EF

Elias Fattal

Professeur de Pharmacotechnie
69 %
Libre accès
118
Documents
Affiliations actuelles
  • Institut Galien Paris-Saclay (IGPS)
  • Institut Galien Paris-Sud (IGPS)
  • Physico-chimie, pharmacotechnie, biopharmacie (PCPB)
Contact

Publications

Publications

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Cobalt: an update review from biokinetic and toxicological data to treatment after internal exposure

Géraldine Landon , Céline Bouvier-Capely , François Fay , Guillaume Phan , E. Fattal

Health Physics, In press, 130 (1), pp.111-125. ⟨10.1097/hp.0000000000002005⟩

Article dans une revue hal-05186310v1
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Inhibition of TRAP1 in the C-terminal domain influences mitochondria properties and breast cancer cell metabolism

Clélia Mathieu , Jessica Ristow Branco , Patricia Zancan , Catherine Brenner , Samir Messaoudi et al.

Biomedicine and Pharmacotherapy, 2026, 196, pp.119060. ⟨10.1016/j.biopha.2026.119060⟩

Article dans une revue hal-05524058v1
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Selective mRNA Delivery to Activated Macrophages via Hyaluronic Acid-Functionalized Lipid Nanoparticles with Optimized PEGylation

Mengyuan Cao , François Fay , Adrouchan Hotier , Séverine Domenichini , Lucile Alexandre et al.

Biomacromolecules, 2026, ⟨10.1021/acs.biomac.5c02390⟩

Article dans une revue hal-05504529v1
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Pulmonary Delivery of siRNA Anti‐TNFα‐loaded Lipid Nanoparticles for Rapid Recovery in Murine Acute Lung Injury

Qinglin Wang , Jihana Achour , Laila Emam , Younes Louaguenouni , Catherine Cailleau et al.

Advanced Healthcare Materials, 2025, 14 (29), pp.e00695. ⟨10.1002/adhm.202500695⟩

Article dans une revue hal-05237521v1
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Precision engineering of macrophage reprogramming with RNA interference-loaded lipid nanoparticles: a game-changer in cancer immunotherapy

Sezen Gül , Juliette Vergnaud , François Fay , Elias Fattal

Drug Delivery and Translational Research, In press, ⟨10.1007/s13346-025-01970-1⟩

Article dans une revue hal-05272960v1
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Deciphering the role of polyethylene glycol-lipid anchors in siRNA-LNP efficacy for P2y2 inhibition in bone marrow-derived macrophages

Sezen Gül , Juliette Vergnaud , Qinglin Wang , Mélanie Hery , Jhon Mino et al.

International Journal of Pharmaceutics, 2025, 684, pp.126186. ⟨10.1016/j.ijpharm.2025.126186⟩

Article dans une revue hal-05322517v1
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Robust micelles formulation to improve systemic corticosteroid therapy in sepsis in multiple healthcare systems

Younes Louaguenouni , Qinglin Wang , Thomas Baticle , Catherine Cailleau , Elodie Lamy et al.

Journal of Controlled Release, 2025, 381, pp.113635. ⟨10.1016/j.jconrel.2025.113635⟩

Article dans une revue hal-05029253v1
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Nanoparticle-based approaches for sepsis treatment: Current trends and perspectives

Younes Louaguenouni , Arnaud Mansart , Djillali Annane , Elias Fattal , François Fay

Journal of Controlled Release, 2025, 386, pp.114139. ⟨10.1016/j.jconrel.2025.114139⟩

Article dans une revue (article de synthèse) hal-05324488v1
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Poly(malic acid) Nanoconjugates of Pyrazinoic Acid for Lung Delivery in the Treatment of Tuberculosis

Thi Hong van Nguyen , Nicolas Tsapis , Lynda Benrabah , Boris Gouilleux , Jean-Pierre Baltaze et al.

Bioconjugate Chemistry, In press, Online ahead of print. ⟨10.1021/acs.bioconjchem.4c00335⟩

Article dans une revue hal-04735909v1

Bisphosphonate Liposomes for Cobalt and Strontium Decorporation ?

Geraldine Landon , Guillaume Phan , François Fay , David Suhard , David Broggio et al.

Health Physics, 2024, 127 (4), pp.463-475. ⟨10.1097/HP.0000000000001812⟩

Article dans une revue irsn-04530091v1
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Poly(malic acid)-budesonide nanoconjugates embedded in microparticles for lung administration

Barbara Tessier , Laurence Moine , Arnaud Peramo , Nicolas Tsapis , Elias Fattal

Drug Delivery and Translational Research, In press, ⟨10.1007/s13346-024-01571-4⟩

Article dans une revue hal-04520623v1
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Overcoming Solubility Challenges: Liposomal isoCoQ‐Carbazole as a Promising Anti‐Tumor Agent for Inoperable and Radiation‐Insensitive cancers

Diana Lamaa , Catherine Cailleau , Juliette Vergnaud , Julie Mougin , Jérôme Bignon et al.

ChemBioChem, 2024, 25 (10), pp.e202400062. ⟨10.1002/cbic.202400062⟩

Article dans une revue hal-04569859v1
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Amphiphilic phosphorus dendrons-associated with anti-inflammatory siRNA reduce symptoms in murine collagen-induced arthritis

Zhibo Yu , Nicolas Tsapis , François Fay , Liang Chen , Andrii Karpus et al.

Biomacromolecules, 2023, 24 (2), pp.667-677. ⟨10.1021/acs.biomac.2c01117⟩

Article dans une revue hal-04101289v1
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Emerging nanoparticle platforms to improve the administration of glucocorticoids

Barbara Tessier , Nicolas Tsapis , Elias Fattal , Laurence Moine

Journal of Controlled Release, 2023, 358, pp.273-292. ⟨10.1016/j.jconrel.2023.04.039⟩

Article dans une revue hal-04101293v1
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Hyaluronic acid-conjugated liposomes loaded with dexamethasone: A promising approach for the treatment of inflammatory diseases

Kamila Bohne Japiassu , Francois Fay , Alessandro Marengo , Sebastião A Mendanha , Catherine Cailleau et al.

International Journal of Pharmaceutics, 2023, 639, pp.122946. ⟨10.1016/j.ijpharm.2023.122946⟩

Article dans une revue hal-04173093v1
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Diclofenac prodrugs nanoparticles: an alternative and efficient treatment for rheumatoid arthritis?

Saadat Hussain , Mujeeb Ur-Rehman , Aqsa Arif , Catherine Cailleau , Cynthia Gillet et al.

International Journal of Pharmaceutics, 2023, 643, pp.123227. ⟨10.1016/j.ijpharm.2023.123227⟩

Article dans une revue hal-04172731v1
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Liposomal AntagomiR‐155‐5p restores anti‐inflammatory macrophages and improves arthritis in pre‐clinical models of Rheumatoid arthritis

Audrey Paoletti , Bineta Ly , Catherine Cailleau , Fan Gao , Marie Péan de Ponfilly-Sotier et al.

Arthritis & rheumatology, 2023, ⟨10.1002/art.42665⟩

Article dans une revue hal-04220797v1
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PLA-PEG forming worm-like nanoparticles despite unfavorable packing parameter: Formation mechanism, thermal stability and potential for cell internalization

Baptiste Robin , Ludivine Mousnier , Hung Lê , Nadège Grabowski , David Chapron et al.

International Journal of Pharmaceutics, 2023, 643, pp.123263. ⟨10.1016/j.ijpharm.2023.123263⟩

Article dans une revue hal-04172728v1
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Resolution of MoS 2 Nanosheets‐Induced Pulmonary Inflammation Driven by Nanoscale Intracellular Transformation and Extracellular‐Vesicle Shuttles

Nathaly Ortiz Peña , Kondareddy Cherukula , Benjamin Even , Dingkun Ji , Sarah Razafindrakoto et al.

Advanced Materials, 2023, 35 (13), pp.2209615. ⟨10.1002/adma.202209615⟩

Article dans une revue hal-04076624v1
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Nanotechnologies and controlled release formulations for the administration of bisphosphonates and their potential in radiation protection

Geraldine Landon , Guillaume Phan , François Fay , Céline Bouvier-Capely , Elias Fattal

Journal of Drug Delivery Science and Technology, 2023, 90, pp.105154. ⟨10.1016/j.jddst.2023.105154⟩

Article dans une revue hal-04280424v1
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Modulation of release and pharmacokinetics from nanoscale lipid prodrugs of dexamethasone with variable linkage chemistry

Mujeeb Ur-Rehman , Franceline Reynaud , Sinda Lepetre , Sonia Abreu , Pierre Chaminade et al.

Journal of Controlled Release, 2023, 360, pp.293-303. ⟨10.1016/j.jconrel.2023.06.031⟩

Article dans une revue (article de synthèse) hal-04157123v1
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Targeted nanotherapy with everolimus reduces inflammation and fibrosis in scleroderma‐related interstitial lung disease developed by PSGL‐1 deficient mice

Elena González-Sánchez , Antonio Muñoz-Callejas , Javier Gómez-Román , Esther San Antonio , Alessandro Marengo et al.

British Journal of Pharmacology, 2022, 179 (18), pp.4534-4548. ⟨10.1111/bph.15898⟩

Article dans une revue hal-03786904v1

Characterization of the physicochemical interactions between exenatide and two intestinal permeation enhancers: Sodium caprate (C10) and salcaprozate sodium (SNAC)

Caroline Twarog , Elias Fattal , Magali Noiray , Brigitte Illel , David Brayden et al.

International Journal of Pharmaceutics, 2022, 626, pp.122131. ⟨10.1016/j.ijpharm.2022.122131⟩

Article dans une revue hal-04305542v1
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Improving dexamethasone drug loading and efficacy in treating arthritis through a lipophilic prodrug entrapped into PLGA-PEG nanoparticles

Rosana Simón-Vázquez , Nicolas Tsapis , Mathilde Lorscheider , Ainhoa Rodríguez , Patricia Calleja et al.

Drug Delivery and Translational Research, 2022, 12 (5), pp.1270-1284. ⟨10.1007/s13346-021-01112-3⟩

Article dans une revue hal-04354571v1
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Interplay between mucus mobility and alveolar macrophage targeting of surface-modified liposomes

Kamila Bohne Japiassu , Francois Fay , Alessandro Marengo , Younès Louaguenouni , Catherine Cailleau et al.

Journal of Controlled Release, 2022, 352, pp.15-24. ⟨10.1016/j.jconrel.2022.10.006⟩

Article dans une revue hal-03853759v2
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Mannosylation Of Budesonide Palmitate Nanoprodrugs For Improved Macrophage Targeting

Ludmila Pinheiro Do Nascimento , Nicolas Tsapis , Franceline Reynaud , Didier Desmaële , Laurence Moine et al.

European Journal of Pharmaceutics and Biopharmaceutics, 2022, 170, pp.112-120. ⟨10.1016/j.ejpb.2021.12.001⟩

Article dans une revue hal-03475936v1
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Synthesis and antiproliferative activity of 6BrCaQ-TPP conjugates for targeting the mitochondrial heat shock protein TRAP1

Clelia Mathieu , Quentin Chamayou , Thi Thanh Hyen Luong , Delphine Naud , Florence Mahuteau-Betzer et al.

European Journal of Medicinal Chemistry, 2022, 229, pp.114052. ⟨10.1016/j.ejmech.2021.114052⟩

Article dans une revue hal-03795373v1
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Liposomes Loaded with Everolimus and Coated with Hyaluronic Acid: A Promising Approach for Lung Fibrosis

Laura Pandolfi , Alessandro Marengo , Kamila Bohne Japiassu , Vanessa Frangipane , Nicolas Tsapis et al.

International Journal of Molecular Sciences, 2021, 22 (14), pp.7743. ⟨10.3390/ijms22147743⟩

Article dans une revue hal-03367005v1
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Interspecies comparison of plasma metabolism and sample stabilization for quantitative bioanalyses: Application to (R)-CE3F4 in preclinical development, including metabolite identification by high-resolution mass spectrometry

Balthazar Toussaint , Hervé Hillaireau , Emmanuel Jaccoulet , Catherine Cailleau , Pauline Legrand et al.

Journal of Chromatography B - Analytical Technologies in the Biomedical and Life Sciences, 2021, 1183, pp.122943. ⟨10.1016/j.jchromb.2021.122943⟩

Article dans une revue hal-04241640v1
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Stability, pharmacokinetics, and biodistribution in mice of the EPAC1 inhibitor (R)-CE3F4 entrapped in liposomes and lipid nanocapsules

Balthazar Toussaint , Hervé Hillaireau , Catherine Cailleau , Yves Ambroise , Elias Fattal

International Journal of Pharmaceutics, 2021, 610, pp.121213. ⟨10.1016/j.ijpharm.2021.121213⟩

Article dans une revue hal-04241642v1
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Combining dexamethasone and TNF-α siRNA within the same nanoparticles to enhance anti-inflammatory effect

Serra Gürcan , Nicolas Tsapis , Franceline Reynaud , Stéphanie Denis , Juliette Vergnaud et al.

International Journal of Pharmaceutics, 2021, 598, pp.120381. ⟨10.1016/j.ijpharm.2021.120381⟩

Article dans une revue hal-03215959v1

Comparison of the effects of the intestinal permeation enhancers, SNAC and sodium caprate (C10): Isolated rat intestinal mucosae and sacs

Caroline Twarog , Fiona Mccartney , Sabine Harrison , Brigitte Illel , Elias Fattal et al.

European Journal of Pharmaceutical Sciences, 2021, 158, pp.105685. ⟨10.1016/j.ejps.2020.105685⟩

Article dans une revue hal-04247571v1
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Nanomedicine-based delivery strategies for nucleic acid gene inhibitors in inflammatory diseases

Elias Fattal , François Fay

Advanced Drug Delivery Reviews, 2021, 175, pp.113809. ⟨10.1016/j.addr.2021.05.019⟩

Article dans une revue hal-04247580v1
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Tiny dexamethasone palmitate nanoparticles for intravitreal injection: optimization and in vivo evaluation

Romain Canioni , Franceline Reynaud , Thais Leite-Nascimento , Claire Gueutin , Nicolas Guiblin et al.

International Journal of Pharmaceutics, 2021, 600, pp.120509. ⟨10.1016/j.ijpharm.2021.120509⟩

Article dans une revue hal-03184392v1

Development of purified glycogen derivatives as siRNA nanovectors

Giuseppe Francesco Racaniello , Valentino Laquintana , Juliette Vergnaud , Angela Lopedota , Annalisa Cutrignelli et al.

International Journal of Pharmaceutics, 2021, 608, pp.121128. ⟨10.1016/j.ijpharm.2021.121128⟩

Article dans une revue hal-04247560v1

Nanotoxicology at the particle/micelle frontier: influence of core-polymerization on the intracellular distribution, cytotoxicity and genotoxicity of polydiacetylene micelles

Federica Costamagna , Hervé Hillaireau , Juliette Vergnaud-Gauduchon , Damien Clarisse , Lucie Jamgotchian et al.

Nanoscale, 2020, 12 (4), pp.2452-2463. ⟨10.1039/C9NR08714A⟩

Article dans une revue hal-02430885v1
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TREATMENT OF ACUTE LUNG INFLAMMATION BY PULMONARY DELIVERY OF ANTI-TNF-alpha SIRNA WITH PAMAM DENDRIMERS IN A MURINE MODEL

Adam Bohr , Nicolas Tsapis , Camilla Foged , Ilaria Andreana , Mingshi Yang et al.

European Journal of Pharmaceutics and Biopharmaceutics, 2020, 156, pp.114-120. ⟨10.1016/j.ejpb.2020.08.009⟩

Article dans une revue hal-02997033v1

A head-to-head Caco-2 assay comparison of the mechanisms of action of the intestinal permeation enhancers: SNAC and sodium caprate (C10)

Caroline Twarog , Kai Liu , Peter O'Brien , Kenneth Dawson , Elias Fattal et al.

European Journal of Pharmaceutics and Biopharmaceutics, 2020, 152, pp.95-107. ⟨10.1016/j.ejpb.2020.04.023⟩

Article dans une revue hal-04247658v1
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Nanomedicines for the delivery of glucocorticoids and nucleic acids as potential alternatives in the treatment of rheumatoid arthritis

Zhibo Yu , Franceline Reynaud , Mathilde Lorscheider , Nicolas Tsapis , Elias Fattal

Wiley Interdisciplinary Reviews: Nanomedicine and Nanobiotechnology, In press, ⟨10.1002/wnan.1630⟩

Article dans une revue hal-02893397v1

Synchronous insight of in vitro and in vivo biological activities of Sambucus nigra L. extracts for industrial uses

Ana Henriques Mota , Joana Andrade , Maria João Rodrigues , Luísa Custódio , Maria Rosário Bronze et al.

Industrial Crops and Products, 2020, 154, pp.112709. ⟨10.1016/j.indcrop.2020.112709⟩

Article dans une revue hal-04247534v1
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Controlled delivery of follicle-stimulating hormone in cattle

Quentin Deguettes , Elias Fattal , Marinette Moreau , Elodie Lego , Amélie Bochot

International Journal of Pharmaceutics, 2020, 590, pp.119904 -. ⟨10.1016/j.ijpharm.2020.119904⟩

Article dans une revue hal-03493591v1
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Stratégies thérapeutiques pour l’application clinique des ARN interférents

E. Fattal

Bulletin de l'Académie Nationale de Médecine, 2020, 204, pp.1088 - 1097. ⟨10.1016/j.banm.2020.06.013⟩

Article dans une revue hal-03493848v1

Nanotechnologies for Medical Devices: Potentialities and Risks

Arnaud Pallotta , Igor Clarot , Jonathan Sobocinski , Elias Fattal , Ariane Boudier

ACS Applied Bio Materials, 2019, 2 (1), pp.1-13. ⟨10.1021/acsabm.8b00612⟩

Article dans une revue hal-01976441v1
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Pyrazinoic acid-Poly(malic acid) biodegradable nanoconjugate for efficient intracellular delivery

Simone Pinto Carneiro , Laurence Moine , Barbara Tessier , Valérie Nicolas , Orlando David Henrique dos Santos et al.

Precision Nanomedicine, 2019, 2 (3), pp.303-317. ⟨10.33218/prnano2(3).190523.1⟩

Article dans une revue hal-02331736v1
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Biodegradable Pickering emulsions of Lipiodol for liver trans-arterial chemo-embolization

Frédéric Deschamps , Thomas Isoardo , Stéphanie Denis , Nicolas Tsapis , Lambros Tselikas et al.

Acta Biomaterialia, 2019, 87, pp.177-186. ⟨10.1016/j.actbio.2019.01.054⟩

Article dans une revue hal-02323562v1
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Dexamethasone palmitate nanoparticles: An efficient treatment for rheumatoid arthritis

Mathilde Lorscheider , Nicolas Tsapis , Mujeeb Ur-Rehman , Françoise Gaudin , Ivana Stolfa et al.

Journal of Controlled Release, 2019, 296, pp.179-189. ⟨10.1016/j.jconrel.2019.01.015⟩

Article dans une revue hal-02323608v1

Intestinal Permeation Enhancers for Oral Delivery of Macromolecules: A Comparison between Salcaprozate Sodium (SNAC) and Sodium Caprate (C10)

Caroline Twarog , Sarinj Fattah , Joanne Heade , Sam Maher , Elias Fattal et al. Article dans une revue hal-04352166v1

Design of Inhalable Solid Dosage Forms of Budesonide and Theophylline for Pulmonary Combination Therapy

Donglei Leng , Eric Ofosu Kissi , Korbinian Löbmann , Kaushik Thanki , Elias Fattal et al.

AAPS PharmSciTech, 2019, 20 (3), pp.137. ⟨10.1208/s12249-019-1344-9⟩

Article dans une revue hal-04247666v1
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Pickering emulsions: Preparation processes, key parameters governing their properties and potential for pharmaceutical applications

Claire Albert , Mohamed Beladjine , Nicolas Tsapis , Elias Fattal , Florence Agnely et al.

Journal of Controlled Release, 2019, 309, pp.302-332. ⟨10.1016/j.jconrel.2019.07.003⟩

Article dans une revue hal-02330281v1
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Immunotoxicity of poly (lactic-co-glycolic acid) nanoparticles: influence of surface properties on dendritic cell activation

S. Barillet , E. Fattal , S. Mura , N. Tsapis , M. Pallardy et al.

Nanotoxicology, 2019, 13 (5), pp.606-622. ⟨10.1080/17435390.2018.1564078⟩

Article dans une revue hal-02323703v2

Hyaluronic Acid–Decorated Liposomes as Innovative Targeted Delivery System for Lung Fibrotic Cells

Laura Pandolfi , Vanessa Frangipane , Claudia Bocca , Alessandro Marengo , Erika Tarro Genta et al. Article dans une revue hal-04352161v1
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Nanoscale Lipophilic Prodrugs of Dexamethasone with Enhanced Pharmacokinetics

Mathilde Lorscheider , Nicolas Tsapis , Rosana Simón-Vázquez , Nicolas Guiblin , Noureddine Ghermani et al.

Molecular Pharmaceutics, 2019, 16 (7), pp.2999-3010. ⟨10.1021/acs.molpharmaceut.9b00237⟩

Article dans une revue hal-02323659v1
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Pancreatic cancer stem cell proliferation is strongly inhibited by diethyldithiocarbamate-copper complex loaded into hyaluronic acid decorated liposomes

Alessandro Marengo , Stefania Forciniti , Ilaria Dando , Elisa Dalla Pozza , Barbara Stella et al.

Biochimica et Biophysica Acta (BBA) - General Subjects, 2019, 1863 (1), pp.61-72. ⟨10.1016/j.bbagen.2018.09.018⟩

Article dans une revue hal-02323431v1
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Formulation and comparison of spray dried non-porous and large porous particles containing meloxicam for pulmonary drug delivery

Anita Chvatal , Rita Ambrus , Petra Party , Gábor Katona , Orsolya Jójárt-Laczkovich et al.

International Journal of Pharmaceutics, 2019, 559, pp.68-75. ⟨10.1016/j.ijpharm.2019.01.034⟩

Article dans une revue hal-02323410v1

Encapsulation of echinomycin in cyclodextrin inclusion complexes into liposomes: in vitro anti-proliferative and anti-invasive activity in glioblastoma

Walhan Alshaer , Manar Zraikat , Amer Amer , Hamdi Nsairat , Zainab Lafi et al.

RSC Advances, 2019, 9 (53), pp.30976-30988. ⟨10.1039/C9RA05636J⟩

Article dans une revue hal-04247682v1
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From Poly(Alkyl Cyanoacrylate) to Squalene as Core Material to Design Nanomedicines

Simona Mura , Elias Fattal , Julien Nicolas

Journal of Drug Targeting, 2019, 27 (5-6), pp.470-501. ⟨10.1080/1061186X.2019.1579822⟩

Article dans une revue hal-02323788v1
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Cancer drug resistance: rationale for drug delivery systems and targeted inhibition of HSP90 family proteins

Clélia Mathieu , Samir Messaoudi , Elias Fattal , Juliette Vergnaud-Gauduchon

Cancer Drug Resistance, 2019, ⟨10.20517/cdr.2019.26⟩

Article dans une revue hal-02396633v1

Hyaluronated liposomes containing H2S-releasing doxorubicin are effective against P-glycoprotein-positive/doxorubicin-resistant osteosarcoma cells and xenografts

Elena Gazzano , Ilaria Buondonno , Alessandro Marengo , Barbara Rolando , Konstantin Chegaev et al.

Cancer Letters, 2019, ⟨10.1016/j.canlet.2019.04.029⟩

Article dans une revue hal-04352164v1

Restructuration kinetics of amphiphilic intraocular lenses during aging

Lionel Tortolano , Johanna Saunier , Senda Hammami , Katia Manerlax , Houssem Matmati et al.

Colloids and Surfaces B: Biointerfaces, 2018, 161, pp.420-432. ⟨10.1016/j.colsurfb.2017.11.007⟩

Article dans une revue hal-04352158v1
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Elucidating the role of surface chemistry on cationic phosphorus dendrimer–siRNA complexation

Marco A. Deriu , N. Tsapis , M. Noiray , G. Grasso , Nabil El brahmi et al.

Nanoscale, 2018, 10 (23), pp.10952-10962. ⟨10.1039/C8NR01928B⟩

Article dans une revue hal-01957985v1

Bare and Sterically Stabilized PLGA Nanoparticles for the Stabilization of Pickering Emulsions

Claire Albert , Nicolas Huang , Nicolas Tsapis , Sandrine Geiger , Véronique Rosilio et al.

Langmuir, 2018, 34 (46), pp.13935-13945. ⟨10.1021/acs.langmuir.8b02558⟩

Article dans une revue hal-04269455v1

Antitumor activity of nanoliposomes encapsulating the novobiocin analog 6BrCaQ in a triple-negative breast cancer model in mice

Félix Sauvage , Elias Fattal , Walhan Al-Shaer , Stéphanie Denis , Emilie Brotin et al.

Cancer Letters, 2018, 432, pp.103-111. ⟨10.1016/j.canlet.2018.06.001⟩

Article dans une revue istex inserm-02096216v1
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Protection against Clostridium difficile infection in a hamster model by oral vaccination using flagellin FliC-loaded pectin beads

J. F. Bruxelle , N. Tsapis , S. Hoys , A. Collignon , Claire Janoir et al.

Vaccine, 2018, 36 (40), pp.6017-6021. ⟨10.1016/j.vaccine.2018.08.013⟩

Article dans une revue hal-02323737v1

Engineering of budesonide-loaded lipid-polymer hybrid nanoparticles using a quality-by-design approach

Donglei Leng , Kaushik Thanki , Elias Fattal , Camilla Foged , Mingshi Yang

International Journal of Pharmaceutics, 2018, 548 (2), pp.740-746. ⟨10.1016/j.ijpharm.2017.08.094⟩

Article dans une revue hal-04352157v1
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Dexamethasone palmitate large porous particles: A controlled release formulation for lung delivery of corticosteroids

Alain N'Guessan , Elias Fattal , Claire Gueutin , Armand Koffi , Nicolas Tsapis et al.

European Journal of Pharmaceutical Sciences, 2018, 113, pp.185-192. ⟨10.1016/j.ejps.2017.09.013⟩

Article dans une revue hal-02323727v1
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Bare and Sterically Stabilized PLGA Nanoparticles for the Stabilization of Pickering Emulsions

Claire Albert , Nicolas Huang , Nicolas Tsapis , Sandrine Geiger , Véronique Rosilio et al.

Langmuir, 2018, 34 (46), pp.13935-13945. ⟨10.1021/acs.langmuir.8b02558⟩

Article dans une revue hal-01990240v1

Aptamer-guided nanomedicines for anticancer drug delivery

Walhan Alshaer , Hervé Hillaireau , Elias Fattal

Advanced Drug Delivery Reviews, 2018, 134, pp.122-137. ⟨10.1016/j.addr.2018.09.011⟩

Article dans une revue hal-04252726v1
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PLA-PEG Nanoparticles Improve the Anti-Inflammatory Effect of Rosiglitazone on Macrophages by Enhancing Drug Uptake Compared to Free Rosiglitazone

Giovanna Giacalone , Nicolas Tsapis , Ludivine Mousnier , Hélène Chacun , Elias Fattal

Materials, 2018, 11 (10), pp.1845. ⟨10.3390/ma11101845⟩

Article dans une revue hal-01990253v1

Aptamer-guided siRNA-loaded nanomedicines for systemic gene silencing in CD-44 expressing murine triple-negative breast cancer model

Walhan Alshaer , Hervé Hillaireau , Juliette Vergnaud , Simona Mura , Félix Sauvage et al.

Journal of Controlled Release, 2018, 271, pp.98-106. ⟨10.1016/j.jconrel.2017.12.022⟩

Article dans une revue hal-04252728v1
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Anti-Inflammatory effect of anti-TNF-α SiRNA cationic phosphorus dendrimer nanocomplexes administered intranasally in a murine acute lung injury model

Adam Bohr , N. Tsapis , I. Andreana , A. Chamarat , C. Foged et al.

Biomacromolecules, 2017, 18 (8), pp.2379-2388. ⟨10.1021/acs.biomac.7b00572⟩

Article dans une revue hal-01945636v1

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Article dans une revue inserm-02438401v1
Deposit thumbnail

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Article dans une revue inserm-02438261v1

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Deposit thumbnail

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Article dans une revue istex hal-04738841v1

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Article dans une revue hal-03110823v1
Deposit thumbnail

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Article dans une revue (article de synthèse) hal-04101325v1
Deposit thumbnail

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Article dans une revue hal-04101335v1
Deposit thumbnail

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Article dans une revue hal-04101322v1

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Deposit thumbnail

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Deposit thumbnail

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Article dans une revue hal-04101331v1
Deposit thumbnail

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Article dans une revue hal-04101306v1
Deposit thumbnail

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Deposit thumbnail

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Article dans une revue hal-04101301v1

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Article dans une revue istex hal-02962933v1
Deposit thumbnail

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Article dans une revue hal-04101317v1

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Article dans une revue istex hal-01762016v1

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Article dans une revue istex hal-02972646v1

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Article dans une revue istex hal-02330046v1

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Article dans une revue hal-02507538v1

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P. Fritsch , A.-L. Sérandour , O. Grémy , B. Le Gall , G. Phan et al.

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Article dans une revue istex hal-00360291v1

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Maillard S , Gauduchon J , Marsaud V , Gouilleux F , Connault E et al.

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Innovative drug delivery nanosystems improve the anti-tumor activity in vitro and in vivo of anti-estrogens in human breast cancer and multiple myeloma

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Article dans une revue inserm-02532838v1

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C Le Visage , F Quaglia , M Dreux , S Ounnar , P Breton et al.

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Article dans une revue istex hal-03298639v1
Deposit thumbnail

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Article dans une revue hal-03222435v1