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Aurones as new modulators of hypoxia inducible factor-1 (HIF-1) to prevent cardiac cell death
Léa Di Maria
,
Brayan Roulier
,
Morane Beaumet
,
Romain Haudecoeur
,
Ahcène Boumendjel
et al.
Article dans une revue
hal-05234686v1
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Bistable and Water‐Operable Hemiindigo Photoswitches Allow Optical Control of Acetylcholinesterase Activity with Visible Light
Letícia da Mata Lazinski
,
Morane Beaumet
,
Frédérique Loiseau
,
Cyril Goudet
,
Martial Boggio‐pasqua
et al.
Article dans une revue
hal-05339073v1
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Tyrosinase Inhibition and Antimelanogenic Effects of Resorcinol‐Containing Compounds
Morane Beaumet
,
Leticia M Lazinski
,
Marc Maresca
,
Romain Haudecoeur
Article dans une revue
hal-04768568v1
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Design and synthesis of 4-amino-2',4'-dihydroxyindanone derivatives as potent inhibitors of tyrosinase and melanin biosynthesis in human melanoma cells
Leticia Lazinski
,
Morane Beaumet
,
Brayan Roulier
,
Rémy Gay
,
Guy Royal
et al.
Article dans une revue
hal-04768565v1
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Expanding Chemical Frontiers: Approaches for Generating Diverse and Bioactive Natural Product-Like Compounds Libraries from Extracts
Aurélien Beato
,
Romain Haudecoeur
,
Benjamin Boucherle
,
Marine Peuchmaur
Article dans une revue
(article de synthèse)
hal-04604571v1
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Aurones and derivatives as promising New Delhi metallo-β-lactamase (NDM-1) inhibitors
Jérémy Caburet
,
Federica Verdirosa
,
Matis Moretti
,
Brayan Roulier
,
Giorgia Simoncelli
et al.
Article dans une revue
hal-04429770v1
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Design and Synthesis of Novel Amino and Acetamidoaurones with Antimicrobial Activities
Attilio Di Maio
,
Hamza Olleik
,
Elise Courvoisier-Dezord
,
Sophie Guillier
,
Fabienne Neulat-Ripoll
et al.
Article dans une revue
hal-04588387v1
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Catechol-mimicking transition-state analogues as non-oxidizable inhibitors of tyrosinases
Morane Beaumet
,
Leticia Lazinski
,
Marc Maresca
,
Romain Haudecoeur
Article dans une revue
hal-04768562v1
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Resorcinol-based hemiindigoid derivatives as human tyrosinase inhibitors and melanogenesis suppressors in human melanoma cells
Brayan Roulier
,
Inbal Rush
,
Leticia Lazinski
,
Basile Pérès
,
Hamza Olleik
et al.
Article dans une revue
hal-03998028v1
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Bioactive Aurones, Indanones, and Other Hemiindigoid Scaffolds: Medicinal Chemistry and Photopharmacology Perspectives
Leticia Lazinski
,
Guy Royal
,
Maxime Robin
,
Marc Maresca
,
Romain Haudecoeur
Article dans une revue
hal-03826221v1
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β-Carboline as a Privileged Scaffold for Multitarget Strategies in Alzheimer's Disease Therapy
Aurélien Beato
,
Anthonin Gori
,
Benjamin Boucherle
,
Marine Peuchmaur
,
Romain Haudecoeur
Article dans une revue
hal-04020932v1
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Targeting different binding sites in the CFTR structures allows to synergistically potentiate channel activity
Lionel Froux
,
Ahmad Elbahnsi
,
Benjamin Boucherle
,
Arnaud Billet
,
Nesrine Baatallah
et al.
Article dans une revue
hal-02924784v1
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Advances in the Design of Genuine Human Tyrosinase Inhibitors for Targeting Melanogenesis and Related Pigmentations
Brayan Roulier
,
Basile Pérès
,
Romain Haudecoeur
Article dans une revue
hal-04768552v1
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Aurone derivatives as promising antibacterial agents against resistant Gram-positive pathogens
Hamza Olleik
,
Samir Yahiaoui
,
Brayan Roulier
,
Elise Courvoisier-Dezord
,
Josette Perrier
et al.
Article dans une revue
hal-01988325v1
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Glycosyl-Substituted Dicarboxylates as Detergents for the Extraction, Overstabilization, and Crystallization of Membrane Proteins
Kim-Anh Nguyen
,
Marine Peuchmaur
,
Sandrine Magnard
,
Romain Haudecoeur
,
Cédric Boyère
et al.
Article dans une revue
hal-02329303v1
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Piperidinyl-embeded chalcones possessing anti PI3K delta inhibitory properties exhibit anti-atopic properties in preclinical models
Charles Dumontet
,
Guillaume Beck
,
Fabrice Gardebien
,
Romain Haudecoeur
,
Doriane Mahe
et al.
Article dans une revue
hal-02621220v1
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Traditional uses, phytochemistry and pharmacological properties of African Nauclea species: A review
Romain Haudecoeur
,
Marine Peuchmaur
,
Basile Pérès
,
Maxime Rome
,
Germain Sotoing Taïwe
et al.
Article dans une revue
hal-04019717v1
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2-Hydroxypyridine- N -oxide-Embedded Aurones as Potent Human Tyrosinase Inhibitors
Romain Haudecoeur
,
Marc Carotti
,
Aurélie Gouron
,
Marc Maresca
,
Elina Buitrago
et al.
Article dans une revue
hal-01617843v1
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Nauclea latifolia: biological activity and alkaloid phytochemistry of a West African tree
Benjamin Boucherle
,
Romain Haudecoeur
,
Emerson Ferreira Queiroz
,
Michel de Waard
,
Jean-Luc Wolfender
et al.
Article dans une revue
hal-02141583v1
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Are Human Tyrosinase and Related Proteins Suitable Targets for Melanoma Therapy?
Elina Buitrago
,
Renaud M Hardré
,
Romain Haudecoeur
,
Hélène Jamet
,
Catherine Belle
et al.
Article dans une revue
istex
hal-01644550v1
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Recombinant Tyrosinase from Polyporus arcularius : Overproduction in Escherichia coli , Characterization, and Use in a Study of Aurones as Tyrosinase Effectors
Eva Marková
,
Michael Kotik
,
Alena Křenková
,
Petr Man
,
Romain Haudecoeur
et al.
Article dans une revue
hal-01948810v1
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Synthetic G-Quartets as Versatile Nanotools for the Luminescent Detection of G-Quadruplexes
Aurélien Laguerre
,
Marine Levillain
,
Loïc Stefan
,
Romain Haudecoeur
,
Fares Katranji
et al.
Article dans une revue
hal-02125788v1
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Biomimetic synthesis of Tramadol
Florine Lecerf-Schmidt
,
Romain Haudecoeur
,
Basile Peres
,
Marc Ferreira Queiroz
,
Marc Marcourt
et al.
Article dans une revue
hal-01683298v1
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Investigation of Binding-Site Homology between Mushroom and Bacterial Tyrosinases by Using Aurones as Effectors
Romain Haudecoeur
,
Aurélie Gouron
,
Carole Dubois
,
Hélène Jamet
,
Mark Lightbody
et al.
Article dans une revue
istex
hal-01652214v1
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B-ring modified aurones as promising allosteric inhibitors of hepatitis C virus RNA-dependent RNA polymerase
Amel Meguellati
,
Abdelhakim Ahmed-Belkacem
,
Wei Yi
,
Romain Haudecoeur
,
Marie Crouillère
et al.
Article dans une revue
hal-04015683v1
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Multitasking Water-Soluble Synthetic G-Quartets: From Preferential RNA-Quadruplex Interaction to Biocatalytic Activity
Romain Haudecoeur
,
Loïc Stefan
,
David Monchaud
Article dans une revue
istex
hal-02125745v1
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Occurrence of the Synthetic Analgesic Tramadol in an African Medicinal Plant.
Ahcène Boumendjel
,
Germain Sotoing Taïwe
,
Elisabeth Ngo Bum
,
Tanguy Chabrol
,
Chantal Beney
et al.
Article dans une revue
istex
inserm-00874145v1
|
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African tree gets to the root of pain
Ahcène Boumendjel
,
Germain Sotoing Taïwe
,
Elisabeth Ngo Gum
,
Tanguy Chabrol
,
Chantal Beney
et al.
Article dans une revue
hal-01683403v1
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Porphyrin-templated synthetic G-quartet (PorphySQ): a second prototype of G-quartet-based G-quadruplex ligand
Hai-Jun Xu
,
Loïc Stefan
,
Romain Haudecoeur
,
Sophie Vuong
,
Philippe R. Richard
et al.
Article dans une revue
hal-02125728v1
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A Model of Smart G-Quadruplex Ligand
Romain Haudecoeur
,
Loïc Stefan
,
Franck Denat
,
David Monchaud
Article dans une revue
hal-02125742v1
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Discovery of Naturally Occurring Aurones That Are Potent Allosteric Inhibitors of Hepatitis C Virus RNA-Dependent RNA Polymerase.
Romain Haudecoeur
,
Abdelhakim Ahmed-Belkacem
,
Wei Yi
,
Antoine Fortuné
,
Rozenn Brillet
et al.
Article dans une revue
inserm-00618322v1
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|
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Refinement of arylthiosemicarbazone pharmacophore in inhibition of mushroom tyrosinase
Wei Yi
,
Carole Dubois
,
Samir Yahiaoui
,
Romain Haudecoeur
,
Catherine Belle
et al.
Article dans une revue
istex
hal-01655567v1
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