Mélanie Etheve

43
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Publications

Publications

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Synthesis of Bisubstrate Analogues for RNA Methylation Studies using two Transition‐Metal‐Catalyzed Reactions

Dylan Coelho , Laurent Le Corre , Karolina Bartosik , Laura Iannazzo , Emmanuelle Braud et al.
Chemistry - A European Journal, 2023, 29 (44), ⟨10.1002/chem.202301134⟩
Article dans une revue hal-04246592 v1
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PSL Chemical Biology Symposia Third Edition: A Branch of Science in its Explosive Phase

Leeroy Baron , Justine Hadjerci , Leishemba Thoidingjam , Marina Plays , Romain Bucci et al.
ChemBioChem, 2023, 24 (8), pp.e202300093. ⟨10.1002/cbic.202300093⟩
Article dans une revue hal-04092530 v1
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Traceless Staudinger Ligation to Access Stable Aminoacyl- or Peptidyl-Dinucleotide

Camélia Kitoun , Saidbakhrom Saidjalolov , Delphine Bouquet , Fabiola Djago , Quentin Blancart-Remaury et al.
ACS Omega, 2023, 8 (4), pp.3850-3860. ⟨10.1021/acsomega.2c06135⟩
Article dans une revue hal-04294940 v1
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Amino-acyl tXNA as inhibitors or amino acid donors in peptide synthesis

Lauriane Rietmeyer , Inès Li de la Sierra-Gallay , Guy Schepers , Delphine Dorchêne , Laura Iannazzo et al.
Nucleic Acids Research, 2022, ⟨10.1093/nar/gkac1023⟩
Article dans une revue hal-03879768 v1

Synthesis of RNA-cofactor conjugates and structural exploration of RNA recognition by an m6A RNA methyltransferase

Vincent Meynier , Laura Iannazzo , Marjorie Catala , Stephanie Oerum , Emmanuelle Braud et al.
Nucleic Acids Research, 2022, ⟨10.1093/nar/gkac354⟩
Article dans une revue hal-03689976 v1
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Enzymatic synthesis of vancomycin-modified DNA

Chiara Figazzolo , Frédéric Bonhomme , Saidbakhrom Saidjalolov , Mélanie Ethève-Quelquejeu , Marcel Hollenstein
Molecules, 2022, 27 (24), pp.8927. ⟨10.3390/molecules27248927⟩
Article dans une revue hal-03927068 v1
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Traceless Staudinger Ligation To Introduce Chemical Diversity on β-Lactamase Inhibitors of Second Generation

Flavie Bouchet , Heiner Atze , Michel Arthur , Mélanie Ethève-Quelquejeu , Laura Iannazzo
Organic Letters, 2021, 23 (20), pp.7755-7758. ⟨10.1021/acs.orglett.1c02741⟩
Article dans une revue hal-03647098 v1
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Synthesis of carbapenems containing peptidoglycanmimetics and inhibition of the cross-linking activity of a transpeptidase of the L,D specificity

Saidbakhrom Saidjalolov , Zainab Edoo , Matthieu Fonvielle , Louis Mayer , Laura Iannazzo et al.
Chemistry - A European Journal, 2021, 27 (10), pp.3542-3551. ⟨10.1002/chem.202004831⟩
Article dans une revue hal-03184204 v1

Traceless Staudinger Ligation for Bioconjugation of RNA

Camélia Kitoun , Matthieu Fonvielle , Michel Arthur , Mélanie Etheve‐quelquejeu , Laura Iannazzo
Current Protocols, 2021, 1 (2), ⟨10.1002/cpz1.42⟩
Article dans une revue hal-03647120 v1
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Partition of tRNAGly isoacceptors between protein and cell-wall peptidoglycan synthesis in Staphylococcus aureus

Lauriane Rietmeyer , Nicolas Fix-Boulier , Chloé Le Fournis , Laura Iannazzo , Camelia Kitoun et al.
Nucleic Acids Research, 2021, 49 (2), pp.684-699. ⟨10.1093/nar/gkaa1242⟩
Article dans une revue hal-03201622 v1
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Click and Release Chemistry for Activity-Based Purification of β-Lactam Targets

Saidbakhrom Saidjalolov , Emmanuelle Braud , Zainab Edoo , Laura Iannazzo , Filippo Rusconi et al.
Chemistry - A European Journal, 2021, 27 (28), pp.7687-7695. ⟨10.1002/chem.202100653⟩
Article dans une revue hal-03281379 v1
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Phosphine-Mediated Bioconjugation of the 3′-End of RNA

Camelia Kitoun , Matthieu Fonvielle , Nicolas Sakkas , Manon Lefresne , Fabiola Djago et al.
Organic Letters, 2020, 22 (20), pp.8034-8038. ⟨10.1021/acs.orglett.0c02982⟩
Article dans une revue hal-02996863 v1
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Microwave-assisted synthesis of 2,5-disubstituted pyrimidine derivatives via Buchwald-Hartwig amination

Bo Li , Mélanie Etheve-Quelquejeu , Expédite Yen-Pon , Christiane Garbay , Huixiong Chen
Tetrahedron Letters, 2020, 61, pp.151406 -. ⟨10.1016/j.tetlet.2019.151406⟩
Article dans une revue hal-03488531 v1

Design and synthesis of a peptide derivative of ametantrone targeting the major groove of the d(GGCGCC) 2 palindromic sequence

Alberto Ongaro , Giovanni Ribaudo , Emmanuelle Braud , Mélanie Ethève-Quelquejeu , Michele de Franco et al.
New Journal of Chemistry, 2020, 44 (9), pp.3624-3631. ⟨10.1039/C9NJ03817E⟩
Article dans une revue hal-03689989 v1
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Diazabicyclooctane Functionalization for Inhibition of β-Lactamases from Enterobacteria

Flavie Bouchet , Heiner Atze , Matthieu Fonvielle , Zainab Edoo , Michel Arthur et al.
Journal of Medicinal Chemistry, 2020, 63 (10), pp.5257-5273. ⟨10.1021/acs.jmedchem.9b02125⟩
Article dans une revue hal-03646829 v2
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Raman reporters derived from aryl diazonium salts for SERS encoded-nanoparticles

Yun Luo , Yu Xiao , Delphine Onidas , Laura Iannazzo , Mélanie Ethève-Quelquejeu et al.
Chemical Communications, 2020, 56 (50), pp.6822-6825. ⟨10.1039/d0cc02842h⟩
Article dans une revue hal-03411993 v1
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Synthesis of triazole-linked SAM-adenosine 2 conjugates: functionalization of adenosine at N-1 or N-6 position without protecting groups

Colette Atdjian , Dylan Coelho , Laura Iannazzo , Mélanie Etheve-Quelquejeu , Emmanuelle Braud
Molecules, 2020, 25 (14), pp.3241. ⟨10.3390/molecules25143241⟩
Article dans une revue hal-02915430 v1

The neurobehavioral effects of the designer drug naphyrone – an experimental investigation with pharmacokinetics and concentration/effect relationship in mice

Bruno Mégarbane , Camille Gamblin , Olivier Roussel , Elodie Bouaziz-Amar , Lucie Chevillard et al.
Psychopharmacology, 2020, 237 (7), pp.1943-1957. ⟨10.1007/s00213-020-05510-2⟩
Article dans une revue hal-03823023 v1
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Negative impact of carbapenem methylation on the reactivity of β-lactams for cysteine acylation revealed by quantum calculations and kinetic analyses

Nicholus Bhattacharjee , Sébastien Triboulet , Vincent Dubée , Matthieu Fonvielle , Zainab Edoo et al.
Antimicrobial Agents and Chemotherapy, 2019, 63 (4), pp.e02039-18. ⟨10.1128/AAC.02039-18⟩
Article dans une revue hal-02057268 v1

Is the 3,4-methylendioxypyrovalerone/mephedrone combination responsible for enhanced stimulant effects? A rat study with investigation of the effect/concentration relationships

Nadia Benturquia , Lucie Chevillard , Christophe Poiré , Olivier Roussel , Camille Cohier et al.
Psychopharmacology, 2019, 236 (3), pp.891-901. ⟨10.1007/s00213-018-4962-0⟩
Article dans une revue hal-03823031 v1

Is the 3,4-methylendioxypyrovalerone/mephedrone combination responsible for enhanced stimulant effects? A rat study with investigation of the effect/concentration relationships

Nadia Benturquia , Lucie Chevillard , Christophe Poiré , Olivier Roussel , Camille Cohier et al.
Psychopharmacology, 2019, 236 (3), pp.891-901. ⟨10.1007/s00213-018-4962-0⟩
Article dans une revue hal-03860105 v1

Acute and chronic neurobehavioral effects of the designer drug and bath salt constituent 3,4-methylenedioxypyrovalerone in the rat

Luisa Alessandra Atehortua-Martinez , Cyriaque Masniere , Patrizia Campolongo , Stéphanie Chasseigneaux , Jacques Callebert et al.
Journal of Psychopharmacology, 2019, 33 (3), pp.392-405. ⟨10.1177/0269881118822151⟩
Article dans une revue hal-03860016 v1

Acute and chronic neurobehavioral effects of the designer drug and bath salt constituent 3,4-methylenedioxypyrovalerone in the rat

Luisa Alessandra Atehortua-Martinez , Cyriaque Masniere , Patrizia Campolongo , Stéphanie Chasseigneaux , Jacques Callebert et al.
Journal of Psychopharmacology, 2019, 33 (3), pp.392-405. ⟨10.1177/0269881118822151⟩
Article dans une revue hal-02557840 v1
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Bisubstrate analogues as structural tools to investigate m 6 A methyltransferase active sites

Stephanie Oerum , Marjorie Catala , Colette Atdjian , Franck Brachet , Luc Ponchon et al.
RNA Biology, 2019, 16 (6), pp.798-808. ⟨10.1080/15476286.2019.1589360⟩
Article dans une revue hal-02353503 v1

Acute and chronic neurobehavioral effects of the designer drug and bath salt constituent 3,4-methylenedioxypyrovalerone in the rat

Luisa Alessandra Atehortua-Martinez , Cyriaque Masniere , Patrizia Campolongo , Stéphanie Chasseigneaux , Jacques Callebert et al.
Journal of Psychopharmacology, 2019, 33 (3), pp.392-405. ⟨10.1177/0269881118822151⟩
Article dans une revue hal-03908457 v1

Synthesis of SAM-Adenosine Conjugates for the Study of m 6 A-RNA Methyltransferases

Colette Atdjian , Laura Iannazzo , Emmanuelle Braud , Mélanie Ethève-Quelquejeu
European Journal of Organic Chemistry, 2018, 2018 (32), pp.4411-4425. ⟨10.1002/ejoc.201800798⟩
Article dans une revue hal-02353523 v1
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Synthesis of lipid-carbohydrate-peptidyl-RNA conjugates to explore the limits imposed by the substrate specificity of cell wall enzymes on the acquisition of drug resistance

Matthieu Fonvielle , Ahmed Bouhss , Coralie Hoareau , Delphine Patin , Dominique Mengin-Lecreulx et al.
Chemistry - A European Journal, 2018, 24 (56), pp.14911-14915. ⟨10.1002/chem.201802360⟩
Article dans une revue hal-01962025 v1
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Structure-Based Design, Synthesis, and Characterization of the First Irreversible Inhibitor of Focal Adhesion Kinase

Expédite Yen-Pon , Bo Li , Marta Acebrón-Garcia-De-Eulate , Céline Tomkiewicz-Raulet , John Dawson et al.
ACS Chemical Biology, 2018, 13 (8), pp.2067-2073. ⟨10.1021/acschembio.8b00250⟩
Article dans une revue hal-02196326 v1

Synthesis of SAM-Adenosine Conjugates for the Study of m 6 A-RNA Methyltransferases

Colette Atdjian , Laura Iannazzo , Emmanuelle Braud , Mélanie Ethève-Quelquejeu
European Journal of Organic Chemistry, 2018, 2018 (32), pp.4411-4425. ⟨10.1002/ejoc.201800798⟩
Article dans une revue hal-03689993 v1
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Critical Impact of Peptidoglycan Precursor Amidation on the Activity of l,d -Transpeptidases from Enterococcus faecium and Mycobacterium tuberculosis

Flora Ngadjeua , Emmanuelle Braud , Saidbakhrom Saidjalolov , Laura Iannazzo , Dirk Schnappinger et al.
Chemistry - A European Journal, 2018, 24 (22), pp.5743 - 5747. ⟨10.1002/chem.201706082⟩
Article dans une revue hal-01817697 v1

Synthesis of tRNA analogues containing a terminal ribose locked in the South conformation to study tRNA-dependent enzymes

Laura Iannazzo , Matthieu Fonvielle , Emmanuelle Braud , Hubert Hřebabecký , Eliška Procházková et al.
Organic & Biomolecular Chemistry, 2018, 16 (11), pp.1903-1911. ⟨10.1039/C8OB00019K⟩
Article dans une revue hal-03689994 v1

Is the 3,4-methylendioxypyrovalerone/mephedrone combination responsible for enhanced stimulant effects? A rat study with investigation of the effect/concentration relationships

Nadia Benturquia , Lucie Chevillard , Christophe Poiré , Olivier Roussel , Camille Cohier et al.
Psychopharmacology, 2018, ⟨10.1007/s00213-018-4962-0⟩
Article dans une revue hal-01899917 v1

Synthesis of SAM-Adenosine Conjugates for the Study of m 6 A-RNA Methyltransferases

Colette Atdjian , Laura Iannazzo , Emmanuelle Braud , Mélanie Ethève-Quelquejeu
European Journal of Organic Chemistry, 2018, 2018 (32), pp.4411-4425. ⟨10.1002/ejoc.201800798⟩
Article dans une revue hal-03647207 v1

Critical Impact of Peptidoglycan Precursor Amidation on the Activity of l,d -Transpeptidases from Enterococcus faecium and Mycobacterium tuberculosis

Flora Ngadjeua , Emmanuelle Braud , Saidbakhrom Saidjalolov , Laura Iannazzo , Dirk Schnappinger et al.
Chemistry - A European Journal, 2018, 24 (22), pp.5743-5747. ⟨10.1002/chem.201706082⟩
Article dans une revue hal-03647180 v1

Synthesis of Avibactam Derivatives and Activity on β-Lactamases and Peptidoglycan Biosynthesis Enzymes of Mycobacteria

Zainab Edoo , Laura Iannazzo , Fabrice Compain , Inès Li de La Sierra Gallay , Herman Van Tilbeurgh et al.
Chemistry - A European Journal, 2018, 24 (32), pp.8081--8086. ⟨10.1002/chem.201800923⟩
Article dans une revue hal-02177911 v1

Insights into the interaction of high potency inhibitor IRC-083864 with phosphatase CDC25

Manal Sarkis , Maria Miteva , Maria Chiara Dasso Lang , Maryse Jaouen , Marie-Agnès Sari et al.
Proteins: Structure, Function, and Bioinformatics, 2017, 85 (4), pp.593-601. ⟨10.1002/prot.25236⟩
Article dans une revue hal-03684762 v1

Insights into the interaction of high potency inhibitor IRC-083864 with phosphatase CDC25

Manal Sarkis , Maria Miteva , Maria Chiara Dasso Lang , Maryse Jaouen , Marie-Agnès Sari et al.
Proteins: Structure, Function, and Bioinformatics, 2017, 85 (4), pp.593-601. ⟨10.1002/prot.25236⟩
Article dans une revue hal-03689998 v1

Electrophilic RNA for Peptidyl-RNA Synthesis and Site-Specific Cross-Linking with tRNA-Binding Enzymes.

Matthieu Fonvielle , Nicolas Sakkas , Laura Iannazzo , Chloé Le fournis , Delphine Patin et al.
Angewandte Chemie International Edition, 2016, 55 (43), pp.13553-13557. ⟨10.1002/anie.201606843⟩
Article dans une revue istex hal-01440830 v1

Monitoring of reversible boronic acid–diol interactions by fluorine NMR spectroscopy in aqueous media

Laura Iannazzo , Erica Benedetti , Marjorie Catala , Mélanie Etheve-Quelquejeu , Carine Tisné et al.
Organic & Biomolecular Chemistry, 2015, 13 (33), pp.8817-8821. ⟨10.1039/c5ob01362c⟩
Article dans une revue hal-03544508 v1

Kinetic features of L,D-transpeptidase inactivation critical for β-lactam antibacterial activity.

Sébastien Triboulet , Vincent Dubée , Lauriane Lecoq , Catherine M Bougault , Jean-Luc Mainardi et al.
PLoS ONE, 2013, 8 (7), pp.e67831. ⟨10.1371/journal.pone.0067831⟩
Article dans une revue hal-01321589 v1

Fluoro-C-glycosides and fluoro-carbasugars, hydrolytically stable and synthetically challenging glycomimetics

Eric Leclerc , Xavier Pannecoucke , Mélanie Etheve-Quelquejeu , M. Sollogoub
Chemical Society Reviews, 2013, 42 (10), pp.4270-4283. ⟨10.1039/c2cs35403a⟩
Article dans une revue hal-00825637 v1

Crystal structure of a chiral binaphthyl porphyrin

Eric Rose , Nicolas Raoul , Mélanie Etheve-Quelquejeu , Emma Gallo , Bernard Boitrel et al.
Journal of Porphyrins and Phthalocyanines, 2012, 16 (3), pp.324-330. ⟨10.1142/S1088424612500393⟩
Article dans une revue hal-00863134 v1

Idiosyncratic features in tRNAs participating in bacterial cell wall synthesis

Régis Villet , Matthieu Fonvielle , Patricia Busca , Maryline Chemama , Antoine P. Maillard et al.
Nucleic Acids Research, 2007, 35 (20), pp.6870-6883. ⟨10.1093/nar/gkm778⟩
Article dans une revue hal-02331010 v1