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Update on the Discovery of Efflux Pump Inhibitors against Critical Priority Gram-Negative Bacteria
Nina Compagne
,
Anais Vieira da Cruz
,
Reinke Müller
,
Ruben C. Hartkoorn
,
Marion Flipo
et al.
Article dans une revue
(article de synthèse)
hal-03970073
v1
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Optimization of pyridylpiperazine-based inhibitors of the Escherichia coli AcrAB-TolC efflux pump
Nina Compagne
,
Juan-Carlos Jiménez-Castellanos
,
Virginie Meurillon
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Elizabeth Pradel
,
Anais Vieira da Cruz
et al.
Article dans une revue
hal-04165261
v1
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Characterization of pyridylpiperazine-based efflux pump inhibitors for Acinetobacter baumannii
Juan-Carlos Jiménez-Castellanos
,
Elizabeth Pradel
,
Nina Compagne
,
Anais Vieira da Cruz
,
Marion Flipo
et al.
Article dans une revue
hal-04397896
v1
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2,6-Disubstituted 7-(naphthalen-2-ylmethyl)-7H-purines as a new class of potent antitubercular agents inhibiting DprE1
Vladimir Finger
,
Tomas Kucera
,
Radka Kafkova
,
Lubica Muckova
,
Rafael Dolezal
et al.
Article dans une revue
hal-04465147
v1
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A Novel Natural Siderophore Antibiotic Conjugate Reveals a Chemical Approach to Macromolecule Coupling
Thibault Caradec
,
Ernesto Anoz-Carbonell
,
Ravil Petrov
,
Muriel Billamboz
,
Kevin Antraygues
et al.
Article dans une revue
hal-04444864
v1
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Regioselective and Stereoselective Synthesis of Parthenolide Analogs by Acyl Nitroso-Ene Reaction and Their Biological Evaluation against Mycobacterium tuberculosis
Bruna Gioia
,
Francesca Ruggieri
,
Alexandre Biela
,
Valérie Landry
,
Pascal Roussel
et al.
Article dans une revue
hal-04339224
v1
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Pyridylpiperazine efflux pump inhibitor boosts in vivo antibiotic efficacy against K. pneumoniae
Anais Vieira da Cruz
,
Juan-Carlos Jiménez-Castellanos
,
Clara Börnsen
,
Laurye van Maele
,
Nina Compagne
et al.
Article dans une revue
hal-04397794
v1
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Pyridylpiperazine-based allosteric inhibitors of RND-type multidrug efflux pumps
Coline Plé
,
Heng-Keat Tam
,
Anais Vieira da Cruz
,
Nina Compagne
,
Juan-Carlos Jiménez-Castellanos
et al.
Article dans une revue
hal-03521512
v1
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Tricyclic SpiroLactams Kill Mycobacteria In Vitro and In Vivo by Inhibiting Type II NADH Dehydrogenases
Sushovan Dam
,
Salia Tangara
,
Claire Hamela
,
Theo Hattabi
,
Léo Faïon
et al.
Article dans une revue
hal-04017354
v1
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Dactylosporolides: Glycosylated Macrolides from Dactylosporangium fulvum
Thibault Caradec
,
Xavier Trivelli
,
Eva Desmecht
,
Veronique Peucelle
,
Ruben Christiaan Hartkoorn
et al.
Article dans une revue
hal-04464884
v1
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Rubrolone production by Dactylosporangium vinaceum: biosynthesis, modulation and possible biological function
Sophie Moureu
,
Thibault Caradec
,
Xavier Trivelli
,
Hervé Drobecq
,
Delphine Beury
et al.
Article dans une revue
hal-03360998
v1
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Intragenic Distribution of IS 6110 in Clinical Mycobacterium tuberculosis Strains: Bioinformatic Evidence for Gene Disruption Leading to Underdiagnosed Antibiotic Resistance
Rudy Antoine
,
Cyril Gaudin
,
Ruben Christiaan Hartkoorn
Article dans une revue
hal-04462804
v1
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Synthesis and Structure–Activity Relationship Studies of C2-Modified Analogs of the Antimycobacterial Natural Product Pyridomycin
Maryline Kienle
,
Patrick Eisenring
,
Barbara Stoessel
,
Oliver Horlacher
,
Samuel Hasler
et al.
Article dans une revue
hal-04462810
v1
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Pyrrolomycins Are Potent Natural Protonophores
Katherine Valderrama
,
Elizabeth Pradel
,
Alexander M. Firsov
,
Hervé Drobecq
,
Hélène Bauderlique-Le Roy
et al.
Article dans une revue
hal-03361019
v1
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Total Synthesis of Ripostatin B and Structure–Activity Relationship Studies on Ripostatin Analogs
Florian Glaus
,
Darija Dedić
,
Priyanka Tare
,
Valakunja Nagaraja
,
Liliana Rodrigues
et al.
Article dans une revue
hal-04462820
v1
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Accelerated microfluidic native chemical ligation at difficult amino acids toward cyclic peptides
Nathalie Ollivier
,
Thomas Toupy
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Ruben Hartkoorn
,
Rémi Desmet
,
Jean-Christophe Monbaliu
et al.
Article dans une revue
hal-02133846
v1
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Characterization of new, efficient Mycobacterium tuberculosis topoisomerase-I inhibitors and their interaction with human ABC multidrug transporters
Csilla Temesszentandrási-Ambrus
,
Szilárd Tóth
,
Rinkee Verma
,
Péter Bánhegyi
,
István Szabadkai
et al.
Article dans une revue
hal-04462816
v1
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A druggable secretory protein maturase of Toxoplasma essential for invasion and egress
Sunil Kumar Dogga
,
Budhaditya Mukherjee
,
Damien Jacot
,
Tobias Kockmann
,
Luca Molino
et al.
Article dans une revue
hal-04462826
v1
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Discovery and Biosynthesis of Gladiolin: A Burkholderia gladioli Antibiotic with Promising Activity against Mycobacterium tuberculosis
Lijiang Song
,
Matthew Jenner
,
Joleen Masschelein
,
Cerith Jones
,
Matthew Bull
et al.
Article dans une revue
hal-04462832
v1
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MoS2/TiO2/SiNW surface as an effective substrate for LDI-MS detection of glucose and glutathione in real samples
Abderrahmane Hamdi
,
Ioana Silvia Hosu
,
Ahmed Addad
,
Ruben Hartkoorn
,
Hervé Drobecq
et al.
Article dans une revue
hal-02133897
v1
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Thiophenecarboxamide Derivatives Activated by EthA Kill Mycobacterium tuberculosis by Inhibiting the CTP Synthetase PyrG
Giorgia Mori
,
Laurent Chiarelli
,
Marta Esposito
,
Vadim Makarov
,
Marco Bellinzoni
et al.
Article dans une revue
pasteur-03096090
v1
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