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            Update on the Discovery of Efflux Pump Inhibitors against Critical Priority Gram-Negative Bacteria
        
                            
                                                                                                            Nina Compagne
                                                                ,
                                                                                                                                Anais Vieira da Cruz
                                                                ,
                                                                                                                                Reinke Müller
                                                                ,
                                                                                                                                Ruben C. Hartkoorn
                                                                ,
                                                                                                                                Marion Flipo
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                             (article de synthèse)
                    
        
        
            
                
                    hal-03970073
                                            v1
                                    
            
        
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            Regioselective and Stereoselective Synthesis of Parthenolide Analogs by Acyl Nitroso-Ene Reaction and Their Biological Evaluation against Mycobacterium tuberculosis
        
                            
                                                                                                            Bruna Gioia
                                                                ,
                                                                                                                                Francesca Ruggieri
                                                                ,
                                                                                                                                Alexandre Biela
                                                                ,
                                                                                                                                Valérie Landry
                                                                ,
                                                                                                                                Pascal Roussel
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-04339224
                                            v1
                                    
            
        
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            Characterization of pyridylpiperazine-based efflux pump inhibitors for Acinetobacter baumannii
        
                            
                                                                                                            Juan-Carlos Jiménez-Castellanos
                                                                ,
                                                                                                                                Elizabeth Pradel
                                                                ,
                                                                                                                                Nina Compagne
                                                                ,
                                                                                                                                Anais Vieira da Cruz
                                                                ,
                                                                                                                                Marion Flipo
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-04397896
                                            v1
                                    
            
        
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            Optimization of pyridylpiperazine-based inhibitors of the Escherichia coli AcrAB-TolC efflux pump
        
                            
                                                                                                            Nina Compagne
                                                                ,
                                                                                                                                Juan-Carlos Jiménez-Castellanos
                                                                ,
                                                                                                                                Virginie Meurillon
                                                                ,
                                                                                                                                Elizabeth Pradel
                                                                ,
                                                                                                                                Anais Vieira da Cruz
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-04165261
                                            v1
                                    
            
        
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            2,6-Disubstituted 7-(naphthalen-2-ylmethyl)-7H-purines as a new class of potent antitubercular agents inhibiting DprE1
        
                            
                                                                                                            Vladimir Finger
                                                                ,
                                                                                                                                Tomas Kucera
                                                                ,
                                                                                                                                Radka Kafkova
                                                                ,
                                                                                                                                Lubica Muckova
                                                                ,
                                                                                                                                Rafael Dolezal
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-04465147
                                            v1
                                    
            
        
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            A Novel Natural Siderophore Antibiotic Conjugate Reveals a Chemical Approach to Macromolecule Coupling
        
                            
                                                                                                            Thibault Caradec
                                                                ,
                                                                                                                                Ernesto Anoz-Carbonell
                                                                ,
                                                                                                                                Ravil Petrov
                                                                ,
                                                                                                                                Muriel Billamboz
                                                                ,
                                                                                                                                Kevin Antraygues
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-04444864
                                            v1
                                    
            
        
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            Pyridylpiperazine efflux pump inhibitor boosts in vivo antibiotic efficacy against K. pneumoniae
        
                            
                                                                                                            Anais Vieira da Cruz
                                                                ,
                                                                                                                                Juan-Carlos Jiménez-Castellanos
                                                                ,
                                                                                                                                Clara Börnsen
                                                                ,
                                                                                                                                Laurye van Maele
                                                                ,
                                                                                                                                Nina Compagne
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-04397794
                                            v1
                                    
            
        
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            Pyridylpiperazine-based allosteric inhibitors of RND-type multidrug efflux pumps
        
                            
                                                                                                            Coline Plé
                                                                ,
                                                                                                                                Heng-Keat Tam
                                                                ,
                                                                                                                                Anais Vieira da Cruz
                                                                ,
                                                                                                                                Nina Compagne
                                                                ,
                                                                                                                                Juan-Carlos Jiménez-Castellanos
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-03521512
                                            v1
                                    
            
        
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            Dactylosporolides: Glycosylated Macrolides from Dactylosporangium fulvum
        
                            
                                                                                                            Thibault Caradec
                                                                ,
                                                                                                                                Xavier Trivelli
                                                                ,
                                                                                                                                Eva Desmecht
                                                                ,
                                                                                                                                Veronique Peucelle
                                                                ,
                                                                                                                                Ruben Christiaan Hartkoorn
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-04464884
                                            v1
                                    
            
        
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            Tricyclic SpiroLactams Kill Mycobacteria In Vitro and In Vivo by Inhibiting Type II NADH Dehydrogenases
        
                            
                                                                                                            Sushovan Dam
                                                                ,
                                                                                                                                Salia Tangara
                                                                ,
                                                                                                                                Claire Hamela
                                                                ,
                                                                                                                                Theo Hattabi
                                                                ,
                                                                                                                                Léo Faïon
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-04017354
                                            v1
                                    
            
        
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            Rubrolone production by Dactylosporangium vinaceum: biosynthesis, modulation and possible biological function
        
                            
                                                                                                            Sophie Moureu
                                                                ,
                                                                                                                                Thibault Caradec
                                                                ,
                                                                                                                                Xavier Trivelli
                                                                ,
                                                                                                                                Hervé Drobecq
                                                                ,
                                                                                                                                Delphine Beury
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-03360998
                                            v1
                                    
            
        
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            Intragenic Distribution of IS 6110 in Clinical Mycobacterium tuberculosis Strains: Bioinformatic Evidence for Gene Disruption Leading to Underdiagnosed Antibiotic Resistance
        
                            
                                                                                                            Rudy Antoine
                                                                ,
                                                                                                                                Cyril Gaudin
                                                                ,
                                                                                                                                Ruben Christiaan Hartkoorn
                                                                                    
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-04462804
                                            v1
                                    
            
        
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            Synthesis and Structure–Activity Relationship Studies of C2-Modified Analogs of the Antimycobacterial Natural Product Pyridomycin
        
                            
                                                                                                            Maryline Kienle
                                                                ,
                                                                                                                                Patrick Eisenring
                                                                ,
                                                                                                                                Barbara Stoessel
                                                                ,
                                                                                                                                Oliver Horlacher
                                                                ,
                                                                                                                                Samuel Hasler
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-04462810
                                            v1
                                    
            
        
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            Pyrrolomycins Are Potent Natural Protonophores
        
                            
                                                                                                            Katherine Valderrama
                                                                ,
                                                                                                                                Elizabeth Pradel
                                                                ,
                                                                                                                                Alexander M. Firsov
                                                                ,
                                                                                                                                Hervé Drobecq
                                                                ,
                                                                                                                                Hélène Bauderlique-Le Roy
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-03361019
                                            v1
                                    
            
        
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            Accelerated microfluidic native chemical ligation at difficult amino acids toward cyclic peptides
        
                            
                                                                                                            Nathalie Ollivier
                                                                ,
                                                                                                                                Thomas Toupy
                                                                ,
                                                                                                                                Ruben Hartkoorn
                                                                ,
                                                                                                                                Rémi Desmet
                                                                ,
                                                                                                                                Jean-Christophe Monbaliu
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-02133846
                                            v1
                                    
            
        
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            Total Synthesis of Ripostatin B and Structure–Activity Relationship Studies on Ripostatin Analogs
        
                            
                                                                                                            Florian Glaus
                                                                ,
                                                                                                                                Darija Dedić
                                                                ,
                                                                                                                                Priyanka Tare
                                                                ,
                                                                                                                                Valakunja Nagaraja
                                                                ,
                                                                                                                                Liliana Rodrigues
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-04462820
                                            v1
                                    
            
        
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            Characterization of new, efficient Mycobacterium tuberculosis topoisomerase-I inhibitors and their interaction with human ABC multidrug transporters
        
                            
                                                                                                            Csilla Temesszentandrási-Ambrus
                                                                ,
                                                                                                                                Szilárd Tóth
                                                                ,
                                                                                                                                Rinkee Verma
                                                                ,
                                                                                                                                Péter Bánhegyi
                                                                ,
                                                                                                                                István Szabadkai
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-04462816
                                            v1
                                    
            
        
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            A druggable secretory protein maturase of Toxoplasma essential for invasion and egress
        
                            
                                                                                                            Sunil Kumar Dogga
                                                                ,
                                                                                                                                Budhaditya Mukherjee
                                                                ,
                                                                                                                                Damien Jacot
                                                                ,
                                                                                                                                Tobias Kockmann
                                                                ,
                                                                                                                                Luca Molino
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-04462826
                                            v1
                                    
            
        
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            Discovery and Biosynthesis of Gladiolin: A Burkholderia gladioli Antibiotic with Promising Activity against Mycobacterium tuberculosis
        
                            
                                                                                                            Lijiang Song
                                                                ,
                                                                                                                                Matthew Jenner
                                                                ,
                                                                                                                                Joleen Masschelein
                                                                ,
                                                                                                                                Cerith Jones
                                                                ,
                                                                                                                                Matthew Bull
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-04462832
                                            v1
                                    
            
        
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            MoS2/TiO2/SiNW surface as an effective substrate for LDI-MS detection of glucose and glutathione in real samples
        
                            
                                                                                                            Abderrahmane Hamdi
                                                                ,
                                                                                                                                Ioana Silvia Hosu
                                                                ,
                                                                                                                                Ahmed Addad
                                                                ,
                                                                                                                                Ruben Hartkoorn
                                                                ,
                                                                                                                                Hervé Drobecq
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    hal-02133897
                                            v1
                                    
            
        
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            Thiophenecarboxamide Derivatives Activated by EthA Kill Mycobacterium tuberculosis by Inhibiting the CTP Synthetase PyrG
        
                            
                                                                                                            Giorgia Mori
                                                                ,
                                                                                                                                Laurent Chiarelli
                                                                ,
                                                                                                                                Marta Esposito
                                                                ,
                                                                                                                                Vadim Makarov
                                                                ,
                                                                                                                                Marco Bellinzoni
                                                                                            et al.
                            
                 
                            
                 Article dans une revue
                    
        
        
            
                
                    pasteur-03096090
                                            v1
                                    
            
        
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