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Identifying Potent Nonsense-Mediated mRNA Decay Inhibitors with a Novel Screening System
Julie Carrard
,
Fiona Ratajczak
,
Joséphine Elsens
,
Catherine Leroy
,
Rebekah Kong
et al.
Article dans une revue
hal-04250857
v1
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Exatecan Antibody Drug Conjugates Based on a Hydrophilic Polysarcosine Drug-Linker Platform
Louise Conilh
,
Guy Fournet
,
Eric Fourmaux
,
Angélique Murcia
,
Eva-Laure Matera
et al.
Article dans une revue
hal-03215941
v1
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Monomethyl Auristatin E Grafted-Liposomes to Target Prostate Tumor Cell Lines
Ariana Abawi
,
Xiaoyi Wang
,
Julien Bompard
,
Anna Bérot
,
Valentina Andretto
et al.
Article dans une revue
(article de synthèse)
hal-04851780
v1
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Monodisperse polysarcosine-based highly-loaded antibody-drug conjugates
Warren Viricel
,
Guy Fournet
,
Sabine Beaumel
,
Emeline Perrial
,
Sébastien Papot
et al.
Article dans une revue
hal-02134857
v1
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Room-Temperature and Transition-Metal-Free Intramolecular α-Arylation of Ketones: A Mild Access to Tetracyclic Indoles and 7-Azaindoles
Chérif Adouama
,
María Budén
,
Walter Guerra
,
Marcelo Puiatti
,
Benoît Joseph
et al.
Article dans une revue
hal-03093867
v1
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Targeting RNA structure in SMN2 reverses spinal muscular atrophy molecular phenotypes
Amparo Garcia-Lopez
,
Francesca Tessaro
,
Hendrik R A Jonker
,
Anna Wacker
,
Christian Richter
et al.
Article dans une revue
hal-02115789
v1
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Correction: Characterization of Transglutaminase 2 activity inhibitors in monocytes in vitro and their effect in a mouse model for multiple sclerosis
Navina Chrobok
,
John Bol
,
Cornelis Jongenelen
,
John Brevé
,
Said El Alaoui
et al.
Article dans une revue
hal-02134577
v1
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Room-Temperature and Transition-Metal-Free Intramolecular α-Arylation of Ketones: A Mild Access to Tetracyclic Indoles and 7-Azaindoles
Chérif Adouama
,
María Budén
,
Walter Guerra
,
Marcelo Puiatti
,
Benoît Joseph
et al.
Article dans une revue
hal-02134648
v1
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Synthesis and biological evaluation of tetrahydro[1,4]diazepino[1,2-a]indol-1-ones as cyclin-dependent kinase inhibitors
Putey Aurelien
,
Fournet Guy
,
Olivier Lozach
,
Lionel Perrin
,
Meijer Laurent
et al.
European Journal of Medicinal Chemistry, 2014, 83, pp.617-629
Article dans une revue
hal-01147615
v1
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Impact of meriolins, a new class of cyclin-dependent kinase inhibitors, on malignant glioma proliferation and neo-angiogenesis.
Marie Jarry
,
Céline Lecointre
,
Céline Malleval
,
Laurence Desrues
,
Marie-Thérèse Schouft
et al.
Neuro-Oncology, 2014, 16 (11), pp.1484-98
Article dans une revue
hal-01109355
v1
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New 1-arylindoles based serotonin 5-HT7 entagonists. Synthesis and binding evaluation studies
Charlène Sagnes
,
Guy Fournet
,
Grzegorz Satala
,
Andrzej J. Bojarski
,
Benoît Joseph
European Journal of Medicinal Chemistry, 2014, 75, pp.159-168
Article dans une revue
hal-01147626
v1
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Recent advances in the synthesis and properties of 4-, 5-, 6- or 7-azaindoles
Jean-Yves Mérour
,
Sylvain Routier
,
Franck Suzenet
,
Benoît Joseph
Article dans une revue
istex
hal-04451515
v1
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Inhibition of hepatitis C virus NS5B polymerase by S-trityl-L-cysteine derivatives.
Daniel B Nichols
,
Guy Fournet
,
K. R. Gurukumar
,
Amartya Basu
,
Jin-Ching Lee
et al.
Article dans une revue
hal-00691431
v1
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Targeting low molecular weight cyclin E (LMW-E) in breast cancer.
Angela Nanos-Webb
,
Natalie A Jabbour
,
Asha S Multani
,
Hannah Wingate
,
Nassima Oumata
et al.
Article dans une revue
hal-00691433
v1
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Unexpected matrix interactions in liquid secondary ion mass spectrometry of two pyranosyl mercaptans
Christian Gardrat
,
Benoît Joseph
,
Christiane Vitry
,
Alain Castellan
,
Patrick Rollin
Rapid Communications in Mass Spectrometry, 2011, 25 (10), pp.1399-1406. ⟨10.1002/rcm.4998⟩
Article dans une revue
istex
hal-00677750
v1
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Structure-activity relationship and multidrug resistance study of new S-trityl-L-cysteine derivatives as inhibitors of Eg5.
Hung Yi Kristal Kaan
,
Johanna Weiss
,
Dominik Menger
,
Venkatasubramanian Ulaganathan
,
Katarzyna Tkocz
et al.
Article dans une revue
hal-00691439
v1
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New insights into homopiperazine-based 5-HT1A/5-HT7R ligands: synthesis and biological evaluation.
Eduard Badarau
,
Aurélien Putey
,
Franck Suzenet
,
Benoit Joseph
,
Andrzej Bojarski
et al.
Article dans une revue
hal-00691441
v1
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Synthesis of 2-, 3-, and 4-Substituted Pyrido[2,3-b]indoles by C-N, C-O, and C-C(sp) Bond Formation
Cédric Schneider
,
David Goyard
,
David Gueyrard
,
Benoît Joseph
,
Peter Goekjian
Article dans une revue
istex
hal-02351724
v1
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Chemoselective functionalization of α-carbolines at the C-2, C-3, C-4, and C-6 positions using Suzuki–Miyaura reactions
Cédric Schneider
,
David Gueyrard
,
Benoît Joseph
,
Peter Goekjian
Article dans une revue
hal-02351645
v1
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Pyrazolo[1,5-a]-1,3,5-triazine as a purine bioisostere: access to potent cyclin-dependent kinase inhibitor (R)-roscovitine analogue.
Florence Popowycz
,
Guy Fournet
,
Cédric Schneider
,
Karima Bettayeb
,
Yoan Ferandin
et al.
Article dans une revue
hal-00416036
v1
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Indolobenzazepin-7-ones and 6-, 8-, and 9-membered ring derivatives as tubulin polymerization inhibitors: synthesis and structure--activity relationship studies.
Aurélien Putey
,
Florence Popowycz
,
Quoc-Tuan Do
,
Philippe Bernard
,
Sandeep K Talapatra
et al.
Article dans une revue
hal-00691446
v1
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Synthesis and antiproliferative evaluation of pyrazolo[1,5-a]-1,3,5-triazine myoseverin derivatives.
Florence Popowycz
,
Cédric Schneider
,
Salvatore Debonis
,
Dimitrios Skoufias
,
Frank Kozielski
et al.
Article dans une revue
istex
hal-00691448
v1
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Meriolins (3-(pyrimidin-4-yl)-7-azaindoles): synthesis, kinase inhibitory activity, cellular effects, and structure of a CDK2/cyclin A/meriolin complex.
Aude Echalier
,
Karima Bettayeb
,
Yoan Ferandin
,
Olivier Lozach
,
Monique Clément
et al.
Article dans une revue
istex
hal-00319787
v1
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Synthesis and reactivity of 7-azaindole (1H-pyrrolo[2,3-b]pyridine)
Florence Popowycz
,
Sylvain Routier
,
Benoît Joseph
,
Jean-Yves Mérour
Article dans une revue
istex
hal-04451569
v1
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Synthesis and antiproliferative activity of clausine E, mukonine, and koenoline bioisosteres
François Liger
,
Florence Popowycz
,
Thierry Besson
,
Laurent Picot
,
Carlos Galmarini
et al.
Article dans une revue
istex
hal-02357763
v1
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Synthesis of 6-Substituted Pyrido[2,3- b ]indoles by Electrophilic Substitution
Cédric Schneider
,
David Gueyrard
,
Florence Popowycz
,
Benoît Joseph
,
Peter Goekjian
Article dans une revue
hal-02380611
v1
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