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Introduction of Structural Diversity at the C2 Position of Unsaturated Iminosugars through Palladium‐Catalyzed Cross‐Coupling Reactions
Quentin Joachim
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Delphine Carry
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Mattéo Di Pasquale
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Jérôme Marrot
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Suzuka Yamamoto
et al.
Article dans une revue
(article de synthèse)
hal-05326462
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Addition of Lithiated 1,3-Dithiane and Nitronate to Sugar-Derived Imines: Synthesis of Homoiminosugars and Pipecolic Acid Analogues
Thanh Van Tran
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Jérôme Marrot
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Suzuka Yamamoto
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Kosuke Yoshimura
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Isabelle Gillaizeau
et al.
Article dans une revue
hal-05248874
v1
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Addition of Lithiated 1,3-Dithiane and Nitronate to Sugar-Derived Imines: Synthesis of Homoiminosugars and Pipecolic Acid Analogues
Thanh Van Tran
,
Jérôme Marrot
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Suzuka Yamamoto
,
Kosuke Yoshimura
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Isabelle Gillaizeau
et al.
Article dans une revue
hal-05326469
v1
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Glycosylium Ions in Superacid Mimic the Transition State of Enzyme Reactions
Mathilde Armand
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Alba Nin-Hill
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Ana Ardá
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Emanuela Berrino
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Jérôme Désiré
et al.
Article dans une revue
hal-05326476
v1
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Glycosylium Ions in Superacid Mimic the Transition State of Enzyme Reactions
Mathilde Armand
,
Alba Nin-Hill
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Ana Ardá
,
Emanuela Berrino
,
Jérôme Désiré
et al.
Article dans une revue
hal-05176253
v1
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Evaluation of nonnatural L-iminosugar C,C-glycosides, a new class of C-branched iminosugars, as glycosidase inhibitors
Jérôme Désiré
,
Zakaria Debbah
,
David Gueyrard
,
Jérôme Marrot
,
Yves Blériot
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Article dans une revue
(article de synthèse)
hal-05326478
v1
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Evaluation of nonnatural L-iminosugar C,C-glycosides, a new class of C-branched iminosugars, as glycosidase inhibitors
Jérôme Désiré
,
Zakaria Debbah
,
David Gueyrard
,
Jérôme Marrot
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Yves Blériot
et al.
Article dans une revue
hal-04542506
v1
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Stereoselective Access to Iminosugar C , C -Glycosides from 6-Azidoketopyranoses
Zakaria Debbah
,
Jérôme Marrot
,
Nicolas Auberger
,
Jérôme Désiré
,
Yves Blériot
Article dans une revue
(article de synthèse)
hal-05326481
v1
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Structural variation of the 3-acetamido-4,5,6-trihydroxyazepane iminosugar through epimerization and C -alkylation leads to low micromolar HexAB and NagZ inhibitors
J. Bouquet
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N. Auberger
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R. Ashmus
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D. King
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A. Bordes
et al.
Article dans une revue
hal-04526197
v1
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Stereoselective Synthesis of 1- C -Diethylphosphonomethyl and -difluoromethyl Iminosugars from Sugar Lactams
Thanh Van Tran
,
Jérôme Désiré
,
Nicolas Auberger
,
Yves Blériot
Article dans une revue
hal-03953681
v1
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Synthesis, conformational analysis and glycosidase inhibition of bicyclic nojirimycin C-glycosides based on an octahydrofuro[3,2-b]pyridine motif
Jérôme Désiré
,
Quentin Foucart
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Ana Poveda
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Gurvan Gourlaouen
,
Yuna Shimadate
et al.
Article dans une revue
hal-04542825
v1
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Stereoselective Access to Iminosugar C, C-Glycosides from 6-Azidoketopyranoses
Zakaria Debbah
,
Jérôme C. Marrot
,
Nicolas Auberger
,
Jérôme Désiré
,
Yves Blériot
Article dans une revue
hal-03775104
v1
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Sugar-Derived Amidines and Congeners: Structures, Glycosidase Inhibition and Applications
Yves Blériot
,
Nicolas Auberger
,
Jérôme Désiré
Article dans une revue
(article de synthèse)
hal-04543430
v1
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Insight into the Ferrier rearrangement by combining flash chemistry and superacids
Naresh Bhuma
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Ludivine Lebedel
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Hiroki Yamashita
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Yutaka Shimizu
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Zahra Abada
et al.
Article dans une revue
hal-03007376
v1
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Synthesis and chelation study of a fluoroionophore and a glycopeptide based on an aza crown iminosugar structure
Alexandra Bordes
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Ana Poveda
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Nathalie Fontelle
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Ana Ardá
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Jérôme Guillard
et al.
Article dans une revue
hal-04336072
v1
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Iminosugar-C-glycosides work as pharmacological chaperones of NAGLU, a glycosidase involved in MPS IIIB rare disease
Sha Zhu
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Yerri Jagadeesh
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Anh Tuan Tran
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Alisdair Boraston
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Dominic S Alonzi
et al.
Article dans une revue
hal-03256952
v1
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Synthesis, Conformational Analysis, and Complexation Study of an Iminosugar-Aza-Crown, a Sweet Chiral Cyclam Analog
Alexandra Bordes
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Ana Poveda
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Thibault Troadec
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Antonio Franconetti
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Ana Arda
et al.
Article dans une revue
hal-02504835
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Synthesis and glycosidase inhibition of conformationally locked DNJ and DMJ derivatives exploiting a 2-oxo- C -allyl iminosugar
Quentin Foucart
,
Yuna Shimadate
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Jérôme Marrot
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Atsushi Kato
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Jérôme Désiré
et al.
Article dans une revue
hal-04418307
v1
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Site-Selective Debenzylation of C -Allyl Iminosugars Enables Their Stereocontroled Structure Diversification at the C-2 Position
Quentin Foucart
,
Jérôme Marrot
,
Jérôme Désiré
,
Yves Blériot
Article dans une revue
hal-04418300
v1
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2-Acetamido-2-deoxy- l -iminosugar C -Alkyl and C -Aryl Glycosides: Synthesis and Glycosidase Inhibition
Balkis Eddhif
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Justin Lange
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Nadia Guignard
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Yann Batonneau
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Jonathan A. Clarhaut
et al.
Article dans une revue
hal-02172201
v1
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Selective trihydroxylated azepane inhibitors of NagZ, a glycosidase involved in Pseudomonas aeruginosa resistance to β-lactam antibiotics
Jaufret Bouquet
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Dustin King
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G. Vadlamani
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G. Benzie
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Bogdan Iorga
et al.
Article dans une revue
hal-02176734
v1
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Conformational flexibility of the glycosidase NagZ allows it to bind structurally diverse inhibitors to suppress β-lactam antibiotic resistance
Grishma Vadlamani
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Keith A Stubbs
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Jerome Desire
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Yves Blériot
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David J. Vocadlo
et al.
Article dans une revue
hal-02176780
v1
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HF-Induced Intramolecular C -Arylation and C -Alkylation/Fluorination of 2-Aminoglycopyranoses
Nicolas Probst
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Amélie Martin
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Jérôme Désiré
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Agnès Mingot
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Jerome Marrot
et al.
Article dans une revue
hal-01743477
v1
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Multivalency To Inhibit and Discriminate Hexosaminidases
Dimitri Alvarez-Dorta
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Dustin King
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Thibaut Legigan
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Daisuke Ide
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Isao Adachi
et al.
Article dans une revue
hal-01744683
v1
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In silico analyses of essential interactions of iminosugars with the Hex A active site and evaluation of their pharmacological chaperone effects for Tay–Sachs disease
Atsushi Kato
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Izumi Nakagome
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Shinpei Nakagawa
,
Kyoko Kinami
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Isao Adachi
et al.
Article dans une revue
hal-02176719
v1
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Catching elusive glycosyl cations in a condensed phase with HF/SbF₅ superacid
A. Martin
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A. Arda
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J. Désiré
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A. Martin-Mingot
,
N. Probst
et al.
Article dans une revue
hal-01505628
v1
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gamma-Aminoalcohol rearrangement applied to pentahydroxylated azepanes provides pyrrolidines epimeric to homoDMDP
Y. Jagadeesh
,
A.T. Tuan
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B. Luo
,
A. Auberger
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J. Desire
et al.
Article dans une revue
hal-01340188
v1
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Synthesis of pyrrolidine-based analogues of 2-acetamidosugars as N-acetyl glucosaminidase inhibitors
Anh Tuan Tran
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Bo Luo
,
Jagadeesh Yerri
,
Nicolas Auberger
,
Jérôme Désiré
et al.
Article dans une revue
hal-01136039
v1
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Synthetic deoxynojirimycin derivatives bearing a thiolated, fluorinated or unsaturated N-alkyl chain: identification of potent α-glucosidase and trehalase inhibitors as well as F508del-CFTR correctors.
V. Cendret
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T. Legigan
,
A. Martin-Mingot
,
S. Thibaudeau
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I. Adachi
et al.
Article dans une revue
hal-01500682
v1
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γ-Aminoalcohol rearrangement applied to pentahydroxylated azepanes provides pyrrolidines epimeric to homoDMDP
Y. Jagadeesh
,
A. Tran
,
B. Luo
,
N. Auberger
,
J. Désiré
et al.
Article dans une revue
hal-04543396
v1
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Superacid and thiol-ene reactions for access to psammaplin analogues with HDAC inhibition activities
Fatima El Bahhaj
,
Jerome Desire
,
Christophe Blanquart
,
Nadine Martinet
,
Vincent Zwick
et al.
Article dans une revue
istex
hal-01314516
v1
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Synthesis of 1,2-trans-2-Acetamido-2-deoxyhomoiminosugars
Yves Blériot
,
Anh Tuan Tran
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Giuseppe Prencipe
,
Jagadeesh Yerri
,
Nicolas Auberger
et al.
Article dans une revue
hal-01315627
v1
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N- and C-alkylation of seven-membered iminosugars generates potent glucocerebrosidase inhibitors and F508del-CFTR correctors
J. Désiré
,
M. Mondon
,
N. Fontelle
,
S. Nakagawa
,
Y. Hirokami
et al.
Article dans une revue
hal-01311606
v1
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Synthesis of 1,2-cis-Homoiminosugars Derived from GlcNAc and GalNAc Exploiting a β-Amino Alcohol Skeletal Rearrangement
Yves Blériot
,
Nicolas Auberger
,
Jagadeesh Yerri
,
Charles Gauthier
,
Giuseppe Prencipe
et al.
Article dans une revue
hal-01315083
v1
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Novel imino sugar α-glucosidase inhibitors as antiviral drugs
J.D. Howe
,
N. Smith
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L.J. Marvin
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N. Ardes-Guillot
,
J. Désiré
et al.
Article dans une revue
istex
hal-00932306
v1
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Cyclodextrin-glycerol dimers: synthesis and NMR conformational analysis
V. Legros
,
C. Vanhaverbeke
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F. Souard
,
C. Len
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J. Désiré
Article dans une revue
istex
hal-00934169
v1
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Novel imino sugar α-glucosidase inhibitors as antiviral compounds.
J. D. Howe
,
N. Smith
,
M. J.-R. Lee
,
N. Ardes-Guisot
,
B. Vauzeilles
et al.
Article dans une revue
istex
hal-00856804
v1
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Access to l- and d-Iminosugar C-Glycosides from a d-gluco-Derived 6-Azidolactol Exploiting a Ring Isomerization/Alkylation Strategy.
Martine Mondon
,
Nathalie Fontelle
,
Jérôme Désiré
,
Frédéric Lecornué
,
Jérôme Guillard
et al.
Article dans une revue
hal-00669930
v1
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Synthesis and conformational analysis of bicyclic mimics of alpha- and beta-D-glucopyranosides adopting the biologically relevant 2,5B conformation
L. Amorim
,
Farias Marcelo
,
J. Désiré
,
M. Sollogoub
,
J. Jimenez-Barbero
et al.
Article dans une revue
istex
hal-00834859
v1
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A Peptide Nucleic Acid-Aminosugar Conjugate Targeting Transactivation Response Element of HIV-1 RNA Genome Shows a High Bioavailability in Human Cells and Strongly Inhibits Tat-Mediated Transactivation of HIV-1 Transcription
I. Das
,
J. Désiré
,
D. Manvar
,
I. Baussanne
,
V.N. Pandey
et al.
Article dans une revue
hal-00838407
v1
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Toward the Supramolecular Cyclodextrin Dimers Using Nucleobase Pairs
Vanessa Legros
,
Florian Hamon
,
Bruno Violeau
,
Frédéric Turpin
,
Florence Djedaini-Pilard
et al.
Article dans une revue
hal-02944637
v1
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Anti-retroviral and cytostatic activity of 2',3'-dideoxyribonucleotide 3'-disulfides.
Béatrice Gerland
,
Jerome Desire
,
Jan Balzarini
,
Jean Luc Decout
Article dans une revue
istex
hal-00383176
v1
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Covalently bonded DNA aptamer chiral stationary phase for the chromatographic resolution of adenosine.
J. Ruta
,
Corinne Ravelet
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J. Désiré
,
Jean Luc Decout
,
E. Peyrin
Article dans une revue
istex
hal-00383152
v1
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Mechanism of RNA cleavage catalyzed by sequence specific polyamide nucleic acid-neamine conjugate.
B. Chaubey
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S. Tripathi
,
Jerome Desire
,
I. Baussanne
,
Jean Luc Decout
et al.
Article dans une revue
hal-00383208
v1
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Direct preparation of nucleoside vinyl disulfides from 2-(trimethylsilyl)ethyl sulfides, an access to vinylthiols.
Jean Luc Decout
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J. Désiré
,
Béatrice Gerland
,
Michel Lepoivre
Organic Letters, 2007, pp.3021-3023
Article dans une revue
hal-00382953
v1
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Neamine dimers targeting the HIV-1 TAR RNA.
Emmanuel Riguet
,
Jerome Desire
,
Oliver Boden
,
Verena Ludwig
,
Michael Göbel
et al.
Bioorganic and Medicinal Chemistry Letters, 2005, 15, pp.4651-4655
Article dans une revue
hal-00382910
v1
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Neamine dimers targeting the HIV-1 TAR RNA.
Jean Luc Decout
,
J. Désiré
,
E. Riguet
,
O. Boden
,
V. Ludwig
et al.
Article dans une revue
istex
hal-00123107
v1
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Imino glycals in synthesis : preparation of novel deoxymannojirimycin analogues
J. Désiré
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M. Shipman
Article dans une revue
hal-00123045
v1
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