Pascal VERDIE

53
Documents
Affiliation actuelle
  • Université de Montpellier (UM)
Identifiants chercheurs

Publications

Publications

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Development of Low-Nanomolar Covalent Epoxide Inhibitors of Tubulin Detyrosinating Enzymes VASH1&2

Anthony Feral , Guillaume Marcellin , Yoann Lannay , Camille Hennebert , Yazid Souf et al.

Journal of Medicinal Chemistry, 2025, 68 (17), pp.18335-18355. ⟨10.1021/acs.jmedchem.5c00980⟩

Article dans une revue hal-05328434v1

Study of the impact of histidine configuration and position on analytical separation of tripeptides

Ella Tyson , Elodie Carretero , Pascal Verdié , Christine Enjalbal , Yoann Ladner

Journal of Chromatography A, 2025, 1759, pp.466202. ⟨10.1016/j.chroma.2025.466202⟩

Article dans une revue hal-05184470v1
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Targeting a lineage-specific PI3Kɣ–Akt signaling module in acute myeloid leukemia using a heterobifunctional degrader molecule

Lois Kelly , Justine Rutter , Kevin Lin , Frank Ling , Matthieu Duchmann et al.

Nature Cancer, In press, Online ahead of print. ⟨10.1038/s43018-024-00782-5⟩

Article dans une revue hal-04598240v1
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Amelogenin-Derived Peptide (ADP-5) Hydrogel for Periodontal Regeneration: An In Vitro Study on Periodontal Cells Cytocompatibility, Remineralization and Inflammatory Profile

Nina Attik , Xavier Garric , Audrey Bethry , Gilles Subra , Charlène Chevalier et al.

Journal of Functional Biomaterials, 2023, 14 (2), pp.53. ⟨10.3390/jfb14020053⟩

Article dans une revue hal-04628797v1

The C-terminal pentapeptide acein analogue (JMV3315) stimulates dopamine release in the brain

Charlène Lucas-Valmalle , Gilles Subra , Pascal Verdié , Marie-Lou Kemel , Valérie Daugé et al.

Australian Journal of Chemistry, 2023, 76 (8), pp.448-454. ⟨10.1071/CH22232⟩

Article dans une revue hal-04604961v1
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Fast and Cost‐Efficient 17 O‐Isotopic Labeling of Carboxylic Groups in Biomolecules: From Free Amino Acids to Peptide Chains

Jessica Špačková , Ieva Goldberga , Rishit Yadav , Guillaume Cazals , Aurélien Lebrun et al.

Chemistry - A European Journal, 2023, 29 (10), pp.e202203014. ⟨10.1002/chem.202203014⟩

Article dans une revue hal-04002744v1
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Structural insights into recognition of chemokine receptors by Staphylococcus aureus leukotoxins

Paul Lambey , Omolade Otun , Xiaojing Cong , François Hoh , Luc Brunel et al.

eLife, 2022, 11, pp.e72555. ⟨10.7554/eLife.72555⟩

Article dans une revue hal-03754372v1
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Peptide-guided self-assembly of polyethylene glycol-b-poly(ε-caprolactone-g-peptide) block copolymers

Ayman El Jundi , Matthias Mayor , Enrique Folgado , Chaimaa Gomri , Belkacem Tarek Benkhaled et al.

European Polymer Journal, 2022, 176, pp.111386. ⟨10.1016/j.eurpolymj.2022.111386⟩

Article dans une revue hal-04065895v1
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Potent Lys Patch-containing Stapled Peptides Targeting PCSK9

Kevin Bourbiaux , Baptiste Legrand , Pascal Verdié , Sergio Mallart , Géraldine Manette et al.

Journal of Medicinal Chemistry, 2021, 64 (15), pp.10834-10848. ⟨10.1021/acs.jmedchem.0c02051⟩

Article dans une revue hal-03371411v1
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Active Targeted Nanoemulsions for Repurposing of Tegaserod in Alzheimer’s Disease Treatment

Line Séguy , Léna Guyon , Manon Maurel , Pascal Verdié , Audrey Davis et al.

Pharmaceutics, 2021, 13 (10), pp.1626. ⟨10.3390/pharmaceutics13101626⟩

Article dans une revue hal-04570312v1
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Star-poly(lactide)-peptide hybrid networks as bioactive materials

L.V. Arsenie , Coline Pinese , Audrey Bethry , L. Valot , P. Verdie et al.

European Polymer Journal, 2020, 139, pp.109990 -. ⟨10.1016/j.eurpolymj.2020.109990⟩

Article dans une revue hal-03491991v1

JMV5656, a short synthetic derivative of TLQP-21, alleviates acid-induced lung injury and fibrosis in mice

Vanessa Zambelli , Laura Rizzi , Paolo Delvecchio , Elena Bresciani , Laura Molteni et al.

Pulmonary Pharmacology and Therapeutics, 2020, 62, pp.101916. ⟨10.1016/j.pupt.2020.101916⟩

Article dans une revue hal-04549706v1

A Short SOX9 Peptide Mimics SOX9 Tumor Suppressor Activity and Is Sufficient to Inhibit Colon Cancer Cell Growth

Philippe Blache , Lucile Canterel-Thouennon , Muriel Busson , Pascal Verdié , Gilles Subra et al.

Molecular Cancer Therapeutics, 2019, 18 (8), pp.1386-1395. ⟨10.1158/1535-7163.MCT-18-1149⟩

Article dans une revue hal-04830489v1

Site-specific grafting on titanium surfaces with hybrid temporin antibacterial peptides

Nicolas Masurier , Jean-Baptiste Tissot , Douae Boukhriss , Said Jebors , Coline Pinese et al.

Journal of materials chemistry‎ B, 2018, 6 (12), pp.1782 - 1790. ⟨10.1039/c8tb00051d⟩

Article dans une revue hal-01742222v1
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STIM Proteins and Orai Ca2+ Channels Are Involved in the Intracellular Pathways Activated by TLQP-21 in RAW264.7 Macrophages

Laura Molteni , Laura Rizzi , Elena Bresciani , Ramona Meanti , Jean-Alain Fehrentz et al.

Frontiers in Pharmacology, 2018, 9, ⟨10.3389/fphar.2018.01386⟩

Article dans une revue hal-02871099v1
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Study of the Tissue Distribution of TLQP-21 in Mice Using [18F]JMV5763, a Radiolabeled Analog Prepared via [18F]Aluminum Fluoride Chelation Chemistry

Elia Turolla , Silvia Valtorta , Elena Bresciani , Jean-Alain Fehrentz , Liliana Giuliano et al.

Frontiers in Pharmacology, 2018, 9, ⟨10.3389/fphar.2018.01274⟩

Article dans une revue hal-02871096v1
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Peptide synthesis: ball-milling, in solution, or on solid support, what is the best strategy?

Ophélie Maurin , Pascal Verdié , Gilles Subra , Frédéric Lamaty , Jean Martinez et al.

Beilstein Journal of Organic Chemistry, 2017, 13, pp.2087-2093. ⟨10.3762/bjoc.13.206⟩

Article dans une revue hal-02336152v1

Bioactive peptides grafted silicone dressings: A simple and specific method

Coline Pinese , Said Jebors , Pierre-Emmanuel Stoebner , Vincent Humblot , Pascal Verdié et al.

Materials Today Chemistry, 2017, 4, pp.73-83. ⟨10.1016/j.mtchem.2017.02.007⟩

Article dans une revue hal-01496701v1
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Systemic Delivery of Tumor-Targeted Bax-Derived Membrane-Active Peptides for the Treatment of Melanoma Tumors in a Humanized SCID Mouse Model

Anastassia Karageorgis , Michaël Claron , Romain Jugé , Caroline Aspord , Fabien Thoreau et al.

Molecular Therapy, 2017, 25 (2), pp.534-546. ⟨10.1016/j.ymthe.2016.11.002⟩

Article dans une revue hal-02000186v1
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Sol-gel synthesis of collagen-inspired peptide hydrogel

Cécile Echalier , Said Jebors , Guillaume Laconde , Luc Brunel , Pascal Verdié et al.

Materials Today, 2017, 20 (2), pp.59-66. ⟨10.1016/j.mattod.2017.02.001⟩

Article dans une revue hal-01516237v1

[Erratum for] "Palatability Can Drive Feeding Independent of AgRP Neurons

Raphael Georges Denis , Aurélie Joly-Amado , Emily Webber , Fanny Langlet , Marie Schaeffer et al.

Cell Metabolism, 2017, 25 (4), pp.975. ⟨10.1016/j.cmet.2017.03.001⟩

Article dans une revue hal-02067393v1
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Pharmacological and Biochemical Characterization of TLQP-21 Activation of a Binding Site on CHO Cells

Laura Molteni , Laura Rizzi , Elena Bresciani , Roberta Possenti , Pamela Petrocchi Passeri et al.

Frontiers in Pharmacology, 2017, 8, pp.167. ⟨10.3389/fphar.2017.00167⟩

Article dans une revue hal-02871330v1
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JMV5656, A Novel Derivative of TLQP-21, Triggers the Activation of a Calcium-Dependent Potassium Outward Current in Microglial Cells

Ilaria Rivolta , Anna Binda , Laura Molteni , Laura Rizzi , Elena Bresciani et al.

Frontiers in Cellular Neuroscience, 2017, 11, pp.41. ⟨10.3389/fncel.2017.00041⟩

Article dans une revue hal-02871317v1

A switchable stapled peptide

Aleksandra Kalistratova , Baptiste Legrand , Pascal Verdié , Emilia Naydenova , Muriel Amblard et al.

Journal of Peptide Science, 2016, 22 (3), pp.143-148. ⟨10.1002/psc.2851⟩

Article dans une revue istex hal-03564342v1

Solid-Supported Synthesis and 5-HT 7 /5-HT 1A Receptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1 H )-one

Katarzyna Grychowska , Nicolas Masurier , Pascal Verdié , Grzegorz Satała , Andrzej Bojarski et al.

Chemical Biology and Drug Design, 2015, 86 (4), pp.697-703. ⟨10.1111/cbdd.12539⟩

Article dans une revue istex hal-03564059v1
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Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling

Céline M'Kadmi , Jean-Philippe Leyris , Lauriane Onfroy , Céline Galés , Aude Saulière et al.

Journal of Biological Chemistry, 2015, 290 (45), pp.27021-27039. ⟨10.1074/jbc.M115.659250⟩

Article dans une revue hal-03564155v1
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Palatability Can Drive Feeding Independent of AgRP Neurons

Raphael Georges Denis , Aurélie Joly-Amado , Emily Webber , Fanny Langlet , Marie Schaeffer et al.

Cell Metabolism, 2015, 22 (4), pp.646-657. ⟨10.1016/j.cmet.2015.07.011⟩

Article dans une revue hal-02067347v1

N- and O-acetylation of threonine residues in the context of proteomics.

Jean-Baptiste Boyer , Alain Dedieu , J. Armengaud , Pascal Verdié , Gilles Subra et al.

Journal of Proteomics, 2014, 108, pp.369-372. ⟨10.1016/j.jprot.2014.06.005⟩

Article dans une revue istex hal-01025681v1

Solid-supported synthesis, molecular modeling, and biological activity of long-chain arylpiperazine derivatives with cyclic amino acid amide fragments as 5-HT7 and 5-HT1A receptor ligands

Vittorio Canale , Paweł Guzik , Rafał Kurczab , Pascal Verdie , Grzegorz Satała et al.

European Journal of Medicinal Chemistry, 2014, 78, pp.10-22. ⟨10.1016/j.ejmech.2014.03.005⟩

Article dans une revue hal-03563396v1

How ligands and signalling proteins affect G-protein-coupled receptors' conformational landscape

Sophie Mary , Jean-Alain Fehrentz , Marjorie Damian , Pascal Verdie , Jean Martinez et al.

Biochemical Society Transactions, 2013, 41 (1), pp.144-147. ⟨10.1042/BST20120267⟩

Article dans une revue hal-02871941v1

Microwave-Mediated Reduction of Disulfide Bridges with Supported (Tris(2-carboxyethyl)phosphine) as Resin-Bound Reducing Agent

Guillaume Miralles , Pascal Verdié , Karine Puget , Amélie Maurras , Jean Martinez et al.

ACS Combinatorial Science, 2013, 15 (4), pp.169-173. ⟨10.1021/co300104k⟩

Article dans une revue hal-03563025v1

Rapid sensing of circulating ghrelin by hypothalamic appetite-modifying neurons.

Marie Schaeffer , Fanny Langlet , Chrystel Lafont , François Molino , David J Hodson et al.

Proceedings of the National Academy of Sciences of the United States of America, 2013, 110 (4), pp.1512-7. ⟨10.1073/pnas.1212137110⟩

Article dans une revue hal-00796900v1

Heating and microwave assisted SPPS of C-terminal acid peptides on trityl resin: The truth behind the yield

Cécile Echalier , Soultan Al-Halifa , Aude Kreiter , Christine Enjalbal , Pierre Sanchez et al.

Amino Acids, 2013, 45 (6), pp.1395-1403. ⟨10.1007/s00726-013-1604-z⟩

Article dans une revue istex hal-01563742v1

Ghrelin Receptor Ligands: Design and Synthesis of Pseudopeptides and Peptidomimetics.

Aline Moulin , Luc Brunel , Pascal Verdié , Laurent Gavara , Jean Martinez et al.

Current Chemical Biology, 2013, 3 (7), pp.000-000. ⟨10.2174/2212796807999131128125920⟩

Article dans une revue istex hal-01089074v1
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Heterodimerization with Its Splice Variant Blocks the Ghrelin Receptor 1a in a Non-signaling Conformation

Sophie Mary , Jean-Alain Fehrentz , Marjorie Damian , Gérald Gaibelet , Hélène Orcel et al.

Journal of Biological Chemistry, 2013, 288 (34), pp.24656-24665. ⟨10.1074/jbc.M113.453423⟩

Article dans une revue hal-02871944v1

Biophysical characterization of a binding site for TLQP-21, a naturally occurring peptide which induces resistance to obesity

V. Cassina , A. Torsello , A. Tempestini , D. Salerno , D. Brogioli et al.

Biochimica et Biophysica Acta:Biomembranes, 2013, 1828 (2), pp.455-460. ⟨10.1016/j.bbamem.2012.10.023⟩

Article dans une revue hal-02871939v1

The pipecolic linker—an acid-labile handle for derivatization of secondary amines on a solid-support. Part 3

Paweł Zajdel , Nicolas Masurier , Vittorio Canale , Pascal Verdie , Muriel Amblard et al.

Tetrahedron Letters, 2013, 54 (8), pp.998-1002. ⟨10.1016/j.tetlet.2012.12.036⟩

Article dans une revue istex hal-03563368v1

Supported oligomethionine sulfoxide and Ellman's reagent for cysteine bridges formation

Luisa Ronga , Pascal Verdié , Pierre Sanchez , Christine Enjalbal , Amélie Maurras et al.

Amino Acids, 2013, 44 (2), pp.733-742. ⟨10.1007/s00726-012-1397-5⟩

Article dans une revue istex hal-01563741v1
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High Constitutive Activity Is an Intrinsic Feature of Ghrelin Receptor Protein. A study with a functional monomeric GHS-R1a receptor reconstitued in lipid discs

Marjorie Damian , Jacky Marie , Jean-Philippe Leyris , Jean-Alain Fehrentz , Pascal Verdie et al.

Journal of Biological Chemistry, 2012, 287 (6), pp.3630-3641. ⟨10.1074/jbc.M111.288324⟩

Article dans une revue hal-00713589v1

Oxyfold: A simple and efficient solid-supported reagent for disulfide bond formation

P. Verdié , Luisa Ronga , M. Cristau , M. Amblard , S. Cantel et al.

Chemistry - An Asian Journal, 2011, 6 (9), pp.2382-2389. ⟨10.1002/asia.201100202⟩

Article dans une revue istex hal-01563744v1

cis-Apa: A Practical Linker for the Microwave-Assisted Preparation of Cyclic Pseudopeptides via RCM Cyclative Cleavage

Alice Baron , Pascal Verdié , Jean Martinez , Frédéric Lamaty

Journal of Organic Chemistry, 2011, 76 (3), pp.766-772. ⟨10.1021/jo101629v⟩

Article dans une revue hal-00564151v1
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From Polyesters to Polyamides Via ON Acyl Migration: An Original Multi-Transfer Reaction

Julien Tailhades , Sébastien Blanquer , Benjamin Nottelet , Jean Coudane , Gilles Subra et al.

Macromolecular Rapid Communications, 2011, 32 (12), pp.876 - 880. ⟨10.1002/marc.201100235⟩

Article dans une revue istex hal-01833151v1

Sequencing Lys-N Proteolytic Peptides by ESI and MALDI Tandem Mass Spectrometry

Mathieu Dupré , Sonia Cantel , Pascal Verdié , Jean Martinez , Christine Enjalbal

Journal of The American Society for Mass Spectrometry, 2011, 22, pp.265-279. ⟨10.1007/s13361-010-0022-7⟩

Article dans une revue hal-00580756v1

Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a

Jean-Philippe Leyris , Thomas Roux , Eric Trinquet , Pascal Verdié , Jean-Alain Fehrentz et al.

Analytical Biochemistry, 2011, 408, pp.253-262. ⟨10.1016/j.ab.2010.09.030⟩

Article dans une revue istex hal-00534262v1

Sulfonamides with the N-alkyl-N'-dialkylguaninidine moiety as 5-HT7 receptor ligands

Pawel Zajdel , Gilles Subra , Pascal Verdié , Ewa Gabzdyl , Andrzej J. Bojarski et al.

Bioorganic and Medicinal Chemistry Letters, 2009, 19, pp.4827-4831. ⟨10.1016/j.bmcl.2009.06.038⟩

Article dans une revue hal-00411218v1

The influence of an ethylene spacer of the 5-HT1A and 5-HT2A receptor affinity of arylpiperazine derivatives of amides with N-acylated amino acids and 3-differently substituted pyrrolidine-2,5-diones

Pawel Zajdel , Gilles Subra , Pascal Verdie , Andrzej J. Bojarski , Beata Duszynska et al.

European Journal of Medicinal Chemistry, 2009, 44, pp.800-808. ⟨10.1016/j.ejmech.2008.05.021⟩

Article dans une revue hal-00411106v1

Solid-phase synthesis of 5-arylhistidines via a microwave-assisted Suzuki-Miyaura cross-coupling

Vanessa Cerezo , Muriel Amblard , Jean Martinez , Pascal Verdié , Marta Planas et al.

Tetrahedron, 2008, 64, pp.10538-10545. ⟨10.1016/j.tet.2008.08.077⟩

Article dans une revue istex hal-00411015v1

Valuable Versatile Reactivity of Thiaisatoic Anhydrides: Expedient Solid-Phases Synthesis of Thieno[1,4]Diazepine-2,5-diones

Yann Brouillette , Pascal Verdié , Jean Martinez

SYNLETT, 2008, 15, pp.2360-2364. ⟨10.1055/s-2008-1078210⟩

Article dans une revue hal-00341629v1

Solid-Phase Synthesis of 4-methylcarboxy-1,4-benzodiazepine-2,5-diones

Pascal Verdié , Gilles Subra , Marie-Christine Averlant-Petit , Muriel Amblard , Jean Martinez

Journal of Combinatorial Chemistry, 2008, 10 (6), pp.869-874. ⟨10.1021/cc800085d⟩

Article dans une revue hal-00411034v1

Marrying sol-gel and peptide chemistry to design bioactive materials

Gilles Subra , Cécile Echalier , Ahmad Mehdi , Margaux Clavié , Mathilde Guerin et al.

Turku Biomaterials Days 2024, Oct 2024, Turku, Finland

Communication dans un congrès hal-04891598v1

Designing biomimetic materials from silylated amino acids, peptides and proteins.

Gilles Subra , Cécile Echalier , Margaux Clavié , Pascal Verdié , Muriel Amblard et al.

European Peptide Synthesis Conference 2023, Feb 2023, Leeds, United Kingdom

Communication dans un congrès hal-04891483v1