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Straightforward Access to a New Class of Dual DYRK1A/CLK1 Inhibitors Possessing a Simple Dihydroquinoline Core
Mihaela-Liliana Ţînţaş
,
Ludovic Peauger
,
Florent Alix
,
Cyril Papamicaël
,
Thierry Besson
Journal articles
hal-03922046v1
|
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Review on the Synthesis and Therapeutic Potential of Pyrido[2,3-d], [3,2-d], [3,4-d] and [4,3-d]pyrimidine Derivatives
Joana F. Campos
,
Thierry Besson
,
Sabine Berteina-Raboin
Journal articles
hal-03890845v1
|
|
A skills framework integrating professionally relevant medicinal chemistry proficiencies to strengthen the contemporary practice of pharmacy
C. Decombat
,
O. Duval
,
T. Besson
,
L. Bourel
,
M. Pudlo
Journal articles
hal-03581421v1
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Copper-Catalyzed C–H Arylation of Fused-Pyrimidinone Derivatives Using Diaryliodonium Salts
Alexandra Pacheco-Benichou
,
Eugénie Ivendengani
,
Ioannis Kostakis
,
Thierry Besson
,
Corinne Fruit
Journal articles
hal-03117643v1
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DYRK1A regulates B cell acute lymphoblastic leukemia through phosphorylation of FOXO1 and STAT3
Rahul Bhansali
,
Malini Rammohan
,
Paul Lee
,
Anouchka Laurent
,
Qiang Wen
Journal articles
hal-03117656v1
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Demonstration of Green Solvent Performance on O,S,N-Heterocycles Synthesis: Metal-Free Click Chemistry and Buchwald—Hartwig Coupling
Joana Campos
,
Manon Cailler
,
Remi Claudel
,
Benjamin Prot
,
Sabine Berteina-Raboin
Journal articles
hal-03190807v1
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Recent Advances in Transition-Metal-Free Late-Stage C-H and N-H Arylation of Heteroarenes Using Diaryliodonium Salts
Thierry Besson
,
Corinne Fruit
Journal articles
hal-03358321v1
|
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Synthesis of Benzo-Fused 11H-Pyrido[2,1-b]quinazolin-11-ones by a Buchwald–Hartwig Coupling/Pyridine Dearomatization Sequence in Eucalyptol
Joana Campos
,
Alexandra Pacheco-Benichou
,
Corinne Fruit
,
Thierry Besson
,
Sabine Berteina-Raboin
Journal articles
hal-03001681v1
|
|
Diaryliodoniums Salts as Coupling Partners for Transition-Metal Catalyzed C- and N-Arylation of Heteroarenes
Alexandra Pacheco-Benichou
,
Thierry Besson
,
Corinne Fruit
Journal articles
hal-02557380v1
|
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Exploring Kinase Inhibition Properties of 9H-pyrimido[5,4-b]- and [4,5-b]indol-4-amine Derivatives
Yvonnick Loidreau
,
Carole Dubouilh-Benard
,
Marie-Renée Nourrisson
,
Nadège Loaëc
,
Laurent Meijer
Journal articles
hal-02612282v1
|
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Microwave-Assisted Synthesis of Potential Bioactive Benzo-, Pyrido- or Pyrazino-thieno[3,2-d]pyrimidin-4-amine Analogs of MPC-6827
Yvonnick Loidreau
,
Marie-Renée Nourrisson
,
Corinne Fruit
,
Cécile Corbière
,
Pascal Marchand
Journal articles
hal-03001666v1
|
|
26th Annual GP2A Medicinal Chemistry Conference & 32nd Journées Franco-Belges de Pharmacochimie
Patrick Dallemagne
,
Christophe Rochais
,
Pascal Marchand
,
Thierry Besson
Journal articles
hal-02330438v1
|
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Harnessing a Novel Dyrk1a-Ablim2-MKL1 Regulatory Module in Megakaryocyte Morphogenesis to Enable Scalable Platelet "Pharming"
Kamaleldin Elagib
,
Ashton Brock
,
Goar Mosoyan
,
Cara Clementelli
,
Lorrie Delehanty
Journal articles
hal-02384958v1
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DYRK1A Is Regulated By Oncogenic KMT2A and Required for Survival of KMT2A-Rearranged Acute Lymphoblastic Leukemia
Christian Hurtz
,
Gerald Wertheim
,
Rahul Bhansali
,
Anne Lehman
,
Grace Jeschke
Journal articles
hal-02417476v1
|
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Biological Characterization of 8-Cyclopropyl-2-(pyridin-3-yl)thiazolo[5,4-f]quinazolin-9(8H)-one, a Promising Inhibitor of DYRK1A
Corinne Fruit
,
Florence Couly
,
Rahul Bhansali
,
Malini Rammohan
,
Mattias F. Lindberg
Journal articles
hal-02417254v1
|
|
Crystal Structure of 6,7-Dihydro-5a,7a,13,14-tetraaza-pentaphene-5,8-dione
Jean Guillon
,
Maria de Fatima Pereira-Rosenfeld
,
Noël Pinaud
,
Thierry Besson
,
Valérie Thiéry
Journal articles
hal-02330806v1
|
|
Synthesis of 2-Mercapto-(2-Oxoindolin-3-Ylidene)Acetonitriles from 3-(4-Chloro-5H-1,2,3-Dithiazol-5-Ylidene)Indolin-2-ones
Boris Letribot
,
Régis Delatouche
,
Hervé Rouillard
,
Antoine Bonnet
,
Jean-René Chérouvrier
Journal articles
hal-02197268v1
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The Chromosome 21 Kinase DYRK1A and Its Substrate FOXO1 Constitute a Novel Therapeutic Pathway in B-ALL
Rahul Bhansali
,
Malini Rammohan
,
Ji Heon Paul Lee
,
Sebastien Malinge
,
Yi-Chien Tsai
Journal articles
hal-02384966v1
|
|
Development of Kinase Inhibitors via Metal-Catalyzed C–H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies
Florence Couly
,
Marine Harari
,
Carole Dubouilh-Benard
,
Laëtitia Bailly
,
Emilie Petit
Journal articles
hal-02024491v1
|
|
Dual-specificity tyrosine phosphorylation-regulated kinase 1A (DYRK1A) inhibitors: a survey of recent patent literature
T.L. Nguyen
,
Corinne Fruit
,
Y. Hérault
,
L. Meijer
,
Thierry Besson
Journal articles
hal-02046302v1
|
|
Late-Stage C-H Arylation of Thiazolo[5,4- f ]quinazolin-9(8 H)-one Backbone: Synthesis of an Array of Potential Kinase Inhibitors
Florence Couly
,
Carole Dubouilh-Benard
,
Thierry Besson
,
Corinne Fruit
Journal articles
hal-02046272v1
|
|
An Unusual Binding Model of the Methyl 9-Anilinothiazolo[5,4-f] quinazoline-2-carbimidates (EHT 1610 and EHT 5372) Confers High Selectivity for Dual-Specificity Tyrosine Phosphorylation-Regulated Kinases
A. Chaikuad
,
J. Diharce
,
M. Schröder
,
Alicia Foucourt
,
B. Leblond
Journal articles
hal-02046195v1
|
|
Efficient Microwave-Assisted Synthesis of Methyl 4- or 5-Nitroanthranilate
Julien Godeau
,
Anthony Martinet
,
Vincent Levacher
,
Corinne Fruit
,
Thierry Besson
Journal articles
hal-02046207v1
|
|
Synthesis of bioactive 2-(arylamino)thiazolo[5,4-f]-quinazolin-9-ones via the Hügershoff reaction or Cu- catalyzed intramolecular C-S bond formation
Damien Hédou
,
Carole Dubouilh-Benard
,
N. Loaëc
,
L. Meijer
,
Corinne Fruit
Journal articles
hal-02046212v1
|
|
Synthesis of Thiazolo[5,4-f]quinazolin-9(8H)-ones as Multi-Target Directed Ligands of Ser/Thr Kinases
Damien Hédou
,
Julien Godeau
,
N. Loaëc
,
L. Meijer
,
Corinne Fruit
Journal articles
hal-02046213v1
|
|
Recent Developments in Microwave-Assisted Metal-Catalyzed C-H Functionalization of Heteroarenes for Medicinal Chemistry and Material Applications
Thierry Besson
,
Corinne Fruit
Journal articles
hal-02046186v1
|
|
Pd-Catalyzed and Copper Assisted Regioselective Sequential C2 and C7 Arylation of Thiazolo[5,4-f]quinazolin-9(8H)-one with Aryl Halides
Marine Harari
,
Florence Couly
,
Corinne Fruit
,
Thierry Besson
Journal articles
hal-02046211v1
|
|
A novel DYRK1A (Dual specificity tyrosine phosphorylation‐regulated kinase 1A) inhibitor for the treatment of Alzheimer's disease: effect on Tau and amyloid pathologies in vitro
S. Coutadeur
,
H. Benyamine
,
L. Delalonde
,
C. de Oliveira
,
B. Leblond
Journal articles
hal-02046148v1
|
|
Synthesis and molecular modelling studies of 8-arylpyrido[3',2':4,5thieno[3,2-d]pyrimidin-4-amines as multitarget Ser/Thr kinases inhibitors
Yvonnick Loidreau
,
Emmanuel Deau
,
Pascal Marchand
,
Marie-Renée Nourrisson
,
Cédric Logé
Journal articles
hal-01135195v1
|
|
Synthesis of polyfunctionalized benzo[d]thiazoles as novel anthranilic acid derivatives
Damien Hédou
,
Marine Harari
,
Julien Godeau
,
Carole Dubouilh-Benard
,
Corinne Fruit
Journal articles
hal-01160622v1
|
|
Cu/Pd-catalyzed C-2-H arylation of quinazolin-4(3H)-ones with (hetero)aryl halides
Julien Godeau
,
Marine Harari
,
Sylvain Laclef
,
Emmanuel Deau
,
Corinne Fruit
Journal articles
hal-02046152v1
|
|
Ligand-Free Pd-Catalyzed and Copper-Assisted C−H Arylation ofQuinazolin-4-ones with Aryl Iodides under Microwave Heating
Sylvain Laclef
,
Marine Harari
,
Julien Godeau
,
Isabelle Schmitz-Afonso
,
Laurent Bischoff
Journal articles
hal-01141150v1
|
|
DYRK1A controls the transition from proliferation to quiescence during lymphoid development by destabilizing Cyclin D3
B. J. Thompson
,
R. Bhansali
,
L. Diebold
,
D. E. Cook
,
L. Stolzenburg
Journal articles
hal-01160621v1
|
|
Rational multistep synthesis of a novel polyfunctionalized benzo[d]thiazole and its thiazolo[5,4-b]pyridine analogue
Damien Hédou
,
Emmanuel Deau
,
Marine Harari
,
Morgane Sanselme
,
Corinne Fruit
Journal articles
hal-01141181v1
|
|
Design and Synthesis of Thiazolo[5,4-f]quinazolines as DYRK1A Inhibitors, Part I
Alicia Foucourt
,
Damien Hédou
,
Carole Dubouilh-Benard
,
Laurent Désiré
,
Anne-Sophie Casagrande
Journal articles
hal-01141172v1
|
|
Design and Synthesis of Thiazolo[5,4-f]quinazolines as DYRK1A Inhibitors, Part II
Alicia Foucourt
,
Damien Hédou
,
Carole Dubouilh-Benard
,
Angelique Girard
,
Thierry Taverne
Journal articles
hal-01135223v1
|
|
Microwave-assisted synthesis of novel N-(4-phenylthiazol-2-yl)-benzo[d]thiazole-, thiazolo[4,5-b]pyridine-, thiazolo[5,4-b]pyridine- and benzo[d]oxazole-2-carboximidamides inspired by marine topsentines and nortopsentines
Emmanuel Deau
,
Carole Dubouilh-Benard
,
Vincent Levacher
,
Thierry Besson
Journal articles
hal-01141178v1
|
|
Efficient new synthesis of N-arylbenzo[b]furo[3,2-d]pyrimidin-4-amines and their benzo[b]thieno[3,2-d]pyrimidin-4-amine analogues via a microwave-assisted Dimroth rearrangement
Yvonnick Loidreau
,
Carole Dubouilh-Benard
,
Pascal Marchand
,
Marie-Renée Nourrisson
,
Muriel Duflos
Journal articles
hal-01015485v1
|
|
Discovery of a Novel Broad-Spectrum Antifungal Agent Derived from Albaconazole
Rémi Guillon
,
Fabrice Pagniez
,
Carine Picot
,
Damien Hédou
,
Alain Tonnerre
Journal articles
hal-01015468v1
|
|
Synthesis of novel 7-substituted pyrido[2',3':4,5]furo[3,2-d]pyrimidin-4-amines and their N-aryl analogues and evaluation of their inhibitory activity against Ser/Thr kinases.
Emmanuel Deau
,
Yvonnick Loidreau
,
Pascal Marchand
,
Marie-Renée Nourrisson
,
Nadège Loaëc
Journal articles
hal-00997420v1
|
|
Developments in Meyers' lactamization methodology: en route to bi(hetero)aryl structures with defined axial chirality.
Svetlana Postikova
,
Mohamad Sabbah
,
Daniel Wightman
,
Ich Tuan Nguyen
,
Morgane Sanselme
Journal articles
hal-00997427v1
|
|
Synthesis and biological evaluation of N-aryl-7-methoxybenzo[b]furo[3,2-d]pyrimidin-4-amines and their N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amine analogues as dual inhibitors of CLK1 and DYRK1A kinases.
Yvonnick Loidreau
,
Pascal Marchand
,
Carole Dubouilh-Benard
,
Marie-Renée Nourrisson
,
Muriel Duflos
Journal articles
hal-00997416v1
|
|
Suzuki cross-coupling of 5-bromothieno[2,3-b]pyridines for the convenient synthesis of 8-arylpyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-amines
Yvonnick Loidreau
,
Vincent Levacher
,
Thierry Besson
Journal articles
hal-01015472v1
|
|
Convenient one-pot synthesis of N3-substituted pyrido[2,3-d]-, pyrido[3,4-d]-, pyrido[4,3-d]-pyrimidin-4(3H)-ones, and quinazolin-4(3H)-ones analogs
Emmanuel Deau
,
Damien Hédou
,
Elizabeth Chosson
,
Vincent Levacher
,
Thierry Besson
Journal articles
hal-01015451v1
|
|
Novel synthesis of angular thiazolo[5,4-f] and [4,5-h]quinazolines, preparation of their linear thiazolo[4,5-g] and [5,4-g]quinazoline analogs
Damien Hédou
,
Rémi Guillon
,
Charlotte Lecointe
,
Cédric Logé
,
Elizabeth Chosson
Journal articles
hal-01015586v1
|
|
Microwave-Assisted [3+2] Cycloaddition and Suzuki-Miyaura Cross-Coupling for a Concise Access to Polyaromatic Scaffolds
Damien Hédou
,
Emmanuel Deau
,
Carole Dubouilh-Benard
,
Morgane Sanselme
,
Anthony Martinet
Journal articles
hal-01015445v1
|
|
Synthesis and biological evaluation of N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amines and their pyrido and pyrazino analogues as Ser/Thr kinase inhibitors
Yvonnick Loidreau
,
Pascal Marchand
,
Carole Dubouilh-Benard
,
Marie-Renée Nourrisson
,
Muriel Duflos
Journal articles
hal-02357785v1
|
|
First synthesis of 4-aminopyrido[2′,3′:4,5]furo[3,2-d]pyrimidines
Yvonnick Loidreau
,
Pascal Marchand
,
Carole Dubouilh-Benard
,
Marie-Renée Nourrisson
,
Muriel Duflos
Journal articles
hal-01016753v1
|
|
Study of N1-alkylation of indoles from the reaction of 2(or 3)-aminoindole-3-(or 2)carbonitriles with DMF-dialkylacetals
Yvonnick Loidreau
,
Sigismund Melissen
,
Vincent Levacher
,
Cédric Logé
,
Jérôme Graton
Journal articles
hal-00997070v1
|
|
Synthesis of novel 7-oxo and 7-hydroxy trifluoroallocolchicinoids with cytotoxic effect
Elizabeth Chosson
,
Francesca Santoro
,
Christophe Rochais
,
Jana Sopkova-de Oliveira Santos
,
Rémi Legay
Journal articles
hal-02357753v1
|
|
Microwave-assisted thermal decomposition of formamide: a tool for coupling a pyrimidine ring with an aromatic partner
Yvonnick Loidreau
,
Thierry Besson
Journal articles
hal-01018135v1
|
|
Structure of Pb2+/dCMP and Pb2+/CMP complexes as characterized by tandem mass spectrometry and IRMPD spectroscopy
Jean-Yves Salpin
,
Létitia Gamiette
,
Jeanine Tortajada
,
Thierry Besson
,
Philippe Maître
Journal articles
hal-00619188v1
|
|
Binaphthyl platform as starting materials for the preparation of electron rich benzo[g,h,i]perylenes. Application to molecular architectures based on amino benzo[g,h,i]perylenes and carborane combinations.
Grégory Pieters
,
Anne Gaucher
,
Damien Prim
,
Thierry Besson
,
José Giner Planas
Journal articles
hal-01018301v1
|
|
Microwave-accelerated Dimroth rearrangement for the synthesis of 4-anilino-6-nitroquinazolines. Application to an efficient synthesis of a microtubule destabilizing agent.
Alicia Foucourt
,
Carole Dubouilh-Benard
,
Elizabeth Chosson
,
Cecile Corbiere
,
Catherine Buquet
Journal articles
hal-01020796v1
|
|
Erymildbraedin A and B, two novel cytotoxic dimethylpyrano-isoflavones from the stem bark of Erythrina mildbraedii: evaluation of their activity toward endocrine cancer cells.
Ruben F Tchokouaha
,
Xanthippi Alexi
,
Elizabeth Chosson
,
Thierry Besson
,
Alexios-Leandros Skaltsounis
Journal articles
hal-01020552v1
|
|
First synthesis of 2-aminosubstituted-2-perfluoroalkyl-3,6-dihydro-2H-thiopyrans by hetero-Diels-Alder reactions of fluorinated thioamides under microwave heating
Sergey S Mikhailichenko
,
J.-P. Bouillon
,
Thierry Besson
,
Yuryi G Shermolovich
Journal articles
hal-01019603v1
|
|
Synthesis and antitumoral activity of novel thiazolobenzotriazole, thiazoloindolo[3,2-c]quinoline and quinolinoquinoline derivatives
Anne Beauchard
,
Alexis Jaunet
,
Laurence Murillo
,
Brigitte Baldeyrou
,
Amélie Lansiaux
Journal articles
hal-01449310v1
|
|
Synthesis and kinase inhibitory activity of novel substituted indigoids.
Anne Beauchard
,
Hélène Laborie
,
Hervé Rouillard
,
Olivier Lozach
,
Yoan Ferandin
Journal articles
hal-00416031v1
|
|
Synthesis and kinase inhibitory activity of novel substituted indigoids
Anne Beauchard
,
Helene Laborie
,
Hervé Rouillard
,
Olivier Lozach
,
Yoan Ferandin
Journal articles
hal-02357759v1
|
|
Microwave-assisted synthesis of alpha-ethoxycarbamates
Alexandre Lumbroso
,
Floris Chevallier
,
Isabelle Beaudet
,
Jean-Paul Quintard
,
Thierry Besson
Journal articles
hal-02143508v1
|
|
Structure of electron-capture dissociation fragments from charge-tagged peptides probed by tunable infrared multiple photon dissociation.
Gilles Frison
,
Guillaume van Der Rest
,
Frantisek Turecek
,
Thierry Besson
,
Joël Lemaire
Journal articles
hal-00467063v1
|
|
Synthesis and evaluation of the antimicrobial activity of novel quinazolinones
Maria de Fatima Pereira
,
Romain Chevrot
,
Eric Rosenfeld
,
Valérie Thiéry
,
Thierry Besson
Journal articles
hal-01960717v1
|
|
Novel 9-oxo-thiazolo[5,4-f]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1)/glycogen synthase kinase-3 (GSK-3) inhibitors: Synthesis, biological evaluation and molecular modeling studies
Cédric Logé
,
Alexandra Testard
,
Valérie Thiéry
,
Olivier Lozach
,
Mélina Blairvacq
Journal articles
hal-02357774v1
|
|
Microwave-assisted Synthesis of Novel Thiazolocarbazoles and Evaluation as Potential Anticancer Agents. Part III
Alexandra Testard
,
Laurent Picot
,
Ingrid Fruitier-Arnaudin
,
Jean-Marie Piot
,
Hadjila Chabane
Journal articles
hal-01967795v1
|
|
Tautomerism of uracil probed via IR spectroscopy of singly hydrated uracil.
Joost M. Bakker
,
Thierry Besson
,
Maurizio Brugnara
,
Paolo Tosi
,
Jean-Yves Salpin
Journal articles
hal-00368127v1
|
|
Synthesis of latonduine derivatives via intramolecular Heck coupling reaction
A. Putey
,
L. Joucla
,
L. Picot
,
Thierry Besson
,
B. Joseph.
Tetrahedron, 2007, pp.63, 867
Journal articles
hal-00158714v1
|
|
Synthesis and antiproliferative activity of clausine E, mukonine, and koenoline bioisosteres
François Liger
,
Florence Popowycz
,
Thierry Besson
,
Laurent Picot
,
Carlos Galmarini
Journal articles
hal-02357763v1
|
|
On the origin of some cubebene derivatives — Diels–Alder adducts and the diene structures of solidago compounds
Christopher Jankowski
,
André Pelletier
,
Eduardo Diaz T.
,
Jacqueline M.R Belanger
,
Jocelyn J.R Paré
Journal articles
hal-02357729v1
|
|
Synthesis of novel 2,3-condensed thieno[2,3- d ]pyrimidin-4-ones via Appel's salt chemistry
Maria de Fatima Pereira
,
Valérie Thiéry
,
Thierry Besson
Journal articles
hal-02357738v1
|
|
Synthesis of novel 5-substituted indirubins as protein kinases inhibitors
Anne Beauchard
,
Yoan Ferandin
,
Stéphane Frère
,
Olivier Lozach
,
Mélina Blairvacq
Journal articles
hal-00169371v1
|
|
Thiazolo[5,4-f]quinazolin-9-ones, inhibitors of glycogen synthase kinase-3
Alexandra Testard
,
Cédric Logé
,
Benoît Léger
,
Jean-Michel Robert
,
Olivier Lozach
Journal articles
hal-02357746v1
|
|
Synthesis and evaluation of the antiproliferative activity of novel thiazoloquinazolinone kinases inhibitors.
Alexandra Testard
,
Laurent Picot
,
Olivier Lozach
,
Melina Blairvacq
,
Laurent Meijer
Journal articles
hal-01443570v1
|
|
Eco-Friendly Microwave-Assisted Scaleable Synthesis of 2-Cyanobenzothiazoles via N -Arylimino-1,2,3-dithiazoles
Stéphane Frère
,
Valérie Thiéry
,
Thierry Besson
Journal articles
hal-02357713v1
|
|
Eco-Friendly Microwave-Assisted Scaleable Synthesis of 2-Cyanobenzothiazoles via N -Arylimino-1,2,3-dithiazoles
Valérie Thiéry
,
Thierry Besson
Journal articles
hal-02357727v1
|
|
Efficient solvent-free microwave phosphorylation of microcrystalline cellulose
Natalia Gospodinova
,
Axelle Grelard
,
Marc Jeannin
,
Gabrielle Chitanu
,
Adrian Carpov
Journal articles
hal-02357733v1
|
|
Rapid synthesis of 2-cyanobenzothiazole, isothiocyanate and cyanoformanilide derivatives of dapsone †
Thierry Besson
,
Jérôme Guillard
,
Charles Rees
Journal of the Chemical Society, Perkin Transactions 1, 2000, 4, pp.563-566. ⟨10.1039/a908742g⟩
Journal articles
hal-02357789v1
|
|
Imidazoquinolinethiones from 8-aminoquinolines by a novel peri-participation
Thierry Besson
,
Charles Rees
,
David Roe
,
Valérie Thiéry
Journal of the Chemical Society, Perkin Transactions 1, 2000, 4, pp.555-561. ⟨10.1039/a908952g⟩
Journal articles
hal-02357793v1
|
|
Fe and H2O2 distributions in the upper water column in the Indian sector of the Southern Ocean
Géraldine Sarthou
,
C. Jeandel
,
Laurence Brisset
,
David Amouroux
,
Thierry Besson
Journal articles
hal-00456475v1
|
|
N-(Cyanothioformyl)indoline; a new indoline ring forming reaction
Thierry Besson
,
Gerald Guillaumet
,
Christelle Lamazzi
,
Charles Rees
,
Valérie Thiéry
Journal of the Chemical Society, Perkin Transactions 1, 1998
Journal articles
hal-02357800v1
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Rapid Synthesis of 2-Cyanobenzothiazoles from N -Aryliminodithiazoles Under Microwave Irradiation
Valérie Bénéteau
,
Thierry Besson
,
Charles Rees
Journal articles
hal-02357709v1
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Synthesis of a benzodioxinic analog of 8-methoxypsoralen
Thierry Besson
,
Nicolas Ruiz
,
Gérard Coudert
,
Gerald Guillaumet
Journal articles
hal-02889857v1
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3,1-Benzoxazin-4-ones, 3,1-benzothiazin-4-ones and N-arylcyanothioformamides
Thierry Besson
,
Kumaraswamy Emayan
,
Charles Rees
Journal articles
hal-02357768v1
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Biophysical and biological properties of newly synthesized dioxinocoumarin derivatives
Gabriella Csík
,
Györgyi Rontó
,
Silvano Nocentini
,
Simone Averbeck
,
Dietrich Averbeck
Journal articles
hal-02889856v1
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Convenient synthesis of 5-substituted-6-methoxy or 6-hydroxy-2,3-dihydro-1,4-benzodioxins via lithiated intermediates
Thierry Besson
,
Mohamed Hretani
,
Gérard Coudert
,
Gerald Guillaumet
Journal articles
hal-02889858v1
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Mitsunobu Thiofunctionalization-Part 2. 1 an Expedient Synthesis of Aza-Heterocycle/Thiosugar Hybrids
Thierry Besson
,
Mamdouh Al Neirabeyeh
,
Marie-Claude Viaud
,
Patrick Rollin
Journal articles
hal-02357706v1
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A mild One-Step Procedure for the Synthesis of β-Iodo Epoxides from the Corresponding Epoxy-Alcohols
Thierry Besson
,
Patrick Rollin
Journal articles
hal-02357707v1
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