Pascal VERDIE

Documents

Current affiliations

1100589

Researcher identifiers

pascal-verdie
0000-0002-5807-0293
IdRef : 087809729

Publications

	Targeting a lineage-specific PI3Kɣ–Akt signaling module in acute myeloid leukemia using a heterobifunctional degrader molecule Lois Kelly , Justine Rutter , Kevin Lin , Frank Ling , Matthieu Duchmann Nature Cancer, In press, Online ahead of print. ⟨10.1038/s43018-024-00782-5⟩ Journal articles hal-04598240v1
	Amelogenin-Derived Peptide (ADP-5) Hydrogel for Periodontal Regeneration: An In Vitro Study on Periodontal Cells Cytocompatibility, Remineralization and Inflammatory Profile Nina Attik , Xavier Garric , Audrey Bethry , Gilles Subra , Charlène Chevalier Journal of Functional Biomaterials, 2023, 14 (2), pp.53. ⟨10.3390/jfb14020053⟩ Journal articles hal-04628797v1
	Fast and Cost‐Efficient 17 O‐Isotopic Labeling of Carboxylic Groups in Biomolecules: From Free Amino Acids to Peptide Chains Jessica Špačková , Ieva Goldberga , Rishit Yadav , Guillaume Cazals , Aurélien Lebrun Chemistry - A European Journal, 2023, 29 (10), pp.e202203014. ⟨10.1002/chem.202203014⟩ Journal articles hal-04002744v1
	The C-terminal pentapeptide acein analogue (JMV3315) stimulates dopamine release in the brain Charlène Lucas-Valmalle , Gilles Subra , Pascal Verdié , Marie-Lou Kemel , Valérie Daugé Australian Journal of Chemistry, 2023, 76 (8), pp.448-454. ⟨10.1071/CH22232⟩ Journal articles hal-04604961v1
	Structural insights into recognition of chemokine receptors by Staphylococcus aureus leukotoxins Paul Lambey , Omolade Otun , Xiaojing Cong , François Hoh , Luc Brunel eLife, 2022, 11, pp.e72555. ⟨10.7554/eLife.72555⟩ Journal articles hal-03754372v1
	Peptide-guided self-assembly of polyethylene glycol-b-poly(ε-caprolactone-g-peptide) block copolymers Ayman El Jundi , Matthias Mayor , Enrique Folgado , Chaimaa Gomri , Belkacem Tarek Benkhaled European Polymer Journal, 2022, 176, pp.111386. ⟨10.1016/j.eurpolymj.2022.111386⟩ Journal articles hal-04065895v1
	Potent Lys Patch-containing Stapled Peptides Targeting PCSK9 Kevin Bourbiaux , Baptiste Legrand , Pascal Verdié , Sergio Mallart , Géraldine Manette Journal of Medicinal Chemistry, 2021, 64 (15), pp.10834-10848. ⟨10.1021/acs.jmedchem.0c02051⟩ Journal articles hal-03371411v1
	Active Targeted Nanoemulsions for Repurposing of Tegaserod in Alzheimer’s Disease Treatment Line Séguy , Léna Guyon , Manon Maurel , Pascal Verdié , Audrey Davis Pharmaceutics, 2021, 13 (10), pp.1626. ⟨10.3390/pharmaceutics13101626⟩ Journal articles hal-04570312v1
	JMV5656, a short synthetic derivative of TLQP-21, alleviates acid-induced lung injury and fibrosis in mice Vanessa Zambelli , Laura Rizzi , Paolo Delvecchio , Elena Bresciani , Laura Molteni Pulmonary Pharmacology and Therapeutics, 2020, 62, pp.101916. ⟨10.1016/j.pupt.2020.101916⟩ Journal articles hal-04549706v1
	Star-poly(lactide)-peptide hybrid networks as bioactive materials L.V. Arsenie , Coline Pinese , Audrey Bethry , L. Valot , P. Verdie European Polymer Journal, 2020, 139, pp.109990 -. ⟨10.1016/j.eurpolymj.2020.109990⟩ Journal articles hal-03491991v1
	Site-specific grafting on titanium surfaces with hybrid temporin antibacterial peptides Nicolas Masurier , Jean-Baptiste Tissot , Douae Boukhriss , Said Jebors , Coline Pinese Journal of materials chemistry‎ B, 2018, 6 (12), pp.1782 - 1790. ⟨10.1039/c8tb00051d⟩ Journal articles hal-01742222v1
	STIM Proteins and Orai Ca2+ Channels Are Involved in the Intracellular Pathways Activated by TLQP-21 in RAW264.7 Macrophages Laura Molteni , Laura Rizzi , Elena Bresciani , Ramona Meanti , Jean-Alain Fehrentz Frontiers in Pharmacology, 2018, 9, ⟨10.3389/fphar.2018.01386⟩ Journal articles hal-02871099v1
	Study of the Tissue Distribution of TLQP-21 in Mice Using [18F]JMV5763, a Radiolabeled Analog Prepared via [18F]Aluminum Fluoride Chelation Chemistry Elia Turolla , Silvia Valtorta , Elena Bresciani , Jean-Alain Fehrentz , Liliana Giuliano Frontiers in Pharmacology, 2018, 9, ⟨10.3389/fphar.2018.01274⟩ Journal articles hal-02871096v1
	[Erratum for] "Palatability Can Drive Feeding Independent of AgRP Neurons" Raphael Georges Denis , Aurélie Joly-Amado , Emily Webber , Fanny Langlet , Marie Schaeffer Cell Metabolism, 2017, 25 (4), pp.975. ⟨10.1016/j.cmet.2017.03.001⟩ Journal articles hal-02067393v1
	JMV5656, A Novel Derivative of TLQP-21, Triggers the Activation of a Calcium-Dependent Potassium Outward Current in Microglial Cells Ilaria Rivolta , Anna Binda , Laura Molteni , Laura Rizzi , Elena Bresciani Frontiers in Cellular Neuroscience, 2017, 11, pp.41. ⟨10.3389/fncel.2017.00041⟩ Journal articles hal-02871317v1
	Peptide synthesis: ball-milling, in solution, or on solid support, what is the best strategy? Ophélie Maurin , Pascal Verdié , Gilles Subra , Frédéric Lamaty , Jean Martinez Beilstein Journal of Organic Chemistry, 2017, 13, pp.2087-2093. ⟨10.3762/bjoc.13.206⟩ Journal articles hal-02336152v1
	Pharmacological and Biochemical Characterization of TLQP-21 Activation of a Binding Site on CHO Cells Laura Molteni , Laura Rizzi , Elena Bresciani , Roberta Possenti , Pamela Petrocchi Passeri Frontiers in Pharmacology, 2017, 8, pp.167. ⟨10.3389/fphar.2017.00167⟩ Journal articles hal-02871330v1
	Sol-gel synthesis of collagen-inspired peptide hydrogel Cécile Echalier , Said Jebors , Guillaume Laconde , Luc Brunel , Pascal Verdié Materials Today, 2017, 20 (2), pp.59-66. ⟨10.1016/j.mattod.2017.02.001⟩ Journal articles hal-01516237v1
	Systemic Delivery of Tumor-Targeted Bax-Derived Membrane-Active Peptides for the Treatment of Melanoma Tumors in a Humanized SCID Mouse Model Anastassia Karageorgis , Michaël Claron , Romain Jugé , Caroline Aspord , Fabien Thoreau Molecular Therapy, 2017, 25 (2), pp.534-546. ⟨10.1016/j.ymthe.2016.11.002⟩ Journal articles hal-02000186v1
	Bioactive peptides grafted silicone dressings: A simple and specific method Coline Pinese , Said Jebors , Pierre-Emmanuel Stoebner , Vincent Humblot , Pascal Verdié Materials Today Chemistry, 2017, 4, pp.73-83. ⟨10.1016/j.mtchem.2017.02.007⟩ Journal articles hal-01496701v1
	A switchable stapled peptide Aleksandra Kalistratova , Baptiste Legrand , Pascal Verdié , Emilia Naydenova , Muriel Amblard Journal of Peptide Science, 2016, 22 (3), pp.143-148. ⟨10.1002/psc.2851⟩ Journal articles hal-03564342v1
	Solid-Supported Synthesis and 5-HT 7 /5-HT 1A Receptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1 H )-one Katarzyna Grychowska , Nicolas Masurier , Pascal Verdié , Grzegorz Satała , Andrzej Bojarski Chemical Biology and Drug Design, 2015, 86 (4), pp.697-703. ⟨10.1111/cbdd.12539⟩ Journal articles hal-03564059v1
	Palatability Can Drive Feeding Independent of AgRP Neurons Raphael Georges Denis , Aurélie Joly-Amado , Emily Webber , Fanny Langlet , Marie Schaeffer Cell Metabolism, 2015, 22 (4), pp.646-657. ⟨10.1016/j.cmet.2015.07.011⟩ Journal articles hal-02067347v1
	Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling Céline M'Kadmi , Jean-Philippe Leyris , Lauriane Onfroy , Céline Galés , Aude Saulière Journal of Biological Chemistry, 2015, 290 (45), pp.27021-27039. ⟨10.1074/jbc.M115.659250⟩ Journal articles hal-03564155v1
	N- and O-acetylation of threonine residues in the context of proteomics. Jean-Baptiste Boyer , Alain Dedieu , J. Armengaud , Pascal Verdié , Gilles Subra Journal of Proteomics, 2014, 108, pp.369-372. ⟨10.1016/j.jprot.2014.06.005⟩ Journal articles hal-01025681v1
	Solid-supported synthesis, molecular modeling, and biological activity of long-chain arylpiperazine derivatives with cyclic amino acid amide fragments as 5-HT7 and 5-HT1A receptor ligands Vittorio Canale , Paweł Guzik , Rafał Kurczab , Pascal Verdie , Grzegorz Satała European Journal of Medicinal Chemistry, 2014, 78, pp.10-22. ⟨10.1016/j.ejmech.2014.03.005⟩ Journal articles hal-03563396v1
	Microwave-Mediated Reduction of Disulfide Bridges with Supported (Tris(2-carboxyethyl)phosphine) as Resin-Bound Reducing Agent Guillaume Miralles , Pascal Verdié , Karine Puget , Amélie Maurras , Jean Martinez ACS Combinatorial Science, 2013, 15 (4), pp.169-173. ⟨10.1021/co300104k⟩ Journal articles hal-03563025v1
	How ligands and signalling proteins affect G-protein-coupled receptors' conformational landscape Sophie Mary , Jean-Alain Fehrentz , Marjorie Damian , Pascal Verdie , Jean Martinez Biochemical Society Transactions, 2013, 41 (1), pp.144-147. ⟨10.1042/BST20120267⟩ Journal articles hal-02871941v1
	Supported oligomethionine sulfoxide and Ellman's reagent for cysteine bridges formation Luisa Ronga , Pascal Verdié , Pierre Sanchez , Christine Enjalbal , Amélie Maurras Amino Acids, 2013, 44 (2), pp.733-742. ⟨10.1007/s00726-012-1397-5⟩ Journal articles hal-01563741v1
	Heating and microwave assisted SPPS of C-terminal acid peptides on trityl resin: The truth behind the yield Cécile Echalier , Soultan Al-Halifa , Aude Kreiter , Christine Enjalbal , Pierre Sanchez Amino Acids, 2013, 45 (6), pp.1395-1403. ⟨10.1007/s00726-013-1604-z⟩ Journal articles hal-01563742v1
	Rapid sensing of circulating ghrelin by hypothalamic appetite-modifying neurons. Marie Schaeffer , Fanny Langlet , Chrystel Lafont , François Molino , David J Hodson Proceedings of the National Academy of Sciences of the United States of America, 2013, 110 (4), pp.1512-7. ⟨10.1073/pnas.1212137110⟩ Journal articles hal-00796900v1
	Heterodimerization with Its Splice Variant Blocks the Ghrelin Receptor 1a in a Non-signaling Conformation Sophie Mary , Jean-Alain Fehrentz , Marjorie Damian , Gérald Gaibelet , Hélène Orcel Journal of Biological Chemistry, 2013, 288 (34), pp.24656-24665. ⟨10.1074/jbc.M113.453423⟩ Journal articles hal-02871944v1
	Ghrelin Receptor Ligands: Design and Synthesis of Pseudopeptides and Peptidomimetics. Aline Moulin , Luc Brunel , Pascal Verdié , Laurent Gavara , Jean Martinez Current Chemical Biology, 2013, 3 (7), pp.000-000. ⟨10.2174/2212796807999131128125920⟩ Journal articles hal-01089074v1
	Biophysical characterization of a binding site for TLQP-21, a naturally occurring peptide which induces resistance to obesity V. Cassina , A. Torsello , A. Tempestini , D. Salerno , D. Brogioli Biochimica et Biophysica Acta:Biomembranes, 2013, 1828 (2), pp.455-460. ⟨10.1016/j.bbamem.2012.10.023⟩ Journal articles hal-02871939v1
	The pipecolic linker—an acid-labile handle for derivatization of secondary amines on a solid-support. Part 3 Paweł Zajdel , Nicolas Masurier , Vittorio Canale , Pascal Verdie , Muriel Amblard Tetrahedron Letters, 2013, 54 (8), pp.998-1002. ⟨10.1016/j.tetlet.2012.12.036⟩ Journal articles hal-03563368v1
	High Constitutive Activity Is an Intrinsic Feature of Ghrelin Receptor Protein. A study with a functional monomeric GHS-R1a receptor reconstitued in lipid discs Marjorie Damian , Jacky Marie , Jean-Philippe Leyris , Jean-Alain Fehrentz , Pascal Verdie Journal of Biological Chemistry, 2012, 287 (6), pp.3630-3641. ⟨10.1074/jbc.M111.288324⟩ Journal articles hal-00713589v1
	From Polyesters to Polyamides Via ON Acyl Migration: An Original Multi-Transfer Reaction Julien Tailhades , Sébastien Blanquer , Benjamin Nottelet , Jean Coudane , Gilles Subra Macromolecular Rapid Communications, 2011, 32 (12), pp.876 - 880. ⟨10.1002/marc.201100235⟩ Journal articles hal-01833151v1
	Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a Jean-Philippe Leyris , Thomas Roux , Eric Trinquet , Pascal Verdié , Jean-Alain Fehrentz Analytical Biochemistry, 2011, 408, pp.253-262. ⟨10.1016/j.ab.2010.09.030⟩ Journal articles hal-00534262v1
	Oxyfold: A simple and efficient solid-supported reagent for disulfide bond formation P. Verdié , Luisa Ronga , M. Cristau , M. Amblard , S. Cantel Chemistry - An Asian Journal, 2011, 6 (9), pp.2382-2389. ⟨10.1002/asia.201100202⟩ Journal articles hal-01563744v1
	Sequencing Lys-N Proteolytic Peptides by ESI and MALDI Tandem Mass Spectrometry Mathieu Dupré , Sonia Cantel , Pascal Verdié , Jean Martinez , Christine Enjalbal Journal of The American Society for Mass Spectrometry, 2011, 22, pp.265-279. ⟨10.1007/s13361-010-0022-7⟩ Journal articles hal-00580756v1
	cis-Apa: A Practical Linker for the Microwave-Assisted Preparation of Cyclic Pseudopeptides via RCM Cyclative Cleavage Alice Baron , Pascal Verdié , Jean Martinez , Frédéric Lamaty Journal of Organic Chemistry, 2011, 76 (3), pp.766-772. ⟨10.1021/jo101629v⟩ Journal articles hal-00564151v1
	Sulfonamides with the N-alkyl-N'-dialkylguaninidine moiety as 5-HT7 receptor ligands Pawel Zajdel , Gilles Subra , Pascal Verdié , Ewa Gabzdyl , Andrzej J. Bojarski Bioorganic and Medicinal Chemistry Letters, 2009, 19, pp.4827-4831. ⟨10.1016/j.bmcl.2009.06.038⟩ Journal articles hal-00411218v1
	The influence of an ethylene spacer of the 5-HT1A and 5-HT2A receptor affinity of arylpiperazine derivatives of amides with N-acylated amino acids and 3-differently substituted pyrrolidine-2,5-diones Pawel Zajdel , Gilles Subra , Pascal Verdie , Andrzej J. Bojarski , Beata Duszynska European Journal of Medicinal Chemistry, 2009, 44, pp.800-808. ⟨10.1016/j.ejmech.2008.05.021⟩ Journal articles hal-00411106v1
	Valuable Versatile Reactivity of Thiaisatoic Anhydrides: Expedient Solid-Phases Synthesis of Thieno[1,4]Diazepine-2,5-diones Yann Brouillette , Pascal Verdié , Jean Martinez SYNLETT, 2008, 15, pp.2360-2364. ⟨10.1055/s-2008-1078210⟩ Journal articles hal-00341629v1
	Solid-Phase Synthesis of 4-methylcarboxy-1,4-benzodiazepine-2,5-diones Pascal Verdié , Gilles Subra , Marie-Christine Averlant-Petit , Muriel Amblard , Jean Martinez Journal of Combinatorial Chemistry, 2008, 10 (6), pp.869-874. ⟨10.1021/cc800085d⟩ Journal articles hal-00411034v1
	Solid-phase synthesis of 5-arylhistidines via a microwave-assisted Suzuki-Miyaura cross-coupling Vanessa Cerezo , Muriel Amblard , Jean Martinez , Pascal Verdié , Marta Planas Tetrahedron, 2008, 64, pp.10538-10545. ⟨10.1016/j.tet.2008.08.077⟩ Journal articles hal-00411015v1

	Fast and cost-efficient approaches for 17O-isotopic labeling of carboxylic groups in biomolecules: from free amino acids to peptide chains Jessica Špačková , Ieva Goldberga , Rishit Yadav , Guillaume Cazals , Aurélien Lebrun 2022 Preprints, Working Papers, ... hal-03846579v1

Pascal VERDIE

Publications

Targeting a lineage-specific PI3Kɣ–Akt signaling module in acute myeloid leukemia using a heterobifunctional degrader molecule

Amelogenin-Derived Peptide (ADP-5) Hydrogel for Periodontal Regeneration: An In Vitro Study on Periodontal Cells Cytocompatibility, Remineralization and Inflammatory Profile

Fast and Cost‐Efficient 17 O‐Isotopic Labeling of Carboxylic Groups in Biomolecules: From Free Amino Acids to Peptide Chains

The C-terminal pentapeptide acein analogue (JMV3315) stimulates dopamine release in the brain

Structural insights into recognition of chemokine receptors by Staphylococcus aureus leukotoxins

Peptide-guided self-assembly of polyethylene glycol-b-poly(ε-caprolactone-g-peptide) block copolymers

Potent Lys Patch-containing Stapled Peptides Targeting PCSK9

Active Targeted Nanoemulsions for Repurposing of Tegaserod in Alzheimer’s Disease Treatment

JMV5656, a short synthetic derivative of TLQP-21, alleviates acid-induced lung injury and fibrosis in mice

Star-poly(lactide)-peptide hybrid networks as bioactive materials

Site-specific grafting on titanium surfaces with hybrid temporin antibacterial peptides

STIM Proteins and Orai Ca2+ Channels Are Involved in the Intracellular Pathways Activated by TLQP-21 in RAW264.7 Macrophages

Study of the Tissue Distribution of TLQP-21 in Mice Using [18F]JMV5763, a Radiolabeled Analog Prepared via [18F]Aluminum Fluoride Chelation Chemistry

[Erratum for] "Palatability Can Drive Feeding Independent of AgRP Neurons"

JMV5656, A Novel Derivative of TLQP-21, Triggers the Activation of a Calcium-Dependent Potassium Outward Current in Microglial Cells

Peptide synthesis: ball-milling, in solution, or on solid support, what is the best strategy?

Pharmacological and Biochemical Characterization of TLQP-21 Activation of a Binding Site on CHO Cells

Sol-gel synthesis of collagen-inspired peptide hydrogel

Systemic Delivery of Tumor-Targeted Bax-Derived Membrane-Active Peptides for the Treatment of Melanoma Tumors in a Humanized SCID Mouse Model

Bioactive peptides grafted silicone dressings: A simple and specific method

A switchable stapled peptide

Solid-Supported Synthesis and 5-HT 7 /5-HT 1A Receptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1 H )-one

Palatability Can Drive Feeding Independent of AgRP Neurons

Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling

N- and O-acetylation of threonine residues in the context of proteomics.

Solid-supported synthesis, molecular modeling, and biological activity of long-chain arylpiperazine derivatives with cyclic amino acid amide fragments as 5-HT7 and 5-HT1A receptor ligands

Microwave-Mediated Reduction of Disulfide Bridges with Supported (Tris(2-carboxyethyl)phosphine) as Resin-Bound Reducing Agent

How ligands and signalling proteins affect G-protein-coupled receptors' conformational landscape

Supported oligomethionine sulfoxide and Ellman's reagent for cysteine bridges formation

Heating and microwave assisted SPPS of C-terminal acid peptides on trityl resin: The truth behind the yield

Rapid sensing of circulating ghrelin by hypothalamic appetite-modifying neurons.

Heterodimerization with Its Splice Variant Blocks the Ghrelin Receptor 1a in a Non-signaling Conformation

Ghrelin Receptor Ligands: Design and Synthesis of Pseudopeptides and Peptidomimetics.

Biophysical characterization of a binding site for TLQP-21, a naturally occurring peptide which induces resistance to obesity

The pipecolic linker—an acid-labile handle for derivatization of secondary amines on a solid-support. Part 3

High Constitutive Activity Is an Intrinsic Feature of Ghrelin Receptor Protein. A study with a functional monomeric GHS-R1a receptor reconstitued in lipid discs

From Polyesters to Polyamides Via ON Acyl Migration: An Original Multi-Transfer Reaction

Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a

Oxyfold: A simple and efficient solid-supported reagent for disulfide bond formation

Sequencing Lys-N Proteolytic Peptides by ESI and MALDI Tandem Mass Spectrometry

cis-Apa: A Practical Linker for the Microwave-Assisted Preparation of Cyclic Pseudopeptides via RCM Cyclative Cleavage

Sulfonamides with the N-alkyl-N'-dialkylguaninidine moiety as 5-HT7 receptor ligands

The influence of an ethylene spacer of the 5-HT1A and 5-HT2A receptor affinity of arylpiperazine derivatives of amides with N-acylated amino acids and 3-differently substituted pyrrolidine-2,5-diones

Valuable Versatile Reactivity of Thiaisatoic Anhydrides: Expedient Solid-Phases Synthesis of Thieno[1,4]Diazepine-2,5-diones

Solid-Phase Synthesis of 4-methylcarboxy-1,4-benzodiazepine-2,5-diones

Solid-phase synthesis of 5-arylhistidines via a microwave-assisted Suzuki-Miyaura cross-coupling

Fast and cost-efficient approaches for 17O-isotopic labeling of carboxylic groups in biomolecules: from free amino acids to peptide chains