006-0310-4⟩
Article dans une revue istex hal-04830750 v1

In vivo imaging of tumour angiogenesis in mice with the alpha(v)beta (3) integrin-targeted tracer (99m)Tc-RAFT-RGD.

Lucie Sancey , Valérie Ardisson , Laurent Riou , Mitra Ahmadi , Danièle Marti-Batlle et al.
European Journal of Nuclear Medicine and Molecular Imaging, 2007, 34 (12), pp.2037-47. ⟨10.1007/s00259-007-0497-z⟩
Article dans une revue istex inserm-00176669 v1

Fluorescent ADP Sensing in Physiological Conditions Based on Cooperative Inhibition of a Miniature Esterase.

Laurent Vial , Pascal Dumy
Journal of the American Chemical Society, 2007, 129, pp.4884-4885. ⟨10.1021/ja070734c⟩
Article dans une revue hal-00169780 v1
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In vivo optical imaging of integrin alphaV-beta3 in mice using multivalent or monovalent cRGD targeting vectors.

Zhao-Hui Jin , Véronique Josserand , Stéphanie Foillard , Didier Boturyn , Pascal Dumy et al.
Molecular Cancer, 2007, 6, pp.41. ⟨10.1186/1476-4598-6-41⟩
Article dans une revue inserm-00176674 v1

alpha and beta-Fucopyranosyl oxyamines : key intermediates for the preparation of fucose-containing glycoconjugates by oxime ligation.

Vincent Dulery , Olivier Renaudet , Christian Philouze , Pascal Dumy
Carbohydrate Research, 2007, 342, pp.894-900. ⟨10.1016/j.carres.2007.02.003⟩
Article dans une revue istex hal-00169781 v1

RAFT Nano‐constructs: surfing to biological applications

Didier Boturyn , Éric Defrancq , Gunnar Dolphin , Julian Garcia , Pierre Labbe et al.
Journal of Peptide Science, 2007, 14 (2), pp.224-240. ⟨10.1002/psc.964⟩
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In Vivo Noninvasive Optical Imaging of Receptor-Mediated RGD Internalization Using Self-Quenched Cy5-Labeled RAFT-c(-RGDfK-)(4)

Zhao-Hui Jin , Veronique Josserand , Jesus Razkin , Elisabeth Garanger , Didier Boturyn et al.
Molecular Imaging, 2007, 6, pp.43-55. ⟨10.2310/7290.2007.00002⟩
Article dans une revue hal-00169559 v1
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Structure-based design of small peptide inhibitors of protein-kinase CK2 subunit interaction

Béatrice Laudet , Caroline Barette , Vincent Dulery , Olivier Renaudet , Pascal Dumy et al.
Biochemical Journal, 2007, 408 (3), pp.363-373. ⟨10.1042/BJ20070825⟩
Article dans une revue hal-00478835 v1

Ethoxyethylidene protecting group prevents N-overacylation in aminooxy peptide synthesis

Vincent Duléry , Olivier Renaudet , Pascal Dumy
Tetrahedron, 2007, 63 (48), pp.11952-11958. ⟨10.1016/j.tet.2007.09.015⟩
Article dans une revue istex hal-04830424 v1

Aldehydic Oligonucleotide: A Key Intermediate for the Preparation of Oligonucleotide Conjugates Through Oxime Bond Formation

Nicolas Spinelli , Yogendra Singh , Éric Defrancq , Pascal Dumy
Nucleosides, Nucleotides and Nucleic Acids, 2007, 26 (8-9), pp.883-887. ⟨10.1080/15257770701505436⟩
Article dans une revue hal-04823327 v1

In vivo optical imaging of integrin alphaV-beta3 in mice using multivalent or monovalent cRGD targeting vectors

Zhao-Hui Jin , V. Josserand , Stephanie Foillard , Didier Boturyn , Pascal Dumy et al.
Molecular Cancer, 2007, 6, pp.41
Article dans une revue hal-00174215 v1

Dipyrido[3 , 2-a : 2' , 3'-c]quinolino[3 , 2-j]phenazine (dpqp-OH) - Synthesis , characterization and DNA interaction of the corresponding Ru(II) complex.

Laurent Bouffier , Martine Demeunynck , Pascal Dumy , Cecile Moucheron , Mesmaeker Kirsch-De
Inorganica Chimica Acta, 2007, 360, pp.3162-3168
Article dans une revue hal-00174218 v1
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Activatable probes for non invasive small animal fluorescence imaging

Isabelle Texier , Jesus Razkin , Veronique Josserand , Didier Boturyn , Pascal Dumy et al.
Nuclear Instruments and Methods in Physics Research, 2007, 571, pp.165-168
Article dans une revue inserm-00331940 v1

Model peptides based on the binding loop of the copper metallochaperone Atx1: selectivity of the consensus sequence MxCxxC for metal ions Hg(II), Cu(I), Cd(II), Pb(II), and Zn(II).

Pierre Rousselot-Pailley , Olivier Sénèque , Colette Lebrun , Serge Crouzy , Didier Boturyn et al.
Inorganic Chemistry, 2006, 45 (14), pp.5510-20. ⟨10.1021/ic060430b⟩
Article dans une revue istex hal-00394430 v1

Activatable fluorescent probes for tumour-targeting imaging in live mice.

Jesus Razkin , Véronique Josserand , Didier Boturyn , Zhao-Hui Jin , Pascal Dumy et al.
ChemMedChem, 2006, 1 (10), pp.1069-72. ⟨10.1002/cmdc.200600118⟩
Article dans une revue istex inserm-00176684 v1
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Electrochemical detection of<i> Arachis hypogaea</i> (peanut) agglutinin binding to monovalent and clustered lactosyl motifs immobilized on a polypyrrole film

Marie-Pierre Dubois , Chantal Gondran , Olivier Renaudet , Pascal Dumy , Hugues Driguez et al.
Chemical Communications, 2005, 34, pp.4318-4320. ⟨10.1039/B506699A⟩
Article dans une revue hal-00305938 v1

Hybridization properties and enzymatic replication of oligonucleotides containing the photocleavable 7-nitroindole base analog

C. Crey-Desbiolles , N. Berthet , M. Kotera , P. Dumy
Nucleic Acids Research, 2005, 33, pp.1532-1543
Article dans une revue hal-00129836 v1

Chemoselective Assembly and Immunological Evaluation of Multiepitopic Glycoconjugates Bearing Clustered Tn Antigen as Synthetic Anticancer Vaccines

Saulius Grigalevicius , Sabine Chierici , Olivier Renaudet , Richard Lo-Man , Edith Dériaud et al.
Bioconjugate Chemistry, 2005, 16 (5), pp.1149-1159. ⟨10.1021/bc050010v⟩
Article dans une revue istex hal-04398355 v1

2'-Deoxyribonolactone lesion produces G&gt;A transitions in Escherichia coli

V. Faure , Pascal Dumy , M. Saparbaev
Nucleic Acids Research, 2004, 32 (9), pp.2937-2946. ⟨10.1093/nar/gkh622⟩
Article dans une revue hal-04980658 v1

Layer-by-layer deposition of chitosan derivatives and DNA on gold surfaces for the development of biorecognition layers

M.L. Pedano , L. Martel , Jacques Desbrieres , E. Defrancq , P. Dumy et al.
Anal. Lett., 2004, pp.2235-2250
Article dans une revue hal-00306770 v1

A case study of 2,2-dimethylthiazolidine as locked cis proline amide bond: synthesis, NMR and molecular modeling studies of a δ-conotoxin EVIA peptide analog

Sabine Chierici , Muriel Jourdan , Mélanie Figuet , Pascal Dumy
Organic & Biomolecular Chemistry, 2004, 2 (17), pp.2437-2441. ⟨10.1039/B408325C⟩
Article dans une revue hal-04398391 v1

Reactivity of Pyrido[4 , 3 , 2-kl]acridines : Regioselective Formation of 6-Substituted Derivatives.

Laurent Bouffier , Martine Demeunynck , Anne Milet , Pascal Dumy
Journal of Organic Chemistry, 2004, 69, pp.8144-8147
Article dans une revue hal-00071546 v1

Template Assembled Synthetic Proteins (TASP) as Functional Mimetics of Proteins

Manfred Mutter , Pascal Dumy , Patrick Garrouste , Christian Lehmann , Marc Mathieu et al.
Angewandte Chemie International Edition, 2003, 35 (13-14), pp.1482-1485. ⟨10.1002/anie.199614821⟩
Article dans une revue hal-04834187 v1

Pseudo-Prolines as a Molecular Hinge: Reversible Induction of cis Amide Bonds into Peptide Backbones

Pascal Dumy , Michael Keller , Declan Ryan , Barbara Rohwedder , Torsten Wöhr et al.
Journal of the American Chemical Society, 1997, 119 (5), pp.918-925. ⟨10.1021/ja962780a⟩
Article dans une revue istex hal-04833482 v1

Synthesis of Glycopeptides and Lipopeptides by Chemoselective Ligation

Stefano Cervigni , Manfred Mutter , Pascal Dumy
Angewandte Chemie International Edition, 1996, 35 (11), pp.1230-1232. ⟨10.1002/anie.199612301⟩
Article dans une revue istex hal-04836293 v1
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Reversible oriented immobilization of histidine-tagged proteins on gold surfaces using a chelator thioalkane

Thomas Keller , Claus Duschl , Dietmar Kröger , Anne-Françoise Sévin-Landais , Horst Vogel et al.
Supramolecular Science, 1995, 2 (3-4), pp.155-160. ⟨10.1016/0968-5677(96)89670-2⟩
Article dans une revue istex hal-04836559 v1

A rational approach to the synthesis of phosphonamidate peptides

Dominique Maffre-Lafon , Pascal Dumy , Roger Escale , Jean Pierre Vidal , Jean Pierre Girard et al.
Letters in Peptide Science, 1994, 1 (1), pp.51-55. ⟨10.1007/BF00132762⟩
Article dans une revue istex hal-04690800 v1