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Contribution of Professor Charles Rees to the development of the chemistry of disulfur dichloride
Thierry Besson
,
Lidia S Konstntinova
,
Panayiotis A Koutentis
,
Oleg A Rakitin
,
Sivaprasad Sivadasan
ARKIVOC - Online Journal of Organic Chemistry, 2024, Commemorative Issue in Honor of Prof. Alan R. Katritzky and Prof. Charles Rees on the occasion of the 25th anniversary of the first publication of Arkivoc (Archive for Organic Chemistry), 2024 (1), ⟨10.24820/ark.5550190.p012.136⟩
Article dans une revue
hal-04432826v1
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Contribution of Professor Charles W. Rees to the development of the chemistry of disulfur dichloride
Thierry Besson
,
Lidia Konstantinova
,
Panayiotis Koutentis
,
Oleg Rakitin
,
Sivaprasad Sivadasan
Article dans une revue
hal-04435494v1
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Photocatalyst-Free, Visible-Light-Mediated C–H Perfluoroalkylation of Quinazolin-4(3H)-ones with perfluoroalkyl Iodides
Thomas Delouche
,
Abdoul Gadiry-Diallo
,
Thierry Besson
,
Sensuke Ogoshi
,
Corinne Fruit
Article dans une revue
hal-04421057v1
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Synthesis of Trifunctional Thiazole-Fused Anthranilonitrile and Anthranilic Acid Derivatives
Nathan Broudic
,
Alexandra Pacheco-Benichou
,
Corinne Fruit
,
Thierry Besson
Article dans une revue
hal-04421061v1
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Straightforward Access to a New Class of Dual DYRK1A/CLK1 Inhibitors Possessing a Simple Dihydroquinoline Core
Mihaela-Liliana Ţînţaş
,
Ludovic Peauger
,
Florent Alix
,
Cyril Papamicaël
,
Thierry Besson
Article dans une revue
hal-03922046v1
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Review on the Synthesis and Therapeutic Potential of Pyrido[2,3-d], [3,2-d], [3,4-d] and [4,3-d]pyrimidine Derivatives
Joana F. Campos
,
Thierry Besson
,
Sabine Berteina-Raboin
Article dans une revue
hal-03890845v1
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A skills framework integrating professionally relevant medicinal chemistry proficiencies to strengthen the contemporary practice of pharmacy
C. Decombat
,
O. Duval
,
T. Besson
,
L. Bourel
,
M. Pudlo
Article dans une revue
hal-03581421v1
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Copper-Catalyzed C–H Arylation of Fused-Pyrimidinone Derivatives Using Diaryliodonium Salts
Alexandra Pacheco-Benichou
,
Eugénie Ivendengani
,
Ioannis Kostakis
,
Thierry Besson
,
Corinne Fruit
Article dans une revue
hal-03117643v1
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Recent Advances in Transition-Metal-Free Late-Stage C-H and N-H Arylation of Heteroarenes Using Diaryliodonium Salts
Thierry Besson
,
Corinne Fruit
Article dans une revue
hal-03358321v1
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DYRK1A regulates B cell acute lymphoblastic leukemia through phosphorylation of FOXO1 and STAT3
Rahul Bhansali
,
Malini Rammohan
,
Paul Lee
,
Anouchka Laurent
,
Qiang Wen
Article dans une revue
hal-03117656v1
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Demonstration of Green Solvent Performance on O,S,N-Heterocycles Synthesis: Metal-Free Click Chemistry and Buchwald—Hartwig Coupling
Joana Campos
,
Manon Cailler
,
Remi Claudel
,
Benjamin Prot
,
Sabine Berteina-Raboin
Article dans une revue
hal-03190807v1
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Exploring Kinase Inhibition Properties of 9H-pyrimido[5,4-b]- and [4,5-b]indol-4-amine Derivatives
Yvonnick Loidreau
,
Carole Dubouilh-Benard
,
Marie-Renée Nourrisson
,
Nadège Loaëc
,
Laurent Meijer
Article dans une revue
hal-02612282v1
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Diaryliodoniums Salts as Coupling Partners for Transition-Metal Catalyzed C- and N-Arylation of Heteroarenes
Alexandra Pacheco-Benichou
,
Thierry Besson
,
Corinne Fruit
Article dans une revue
hal-02557380v1
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Microwave-Assisted Synthesis of Potential Bioactive Benzo-, Pyrido- or Pyrazino-thieno[3,2-d]pyrimidin-4-amine Analogs of MPC-6827
Yvonnick Loidreau
,
Marie-Renée Nourrisson
,
Corinne Fruit
,
Cécile Corbière
,
Pascal Marchand
Article dans une revue
hal-03001666v1
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Synthesis of Benzo-Fused 11H-Pyrido[2,1-b]quinazolin-11-ones by a Buchwald–Hartwig Coupling/Pyridine Dearomatization Sequence in Eucalyptol
Joana Campos
,
Alexandra Pacheco-Benichou
,
Corinne Fruit
,
Thierry Besson
,
Sabine Berteina-Raboin
Article dans une revue
hal-03001681v1
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26th Annual GP2A Medicinal Chemistry Conference & 32nd Journées Franco-Belges de Pharmacochimie
Patrick Dallemagne
,
Christophe Rochais
,
Pascal Marchand
,
Thierry Besson
Article dans une revue
hal-02330438v1
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Crystal Structure of 6,7-Dihydro-5a,7a,13,14-tetraaza-pentaphene-5,8-dione
Jean Guillon
,
Maria de Fatima Pereira-Rosenfeld
,
Noël Pinaud
,
Thierry Besson
,
Valérie Thiéry
Article dans une revue
hal-02330806v1
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DYRK1A Is Regulated By Oncogenic KMT2A and Required for Survival of KMT2A-Rearranged Acute Lymphoblastic Leukemia
Christian Hurtz
,
Gerald Wertheim
,
Rahul Bhansali
,
Anne Lehman
,
Grace Jeschke
Article dans une revue
hal-02417476v1
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Biological Characterization of 8-Cyclopropyl-2-(pyridin-3-yl)thiazolo[5,4-f]quinazolin-9(8H)-one, a Promising Inhibitor of DYRK1A
Corinne Fruit
,
Florence Couly
,
Rahul Bhansali
,
Malini Rammohan
,
Mattias F. Lindberg
Article dans une revue
hal-02417254v1
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Harnessing a Novel Dyrk1a-Ablim2-MKL1 Regulatory Module in Megakaryocyte Morphogenesis to Enable Scalable Platelet "Pharming"
Kamaleldin Elagib
,
Ashton Brock
,
Goar Mosoyan
,
Cara Clementelli
,
Lorrie Delehanty
Article dans une revue
hal-02384958v1
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The Chromosome 21 Kinase DYRK1A and Its Substrate FOXO1 Constitute a Novel Therapeutic Pathway in B-ALL
Rahul Bhansali
,
Malini Rammohan
,
Ji Heon Paul Lee
,
Sebastien Malinge
,
Yi-Chien Tsai
Article dans une revue
hal-02384966v1
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Development of Kinase Inhibitors via Metal-Catalyzed C–H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies
Florence Couly
,
Marine Harari
,
Carole Dubouilh-Benard
,
Laëtitia Bailly
,
Emilie Petit
Article dans une revue
hal-02024491v1
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Synthesis of 2-Mercapto-(2-Oxoindolin-3-Ylidene)Acetonitriles from 3-(4-Chloro-5H-1,2,3-Dithiazol-5-Ylidene)Indolin-2-ones
Boris Letribot
,
Régis Delatouche
,
Hervé Rouillard
,
Antoine Bonnet
,
Jean-René Chérouvrier
Article dans une revue
hal-02197268v1
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Late-Stage C-H Arylation of Thiazolo[5,4- f ]quinazolin-9(8 H)-one Backbone: Synthesis of an Array of Potential Kinase Inhibitors
Florence Couly
,
Carole Dubouilh-Benard
,
Thierry Besson
,
Corinne Fruit
Article dans une revue
hal-02046272v1
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Dual-specificity tyrosine phosphorylation-regulated kinase 1A (DYRK1A) inhibitors: a survey of recent patent literature
T.L. Nguyen
,
Corinne Fruit
,
Y. Hérault
,
L. Meijer
,
Thierry Besson
Article dans une revue
hal-02046302v1
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Recent Developments in Microwave-Assisted Metal-Catalyzed C-H Functionalization of Heteroarenes for Medicinal Chemistry and Material Applications
Thierry Besson
,
Corinne Fruit
Article dans une revue
hal-02046186v1
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Pd-Catalyzed and Copper Assisted Regioselective Sequential C2 and C7 Arylation of Thiazolo[5,4-f]quinazolin-9(8H)-one with Aryl Halides
Marine Harari
,
Florence Couly
,
Corinne Fruit
,
Thierry Besson
Article dans une revue
hal-02046211v1
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Synthesis of bioactive 2-(arylamino)thiazolo[5,4-f]-quinazolin-9-ones via the Hügershoff reaction or Cu- catalyzed intramolecular C-S bond formation
Damien Hédou
,
Carole Dubouilh-Benard
,
N. Loaëc
,
L. Meijer
,
Corinne Fruit
Article dans une revue
hal-02046212v1
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Synthesis of Thiazolo[5,4-f]quinazolin-9(8H)-ones as Multi-Target Directed Ligands of Ser/Thr Kinases
Damien Hédou
,
Julien Godeau
,
N. Loaëc
,
L. Meijer
,
Corinne Fruit
Article dans une revue
hal-02046213v1
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Efficient Microwave-Assisted Synthesis of Methyl 4- or 5-Nitroanthranilate
Julien Godeau
,
Anthony Martinet
,
Vincent Levacher
,
Corinne Fruit
,
Thierry Besson
Article dans une revue
hal-02046207v1
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An Unusual Binding Model of the Methyl 9-Anilinothiazolo[5,4-f] quinazoline-2-carbimidates (EHT 1610 and EHT 5372) Confers High Selectivity for Dual-Specificity Tyrosine Phosphorylation-Regulated Kinases
A. Chaikuad
,
J. Diharce
,
M. Schröder
,
Alicia Foucourt
,
B. Leblond
Article dans une revue
hal-02046195v1
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Ligand-Free Pd-Catalyzed and Copper-Assisted C−H Arylation ofQuinazolin-4-ones with Aryl Iodides under Microwave Heating
Sylvain Laclef
,
Marine Harari
,
Julien Godeau
,
Isabelle Schmitz-Afonso
,
Laurent Bischoff
Article dans une revue
hal-01141150v1
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A novel DYRK1A (Dual specificity tyrosine phosphorylation‐regulated kinase 1A) inhibitor for the treatment of Alzheimer's disease: effect on Tau and amyloid pathologies in vitro
S. Coutadeur
,
H. Benyamine
,
L. Delalonde
,
C. de Oliveira
,
B. Leblond
Article dans une revue
hal-02046148v1
|
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Cu/Pd-catalyzed C-2-H arylation of quinazolin-4(3H)-ones with (hetero)aryl halides
Julien Godeau
,
Marine Harari
,
Sylvain Laclef
,
Emmanuel Deau
,
Corinne Fruit
Article dans une revue
hal-02046152v1
|
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Synthesis of polyfunctionalized benzo[d]thiazoles as novel anthranilic acid derivatives
Damien Hédou
,
Marine Harari
,
Julien Godeau
,
Carole Dubouilh-Benard
,
Corinne Fruit
Article dans une revue
hal-01160622v1
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DYRK1A controls the transition from proliferation to quiescence during lymphoid development by destabilizing Cyclin D3
B. J. Thompson
,
R. Bhansali
,
L. Diebold
,
D. E. Cook
,
L. Stolzenburg
Article dans une revue
hal-01160621v1
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Synthesis and molecular modelling studies of 8-arylpyrido[3',2':4,5thieno[3,2-d]pyrimidin-4-amines as multitarget Ser/Thr kinases inhibitors
Yvonnick Loidreau
,
Emmanuel Deau
,
Pascal Marchand
,
Marie-Renée Nourrisson
,
Cédric Logé
Article dans une revue
hal-01135195v1
|
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Microwave-assisted synthesis of novel N-(4-phenylthiazol-2-yl)-benzo[d]thiazole-, thiazolo[4,5-b]pyridine-, thiazolo[5,4-b]pyridine- and benzo[d]oxazole-2-carboximidamides inspired by marine topsentines and nortopsentines
Emmanuel Deau
,
Carole Dubouilh-Benard
,
Vincent Levacher
,
Thierry Besson
Article dans une revue
hal-01141178v1
|
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Rational multistep synthesis of a novel polyfunctionalized benzo[d]thiazole and its thiazolo[5,4-b]pyridine analogue
Damien Hédou
,
Emmanuel Deau
,
Marine Harari
,
Morgane Sanselme
,
Corinne Fruit
Article dans une revue
hal-01141181v1
|
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Design and Synthesis of Thiazolo[5,4-f]quinazolines as DYRK1A Inhibitors, Part I
Alicia Foucourt
,
Damien Hédou
,
Carole Dubouilh-Benard
,
Laurent Désiré
,
Anne-Sophie Casagrande
Article dans une revue
hal-01141172v1
|
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Design and Synthesis of Thiazolo[5,4-f]quinazolines as DYRK1A Inhibitors, Part II
Alicia Foucourt
,
Damien Hédou
,
Carole Dubouilh-Benard
,
Angelique Girard
,
Thierry Taverne
Article dans une revue
hal-01135223v1
|
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Novel synthesis of angular thiazolo[5,4-f] and [4,5-h]quinazolines, preparation of their linear thiazolo[4,5-g] and [5,4-g]quinazoline analogs
Damien Hédou
,
Rémi Guillon
,
Charlotte Lecointe
,
Cédric Logé
,
Elizabeth Chosson
Article dans une revue
hal-01015586v1
|
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Microwave-Assisted [3+2] Cycloaddition and Suzuki-Miyaura Cross-Coupling for a Concise Access to Polyaromatic Scaffolds
Damien Hédou
,
Emmanuel Deau
,
Carole Dubouilh-Benard
,
Morgane Sanselme
,
Anthony Martinet
Article dans une revue
hal-01015445v1
|
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Suzuki cross-coupling of 5-bromothieno[2,3-b]pyridines for the convenient synthesis of 8-arylpyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-amines
Yvonnick Loidreau
,
Vincent Levacher
,
Thierry Besson
Article dans une revue
hal-01015472v1
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Synthesis and biological evaluation of N-aryl-7-methoxybenzo[b]furo[3,2-d]pyrimidin-4-amines and their N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amine analogues as dual inhibitors of CLK1 and DYRK1A kinases.
Yvonnick Loidreau
,
Pascal Marchand
,
Carole Dubouilh-Benard
,
Marie-Renée Nourrisson
,
Muriel Duflos
Article dans une revue
hal-00997416v1
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Efficient new synthesis of N-arylbenzo[b]furo[3,2-d]pyrimidin-4-amines and their benzo[b]thieno[3,2-d]pyrimidin-4-amine analogues via a microwave-assisted Dimroth rearrangement
Yvonnick Loidreau
,
Carole Dubouilh-Benard
,
Pascal Marchand
,
Marie-Renée Nourrisson
,
Muriel Duflos
Article dans une revue
hal-01015485v1
|
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Convenient one-pot synthesis of N3-substituted pyrido[2,3-d]-, pyrido[3,4-d]-, pyrido[4,3-d]-pyrimidin-4(3H)-ones, and quinazolin-4(3H)-ones analogs
Emmanuel Deau
,
Damien Hédou
,
Elizabeth Chosson
,
Vincent Levacher
,
Thierry Besson
Article dans une revue
hal-01015451v1
|
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Developments in Meyers' lactamization methodology: en route to bi(hetero)aryl structures with defined axial chirality.
Svetlana Postikova
,
Mohamad Sabbah
,
Daniel Wightman
,
Ich Tuan Nguyen
,
Morgane Sanselme
Article dans une revue
hal-00997427v1
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Synthesis of novel 7-substituted pyrido[2',3':4,5]furo[3,2-d]pyrimidin-4-amines and their N-aryl analogues and evaluation of their inhibitory activity against Ser/Thr kinases.
Emmanuel Deau
,
Yvonnick Loidreau
,
Pascal Marchand
,
Marie-Renée Nourrisson
,
Nadège Loaëc
Article dans une revue
hal-00997420v1
|
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Discovery of a Novel Broad-Spectrum Antifungal Agent Derived from Albaconazole
Rémi Guillon
,
Fabrice Pagniez
,
Carine Picot
,
Damien Hédou
,
Alain Tonnerre
Article dans une revue
hal-01015468v1
|
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Study of N1-alkylation of indoles from the reaction of 2(or 3)-aminoindole-3-(or 2)carbonitriles with DMF-dialkylacetals
Yvonnick Loidreau
,
Sigismund Melissen
,
Vincent Levacher
,
Cédric Logé
,
Jérôme Graton
Article dans une revue
hal-00997070v1
|
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Synthesis of novel 7-oxo and 7-hydroxy trifluoroallocolchicinoids with cytotoxic effect
Elizabeth Chosson
,
Francesca Santoro
,
Christophe Rochais
,
Jana Sopkova-de Oliveira Santos
,
Rémi Legay
Article dans une revue
hal-02357753v1
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Synthesis and biological evaluation of N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amines and their pyrido and pyrazino analogues as Ser/Thr kinase inhibitors
Yvonnick Loidreau
,
Pascal Marchand
,
Carole Dubouilh-Benard
,
Marie-Renée Nourrisson
,
Muriel Duflos
Article dans une revue
hal-02357785v1
|
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First synthesis of 4-aminopyrido[2′,3′:4,5]furo[3,2-d]pyrimidines
Yvonnick Loidreau
,
Pascal Marchand
,
Carole Dubouilh-Benard
,
Marie-Renée Nourrisson
,
Muriel Duflos
Article dans une revue
hal-01016753v1
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Microwave-assisted thermal decomposition of formamide: a tool for coupling a pyrimidine ring with an aromatic partner
Yvonnick Loidreau
,
Thierry Besson
Article dans une revue
hal-01018135v1
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Binaphthyl platform as starting materials for the preparation of electron rich benzo[g,h,i]perylenes. Application to molecular architectures based on amino benzo[g,h,i]perylenes and carborane combinations.
Grégory Pieters
,
Anne Gaucher
,
Damien Prim
,
Thierry Besson
,
José Giner Planas
Article dans une revue
hal-01018301v1
|
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Structure of Pb2+/dCMP and Pb2+/CMP complexes as characterized by tandem mass spectrometry and IRMPD spectroscopy
Jean-Yves Salpin
,
Létitia Gamiette
,
Jeanine Tortajada
,
Thierry Besson
,
Philippe Maître
Article dans une revue
hal-00619188v1
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First synthesis of 2-aminosubstituted-2-perfluoroalkyl-3,6-dihydro-2H-thiopyrans by hetero-Diels-Alder reactions of fluorinated thioamides under microwave heating
Sergey S Mikhailichenko
,
J.-P. Bouillon
,
Thierry Besson
,
Yuryi G Shermolovich
Article dans une revue
hal-01019603v1
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Erymildbraedin A and B, two novel cytotoxic dimethylpyrano-isoflavones from the stem bark of Erythrina mildbraedii: evaluation of their activity toward endocrine cancer cells.
Ruben F Tchokouaha
,
Xanthippi Alexi
,
Elizabeth Chosson
,
Thierry Besson
,
Alexios-Leandros Skaltsounis
Article dans une revue
hal-01020552v1
|
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Microwave-accelerated Dimroth rearrangement for the synthesis of 4-anilino-6-nitroquinazolines. Application to an efficient synthesis of a microtubule destabilizing agent.
Alicia Foucourt
,
Carole Dubouilh-Benard
,
Elizabeth Chosson
,
Cecile Corbiere
,
Catherine Buquet
Article dans une revue
hal-01020796v1
|
|
Synthesis and kinase inhibitory activity of novel substituted indigoids
Anne Beauchard
,
Helene Laborie
,
Hervé Rouillard
,
Olivier Lozach
,
Yoan Ferandin
Article dans une revue
hal-02357759v1
|
|
Microwave-assisted synthesis of alpha-ethoxycarbamates
Alexandre Lumbroso
,
Floris Chevallier
,
Isabelle Beaudet
,
Jean-Paul Quintard
,
Thierry Besson
Article dans une revue
hal-02143508v1
|
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Synthesis and kinase inhibitory activity of novel substituted indigoids.
Anne Beauchard
,
Hélène Laborie
,
Hervé Rouillard
,
Olivier Lozach
,
Yoan Ferandin
Article dans une revue
hal-00416031v1
|
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Synthesis and antitumoral activity of novel thiazolobenzotriazole, thiazoloindolo[3,2-c]quinoline and quinolinoquinoline derivatives
Anne Beauchard
,
Alexis Jaunet
,
Laurence Murillo
,
Brigitte Baldeyrou
,
Amélie Lansiaux
Article dans une revue
hal-01449310v1
|
|
Synthesis and evaluation of the antimicrobial activity of novel quinazolinones
Maria de Fatima Pereira
,
Romain Chevrot
,
Eric Rosenfeld
,
Valérie Thiéry
,
Thierry Besson
Article dans une revue
hal-01960717v1
|
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Novel 9-oxo-thiazolo[5,4-f]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1)/glycogen synthase kinase-3 (GSK-3) inhibitors: Synthesis, biological evaluation and molecular modeling studies
Cédric Logé
,
Alexandra Testard
,
Valérie Thiéry
,
Olivier Lozach
,
Mélina Blairvacq
Article dans une revue
hal-02357774v1
|
|
Microwave-assisted Synthesis of Novel Thiazolocarbazoles and Evaluation as Potential Anticancer Agents. Part III
Alexandra Testard
,
Laurent Picot
,
Ingrid Fruitier-Arnaudin
,
Jean-Marie Piot
,
Hadjila Chabane
Article dans une revue
hal-01967795v1
|
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Tautomerism of uracil probed via IR spectroscopy of singly hydrated uracil.
Joost M. Bakker
,
Thierry Besson
,
Maurizio Brugnara
,
Paolo Tosi
,
Jean-Yves Salpin
Article dans une revue
hal-00368127v1
|
|
Structure of electron-capture dissociation fragments from charge-tagged peptides probed by tunable infrared multiple photon dissociation.
Gilles Frison
,
Guillaume van Der Rest
,
Frantisek Turecek
,
Thierry Besson
,
Joël Lemaire
Article dans une revue
hal-00467063v1
|
|
Synthesis and antiproliferative activity of clausine E, mukonine, and koenoline bioisosteres
François Liger
,
Florence Popowycz
,
Thierry Besson
,
Laurent Picot
,
Carlos Galmarini
Article dans une revue
hal-02357763v1
|
|
Synthesis of latonduine derivatives via intramolecular Heck coupling reaction
A. Putey
,
L. Joucla
,
L. Picot
,
Thierry Besson
,
B. Joseph.
Tetrahedron, 2007, pp.63, 867
Article dans une revue
hal-00158714v1
|
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On the origin of some cubebene derivatives — Diels–Alder adducts and the diene structures of solidago compounds
Christopher Jankowski
,
André Pelletier
,
Eduardo Diaz T.
,
Jacqueline M.R Belanger
,
Jocelyn J.R Paré
Article dans une revue
hal-02357729v1
|
|
Synthesis of novel 5-substituted indirubins as protein kinases inhibitors
Anne Beauchard
,
Yoan Ferandin
,
Stéphane Frère
,
Olivier Lozach
,
Mélina Blairvacq
Article dans une revue
hal-00169371v1
|
|
Thiazolo[5,4-f]quinazolin-9-ones, inhibitors of glycogen synthase kinase-3
Alexandra Testard
,
Cédric Logé
,
Benoît Léger
,
Jean-Michel Robert
,
Olivier Lozach
Article dans une revue
hal-02357746v1
|
|
Synthesis of novel 2,3-condensed thieno[2,3- d ]pyrimidin-4-ones via Appel's salt chemistry
Maria de Fatima Pereira
,
Valérie Thiéry
,
Thierry Besson
Article dans une revue
hal-02357738v1
|
|
Synthesis and evaluation of the antiproliferative activity of novel thiazoloquinazolinone kinases inhibitors.
Alexandra Testard
,
Laurent Picot
,
Olivier Lozach
,
Melina Blairvacq
,
Laurent Meijer
Article dans une revue
hal-01443570v1
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Eco-Friendly Microwave-Assisted Scaleable Synthesis of 2-Cyanobenzothiazoles via N -Arylimino-1,2,3-dithiazoles
Stéphane Frère
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Valérie Thiéry
,
Thierry Besson
Article dans une revue
hal-02357713v1
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Eco-Friendly Microwave-Assisted Scaleable Synthesis of 2-Cyanobenzothiazoles via N -Arylimino-1,2,3-dithiazoles
Valérie Thiéry
,
Thierry Besson
Article dans une revue
hal-02357727v1
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Efficient solvent-free microwave phosphorylation of microcrystalline cellulose
Natalia Gospodinova
,
Axelle Grelard
,
Marc Jeannin
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Gabrielle Chitanu
,
Adrian Carpov
Article dans une revue
hal-02357733v1
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Rapid synthesis of 2-cyanobenzothiazole, isothiocyanate and cyanoformanilide derivatives of dapsone †
Thierry Besson
,
Jérôme Guillard
,
Charles Rees
Journal of the Chemical Society, Perkin Transactions 1, 2000, 4, pp.563-566. ⟨10.1039/a908742g⟩
Article dans une revue
hal-02357789v1
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Imidazoquinolinethiones from 8-aminoquinolines by a novel peri-participation
Thierry Besson
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Charles Rees
,
David Roe
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Valérie Thiéry
Journal of the Chemical Society, Perkin Transactions 1, 2000, 4, pp.555-561. ⟨10.1039/a908952g⟩
Article dans une revue
hal-02357793v1
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Fe and H2O2 distributions in the upper water column in the Indian sector of the Southern Ocean
Géraldine Sarthou
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C. Jeandel
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Laurence Brisset
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David Amouroux
,
Thierry Besson
Article dans une revue
hal-00456475v1
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N-(Cyanothioformyl)indoline; a new indoline ring forming reaction
Thierry Besson
,
Gerald Guillaumet
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Christelle Lamazzi
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Charles Rees
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Valérie Thiéry
Journal of the Chemical Society, Perkin Transactions 1, 1998
Article dans une revue
hal-02357800v1
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Rapid Synthesis of 2-Cyanobenzothiazoles from N -Aryliminodithiazoles Under Microwave Irradiation
Valérie Bénéteau
,
Thierry Besson
,
Charles Rees
Article dans une revue
hal-02357709v1
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Synthesis of a benzodioxinic analog of 8-methoxypsoralen
Thierry Besson
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Nicolas Ruiz
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Gérard Coudert
,
Gerald Guillaumet
Article dans une revue
hal-02889857v1
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3,1-Benzoxazin-4-ones, 3,1-benzothiazin-4-ones and N-arylcyanothioformamides
Thierry Besson
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Kumaraswamy Emayan
,
Charles Rees
Article dans une revue
hal-02357768v1
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Biophysical and biological properties of newly synthesized dioxinocoumarin derivatives
Gabriella Csík
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Györgyi Rontó
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Silvano Nocentini
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Simone Averbeck
,
Dietrich Averbeck
Article dans une revue
hal-02889856v1
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Convenient synthesis of 5-substituted-6-methoxy or 6-hydroxy-2,3-dihydro-1,4-benzodioxins via lithiated intermediates
Thierry Besson
,
Mohamed Hretani
,
Gérard Coudert
,
Gerald Guillaumet
Article dans une revue
hal-02889858v1
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A mild One-Step Procedure for the Synthesis of β-Iodo Epoxides from the Corresponding Epoxy-Alcohols
Thierry Besson
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Patrick Rollin
Article dans une revue
hal-02357707v1
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Mitsunobu Thiofunctionalization-Part 2. 1 an Expedient Synthesis of Aza-Heterocycle/Thiosugar Hybrids
Thierry Besson
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Mamdouh Al Neirabeyeh
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Marie-Claude Viaud
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Patrick Rollin
Article dans une revue
hal-02357706v1
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